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Métabolisme

Métabolisme

Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.

Sous-catégories appartenant à la catégorie "Métabolisme"

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8626 produits trouvés pour "Métabolisme"

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  • ATP disodium salt

    CAS :
    <p>ATP disodium salt (Adenosine-Triphosphate) is a P2 purinoceptor agonist.</p>
    Formule :C10H14N5O13P3·2Na
    Degré de pureté :97.91% - 99.7%
    Couleur et forme :Solid
    Masse moléculaire :551.14
  • Methazolamide

    CAS :
    <p>Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.</p>
    Formule :C5H8N4O3S2
    Degré de pureté :99.31% - 99.77%
    Couleur et forme :Crystals From Water Solid
    Masse moléculaire :236.27
  • Carbadox

    CAS :
    <p>Carbadox, an antibacterial for swine dysentery and growth promotion, is banned in the UK due to carcinogen and mutagen risks.</p>
    Formule :C11H10N4O4
    Degré de pureté :98.38% - 99.73%
    Couleur et forme :Minute Yellow Crystals Yellow Crystals
    Masse moléculaire :262.22
  • Nitisinone

    CAS :
    <p>Nitisinone (SC0735)(SC0735) is an enzyme 4-hydroxyphenylpyruvate dioxygenase inhibitor.</p>
    Formule :C14H10F3NO5
    Degré de pureté :99.63%
    Couleur et forme :Solid
    Masse moléculaire :329.23
  • PT2399

    CAS :
    <p>PT2399, an oral HIF-2 inhibitor, blocks HIF-2α/1β dimerization, showing strong in vivo antitumor effects.</p>
    Formule :C17H10F5NO4S
    Degré de pureté :98.8% - 99.45%
    Couleur et forme :Solid
    Masse moléculaire :419.32
  • N1-Acetylspermine trihydrochloride

    CAS :
    <p>N1-Acetylspermine trihydrochloride: monoacetylated spermine, aids in bleomycin-A5 uptake studies via SLC22A16.</p>
    Formule :C12H31Cl3N4O
    Degré de pureté :98.79% - 99.93%
    Couleur et forme :Solid
    Masse moléculaire :353.76
  • Naringinase

    CAS :
    <p>Naringinase, with α-L-rhamnosidase and β-D-glucosidase activities, transforms steroids, antibiotics, and glycosides.</p>
    Degré de pureté :98%
    Couleur et forme :Solid
  • Opicapone

    CAS :
    <p>Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).</p>
    Formule :C15H10Cl2N4O6
    Degré de pureté :98.17% - 99.36%
    Couleur et forme :Solid
    Masse moléculaire :413.17
  • Diethylcarbamazine citrate

    CAS :
    <p>Diethylcarbamazine citrate treats filariasis, targeting W. bancrofti and L. loa by inhibiting arachidonic acid in microfilaria.</p>
    Formule :C10H21N3O·C6H8O7
    Degré de pureté :99.61%
    Couleur et forme :White Crystalline Powder And Animals (Epa 1998)
    Masse moléculaire :391.42
  • Mefentrifluconazole

    CAS :
    <p>Mefentrifluconazole: potent, selective oral fungicide; strong CYP51 blocker, weaker on human aromatase; novel azole for broad-spectrum use.</p>
    Formule :C18H15ClF3N3O2
    Degré de pureté :99.88%
    Couleur et forme :Solid
    Masse moléculaire :397.78
  • 3-Pyridinemethanol

    CAS :
    <p>3-Pyridinemethanol (Roniacol) is an alcohol analog of nicotinic acid which is a peripheral vasodilator that causes flushing and may decrease blood pressure.</p>
    Formule :C6H7NO
    Degré de pureté :98.9% - 99.30%
    Couleur et forme :Clear Light Yellow To Yellow Liquid
    Masse moléculaire :109.13
  • Monacolin J

    CAS :
    <p>Monacolin J (Antibiotic MB 530A) is a cholesterol biosynthesis inhibitor.</p>
    Formule :C19H28O4
    Degré de pureté :98.06%
    Couleur et forme :Solid
    Masse moléculaire :320.42
  • ER-000444793

