
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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3-Bromopyruvic acid
CAS :<p>3-Bromopyruvic acid (Hexokinase II Inhibitor II, 3-BP) is a hexokinase II inhibitor with Ki of 2.4 mM for glycolysis/hexokinase inhibition.</p>Formule :C3H3BrO3Degré de pureté :95% - 99.644%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :166.96Fangchinoline
CAS :<p>Fangchinoline (Tetrandrine B) is extracted from Stephania tetrandra S. Moore.</p>Formule :C37H40N2O6Degré de pureté :99.86% - >99.99%Couleur et forme :SolidMasse moléculaire :608.72Lexibulin
CAS :<p>Lexibulin (CYT-997)(CYT-997) is a potent tubulin polymerization inhibitor (IC50: 10-100 nM, in Y cell lines).</p>Formule :C24H30N6O2Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :434.53Cucurbitacin IIb
CAS :<p>Cucurbitacin IIb is an active ingredient in Hemsleyadine, used to treat dysentery and other infections; it has anti-inflammatory effects.</p>Formule :C30H48O7Degré de pureté :98.66% - >99.99%Couleur et forme :SolidMasse moléculaire :520.7Poncirin
CAS :<p>Poncirin inhibits human gastric cancer cell growth and prevents fat formation while boosting bone density and improving structure in osteoporosis mice.</p>Formule :C28H34O14Degré de pureté :99.89% - 99.92%Couleur et forme :SolidMasse moléculaire :594.56Entinostat
CAS :<p>Entinostat (MS-275) is an HDAC class I with oral activity. Entinostat has antitumor activity. Cost-effective and quality-assured.</p>Formule :C21H20N4O3Degré de pureté :98% - 99.74%Couleur et forme :SolidMasse moléculaire :376.41Ligustilide
CAS :<p>3-Butylidene-4,5-dihydrophthalide is an effective constituent extracted from Angelica sinensis.</p>Formule :C12H14O2Degré de pureté :96.03% - 98.14%Couleur et forme :Yellow Brown PowderMasse moléculaire :190.24Dioscin
CAS :<p>Dioscin (Collettiside III) is a saponin with antitumor activities.</p>Formule :C45H72O16Degré de pureté :99.85% - 99.87%Couleur et forme :SolidMasse moléculaire :869.04JIB-04
CAS :<p>JIB-04 (NSC 693627) is a pan-selective Jumonji histone demethylase inhibitor.</p>Formule :C17H13ClN4Degré de pureté :98.02% - 98.87%Couleur et forme :SolidMasse moléculaire :308.76Tebufenozide
CAS :<p>Tebufenozide is a novel nonsteroidal ecdysone agonist. It shows good efficacy and playing an increasingly important role in the control of Lepidopteran pests.</p>Formule :C22H28N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.47Y-320
CAS :<p>Y-320 is a new phenylpyrazoleanilide immunomodulator.</p>Formule :C27H29ClN6O2Degré de pureté :98% - 99.64%Couleur et forme :SolidMasse moléculaire :505.01PIK-75 hydrochloride
CAS :<p>PIK-75 hydrochloride (PIK-75 HCl) is a p110α inhibitor, isoform-specific mutants at Ser773, and potently inhibits DNA-PK with IC50 of 2 nM in cell-free assay.</p>Formule :C16H14BrN5O4S·HClDegré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :488.745-Aminolevulinic acid hydrochloride
CAS :<p>5-Aminolevulinic acid hydrochloride (5-ALA) serves as an intermediate in the body's heme biosynthesis and is the universal precursor of tetrapyrroles.</p>Formule :C5H10ClNO3Degré de pureté :98% - 99.97%Couleur et forme :White To Pale Yellow Crystals OrMasse moléculaire :167.59Pulsatilla saponin D
CAS :<p>Pulsatilla saponin D (Hederacolchiside A) may prevent cancer, hindering cancer cell growth through cell cycle arrest and apoptosis.</p>Formule :C47H76O17Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :913.1Fludarabine Phosphate
