Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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MS1262-C3-amide-C10-amine
<p>MS1262-C3-amide-C10-amine is an E3 Ligase Ligand-Linker conjugate. It includes a GLP ligand targeting the E3 ligase SPOP and a PROTAC linker. This compound can be utilized in designing PROTACs such as example [MS479].</p>Couleur et forme :Odour SolidTKL-IN-1
<p>TKL-IN-1 (compound 7r) serves as an inhibitor of transketolase (Transketolase) and can be utilized as an herbicide. This compound effectively hampers the growth of Digitaria sanguinalis (Ds) and Amaranthus retroflexus (Ar).</p>Formule :C20H12ClN5OS2Couleur et forme :SolidMasse moléculaire :437.93Amiquinsin hydrochloride monohydrate
CAS :<p>Amiquinsin hydrochloride monohydrate is a compound known for its antihypertensive activity. It undergoes metabolism in the body, with its primary metabolite being 4-amino-6,7-dimethoxy-3-quinolineol hydrochloride monohydrate.</p>Formule :C11H15ClN2O3Couleur et forme :SolidMasse moléculaire :258.7DSPE-PEG5000-YIGSR
<p>DSPE-PEG5000-YIGSR is a PEG compound comprised of DSPE and the biomimetic peptide YIGSR. YIGSR interacts with the 67 kDa laminin-binding protein (LBP), enhancing the adhesion and proliferation of various cell types, such as endothelial cells, fibroblasts, and smooth muscle cells. DSPE-PEG5000-YIGSR is applicable for drug delivery.</p>Couleur et forme :Odour SolidL-Arginyl-L-alanine
CAS :<p>L-Arginyl-L-alanine is a dipeptide and acts as a vasodilator derived from vascular smooth muscle. It can elevate the levels of cyclic guanosine monophosphate (cGMP) and nitrite in endothelium-denuded artery rings.</p>Formule :C9H19N5O3Couleur et forme :SolidMasse moléculaire :245.28DSPE-PEG5000-LTLRWVGLMS
<p>DSPE-PEG5000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 serves as a receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG5000-LTLRWVGLMS can be utilized for drug delivery.</p>Couleur et forme :Odour SolidN-Acetyl-Ser-Asp-Lys-Pro TFA
N-Acetyl-Ser-Asp-Lys-Pro (TFA), a bone marrow tetrapeptide, is a specific ACE substrate for angiotensin conversion.Formule :C22H34F3N5O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :601.53Propiverine N-oxide
CAS :<p>Propiverine N-oxide is the primary metabolite of propiverine hydrochloride, and it influences bladder contraction and saliva secretion in miniature pigs.</p>Formule :C23H29NO4Couleur et forme :SolidMasse moléculaire :383.48[pTyr5] EGFR (988-993)
CAS :<p>'[pTyr5] EGFR (988-993) is a phosphorylated peptide from EGFR's Tyr992 site, often bound to inactive PTP1B.</p>Formule :C31H45N6O17PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :804.69GS-704277
CAS :<p>GS-704277, a Remdesivir metabolite, shows potent in vitro effects against COVID-19.</p>Formule :C15H19N6O8PCouleur et forme :SolidMasse moléculaire :442.325Cirsiliol 4′-glucoside
CAS :<p>Cirsiliol 4′-glucoside, a compound extracted from Ruellia tuberosa L., acts as a free radical scavenger and demonstrates potential anti-diabetic activity [1].</p>Formule :C23H24O12Couleur et forme :SolidMasse moléculaire :492.43Menthol glucuronide
CAS :<p>Menthol glucuronide is a metabolite of L-(-)-Menthol, the natural form of Methanol.</p>Formule :C16H28O7Couleur et forme :SolidMasse moléculaire :332.39BDM_92499