    CAS :
    <p>ER-000444793 is a potent mitochondrial permeability transition pore (mPTP) opening inhibitor and it also inhibits mPTP (IC50: 2.8 μM).</p>
    Formule :C23H18N2O2
    Degré de pureté :99.55%
    Couleur et forme :Solid
    Masse moléculaire :354.4
  • LY2183240

    CAS :
    <p>LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM).</p>
    Formule :C17H17N5O
    Degré de pureté :99.26%
    Couleur et forme :Solid
    Masse moléculaire :307.35
  • GW7647

    CAS :
    <p>GW 7647 is an effective and highly selective PPARα agonist. GW 7647 can reduce the production of nitric oxide in macrophages. Cost-effective and quality-assured.</p>
    Formule :C29H46N2O3S
    Degré de pureté :99.3% - 99.34%
    Couleur et forme :Solid
    Masse moléculaire :502.75
  • Amlodipine

    CAS :
    <p>Amlodipine (UK-48340) is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties.</p>
    Formule :C20H25ClN2O5
    Degré de pureté :99.33% - 99.60%
    Couleur et forme :Solid Powder
    Masse moléculaire :408.88
  • N-Desmethyl-Apalutamide

    CAS :
    <p>N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.</p>
    Formule :C20H13F4N5O2S
    Degré de pureté :98.6%
    Couleur et forme :Solid
    Masse moléculaire :463.41
  • HIF-PHD-IN-3

    CAS :
    <p>HIF-PHD-IN-3 is a hiPSC-CM cardioprotective scaffold with potential inhibitory effects on HIF-PHD, regulates heme oxygenase-1, and can be used to study anaemia.</p>
    Formule :C16H13N3OS2
    Degré de pureté :98.12%
    Couleur et forme :Solid
    Masse moléculaire :327.42
  • Mouse PP(Pancreatic Polypeptide) ELISA Kit


    <p>This assay employs the competitive inhibition enzyme immunoassay technique. The microtiter plate provided in this kit has been pre-coated with Mouse PP protein. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Mouse PP. Next, Avidin conjugated to Horseradish Peroxidase (HRP) is added to each microplate well and incubated. After TMB substrate solution is added. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Mouse PP in the samples is then determined by comparing the OD of the samples to the standard curve.</p>
  • Imidacloprid-urea

    CAS :
    <p>Imidacloprid-urea, a byproduct of imidacloprid, may alter its environmental behavior by competing for soil binding sites.</p>
    Formule :C9H10ClN3O
    Degré de pureté :99.89%
    Couleur et forme :Solid
    Masse moléculaire :211.65
  • Sucralose

    CAS :
    <p>Sucralose (Trichlorosucrose), an artificial sweetener, is not degraded by the body, so it is noncaloric.</p>
    Formule :C12H19Cl3O8
    Degré de pureté :99.85% - 99.89%
    Couleur et forme :White To Off White Crystalline Powder White To Off-White Practically Odourless Crystalline Powder
    Masse moléculaire :397.63
  • DPA-714

    CAS :
    <p>DPA-714: a TSPO ligand (Ki=7 nM) with a fluorine atom for PET imaging of inflammation and brain tumors.</p>
    Formule :C22H27FN4O2
    Degré de pureté :99.52%
    Couleur et forme :Solid
    Masse moléculaire :398.47
  • NSP-805

    CAS :
    <p>NSP-805 is a potent and selective guinea pig cardiac phosphodiesterase 3 (PDE3) inhibitor.</p>
    Formule :C17H19N3O2
    Degré de pureté :99.85%
    Couleur et forme :Solid
    Masse moléculaire :297.35
  • CAY10566

    CAS :
    <p>CAY10566 is a potent SCD1 inhibitor, orally bioavailable, with IC50s: HepG2 cells, 7.9nM; mouse, 4.5nM; human, 26nM.</p>
    Formule :C18H17ClFN5O2
    Degré de pureté :99.5% - 99.54%
    Couleur et forme :Solid
    Masse moléculaire :389.81
  • Levamlodipine