CAS :<p>Fludarabine Phosphate (NSC 312887 Phosphate) is a fluorinated nucleotide antimetabolite analog of the antiviral agent vidarabine with antineoplastic activity.</p>Formule :C10H13FN5O7PDegré de pureté :99.25% - 99.78%Couleur et forme :SolidMasse moléculaire :365.21L-Theanine
CAS :<p>L-Theanine, a unique amino acid from Camellia sinensis tea, induces relaxation without drowsiness.</p>Formule :C7H14N2O3Degré de pureté :99.31% - 99.38%Couleur et forme :White Crystals From Ethanol + Water White Crystalline SolidMasse moléculaire :174.2Glaucocalyxin A
CAS :<p>Glaucocalyxin A improves drug delivery, activates apoptosis, inhibits cell growth, with potential as an antiplatelet agent.</p>Formule :C20H28O4Degré de pureté :99.55% - 99.80%Couleur et forme :SolidMasse moléculaire :332.43Phthalazinone pyrazole
CAS :<p>Phthalazinone pyrazole: a potent, selective oral Aurora-A kinase inhibitor, overexpressed in tumors with oncogenic activity.</p>Formule :C18H15N5ODegré de pureté :97.03%Couleur et forme :SolidMasse moléculaire :317.34Pyroxamide
CAS :<p>Pyroxamide is an histone deacetylases (HDACs) inhibitor with antineoplastic properties ( HDAC1;IC50: 0.1-0.2 μM).</p>Formule :C13H19N3O3Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :265.31Pinoresinol
CAS :<p>Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury</p>Formule :C20H22O6Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :358.391-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea
CAS :<p>SC-1 is a a derivative of the multiple tyrosine kinase inhibitor sorafenib.</p>Formule :C21H13ClF3N3O2Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :431.82-Deoxy-D-glucose
CAS :<p>2-Deoxy-D-glucose (2-DG) is an analog of glucose, an inhibitor of glycolysis.</p>Formule :C6H12O5Degré de pureté :99.31% - ≥98%Couleur et forme :White PowderMasse moléculaire :164.16BX-912
CAS :<p>BX-912 inhibits PDK1 with IC50 of 12 nM; over 10x more selective versus C-Kit, EGFR, PKA, PKC.</p>Formule :C20H23BrN8ODegré de pureté :98.29% - 99.34%Couleur et forme :SolidMasse moléculaire :471.35Supinoxin
CAS :<p>Supinoxin (RX-5902) is an oral anti-cancer drug targeting p68 RNA helicase, inducing apoptosis in TNBC cells (IC50: 10-20nM).</p>Formule :C22H24FN5O4Degré de pureté :99.83% - 99.95%Couleur et forme :SolidMasse moléculaire :441.46GDC-0152
CAS :<p>GDC-0152 is a potent inhibitor of IAPs.</p>Formule :C25H34N6O3SDegré de pureté :97.18% - 99.32%Couleur et forme :SolidMasse moléculaire :498.64CCT128930 hydrochloride
CAS :<p>CCT128930 hydrochloride: Potent AKT inhibitor (IC50=6 nM), 28x selective over PKA, 20x over p70S6K, induces cell cycle arrest & DNA damage.</p>Formule :C18H21Cl2N5Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :378.3Lobaplatin
CAS :<p>Lobaplatin (D-19466) (D-19466) is a diastereometric mixture of platinum(II) complexe.</p>Formule :C9H18N2O3PtDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :397.33L-Asparaginase
CAS :<p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>Formule :NADegré de pureté :97%Couleur et forme :SolidMasse moléculaire :N/ASGI-1776
CAS :<p>SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.</p>Formule :C20H22F3N5ODegré de pureté :99.3% - >99.99%Couleur et forme :SolidMasse moléculaire :405.42Elesclomol
CAS :<p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>Formule :C19H20N4O2S2Degré de pureté :97.17% - 99.51%Couleur et forme :SolidMasse moléculaire :400.52Rilmenidine Phosphate
CAS :<p>Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.</p>Formule :C10H19N2O5PDegré de pureté :99.87% - ≥95%Couleur et forme :SolidMasse moléculaire :278.24HO-3867