<p>BDM_92499 is a nanomolar, selective IRAP inhibitor with an IC50 of 3.4 nM. It also inhibits ERAP1 and ERAP2, with IC50 values of 0.46 μM and 4.2 μM, respectively.</p>Couleur et forme :Odour SolidAtocalcitol
CAS :<p>Atocalcitol is a vitamin D analog. It also acts as an agonist of alcitriol receptor.</p>Formule :C32H46O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :494.71Geranylgeranyl pyrophosphate
CAS :<p>Geranylgeranyl pyrophosphate: a metabolite for protein modification and diterpenoid precursor, used in cancer research.</p>Formule :C20H36O7P2Couleur et forme :SolidMasse moléculaire :450.44DL-TBOA ammonium
CAS :<p>DL-TBOA ammonium is a potent EAAT inhibitor with IC50 (6-70 μM) and Ki (3.2-42 μM) against EAAT1-5, blocking [14C]glutamate uptake.</p>Formule :C11H16N2O5Couleur et forme :SolidMasse moléculaire :256.258Orotidine 5′-monophosphate
CAS :<p>Orotidine 5′-monophosphate, a pyrimidine ribonucleoside, functions as an endogenous metabolite in human, E.</p>Formule :C10H13N2O11PCouleur et forme :SolidMasse moléculaire :368.191L-Amino acid oxidase
CAS :<p>L-Amino acid oxidase catalyzes the oxidative deamination of L-amino acids, which have local oxidative effects as well as potent antimicrobial effects.</p>Couleur et forme :SolidPDE5-IN-10
<p>PDE5-IN-10 (compound 4b), a potent phosphodiesterase type 5 (PDE5) inhibitor, exhibits an effective half-maximal inhibitory concentration (IC50) of 20 nM,</p>Formule :C21H20N4O2Couleur et forme :SolidMasse moléculaire :360.419(S)-HOTrE
CAS :<p>9(S)-HOTrE is a plant metabolite and octadecatrienoic acid produced by the action of 5-lipoxygenase (5-LO) on α-linolenic acid.</p>Formule :C18H30O3Couleur et forme :SolidMasse moléculaire :294.434'-Methoxyisoagarotetrol
CAS :<p>4'-Methoxyisoagarotetrol, a chromone derivative, exhibits moderate phosphodiesterase 3A (PDE3A) inhibitory activity with an IC50 value of 54 μM [1].</p>Formule :C18H20O7Couleur et forme :SolidMasse moléculaire :348.35Porcine Factor Xa
CAS :<p>PorcineFactor Xa is obtained by activating purified Porcine Factor X using Russells' Viper Venom, after which the venom is removed.</p>Couleur et forme :SolidTrifluoperazine N-Glucuronide
CAS :<p>Trifluoperazine N-Glucuronide is a metabolite of Trifluoperazine with antidepressant and antipsychotic activity.</p>Formule :C27H32F3N3O6SCouleur et forme :SolidMasse moléculaire :583.62Sinbaglustat
CAS :<p>Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.</p>Formule :C11H23NO4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :233.3cis-Vitamin K1
CAS :<p>Cis-Vitamin K1 is an endogenous metabolite of Vitamin K [1] .</p>Formule :C31H46O2Couleur et forme :SolidMasse moléculaire :450.70(S)-3,4-Dihydroxybutyric acid
CAS :<p>(S)-3,4-Dihydroxybutyric acid is a human urinary metabolite.</p>Formule :C4H8O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :120.1CP-610431
CAS :<p>CP-610431 inhibits ACC1/ACC2 (nonselective) with ~50 nM IC50, potentially aiding metabolic syndrome research.</p>Formule :C30H37N3O2Couleur et forme :SolidMasse moléculaire :471.645IONIS PTP1BRx
CAS :<p>IONIS PTP1BRx (ISIS 404173) acts as an antisense inhibitor of protein tyrosine phosphatase 1B (PTP-1B). This compound exhibits anti-diabetic properties, making it suitable for research into insulin resistance related to obesity and type 2 diabetes.</p>Couleur et forme :SolidVitamin K1 2,3-epoxide
CAS :<p>Vitamin K1 2,3-epoxide (Phylloquinone oxide) is reduced to vitamin k and is involved in the vitamin k cycle.</p>Formule :C31H46O3Degré de pureté :98% - 98.05%Couleur et forme :SolidMasse moléculaire :466.7Methylcardol triene