    CAS :
    <p>Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers.</p>
    Formule :C20H25ClN2O5
    Degré de pureté :97.21%
    Couleur et forme :White Crystal Powder
    Masse moléculaire :408.88
  • Anhydrosimvastatin

    CAS :
    <p>Anhydrosimvastatin (Dehydro simvastatin) is an impurity of Simvastatin. Simvastatin is an HMG-CoA reductase inhibitor.</p>
    Formule :C25H36O4
    Degré de pureté :99.63%
    Couleur et forme :Solid
    Masse moléculaire :400.55
  • Albendazole

    CAS :
    <p>Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations.</p>
    Formule :C12H15N3O2S
    Degré de pureté :98.21% - 98.76%
    Couleur et forme :Colorless Crystals Solid
    Masse moléculaire :265.33
  • Hydralazine hydrochloride

    CAS :
    <p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>
    Formule :C8H9ClN4
    Degré de pureté :99.85% - 99.86%
    Couleur et forme :Yellow Crystals White Crystalline Solid
    Masse moléculaire :196.64
  • N-desmethyl Olanzapine

    CAS :
    <p>N-desmethyl Olanzapine, a metabolite of Olanzapine, is created via CYP1A2 oxidative metabolism.</p>
    Formule :C16H18N4S
    Degré de pureté :99.67%
    Couleur et forme :Solid
    Masse moléculaire :298.41
  • TAME hydrochloride

    CAS :
    <p>TAME hydrochloride (Tos-Arg-OMe HCl) is a kind od amino acid derivatives.</p>
    Formule :C14H23ClN4O4S
    Degré de pureté :99.11% - 99.21%
    Couleur et forme :White Fine Crystalline Powder
    Masse moléculaire :378.87
  • Oltipraz

    CAS :
    <p>Oltipraz (RP 35972) is a synthetic dithiolethione with potential chemopreventive and anti-angiogenic properties.</p>
    Formule :C8H6N2S3
    Degré de pureté :98.79% - 99.77%
    Couleur et forme :Solid
    Masse moléculaire :226.34
  • Tris(2,4-di-tert-butylphenyl)phosphate

    CAS :
    <p>Tris(2,4-di-tert-butylphenyl)phosphate (TDTBPP) inhibits secretory phospholipase A2 (sPLA2) with anti-inflammatory effect. Cost-effective and quality-assured.</p>
    Formule :C42H63O4P
    Degré de pureté :99.73%
    Couleur et forme :Solid
    Masse moléculaire :662.92
  • Ethylvanillin

    CAS :
    <p>Ethylvanillin (Rhodiarome) is a flavorant used in the production of chocolate. It is about three times as potent as vanillin.</p>
    Formule :C9H10O3
    Degré de pureté :99.44%
    Couleur et forme :White - Off White Solid Powder
    Masse moléculaire :166.17
  • N-Desmethyltamoxifen hydrochloride

    CAS :
    <p>N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.</p>
    Formule :C25H28ClNO
    Degré de pureté :99.15%
    Couleur et forme :Solid
    Masse moléculaire :393.95
  • Liarozole

    CAS :
    <p>Liarozole dihydrochloride inhibits CYP450, estrogen, androgen synthesis; an oral drug for prostate cancer/skin disorders.</p>
    Formule :C17H13ClN4
    Degré de pureté :98.31%
    Couleur et forme :Solid
    Masse moléculaire :308.76
  • myo-Inositol, 1,2,3,4,5,6-hexakis(dihydrogen phosphate)

    CAS :
    Formule :C6H18O24P6
    Degré de pureté :%
    Couleur et forme :Liquid
    Masse moléculaire :660.0353

    Ref: IN-DA003TRV

    25g
    26,00€
    100g
    27,00€
    200l
    17.155,00€
    500g
    65,00€
  • Denifanstat

    CAS :
    <p>Denifanstat (FASN-IN-2) is a FASN inhibitor with selective and oral activity. Denifanstat has been used in studies of steatohepatitis. Cost effective and quality assured.</p>
    Formule :C27H29N5O
    Degré de pureté :98.33% - 99.35%
    Couleur et forme :Solid
    Masse moléculaire :439.55
  • Olutasidenib