CAS :<p>HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.</p>Formule :C28H30F2N2O2Degré de pureté :91.18% - 99.21%Couleur et forme :SolidMasse moléculaire :464.55LRRK2-IN-1
CAS :<p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>Formule :C31H38N8O3Degré de pureté :98% - 98.82%Couleur et forme :SolidMasse moléculaire :570.69kauran-16,17-diol
CAS :<p>Kauran-16,17-diol, a natural diterpenoid product, exhibits anti-tumoral and apoptosis-inducing activities by inhibiting NO production in LPS-induced RAW 264.7</p>Formule :C20H34O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :306.48Daphnetin
CAS :<p>Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),</p>Formule :C9H6O4Degré de pureté :97.47% - 99.8%Couleur et forme :SolidMasse moléculaire :178.14S-trityl-L-Cysteine
CAS :<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Formule :C22H21NO2SDegré de pureté :97.02%Couleur et forme :Almost White To Light Yellow Granular PowderMasse moléculaire :363.47NSC 95397
CAS :<p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>Formule :C14H14O4S2Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :310.39Diffractaic Acid
CAS :<p>Diffractaic Acid (NSC 685595) can inhibit LTB4 biosynthesis in A-23187-stimulated bovine PMNL cells with activity value of 8 μM.</p>Formule :C20H22O7Degré de pureté :99.81% - 99.87%Couleur et forme :SolidMasse moléculaire :374.38SKI II
CAS :<p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>Formule :C15H11ClN2OSDegré de pureté :99.34% - 99.93%Couleur et forme :SolidMasse moléculaire :302.78[6]-Gingerol
CAS :<p>[6]-Gingerol ((S)-(+)-[6]Gingerol), an antioxidant, protects HL-60 cells from oxidative stress. It has protective effects for tumors.</p>Formule :C17H26O4Degré de pureté :98% - 99.66%Couleur et forme :Light Yellow OilinessMasse moléculaire :294.39STF-118804
CAS :<p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 <10 nM.</p>Formule :C25H23N3O4SDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :461.53GSK1059615
CAS :<p>GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.</p>Formule :C18H11N3O2SDegré de pureté :99.3% - ≥95%Couleur et forme :SolidMasse moléculaire :333.36GMB-475
CAS :<p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>Formule :C43H46F3N7O7SDegré de pureté :98.78% - >99.99%Couleur et forme :SolidMasse moléculaire :861.932-Hydroxychalcone
CAS :<p>2-Hydroxychalcone (2-(2-Hydroxybenzal)Acetophenone) can be used as antiparasitic hit compounds when Methoxylated. It inhibits invasion of breast cancer cells.</p>Formule :C15H12O2Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :224.25Pracinostat
CAS :<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Formule :C20H30N4O2Degré de pureté :99.15% - 99.67%Couleur et forme :SolidMasse moléculaire :358.48Phellamurin
CAS :<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Formule :C26H30O11Degré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :518.51Astragalin
CAS :<p>Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid.</p>Formule :C21H20O11Degré de pureté :98.8% - ≥95%Couleur et forme :SolidMasse moléculaire :448.38Dinaciclib
CAS :<p>Dinaciclib (SCH 727965) is a CDK inhibitor that selectively inhibits CDK1, CDK2, CDK5, and CDK9 (IC50 = 3/1/1/4 nM).</p>Formule :C21H28N6O2Degré de pureté :98.21% - 99.75%Couleur et forme :SolidMasse moléculaire :396.49Etidronic acid
CAS :<p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>Formule :C2H8O7P2Degré de pureté :99.93% - ≥95%Couleur et forme :Liquid SyrupMasse moléculaire :206.03Nafamostat mesylate