CAS :<p>Methylcardol triene, a phenolic compound present in cashew nut shell liquid, demonstrates α-glucosidase inhibition (IC50= 39.6 µM) and exhibits schistosomicidal properties by eliminating 100% of adult S. mansoni worms within 24 hours at 100 and 200 µM concentrations. Moreover, it serves as a precursor for synthesizing mono- and bis-benzoxazines.</p>Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.496α-Hydroxytamoxifen
CAS :<p>α-Hydroxytamoxifen is a metabolite of tamoxifen. It reacts with DNA and causes the formation of DNA adducts.</p>Formule :C26H29NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.51ZD-2138
CAS :<p>ZD-2138: Selective 5-LOX inhibitor, eases allergen-induced asthma attacks and airway constriction in guinea pigs.</p>Formule :C23H24FNO4Degré de pureté :99.68% - >99.99%Couleur et forme :SolidMasse moléculaire :397.44DSPE-PEG2000-NYZL1
<p>DSPE-PEG2000-NYZL1 is a PEG compound composed of DSPE and NYZL1. NYZL1 has the ability to specifically bind to bladder cancer tissues and cells. DSPE-PEG2000-NYZL1 is suitable for drug delivery applications.</p>Couleur et forme :Odour SolidDSPE-PEG1000-WYRGRL
<p>DSPE-PEG1000-WYRGRL consists of DSPE and a cartilage-targeting peptide (WYRGRL) as a PEG compound. WYRGRL is a type II collagen-targeting peptide that can bind to type II collagen α1. DSPE-PEG1000-WYRGRL is suitable for drug delivery applications.</p>Couleur et forme :Odour SolidhCA/VEGFR-2-IN-4
<p>hCA/VEGFR-2-IN-4 (compound 15b), an indolinylbenzenesulfonamide, serves as a potential dual inhibitor targeting cancer-related human carbonic anhydrases hCA IX/</p>Formule :C22H23FN6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :502.52Myristelaidic Acid
CAS :<p>Myristelaidic Acid is a natural product for research related to life sciences. The catalog number is T37358 and the CAS number is 50286-30-1.</p>Formule :C14H26O2Couleur et forme :SolidMasse moléculaire :226.35ATP ditromethamine
CAS :<p>ATP ditromethamine is key for energy storage, metabolism, and acts as a coenzyme and signaling molecule in immunity and inflammation.</p>Formule :C18H38N7O19P3Couleur et forme :SolidMasse moléculaire :749.45H-Ile-Pro-Pro-OH
CAS :<p>H-Ile-Pro-Pro-OH, a milk-derived peptide, inhibits angiotensin-converting enzyme (ACE)[1] with an IC50 of 5 μM.</p>Formule :C16H27N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :325.4(±)13(14)-DiHDPA
CAS :<p>(±)13(14)-DiHDPA is a metabolite of docosahexaenoic acid that is produced via oxidation by cytochrome P450 epoxygenases.</p>Formule :C22H34O4Couleur et forme :SolidMasse moléculaire :362.51CAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formule :C23H21N5O3SCouleur et forme :SolidMasse moléculaire :447.51Tetrahydrothiophen-3-one
CAS :<p>Tetrahydrothiophen-3-one can be used as food spices.</p>Formule :C4H6OSDegré de pureté :98.67%Couleur et forme :LiquidMasse moléculaire :102.154,12-Dimethoxy-6-(7,8-dihydroxy-7,8-dihydrostyryl)-2-pyrone
CAS :<p>4,12-Dimethoxy-6-(7,8-dihydroxy-7,8-dihydrostyryl)-2-pyrone is a microbial metabolism of yangonin, a major styryl lactone from Piper methysticum.</p>Formule :C14H12O5Degré de pureté :99.67%Couleur et forme :SoildMasse moléculaire :260.24Mersalyl
CAS :<p>Mersalyl is an organic mercurial diuretic.</p>Formule :C13H16HgNNaO6Couleur et forme :SolidMasse moléculaire :505.854N1-Acetylspermine