    CAS :
    <p>Olutasidenib (FT-2102), an IDH1 inhibitor (IC50: 21.2/114 nM), is studied for treating AML/MDS and can cross the blood-brain barrier.</p>
    Formule :C18H15ClN4O2
    Degré de pureté :98.57%
    Couleur et forme :Solid
    Masse moléculaire :354.79
  • IDO-IN-13

    CAS :
    <p>IDO-IN-13 (GS-4361) is a potent indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor (EC50: 17 nM).</p>
    Formule :C26H17F3N4O
    Degré de pureté :99.29%
    Couleur et forme :Solid
    Masse moléculaire :458.43
  • Bezafibrate

    CAS :
    <p>Bezafibrate (BM15075) is an antilipemic agent that lowers CHOLESTEROL and TRIGLYCERIDES.</p>
    Formule :C19H20ClNO4
    Degré de pureté :99.56% - 99.82%
    Couleur et forme :Solid
    Masse moléculaire :361.82
  • Chloramphenicol

    CAS :
    <p>Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.</p>
    Formule :C11H12Cl2N2O5
    Degré de pureté :99.6% - 99.84%
    Couleur et forme :Needles Or Elongated Plates From Water Or Ethylene Dichloride Solid
    Masse moléculaire :323.13
  • BAY-2402234

    CAS :
    <p>BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.</p>
    Formule :C21H18ClF5N4O4
    Degré de pureté :98.9%
    Couleur et forme :Solid
    Masse moléculaire :520.84
  • Hi 76-0079

    CAS :
    <p>Hi 76-0079: HSL inhibitor, IC50=184 nM; potential for obesity and diabetes research.</p>
    Formule :C11H13ClN2O3
    Degré de pureté :99.9%
    Couleur et forme :Soild
    Masse moléculaire :256.69
  • Hydroxycitric acid tripotassium hydrate

    CAS :
    <p>Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits HIF, has antioxidation, anti-inflammation, and anti-tumor effects.</p>
    Formule :C6H7K3O8
    Degré de pureté :99.85%
    Couleur et forme :White Solid Crystalline
    Masse moléculaire :324.41
  • Abiraterone

    CAS :
    <p>Abiraterone (CB-7598) (CB-7598) is an effective steroidal cytochrome P450 17alpha-hydroxylase-17, 20-lyase (CYP17) inhibitor (IC50: 4 nM).</p>
    Formule :C24H31NO
    Degré de pureté :99.18% - 99.93%
    Couleur et forme :White Solid
    Masse moléculaire :349.51
  • Amylase

    CAS :
    <p>Amylase (Diastase) is any one of a group of enzymes which catalyses the breakdown of starch into maltose.</p>
    Formule :NA
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :N/A
  • Moclobemide

    CAS :
    <p>Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.</p>
    Formule :C13H17ClN2O2
    Degré de pureté :99.51% - 99.59%
    Couleur et forme :White To Off-White Solid
    Masse moléculaire :268.74
  • 6-Aminocaproic acid

    CAS :
    <p>6-Aminocaproic acid (EACA) is an antifibrinolytic agent that acts by inhibiting plasminogen activators which have fibrinolytic properties.</p>
    Formule :C6H13NO2
    Degré de pureté :99.55%
    Couleur et forme :Fine White Crystalline Powder Solid
    Masse moléculaire :131.17
  • Norgestimate metabolite Norelgestromin

    CAS :
    <p>Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate), an active metabolites of norgestimate, is a steroidal progestin used in contraceptive patches.</p>
    Formule :C21H29NO2
    Degré de pureté :99.64%
    Couleur et forme :Solid
    Masse moléculaire :327.46
  • CBR-5884

    CAS :
    <p>CBR-5884: active PHGDH inhibitor, IC50=33μM, disrupts serine synthesis, selectively targets high-serine cancers.</p>
    Formule :C14H12N2O4S2
    Degré de pureté :99.97%
    Couleur et forme :Solid
    Masse moléculaire :336.39
  • H-Lys(Tfa)-OH