CAS :<p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>Formule :C19H17N5O2·2CH4O3SDegré de pureté :97.36% - 99.76%Couleur et forme :Tan To Pale Orange SolidMasse moléculaire :539.58KW-2449
CAS :<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Formule :C20H20N4ODegré de pureté :98.43% - 99.69%Couleur et forme :SolidMasse moléculaire :332.4WYC-209
CAS :<p>WYC-209 inhibits proliferation of malignant murine melanoma tumor-repopulating cells (TRCs, IC50: 0.19 uM). It targets the retinoic acid receptor (RAR).</p>Formule :C20H20N2O3SDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :368.45Amentoflavone
CAS :<p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>Formule :C30H18O10Degré de pureté :98.21% - 99.22%Couleur et forme :Odourless Whitish SolidMasse moléculaire :538.46BAY 61-3606
CAS :<p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>Formule :C20H18N6O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :390.4BAY 87-2243
CAS :<p>BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).</p>Formule :C26H26F3N7O2Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :525.53Niraparib tosylate monohyrate
CAS :<p>Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.</p>Formule :C26H30N4O5SDegré de pureté :97.7% - 98.41%Couleur et forme :SolidMasse moléculaire :510.61Sacubitril/Valsartan
CAS :<p>Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for treatment of hypertension and heart failure.</p>Formule :C48H55N6O8Na3·5H2ODegré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :957.99SKI-178
CAS :<p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>Formule :C21H22N4O4Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :394.42Afatinib Dimaleate
CAS :<p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>Formule :C32H33ClFN5O11Degré de pureté :98.11% - 99.87%Couleur et forme :SolidMasse moléculaire :718.08Etretinate
CAS :<p>Etretinate (Ro 10-9359), an oral retinoid, treats psoriasis by promoting cell differentiation and reducing cell growth and inflammation.</p>Formule :C23H30O3Degré de pureté :97.89%Couleur et forme :Crystals Crystalline SolidMasse moléculaire :354.48Sepantronium bromide
CAS :<p>Sepantronium bromide (YM155) is a small-molecule proapoptotic agent with potential antineoplastic activity.</p>Formule :C20H19BrN4O3Degré de pureté :99.68% - 99.85%Couleur et forme :SolidMasse moléculaire :443.26Psoralen
CAS :<p>Psoralen (Ficusin) is a furocoumarin that intercalates with DNA, inhibiting DNA synthesis and cell division.</p>Formule :C11H6O3Degré de pureté :99.3% - 99.87%Couleur et forme :Crystals From Ether Crystalline SolidMasse moléculaire :186.16Clodronate disodium tetrahydrate
CAS :<p>Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.</p>Formule :CH10Cl2Na2O10P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.92CM-272
CAS :<p>CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.</p>Formule :C28H38N4O3Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :478.63Isolongifolene
CAS :<p>Isolongifolene ((-)-Isolongifolene), a tricyclic sesquiterpene isolated from Murraya koenigii, exhibits antioxidant, anti-inflammatory, anticancer, and</p>Formule :C15H24Degré de pureté :90.13% - 99.46%Couleur et forme :Colorless Or Light Yellow LiquidMasse moléculaire :204.35ERK1/2 inhibitor 2
CAS :<p>ERK1/2 inhibitor 2 (ASTX029) is a selective and orally bioavailable ERK 1/2 inhibitor, with potential antineoplastic activity.</p>Formule :C29H31ClFN5O5Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :584.04Trifloxystrobin
