
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(115 produits)
- CDK(546 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(47 produits)
- Dynamine(27 produits)
- Ferroptose(227 produits)
- HSP(180 produits)
- Intégrine(269 produits)
- Kinésine(87 produits)
- LIM Kinase(20 produits)
- Microtubules associés(273 produits)
- PKC(126 produits)
- PLK(25 produits)
- ROCK(62 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(76 produits)
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3908 produits trouvés pour "Cycle cellulaire/point de contrôle"
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Datelliptium chloride hydrochloride
CAS :Datelliptium chloride hydrochloride is a DNA-intercalating agent derived from ellipticine. with anti-tumor activities.
Formule :C23H29Cl2N3ODegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :434.4Favipiravir sodium
CAS :Favipiravir sodium inhibits viral RNA polymerases, effective against flu, West Nile, yellow fever, and more RNA viruses.Formule :C5H4FN3NaO2Couleur et forme :SolidMasse moléculaire :180.09MLS000532223
CAS :MLS000532223 is a selectiveRho family GTPases inhibitor(EC50 : 16 μM to 120 μM).Formule :C15H9NO3Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :251.24Ref: TM-T8473
1mg105,00€5mg250,00€1mL*10mM (DMSO)301,00€10mg401,00€25mg685,00€50mg982,00€100mg1.341,00€Hesperadin
CAS :Hesperadin(IC50=250 nM) effectively inhibits Aurora B.Formule :C29H32N4O3SDegré de pureté :98.04% - 99.44%Couleur et forme :SolidMasse moléculaire :516.65Reversine
CAS :Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).Formule :C21H27N7ODegré de pureté :98% - 99.45%Couleur et forme :SolidMasse moléculaire :393.49Ref: TM-T1825
1mg35,00€2mg50,00€5mg66,00€1mL*10mM (DMSO)66,00€10mg84,00€25mg156,00€50mg212,00€100mg371,00€SB-743921 hydrochloride
CAS :SB-743921 hydrochloride (SB743921 HCl) is an effective inhibitor of kinesin spindle protein, KSP, (Ki =0.1 nM).Formule :C31H34Cl2N2O3Degré de pureté :95.58% - 99.70%Couleur et forme :SolidMasse moléculaire :553.52Ref: TM-T2255
1mg39,00€5mg101,00€1mL*10mM (DMSO)123,00€10mg155,00€25mg263,00€50mg406,00€100mg622,00€500mg1.423,00€BCH001
CAS :BCH001 is a specific small-molecule inhibitor of PAPD5.Formule :C20H15F3N2O5Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :420.34P005091
CAS :P005091 (P5091) is a selective and potent inhibitor of ubiquitin-specific protease 7 (USP7) with EC50 of 4.2 μM.Formule :C12H7Cl2NO3S2Degré de pureté :99.53% - 99.87%Couleur et forme :SolidMasse moléculaire :348.22USP7-IN-8
CAS :Benzamide, 4-[6-amino-4-ethyl-5-(4-hydroxyphenyl)-3-pyridinyl]-N-methyl- is a selective ubiquitin-specific protease 7 (USP7) inhibitor with an IC50 of 1.4 μM.Formule :C21H21N3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :347.41Ref: TM-T9217
1mg46,00€5mg92,00€1mL*10mM (DMSO)100,00€10mg147,00€25mg269,00€50mg389,00€100mg532,00€200mg705,00€XL177A
CAS :XL177A is a selective irreversible USP7 inhibitor(IC50 : 0.34 nM). XL177A elicits cancer cell killing through a p53-dependent mechanism.Formule :C48H57ClN8O5Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :861.47BDP5290
CAS :BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.)Formule :C17H18ClN7ODegré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :371.82Ref: TM-T7301
1mg52,00€2mg77,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg178,00€25mg369,00€50mg535,00€100mg780,00€SAR407899 hydrochloride