CAS :<p>N1-Acetylspermine, an endogenous metabolite found in urine, has applications in leukemia research [1] [2].</p>Formule :C12H28N4OCouleur et forme :SolidMasse moléculaire :244.382-(2',3',4'-Trihydroxybutyl)quinoxaline
CAS :<p>2-(2',3',4'-Trihydroxybutyl)quinoxaline is a food metabolite.</p>Formule :C12H14N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :234.25TSPO/Carbonic Anhydrase Modulator 1
<p>TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.</p>Formule :C35H51N3O3Couleur et forme :SolidMasse moléculaire :561.7985(S)-HPETE
CAS :<p>5(S)-HpETE is a PUFA made by 5-LO from arachidonic acid, metabolized into LTA4, a key leukotriene precursor.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472α-1,3-Galactosyltransferase (GTB)
CAS :<p>alpha-1,3-Galactosyltransferase (GTB) synthesizes α-Gal epitopes by transferring galactose to specific acceptors.</p>Couleur et forme :SolidEpoxide hydrolase
CAS :<p>Epoxide hydrolase, an enzyme responsible for catalyzing the reaction of epoxides with water to convert epoxy groups into diols, plays a crucial role in the metabolism of environmental pollutants and lipids. It is instrumental in detoxification, inflammatory responses, and regulating the health of the cardiovascular system. Additionally, Epoxide hydrolase is used in asymmetric catalytic reactions, such as the asymmetric ring-opening of epoxides, which are important for the synthesis of chiral pharmaceutical molecules.</p>Couleur et forme :SolidThymopentin acetate
CAS :<p>Thymopentin acetate: an immunomodulatory peptide from thymus cells with a 30-sec half-life, boosts T-cell production from hESCs.</p>Formule :C32H53N9O11Couleur et forme :SolidMasse moléculaire :739.82Etavopivat
CAS :<p>Etavopivat activates PKR in RBCs; taken orally, prevents sickling.</p>Formule :C22H23N3O6SCouleur et forme :SolidMasse moléculaire :457.5PTP1B-IN-22
CAS :<p>PTP1B-IN-22 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that inhibits glucose uptake in skeletal muscle L6 myotubes.</p>Formule :C16H12N2O3S2Degré de pureté :98.35%Couleur et forme :SoildMasse moléculaire :344.41ADP-specific glucokinase
CAS :<p>ADP-specific glucokinase, expressed in thermophilic archaea, is an ADP-specific enzyme that catalyzes the conversion of glucose to glucose-6-phosphate, thereby facilitating glycolysis. This enzyme can activate T cells and enhance the phagocytic activity of macrophages. It is used in research related to metabolic disorders, neurological diseases, and tumors.</p>Couleur et forme :SolidZaragozic acid D(2)
CAS :<p>Zaragozic acid D(2) inhibits squalene synthase and ras farnesyl-protein transferase isolated from the keratinophilic fungus Amauroascus niger.</p>Formule :C36H50O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :706.77Hydroorotic acid
CAS :<p>Hydroorotic acid（Dihydroorotic acid） is an endogenous metabolite，a potential biomarker for diabetic nephropathy and adrenal pheochromocytoma.</p>Formule :C5H6N2O4Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :158.11Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS :<p>ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.</p>Formule :C12H10ClNO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :251.67Equilenin
CAS :<p>Equilenin (E 400) is a natural estrogen that is an endocrine disruptor and has been used in breast cancer research.</p>Formule :C18H18O2Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :266.33Raloxifene 6,4'-Bis-β-D-glucuronide