CAS :<p>Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.</p>Formule :C20H19F3N2O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :408.37LY294002
CAS :<p>LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).</p>Formule :C19H17NO3Degré de pureté :98% - 99.96%Couleur et forme :Pale Yellow SolidMasse moléculaire :307.34JKE-1674
CAS :<p>JKE-1674 is an orally active glutathione peroxidase 4 (GPX4) inhibitor and the active metabolite of ML-210.Cost-effective and quality-assured.</p>Formule :C20H20Cl2N4O4Degré de pureté :98.02% - 98.4%Couleur et forme :SolidMasse moléculaire :451.3QNZ
CAS :<p>QNZ (EVP4593) (EVP4593) is an effective inhibitor of NF-κB activation and TNF-α production. The IC50 of QNZ for NF-κB and TNF-α is11 nM and 7 nM, respectively.</p>Formule :C22H20N4ODegré de pureté :99.17% - 99.18%Couleur et forme :White SolidMasse moléculaire :356.42Bardoxolone
CAS :<p>Bardoxolone (CDDO) inhibits iNOS, COX-2 in cells; IC50=0.4nM. Reduces ROS/RNS, DNA damage, & cancer growth; triggers apoptosis & boosts antioxidant genes.</p>Formule :C31H41NO4Degré de pureté :97.9% - 98.97%Couleur et forme :SolidMasse moléculaire :491.66Thalidomide-O-C4-NH2 hydrochloride
CAS :<p>Thalidomide-linker 9: a cereblon ligand, E3 ligase conjugate for PROTAC tech.</p>Formule :C17H20ClN3O5Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :381.81Dihydrocapsaicin
CAS :<p>Dihydrocapsaicin, similar to capsaicin, is an irritant found in Capsicum, used in "pure" capsaicin products at about 10%, activates VR1, and is an antioxidant.</p>Formule :C18H29NO3Degré de pureté :99.61% - ≥95%Couleur et forme :White CrystalMasse moléculaire :307.43Laquinimod sodium
CAS :<p>Laquinimod (ABR-215062) sodium is an oral agent for MS, halting neurodegeneration and inflammation.</p>Formule :C19H16ClN2NaO3Couleur et forme :SolidMasse moléculaire :378.79Thalidomide-PEG4-Propargyl
CAS :<p>Thalidomide-PEG4-Propargyl is a synthetic E3 ligase ligand for PROTAC with a cereblon ligand and linker.</p>Formule :C24H28N2O9Degré de pureté :97.46%Couleur et forme :SolidMasse moléculaire :488.49PFI-1
CAS :<p>PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 μM in a cell-free assay.</p>Formule :C16H17N3O4SDegré de pureté :98.74% - 99.19%Couleur et forme :SolidMasse moléculaire :347.39MCB-613
CAS :<p>MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.</p>Formule :C20H20N2ODegré de pureté :98.17% - 99.754%Couleur et forme :SolidMasse moléculaire :304.39SKLB-163
CAS :<p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>Formule :C18H16ClN3O2S2Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :405.92Fasentin
CAS :<p>Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.</p>Formule :C11H9ClF3NO2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :279.64Mitoxantrone diacetate
CAS :<p>Mitoxantrone diacetate hinders topoisomerase II & PKC, fights tumors & orthopoxviruses (IC50: 8.5μM, EC50: 0.25-0.8μM).</p>Formule :C26H36N4O10Couleur et forme :SolidMasse moléculaire :564.592ONO-8130
CAS :<p>ONO-8130 is an orally available antagonist of EP1 receptor.</p>Formule :C25H28N2O5S2Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :500.63Fedratinib
CAS :<p>Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.</p>Formule :C27H36N6O3SDegré de pureté :97.31% - 99.96%Couleur et forme :SolidMasse moléculaire :524.68Chelerythrine
CAS :<p>1.</p>Formule :C21H18NO4Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :348.37Dimethyl malonate
CAS :<p>Dimethyl Malonate is a Succinate Dehydrogenase inhibitor.</p>Formule :C5H8O4Degré de pureté :≥95%Couleur et forme :LiquidMasse moléculaire :132.11Itanapraced