    CAS :
    <p>H-Lys(Tfa)-OH is an inhibitor of L-lysine cyclodeaminase.</p>
    Formule :C8H13F3N2O3
    Degré de pureté :99.35%
    Couleur et forme :Solid
    Masse moléculaire :242.2
  • Clevidipine

    CAS :
    <p>Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for blood</p>
    Formule :C21H23Cl2NO6
    Degré de pureté :99.40%
    Couleur et forme :Powder
    Masse moléculaire :456.32
  • CPDA

    CAS :
    <p>CPDA is a new potent inhibitor of SH2 domain-containing inositol phosphatase 2 (SHIP2).</p>
    Formule :C20H15ClF2N2O2
    Degré de pureté :98.34%
    Couleur et forme :Solid
    Masse moléculaire :388.8
  • Finasteride

    CAS :
    <p>Finasteride (MK-906) is an oral inhibitor of active testosterone 5-alpha-reductase and Ki value is 10 nM.</p>
    Formule :C23H36N2O2
    Degré de pureté :99.04% - 99.97%
    Couleur et forme :White To Off-White Crystalline Powder
    Masse moléculaire :372.54
  • Gabexate mesylate

    CAS :
    <p>Gabexate mesylate (FOY) inhibits thrombin, plasmin, kallikrein; used for pancreatitis, DIC, hemodialysis anticoagulant.</p>
    Formule :C17H27N3O7S
    Degré de pureté :99.2% - 99.64%
    Couleur et forme :White Crystal
    Masse moléculaire :417.48
  • Vitamin K

    CAS :
    <p>Vitamin K (Kephton) has blood coagulation action and is important for coagulation factors, matrix-Gla protein, and osteocalcin.</p>
    Degré de pureté :97.00% - 99.79%
    Couleur et forme :Solid
  • Topiramate

    CAS :
    <p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>
    Formule :C12H21NO8S
    Degré de pureté :99.79% - 99.92%
    Couleur et forme :White To Off-White Crystalline Powder
    Masse moléculaire :339.36
  • Amlodipine Besylate

    CAS :
    <p>Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker.</p>
    Formule :C26H31ClN2O8S
    Degré de pureté :96.67% - 99.92%
    Couleur et forme :White Powder
    Masse moléculaire :567.05
  • Fenofibrate

    CAS :
    <p>Fenofibrate (Lipanthyl) is a PPARα agonist. Fenofibrate inhibits cytochrome P450 isoforms. Fenofibrate exhibits antihyperlipidemic activity. Cost-effective and quality-assured.</p>
    Formule :C20H21ClO4
    Degré de pureté :99.13% - 99.95%
    Couleur et forme :Crystals From Isopropanol Solid
    Masse moléculaire :360.83
  • EMD57439

    CAS :
    <p>EMD57439 is a selective PDE-III inhibitor, showing no significant increase in c-AMP concentration and producing little change in Ca(50).</p>
    Formule :C22H23N3O4S
    Degré de pureté :99.38% - 99.57%
    Couleur et forme :Solid
    Masse moléculaire :425.5
  • T-0156

    CAS :
    <p>T-0156 is a PEG5 inhibitor that inhibits the hydrolysis of cyclic guanosine monophosphate (cGMP) with low affinity for PDE6, PDE1, PDE2, PDE3 and PDE4.</p>
    Formule :C31H29N5O7
    Degré de pureté :98.53% - 98.76%
    Couleur et forme :Soild
    Masse moléculaire :583.59
  • Mouse PⅠNP(Procollagen Ⅰ N-Terminal Propeptide) ELISA Kit


    <p>This assay employs the competitive inhibition enzyme immunoassay technique. The microtiter plate provided in this kit has been pre-coated with Mouse PⅠNP protein. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Mouse PⅠNP. Next, Avidin conjugated to Horseradish Peroxidase (HRP) is added to each microplate well and incubated. After TMB substrate solution is added. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Mouse PⅠNP in the samples is then determined by comparing the OD of the samples to the standard curve.</p>
  • Vasopressin acetate


    <p>Vasopressin acetate: cyclic nonapeptide synthesized in the hypothalamus, functions as a neurotransmitter via G protein-coupled receptors.</p>
    Degré de pureté :98.11%
    Couleur et forme :Liquid
  • Pyrimethamine