CAS :<p>Raloxifene 6,4'-Bis-β-D-glucuronide is a Raloxifene metabolite. Raloxifene is a selective antagonist of estrogen receptor for the prevention of osteoporosis.</p>Formule :C40H43NO16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :825.83Secaubryenol
CAS :<p>Secaubryenol is a 3,4-secocycloartane triterpenes isolated from Coussarea macrophylla.</p>Formule :C30H48O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.7Amidepsine A
CAS :<p>Amidepsine A is a natural product for research related to life sciences. The catalog number is T22187 and the CAS number is 169181-28-6.</p>Couleur et forme :SolidMasse moléculaire :567.5415α-Hydroxy-6-keto cholesterol
CAS :<p>Yakkasterone is a major metabolite of cholesterol formed during exposure of lung epithelial cells to ozone.</p>Formule :C27H46O3Couleur et forme :SolidMasse moléculaire :418.662Febuxostat Acyl Glucuronide
CAS :<p>Febuxostat acyl glucuronide, a febuxostat metabolite, forms through UGTs catalyzed glucuronidation.</p>Formule :C22H24N2O9SCouleur et forme :SolidMasse moléculaire :492.5Captopril disulfide
CAS :<p>Captopril disulfide, a metabolite of Captopril, is a new antihypertensive agent.</p>Formule :C18H28N2O6S2Couleur et forme :SolidMasse moléculaire :432.56FPI-1523 sodium
CAS :<p>FPI-1523 sodium, avibactam derivative; β-lactamase inhibitor (Kd: CTX-M-15, 4nM; OXA-48, 34nM); PBP2 inhibitor (IC50, 3.2μM); strong antibacterial.</p>Formule :C9H13N4NaO7SDegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :344.27ACAT-IN-10
CAS :<p>ACAT-IN-10, from EP1236468A1 ex. 197, is an ACAT inhibitor with mild NF-κB blocking action.</p>Formule :C35H56N4O5SCouleur et forme :SolidMasse moléculaire :644.92N-Demethylerythromycin A
CAS :<p>N-Demethylerythromycin A, a metabolite of erythromycin from S. erythreus, may contaminate its preparations.</p>Formule :C36H65NO13Couleur et forme :SolidMasse moléculaire :719.9PDE4-IN-13
<p>PDE4-IN-13 is a phosphodiesterase 4 (PDE4) inhibitor exhibiting anti-inflammatory and antioxidant activities, with an half maximal inhibitory concentration (</p>Formule :C20H20O5Couleur et forme :SolidMasse moléculaire :340.37N-Acetylhexosamine kinase (NahK)
CAS :<p>NahK phosphorylates GlcNAc/GalNAc at C1 using ATP to form GlcNAc-1P/GalNAc-1P.</p>Couleur et forme :SolidCholesterol nervonate
CAS :<p>Cholesterol nervonate is a cholesterol ester found in human meibum, used experimentally in synthetic liposomes for biophysics and drug delivery research.</p>Formule :C51H90O2Couleur et forme :SolidMasse moléculaire :735.26Aldosterone-d8
CAS :<p>Aldosterone D8, a deuterium-labeled variant of Aldosterone produced in the adrenal zona glomerulosa, regulates blood pressure.</p>Formule :C21H28O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.49Mevinolinic acid
CAS :<p>Mevinolinic acid is an active metabolite of Lovastatin. Lovastatin is an HMG-CoA reductase inhibitor.</p>Formule :C24H38O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :422.562α-Lactose hydrate
CAS :<p>α-Lactose (hydrate) (α-D-Lactose (hydrate)), the main carbohydrate in mammalian milk, comprises two sugar units: glucose and galactose, and occurs as two</p>Formule :C12H24O12Couleur et forme :SolidMasse moléculaire :360.31DSPE-PEG2000-CREKA