CAS :<p>Itanapraced (CHF5074), a γ-secretase modulator, reduces Aβ42/40 secretion (IC50: 3.6/18.4 μM).</p>Formule :C16H11Cl2FO2Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :325.16Tofacitinib Citrate
CAS :<p>Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).</p>Formule :C22H28N6O8Degré de pureté :99.19% - 99.75%Couleur et forme :SolidMasse moléculaire :504.49Siremadlin
CAS :<p>Siremadlin (NVP-HDM 201) is a potent, orally bioavailable and highly specific p53-MDM2 interaction inhibitor.</p>Formule :C26H24Cl2N6O4Degré de pureté :99.30% - 99.76%Couleur et forme :SolidMasse moléculaire :555.41Meloxicam sodium
CAS :<p>Meloxicam sodium is a non-steroidal anti-inflammatory agent, inhibits COX activity, with IC 50 s of 0.49 μM and 36.6 μM for COX-2 and COX-1, respectively [1].</p>Formule :C14H12N3NaO4S2Couleur et forme :SolidMasse moléculaire :373.383'-Hydroxypterostilbene
CAS :<p>3'-Hydroxypterostilbene suppresses colon cancer cell growth (COLO 205, HCT-116, HT-29) by triggering apoptosis and autophagy, affecting key pathways.</p>Formule :C16H16O4Degré de pureté :98.25% - 99.19%Couleur et forme :SolidMasse moléculaire :272.3Benzoylpaeoniflorin
CAS :<p>1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes.</p>Formule :C30H32O12Degré de pureté :95.86% - 97.28%Couleur et forme :SolidMasse moléculaire :584.57Cinchonine monohydrochloride hydrate
CAS :<p>Cinchonine monohydrochloride hydrate: natural antimalarial, inhibits platelet aggregation & cancer cell growth, blocks fat cell formation.</p>Formule :C19H25ClN2O2Couleur et forme :SolidMasse moléculaire :348.87Ulinastatin
CAS :<p>Ulinastatin is a multivalent Kunitz-type serine protease inhibitor with anti-inflammatory properties.</p>Formule :C13H16O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :220.10994Droxinostat
CAS :<p>Droxinostat (NS 41080) is a selective inhibitor of HDAC, mostly for HDACs 6 and 8 with IC50 of 2.47 μM and 1.46 μM, greater than 8-fold selective against HDAC3</p>Formule :C11H14ClNO3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :243.69RG7112
CAS :<p>RG7112 (RO5045337) (RO5045337) is an orally bioavailable and selective p53-MDM2 inhibitor.</p>Formule :C38H48Cl2N4O4SDegré de pureté :99.66% - 99.9%Couleur et forme :SolidMasse moléculaire :727.788-Bromo-cAMP sodium salt
CAS :<p>8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) is a long-acting derivative of cyclic AMP. 8-Bromo-cAMP is an activator of cyclic AMP-dependent protein kinase.</p>Formule :C10H10BrN5NaO6PDegré de pureté :98% - 99.94%Couleur et forme :Off-White PowderMasse moléculaire :430.08C5 Lenalidomide
CAS :<p>C5 Lenalidomide is an chemical weith inconclusive biological activity.</p>Formule :C13H13N3O3Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :259.26Kinetin riboside
CAS :<p>Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)</p>Formule :C15H17N5O5Degré de pureté :98.17%Couleur et forme :White SolidMasse moléculaire :347.33Dacomitinib
CAS :<p>Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.</p>Formule :C24H25ClFN5O2Degré de pureté :99.4% - 99.72%Couleur et forme :SolidMasse moléculaire :469.94Flupentixol dihydrochloride
CAS :<p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>Formule :C23H27Cl2F3N2OSDegré de pureté :98.76% - >99.99%Couleur et forme :White Or Off-White SolidMasse moléculaire :507.43Shield-1
CAS :<p>Shield-1 is a specific, high-affinity, and cell-permeable ligand for FK506-binding protein 12 (FKBP).Cost-effective and quality-assured.</p>Formule :C42H56N2O10Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :748.9