    CAS :
    <p>Pyrimethamine (Pirimecidan) is a competitive inhibitor of dihydrofolate reductase (DHFR), used as an antimalarial drug.</p>
    Formule :C12H13ClN4
    Degré de pureté :99.67%
    Couleur et forme :Crystals
    Masse moléculaire :248.71
  • Felodipine

    CAS :
    <p>Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor.</p>
    Formule :C18H19Cl2NO4
    Degré de pureté :99.91%
    Couleur et forme :Solid
    Masse moléculaire :384.25
  • 1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium

    CAS :
    <p>1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium, a phosphatidic acid, is a human endogenous metabolite.</p>
    Formule :C35H68NaO8P
    Degré de pureté :99.37%
    Couleur et forme :Solid
    Masse moléculaire :670.87
  • JW 642

    CAS :
    <p>JW 642 inhibits MAGL in mouse, rat, human brains (IC50: 7.6, 14, 3.7 nM).</p>
    Formule :C21H20F6N2O3
    Degré de pureté :99.28%
    Couleur et forme :Solid
    Masse moléculaire :462.39
  • LY195448

    CAS :
    <p>LY 195448 (4-(3-(2-Hydroxy-2-phenyl)ethylamino-3-methylbutyl)benzamide) shows antitumor activity in a mouse tumor model, blocking cells in the mid-stage.</p>
    Formule :C20H26N2O2
    Degré de pureté :98.11% - 99.04%
    Couleur et forme :Solid
    Masse moléculaire :326.43
  • Eliglustat hemitartrate

    CAS :
    <p>Eliglustat hemitartrate (Genz-112638) , with an IC50 of 24 nM, is a specific, potent, oral active glucocerebral glycosidase inhibitor.</p>
    Formule :C25H39N2O7
    Degré de pureté :99.71%
    Couleur et forme :Solid
    Masse moléculaire :479.59
  • Cinepazide maleate

    CAS :
    <p>Cinepazide maleate (MD-67350), a maleate salt form of cinepazide, is a vasodilator.</p>
    Formule :C22H31N3O5·C4H4O4
    Degré de pureté :99.9% - 99.97%
    Couleur et forme :White Or Off-White Crystalline Powder
    Masse moléculaire :533.57
  • ML390

    CAS :
    <p>ML390 exerts its potent differentiation effect on multiple leukemia models.</p>
    Formule :C21H21F3N2O3
    Degré de pureté :99.76%
    Couleur et forme :Solid
    Masse moléculaire :406.4
  • Acetoacetic acid sodium salt

    CAS :
    <p>Acetoacetic acid sodium salt is a metabolite of non-esterified fatty acids, involved in the development of human diabetes.</p>
    Formule :C4H5NaO3
    Degré de pureté :≥98%
    Couleur et forme :Solid
    Masse moléculaire :124.07
  • LDN-212320

    CAS :
    <p>LDN-212320 (OSU-0212320) is a glutamate transporter EAAT2 activator. It also enhances EAAT2 levels by &gt; 6 fold at concentrations &lt; 5 μM after 24 h.</p>
    Formule :C17H15N3S
    Degré de pureté :98.18%
    Couleur et forme :Solid
    Masse moléculaire :293.39
  • VU0359595

    CAS :
    <p>VU0359595 (ML-270) is a selective PLD1 inhibitor with 3.7 nM IC50; &gt;1700x more selective over PLD2, for cancer/diabetes/neurodegenerative research.</p>
    Formule :C25H29BrN4O2
    Degré de pureté :99.79%
    Couleur et forme :Solid
    Masse moléculaire :497.43
  • DL-Propargylglycine HCl

    CAS :
    <p>DL-Propargylglycine HCl (DL-Propargylglycine HCl) is a cystathionine gamma catabolism enzyme inhibitor that can be used in heart failure studies.</p>
    Formule :C5H8ClNO2
    Degré de pureté :>99.99%
    Couleur et forme :Solid
    Masse moléculaire :149.58
  • EC5026