CAS :SAR407899 hydrochloride is a selective, potent and ATP-competitive ROCK inhibitor, with an IC50 of 135 nM for ROCK-2, and Kis of 36 nM and 41 nM for human andFormule :C14H17ClN2O2Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :280.75KenPaullone
CAS :KenPaullone (9-Bromopaullone), a potent CDK1, CDK2 and CDK5 inhibitor, as new enhancer for iTreg cell differentiation.Formule :C16H11BrN2ODegré de pureté :97.14% - 98.99%Couleur et forme :Tan SolidMasse moléculaire :327.18Ref: TM-T2247
1mg35,00€2mg50,00€5mg66,00€1mL*10mM (DMSO)71,00€10mg89,00€25mg178,00€50mg303,00€100mg449,00€500mg1.018,00€GNE-6640
CAS :GNE-6640: non-covalent USP7 inhibitor; IC50s: 0.75 µM (full), 0.43 µM (catalytic), 20.3 µM (USP43), 0.23 µM (Ub-MDM2).Formule :C20H18N4ODegré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :330.38Ref: TM-T5461
1mg66,00€2mg96,00€5mg144,00€1mL*10mM (DMSO)158,00€10mg236,00€25mg507,00€50mg730,00€100mg1.018,00€R-IMPP
CAS :R-IMPP is an inhibitor of PCSK9 translation.Formule :C24H27N3O2Degré de pureté :99.47% - 99.85%Couleur et forme :SolidMasse moléculaire :389.49Ref: TM-T4058
1mg46,00€2mg56,00€1mL*10mM (DMSO)75,00€5mg88,00€10mg140,00€25mg280,00€50mg500,00€100mg718,00€MLCK inhibitor peptide 18 acetate
MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.Formule :C62H109N23O13Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :1384.67ROCK-IN-2
CAS :ROCK-IN-2 (Azaindole 1) is a selective and ATP-competitive ROCK inhibitor with IC50 of 0.6 and 1.1 nM for human ROCK-1 and ROCK-2.Formule :C18H13ClF2N6ODegré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :402.79Ref: TM-TQ0110
1mg108,00€5mg260,00€1mL*10mM (DMSO)353,00€10mg416,00€25mg690,00€50mg964,00€100mg1.305,00€EOAI3402143
CAS :EOAI3402143 inhibits Usp9x and Usp24 activity, increases tumor cell apoptosis.Formule :C25H28Cl2N4O3Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :503.42Ref: TM-T11209
1mg63,00€5mg137,00€1mL*10mM (DMSO)152,00€10mg215,00€25mg423,00€50mg680,00€100mg1.009,00€NSC632839
CAS :NSC-632839 (Ubiquitin Isopeptidase Inhibitor II) is a nonselective isopeptidase inhibitor, which inhibits USP2 (EC50: 45±4 μM), USP7 (EC50: 37±1 μM), and SENP2Formule :C21H22ClNODegré de pureté :99.74% - 99.88%Couleur et forme :SolidMasse moléculaire :339.86Trifluridine/tipiracil hydrochloride mixture
CAS :Trifluridine/tipiracil hydrochloride mixture (TAS-102) is a novel oral combination drug containing trifluridine (TFT) and Tipiracil hydrochloride (TTP) in aFormule :C29H34Cl2F6N8O12Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :871.53Ref: TM-T3658
2mg37,00€5mg54,00€1mL*10mM (DMSO)73,00€10mg93,00€25mg148,00€50mg236,00€100mg358,00€200mg538,00€500mg842,00€LDC4297 hydrochloride
CAS :LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Formule :C23H29ClN8OCouleur et forme :SolidMasse moléculaire :468.98Arg-Gly-Asp TFA (99896-85-2(free base))
Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.Formule :C14H23F3N6O8Degré de pureté :99.2% - ≥98%Couleur et forme :SolidMasse moléculaire :460.36Tempo
CAS :Tempo (2,2,6,6-Tetramethylpiperidinooxy) has a wide range of applications including use as a free radical scavenger, a reagent in organic synthesis and as aFormule :C9H18NODegré de pureté :98.35%Couleur et forme :Orange Crystals Or PowderMasse moléculaire :156.25Netarsudil mesylate