<p>DSPE-PEG3000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide targets tumor cells and tumor vasculature, exhibiting antitumor activity. DSPE-PEG3000-CREKA is useful in drug delivery applications.</p>Couleur et forme :Odour SolidAntibacterial agent 237
<p>Anti bacterial agent 237 (compound Ru-8) acts as a potent antibacterial agent against Staphylococcus aureus, exhibiting minimum inhibitory concentrations (MICs) ranging from 0.78 to 1.56 μg/mL. It works by disrupting bacterial cell membranes, altering their permeability, and inducing the production of reactive oxygen species, which leads to bacterial cell death without promoting resistance. Additionally, Anti bacterial agent 237 demonstrates low hemolytic toxicity towards rabbit erythrocytes and Raw 264.7 cells. It has shown significant antibacterial activity in models of skin wound infections in mice and larval infections by the greater wax moth, effectively combating Staphylococcus aureus infections.</p>Formule :C65H69Cl3N10RuS2Couleur et forme :SolidMasse moléculaire :1261.87Isodihydroauroglaucin
CAS :<p>Isodihydroauroglaucin is a useful organic compound for research related to life sciences. The catalog number is T124274 and the CAS number is 74886-31-0.</p>Formule :C19H24O3Couleur et forme :SolidMasse moléculaire :300.398DSPE-PEG5000-APRPG
<p>DSPE-PEG5000-APRPG is a PEG compound composed of DSPE and the APRPG peptide, utilized for drug delivery.</p>Couleur et forme :Odour Solid11(R)-HETE
CAS :<p>11(R)-HETE aids in oocyte maturation in sea urchins and tentacle regeneration in hydras; it is also made by aspirin-influenced COX-2 and arachidonic acid.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473IP3RPEP6
CAS :<p>IP3RPEP6 serves as a competitive inhibitor of IP3R. Its IC50 values for IP3R1, IP3R2, and IP3R3 are 9.0 μM, 3.9 μM, and 4.3 μM, respectively. This compound does not affect ryanodine receptors and Cx43 hemichannels, and it is capable of modulating intracellular calcium signaling.</p>Formule :C49H79N15O24Couleur et forme :SolidMasse moléculaire :1262.24TAT-cyclo-CLLFVY
CAS :<p>Blocks HIF-1α/β dimerization, not HIF-2α; suppresses VEGF, CAIX in cancer cells; antiangiogenic in HUVECs (IC50 = 1.3 μM).</p>Formule :C111H188N42O24S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2559.1UDP-α-D-Glucose sodium hydrate
<p>UDP-α-D-Glucose sodium hydrate is an endogenous metabolite and a pyrimidine nucleotide sugar, involved in glycosylation reactions during metabolic</p>Formule :C15H24N2Na2O18P2Couleur et forme :SolidMasse moléculaire :628.28Carbonic anhydrase inhibitor 32
<p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>Formule :C17H16N6O3SCouleur et forme :SolidMasse moléculaire :384.41BAY-588
CAS :<p>BAY-588 is an inactive control probe of BAY-876 which is an inhibitor of GLUT1.</p>Formule :C27H25F4N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.51Leucine dehydrogenase
CAS :<p>Leucine dehydrogenase from Bacillus spheroides oxidizes/reduces branched-chain amino acids and their keto analogs.</p>Couleur et forme :SolidBIRM 271
CAS :<p>BIRM 271 is a novel arachidonic acid release inhibitor that blocks leukotriene B4 and platelet-activating factor biosynthesis in human neutrophils.</p>Formule :C21H25N3ODegré de pureté :99.64%Couleur et forme :SoildMasse moléculaire :335.44DSPE-PEG2000-R6H4