    CAS :
    <p>EC5026 (BPN-19186) has the potential to relieve pain by stabilizing natural analgesic and anti-inflammatory mediators.</p>
    Formule :C18H23F4N3O3
    Degré de pureté :96.6% - 99.81%
    Couleur et forme :Solid
    Masse moléculaire :405.39
  • Garadacimab

    CAS :
    <p>Garadacimab (CSL312) is a human IgG4 antibody against FXIIa, used to research hereditary angioedema.</p>
    Degré de pureté :SDS-PAGE:95% SEC-HPLC:99.99%
    Couleur et forme :Liquid
    Masse moléculaire :146.5 kDa
  • L-Carnitine

    CAS :
    <p>L-Carnitine aids fatty acid oxidation in mitochondria for energy, excluding the brain.</p>
    Formule :C7H15NO3
    Degré de pureté :99.29% - 99.94%
    Couleur et forme :White Crystalline Hygroscopic Powder Solid
    Masse moléculaire :161.20
  • Diphenyl phosphate

    CAS :
    <p>Diphenyl phosphate (Phenyl hydrogen phosphate) is capable of gender-specific inhibition of growth and energy metabolism in zebrafish.</p>
    Formule :C12H11O4P
    Degré de pureté :99.95%
    Couleur et forme :Liquid
    Masse moléculaire :250.19
  • G0-C14 HCl


    <p>G0-C14 HCl is a cationic lipid molecule and amphiphilic dendritic macromolecule commonly used in the synthesis of nanoparticles and vaccine delivery.</p>
    Formule :C106H217ClN10O10
    Degré de pureté :99.12%
    Couleur et forme :Solid
    Masse moléculaire :1827.37
  • DHODH-IN-11

    CAS :
    <p>DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.</p>
    Formule :C15H11N3O2
    Degré de pureté :98.14%
    Couleur et forme :Solid
    Masse moléculaire :265.27
  • SBI-797812

    CAS :
    <p>SBI-797812 is structurally similar to active-site directed inhibitor of NAMPT(NAMPT with EC50 of 0.37 μM).</p>
    Formule :C19H22N4O4S
    Degré de pureté :99.31%
    Couleur et forme :Solid
    Masse moléculaire :402.47
  • Mildronate dihydrate

    CAS :
    <p>Mildronate dihydrate is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitine reabsorption.</p>
    Formule :C6H18N2O4
    Degré de pureté :≥98%
    Couleur et forme :Solid
    Masse moléculaire :182.22
  • Cilostazol

    CAS :
    <p>Cilostazol (OPC 21) is a Phosphodiesterase 3 Inhibitor. The mechanism of action of cilostazol is as a Phosphodiesterase 3 Inhibitor.</p>
    Formule :C20H27N5O2
    Degré de pureté :99.58% - 99.90%
    Couleur et forme :Off-White Solid
    Masse moléculaire :369.46
  • Zoxazolamine

    CAS :
    <p>Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant.</p>
    Formule :C7H5ClN2O
    Degré de pureté :99.54%
    Couleur et forme :Light Brown To Yellow-Brown Powder
    Masse moléculaire :168.58
  • Etofylline

    CAS :
    <p>Etofylline (Oxyphylline) is used for difficulty in breathing, asthma, breathing difficulty and other conditions.</p>
    Formule :C9H12N4O3
    Degré de pureté :99.36%
    Couleur et forme :Solid
    Masse moléculaire :224.22
  • Bis(4-cyanophenyl)methanol

    CAS :
    Bis(4-cyanophenyl)methanol (4, 4'-Dicyanobenzhydrol) is a metabolite of Letrozole.
    Formule :C15H10N2O
    Degré de pureté :98.55%
    Couleur et forme :White Or Off-White Crystalline Powder
    Masse moléculaire :234.25
  • Pimobendan

    CAS :
    <p>Pimobendan (UD-CG 115 BS) is a selective inhibitor of PDE3 (IC50: 0.32 μM).</p>
    Formule :C19H18N4O2
    Degré de pureté :99.91%
    Couleur et forme :Solid
    Masse moléculaire :334.37
  • Deferoxamine Mesylate

