
GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(249 productos)
- Receptor adrenérgico(3.018 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(158 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(217 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(23 productos)
- Receptor de glucagón(194 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(327 productos)
- PAFR(14 productos)
- PKA(60 productos)
- Receptor S1P(18 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5983 productos de "GPCR / proteína G"
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Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59Propafenone
CAS:Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.Fórmula:C21H27NO3Pureza:99.02%Forma y color:SolidPeso molecular:341.44Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Palonosetron hydrochloride
CAS:Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Forma y color:White SolidPeso molecular:332.87Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Forma y color:Colorless To Pink SolidPeso molecular:495.53Ref: TM-T1504
5mg34,00€10mg50,00€25mg73,00€50mg92,00€100mg99,00€200mg126,00€1500mg267,00€1mL*10mM (DMSO)35,00€Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:99.87% - 99.93%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Forma y color:SolidPeso molecular:260.3PF429242 dihydrochloride
CAS:PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Fórmula:C25H37Cl2N3O2Pureza:99.68%Forma y color:SolidPeso molecular:482.49Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Fórmula:C15H18ClNS2Pureza:99.97%Forma y color:SolidPeso molecular:311.89Pranazepide
CAS:Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.Fórmula:C26H19FN4O2Pureza:97.43% - 99.53%Forma y color:SolidPeso molecular:438.45Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Fórmula:C17H19N3Pureza:99.98%Forma y color:SolidPeso molecular:265.35Vapreotide acetate
CAS:Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).Fórmula:C59H74N12O11S2Pureza:99.89%Forma y color:SolidPeso molecular:1191.42GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Fórmula:C30H35N3O3Pureza:98.94% - 99.29%Forma y color:SolidPeso molecular:485.62Ref: TM-T11463
2mg39,00€5mg58,00€10mg92,00€25mg177,00€50mg289,00€100mg462,00€200mg655,00€1mL*10mM (DMSO)63,00€Atomoxetine hydrochloride
CAS:Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Fórmula:C17H22ClNOPureza:99.86%Forma y color:White SolidPeso molecular:291.82Tolnaftate
CAS:Tolnaftate (NP-27) is a synthetic antifungal agent.Fórmula:C19H17NOSPureza:98.85%Forma y color:White PowderPeso molecular:307.41(-)-GSK598809 hydrochloride
CAS:(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.
Fórmula:C22H24ClF4N5OSPureza:98.36%Forma y color:SoildPeso molecular:517.97Prostaglandin E1
CAS:Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.Fórmula:C20H34O5Pureza:99.78% - >99.99%Forma y color:SolidPeso molecular:354.48Ref: TM-T1626
1mg34,00€5mg63,00€10mg94,00€25mg167,00€50mg276,00€100mg415,00€200mg595,00€1mL*10mM (DMSO)50,00€Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Forma y color:Crystal PowderPeso molecular:435.31Ramelteon
CAS:Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.Fórmula:C16H21NO2Pureza:97.21% - 99.92%Forma y color:Crystalline SolidPeso molecular:259.34Ref: TM-T1463
2mg42,00€5mg62,00€10mg84,00€25mg129,00€50mg192,00€100mg309,00€500mg485,00€1mL*10mM (DMSO)67,00€Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Fórmula:C12H13NO3Pureza:99.88% - 99.89%Forma y color:White Crystalline Or Crystalline PowdePeso molecular:219.24