<p>DSPE-PEG2000-R6H4 is a PEG compound composed of DSPE and a pH-responsive cell-penetrating peptide (R6H4). The R6H4 component is utilized for pH-responsive anticancer drug delivery. Additionally, DSPE-PEG2000-R6H4 is applicable in drug delivery systems.</p>Couleur et forme :Odour Solidα-Glucosidase-IN-85
<p>α-Glucosidase-IN-85 (Compound 8D1) functions as an inhibitor of α-Glucosidase, with an IC50 of 5.43 μM. This compound is useful for research related to type 2 diabetes.</p>Couleur et forme :Odour SolidO-Desmethyl apixaban
CAS :<p>O-Desmethyl apixaban is a metabolite of Apixaban, a selective Factor Xa inhibitor with Ki of 0.08 nM in humans.</p>Formule :C24H23N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.47DHODH-IN-23
CAS :<p>DHODH-IN-23 is a DHODH inhibitor with oral activity. DHODH-IN-23 is often used in cancer research.</p>Formule :C24H21ClFNO4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :441.88ATX inhibitor 7
CAS :<p>ATX inhibitor 7 is a autotaxin inhibitor and shows good oral exposure.</p>Formule :C21H22F3N7O2Couleur et forme :SolidMasse moléculaire :461.449ZINC77292789
CAS :<p>ZINC77292789 (Fmoc-Thr[GalNAc(Ac)3-α-D]-OH) is a reagent for the preparation of a synthetic MUC1 Glycopeptide Bearing βGalNAc-Thr as a Tn antigen isomer which</p>Formule :C33H38N2O13Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :670.66Sofosbuvir impurity C
CAS :<p>Sofosbuvir impurity C, a less active byproduct, inhibits HCV RNA replication and exhibits strong anti-HCV effects.</p>Formule :C22H29FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.45Lurasidone Metabolite 14283 hydrochloride
CAS :Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone.Formule :C28H37ClN4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :545.14[(3R)-3-Hydroxydodecanoyl]-L-carnitine
CAS :<p>[(3R)-3-Hydroxydodecanoyl]-L-carnitine is an endogenous metabolite[1].</p>Formule :C19H37NO5Couleur et forme :SolidMasse moléculaire :359.50N-acetyl Leukotriene E4
CAS :<p>N-acetyl Leukotriene E4 is an endogenous metabolite of Leukotriene E4, less active than Leukotriene E4, causing constriction of the airways.</p>Formule :C25H39NO6SCouleur et forme :SolidMasse moléculaire :481.653-HIB
CAS :<p>3-HIB is a paracrine regulator of transendothelial fatty acid transport.</p>Formule :C4H7NaO3Couleur et forme :SolidMasse moléculaire :126.09(1R,2R)-MK-8189
CAS :<p>(1R,2R)-MK-8189 is an isomer of MK-8189, a potent and selective pyrimidine PDE10A inhibitor.</p>Formule :C19H22N6OSDegré de pureté :>99.99% - >99.99%Couleur et forme :SoildMasse moléculaire :382.481-Methylhistamine
CAS :<p>2-(1-Methyl-1H-imidazol-4-yl)ethan-1-amine is a histamine metabolite.</p>Formule :C6H11N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :125.1716DSPE-PEG1000-pPB
<p>DSPE-PEG1000-pPB is a PEG compound consisting of DSPE and a cyclic oligopeptide (pPB). The pPB component exhibits a strong binding affinity to PDGFRβ, which is overexpressed in activated hepatic stellate cells (HSC). DSPE-PEG1000-pPB is applicable for drug delivery.</p>Couleur et forme :Odour SolidOphiobolin A
CAS :<p>Ophiobolin A: Fungal metabolite, phytotoxin, inhibits calmodulin-activated phosphodiesterase (IC50: 9μM), with antimicrobial and anticancer properties.</p>Formule :C25H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.559CE(20:5(5Z,8Z,11Z,14Z,17Z)
CAS :CE(20:5(5Z,8Z,11Z,14Z,17Z) is an endogenous metabolite.Formule :C47H74O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :671.09
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