    CAS :
    <p>Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.</p>
    Formule :C26H52N6O11S
    Degré de pureté :94.68% - 99.8%
    Couleur et forme :Solid
    Masse moléculaire :656.79
  • Phenylhydantoin

    CAS :
    <p>5-Phenylhydantoin is a Mephenytoin metabolite with anti-epileptic effects, targeting NVSCs.</p>
    Formule :C9H8N2O2
    Degré de pureté :98.09% - 98.91%
    Couleur et forme :White Solid
    Masse moléculaire :176.17
  • K-604 dihydrochloride

    CAS :
    <p>K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.</p>
    Formule :C23H32Cl2N6OS3
    Degré de pureté :99.10% - 99.74%
    Couleur et forme :Solid
    Masse moléculaire :575.64
  • Cefadroxil

    CAS :
    <p>Cefadroxil (BL-S 578) is a Cephalosporin Antibacterial. The chemical classification of cefadroxil anhydrous is Cephalosporins.</p>
    Formule :C16H17N3O5S
    Degré de pureté :96.22% - 97.54%
    Couleur et forme :Solid
    Masse moléculaire :363.39
  • Mafenide hydrochloride

    CAS :
    <p>Mafenide hydrochloride (4-Aminomethylbenzenesulfonamide hydrochloride) is a sulfonamide that inhibits the enzyme carbonic anhydrase and is used as topical anti-</p>
    Formule :C7H11ClN2O2S
    Degré de pureté :98.34%
    Couleur et forme :Solid
    Masse moléculaire :222.69
  • ML-9

    CAS :
    <p>ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively.</p>
    Formule :C15H18Cl2N2O2S
    Degré de pureté :99.69%
    Couleur et forme :Crystalline Solid
    Masse moléculaire :361.29
  • BAMB-4

    CAS :
    <p>BAMB-4 inhibits ITPKA, impeding lung tumor cell metastasis, with an IC50 of 37 μM.</p>
    Formule :C15H12N2O2
    Degré de pureté :98.57%
    Couleur et forme :Solid
    Masse moléculaire :252.27
  • GSTO1-IN-1

    CAS :
    <p>GSTO1-IN-1 is a potent glutathione S-transferase omega 1 inhibitor (GSTO1; IC50: 31 nM).</p>
    Formule :C10H12Cl2N2O3S
    Degré de pureté :98.11% - 98.45%
    Couleur et forme :Solid
    Masse moléculaire :311.18
  • Rat PP(Pancreatic Polypeptide) ELISA Kit


    <p>This assay employs the competitive inhibition enzyme immunoassay technique. The microtiter plate provided in this kit has been pre-coated with Rat PP protein. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Rat PP. Next, Avidin conjugated to Horseradish Peroxidase (HRP) is added to each microplate well and incubated. After TMB substrate solution is added. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Rat PP in the samples is then determined by comparing the OD of the samples to the standard curve.</p>
  • Arhalofenate

    CAS :
    <p>Arhalofenate (JNJ 39659100) is a selective partial agonist of peroxisome proliferator-activated receptor PPARγ. It is used for the treatment of type 2 diabetes.</p>
    Formule :C19H17ClF3NO4
    Degré de pureté :98.97%
    Couleur et forme :Solid
    Masse moléculaire :415.79
  • (S)-(+)-N-3-Benzylnirvanol

    CAS :
    <p>(S)-(+)-N-3-Benzylnirvanol is a cytochrome P450 CYP2C19 inhibitor with a ki value of 82.5μM for CYP2C9 and 0.25μM for CYP2C19.Cost-effective and quality-assured.</p>
    Formule :C18H18N2O2
    Degré de pureté :98.90%
    Couleur et forme :Soild
    Masse moléculaire :294.35
  • DATPT

    CAS :
    <p>DATPT is a 12WLVSKF17 peptide mimetic molecule with anti-inflammatory and antimicrobial activities.DATPT inhibits the production of reactive oxygen species.</p>
    Formule :C24H39ClN6O3
    Degré de pureté :99.75%
    Couleur et forme :Solid
    Masse moléculaire :495.06