CAS :Netarsudil mesylate (AR-13324 mesylate) is a Rho-related protein kinase inhibitor used to study glaucoma and hypertension.Formule :C30H35N3O9S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :645.74Ref: TM-T10358L2
1mg34,00€5mg66,00€1mL*10mM (DMSO)96,00€10mg105,00€25mg236,00€50mg409,00€100mg700,00€Remdesivir
CAS :Remdesivir (GS-5734) is a nucleoside analog, a broad-spectrum antiviral compound that exerts its activity by inhibiting the RNA-dependent RNA polymerase ofFormule :C27H35N6O8PDegré de pureté :97.62% - 99.98%Couleur et forme :SolidMasse moléculaire :602.58Ref: TM-T7766
1mg108,00€5mg205,00€1mL*10mM (DMSO)268,00€10mg326,00€25mg497,00€50mg663,00€100mg1.063,00€SRPIN340
CAS :SRPIN340 (SRPK inhibitor), a serine/arginine-rich protein kinase (SRPK)-specific inhibitor, is potent for SRPK1 (IC50 = 0.89 uM).Formule :C18H18F3N3ODegré de pureté :99.79% - 99.96%Couleur et forme :SolidMasse moléculaire :349.35Ref: TM-T1954
2mg44,00€5mg65,00€1mL*10mM (DMSO)71,00€10mg100,00€25mg177,00€50mg324,00€100mg421,00€500mg945,00€CKI-7
CAS :CKI-7 is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor.Formule :C11H14Cl3N3O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :358.67Ref: TM-T19913
1mg73,00€5mg128,00€1mL*10mM (DMSO)140,00€10mg185,00€25mg299,00€50mg405,00€100mg545,00€LDN-192960
CAS :LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).Formule :C18H20N2O2SDegré de pureté :99.01% - 99.51%Couleur et forme :SolidMasse moléculaire :328.43Ref: TM-TQ0111
1mg49,00€2mg64,00€5mg92,00€1mL*10mM (DMSO)104,00€10mg152,00€25mg295,00€50mg477,00€100mg763,00€200mg1.018,00€L189
CAS :L189 is a human DNA ligase inhibitor, inhibits hLigI/III/IV (IC50: 5/9/5 μM).Formule :C11H10N4OSDegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :246.29CeMMEC13
CAS :CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).Formule :C19H16N2O4Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :336.34Ref: TM-T6801
1mg34,00€2mg44,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg105,00€25mg230,00€50mg334,00€100mg447,00€Protein kinase inhibitors 1
CAS :Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.Formule :C18H17N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.42SJB2-043
CAS :SJB2-043 is an inhibitor of USP1-UAF1 ( IC50 : 544 nM).Formule :C17H9NO3Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :275.26Indirubin-3'-monoxime
CAS :Indirubin-3'-monoxime (Indirubin-3'-oxime) is a potent inhibitor of GSK3β (IC50: 22 nM) and also inhibits CDKs ( (IC50s: 100/180/250 nM for Cdk5/p35, Cdk1/Formule :C16H11N3O2Degré de pureté :99.55%Couleur et forme :Dark Red SolidMasse moléculaire :277.28USP25/28 inhibitor AZ1
CAS :USP25/28 inhibitor AZ1 is a selective, orally active and non-competitive dual ubiquitin-specific protease USP25/28 inhibitor.Cost-effective and quality-assured.Formule :C17H16BrF4NO2Degré de pureté :99.79% - 99.86%Couleur et forme :SolidMasse moléculaire :422.21Ref: TM-T7685
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg92,00€25mg200,00€50mg304,00€100mg447,00€500mg982,00€WR99210
CAS :WR99210 (BRL 6231 free base) is a DHFR inhibitor with antiparasitic activity.Formule :C14H18Cl3N5O2Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :394.68ID-8
CAS :ID-8, a DYRK inhibitor, sustains embryonic stem cell self-renewal in long-term culture.Formule :C16H14N2O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :298.29AZ191
CAS :AZ191(IC50 of 17 nM) is an effective and specific DYRK1B inhibitor.Formule :C24H27N7ODegré de pureté :98.04% - 99.65%Couleur et forme :SolidMasse moléculaire :429.52Hexapeptide-10 Acetate
Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) is a synthetic peptide.Formule :C30H57N7O10Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :675.81GNF4877
CAS :GNF4877 inhibits DYRK1A/GSK3β (IC50: 6/16 nM), blocks NFATc export, and boosts β-cell growth.Formule :C25H27FN6O4Degré de pureté :98.68% - 99.40%Couleur et forme :SolidMasse moléculaire :494.52AZ3146
CAS :AZ3146 is a selective Mps1 inhibitor with IC50 of ~35 nM.Formule :C24H32N6O3Degré de pureté :97.84% - >99.99%Couleur et forme :SolidMasse moléculaire :452.55USP7/USP47 inhibitor
CAS :USP7/USP47 inhibitor (USP7/47 inhibitor-1) is a selective ubiquitin-specific protease 7/47 (USP7/USP47) inhibitor, with EC50s of 0.42 μM and 1.0 μM,Formule :C18H11Cl2N3O3S3Degré de pureté :98.5% - 98.71%Couleur et forme :SolidMasse moléculaire :484.4Ref: TM-T4338
1mg40,00€1mL*10mM (DMSO)94,00€5mg96,00€10mg152,00€25mg268,00€50mg429,00€100mg703,00€200mg954,00€BSJ-4-116
CAS :BSJ-4-116: potent, selective CDK12 PROTAC, IC50 = 6 nM; downregulates DDR genes, induces premature transcription termination.Formule :C40H49ClN8O8SDegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :837.38ML364
CAS :ML364 is an inhibitor of ubiquitin specific peptidase 2 (USP2) and can be used for the research of breast cancer.Formule :C24H18F3N3O3S2Degré de pureté :99.35% - >99.99%Couleur et forme :SolidMasse moléculaire :517.54CID 2011756
CAS :CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.Formule :C22H21ClN2O3Degré de pureté :98.15% - ≥95%Couleur et forme :SolidMasse moléculaire :396.87GAK inhibitor 49
CAS :GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).Formule :C20H22N2O5Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :370.4Ref: TM-T8535
1mg54,00€5mg111,00€1mL*10mM (DMSO)128,00€10mg177,00€25mg299,00€50mg430,00€100mg587,00€200mg792,00€BI-847325
CAS :BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 values of 4 and 15 nM for human MEK2 and AK-C, respectively.Formule :C29H28N4O2Degré de pureté :97.13% - 97.54%Couleur et forme :SolidMasse moléculaire :464.56GDC0575 monohydrochloride
CAS :GDC0575 (ARRY575), a potent Chk1 inhibitor, IC50 1.2nM, disrupts cell cycle arrest, allowing DNA repair before mitosis.Formule :C16H21BrClN5ODegré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :414.73Ref: TM-T27407
1mg43,00€2mg55,00€5mg80,00€1mL*10mM (DMSO)93,00€10mg103,00€25mg177,00€50mg255,00€100mg356,00€200mg520,00€Aurora kinase inhibitor-2
CAS :Aurora kinase inhibitor-2 (IUN-70219) is a cell-permeable anilinoquinazoline that inhibit the activity of Aurora A (IC50 = 0.39 M).Formule :C23H20N4O3Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :400.43Ref: TM-T9040
1mg63,00€5mg138,00€1mL*10mM (DMSO)150,00€10mg200,00€25mg360,00€50mg532,00€100mg788,00€200mg1.063,00€SR18662
SR18662, improved ML264 derivative, inhibits KLF5 at 4.4 nM IC50; curbs colorectal cancer cell growth and triggers apoptosis.Formule :C16H19Cl2N3O4SDegré de pureté :98.97% - 99.2%Couleur et forme :SolidMasse moléculaire :420.31Ref: TM-T22429
1mg46,00€5mg90,00€1mL*10mM (DMSO)100,00€10mg152,00€25mg295,00€50mg475,00€100mg680,00€200mg888,00€500mg1.378,00€BIO-1211
CAS :BIO-1211 is a more potent inhibitor of α4β1 (VLA-4, IC50 = 4 nM) over α4β7(IC50 = 2 μM).Formule :C36H48N6O9Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :708.8
