Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(196 produits)
- Caséine Kinase(138 produits)
- DHFR(32 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(85 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(134 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(86 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(22 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(45 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9182 produits trouvés pour "Métabolisme"
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Lp-PLA2-IN-3
CAS :Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.Formule :C20H13ClF3N3O3SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :467.85Ref: TM-T11874
1mg90,00€2mg132,00€5mg215,00€10mg340,00€25mg565,00€50mg797,00€100mg1.063,00€500mg2.142,00€1mL*10mM (DMSO)220,00€Sch 34826
CAS :Sch 34826 is a potent, selective neutral endopeptidase inhibitor.Formule :C27H34N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.57NPD-1335
CAS :NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.Formule :C28H29N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.55α-Amylase/α-Glucosidase-IN-2
CAS :α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μMFormule :C22H16ClN5Couleur et forme :SolidMasse moléculaire :385.85D-threo-PPMP hydrochloride
CAS :D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.Formule :C29H51ClN2O3Couleur et forme :SolidMasse moléculaire :511.19Xanthine oxidase-IN-5
CAS :Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.Formule :C18H16FN3O3Couleur et forme :SolidMasse moléculaire :341.34ICI 153110
CAS :ICI 153110: Oral phosphodiesterase inhibitor for treating congestive heart failure, has inotropic, vasodilator effects.Formule :C11H11N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :201.22hCAIX-IN-8
CAS :hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.Formule :C19H16N4O6Couleur et forme :SolidMasse moléculaire :396.35PRRSV/CD163-IN-1
CAS :PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.Formule :C25H24FN5O5S2Couleur et forme :SolidMasse moléculaire :557.62Xanthine oxidase-IN-4
CAS :Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.Formule :C15H13N5O2Couleur et forme :SolidMasse moléculaire :295.3DP00477
CAS :DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.Formule :C17H11ClF3N3OSCouleur et forme :SolidMasse moléculaire :397.8PDE4-IN-11
CAS :PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.Formule :C21H19FN2O2Couleur et forme :SolidMasse moléculaire :350.39ENPP1 inhibitor 43
CAS :ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.Formule :C16H18N6O3SCouleur et forme :SolidMasse moléculaire :374.42MY33-3 hydrochloride
CAS :MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.Formule :C16H14ClF6NS2Couleur et forme :SolidMasse moléculaire :433.86hCAXII-IN-1
CAS :hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.Formule :C20H17NO5Couleur et forme :SolidMasse moléculaire :351.3524(S),25-Epoxycholesterol
CAS :24(S),25-Epoxycholesterol is an oxysterol agonist of the liver X receptor.Formule :C27H44O2Couleur et forme :SolidMasse moléculaire :400.64FABP-IN-2
CAS :FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.Formule :C25H21ClN2O3Couleur et forme :SolidMasse moléculaire :432.9A-908292
CAS :A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.Formule :C18H20N2O4SCouleur et forme :SolidMasse moléculaire :360.43Arasertaconazole
CAS :Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.Formule :C20H15Cl3N2OSCouleur et forme :SolidMasse moléculaire :437.77IDO1-IN-15
CAS :IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.Formule :C13H14BrFN6O3Couleur et forme :SolidMasse moléculaire :401.19Carbonic anhydrase inhibitor 7
CAS :Potent hCA inhibitor; targets hCA IX, II, XII, I with Ki: 6.5, 7.1, 72.1, 255.8 nM respectively.Formule :C23H17N3O5SCouleur et forme :SolidMasse moléculaire :447.46hCA IX-IN-2
hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferativeFormule :C23H24N2O4STeCouleur et forme :SolidMasse moléculaire :552.11Spirapril
CAS :Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.Formule :C22H30N2O5S2Couleur et forme :SolidMasse moléculaire :466.613,3-Dimethyl-1-butanol
CAS :3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.Formule :C6H14OCouleur et forme :SolidMasse moléculaire :102.17α-Glucosidase-IN-21
CAS :α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.Formule :C24H23NO2SCouleur et forme :SolidMasse moléculaire :389.51Antitumor agent-88
CAS :Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).Formule :C23H30N2O7SCouleur et forme :SolidMasse moléculaire :478.56PKM2 activator 4
CAS :PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.Formule :C16H16N2O4SCouleur et forme :SolidMasse moléculaire :332.37Fmoc-5-aminopentanoic acid
CAS :Fmoc-5-aminopentanoic acid: alkane, Fmoc-protected amine, carboxyl group, PROTAC linker, deprotects to free amine, forms amides with activators.Formule :C20H21NO4Couleur et forme :SolidMasse moléculaire :339.39hCAIX-IN-14
CAS :hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .Formule :C11H17ClN6O2SCouleur et forme :SolidMasse moléculaire :332.81ATX inhibitor 8
CAS :ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).Formule :C28H26N10OCouleur et forme :SolidMasse moléculaire :518.57hCAIX-IN-3
CAS :hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.Formule :C21H21BrN6O4SCouleur et forme :SolidMasse moléculaire :533.4CP 80633
CAS :CP 80633 is a PDE4 inhibitor.Formule :C18H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :316.39PDE11-IN-1
CAS :PDE11-IN-1 is a PDE11 inhibitor and can be used for adrenal insufficiency research [1].Formule :C16H10ClN3O3SCouleur et forme :SolidMasse moléculaire :359.79mEH-IN-1
CAS :mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.Formule :C16H17F6NOSCouleur et forme :SolidMasse moléculaire :385.37SYN20028567
CAS :SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].Formule :C20H29N3O3SCouleur et forme :SolidMasse moléculaire :391.53FAAH-IN-7
FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.Formule :C26H29N3O4Couleur et forme :SolidMasse moléculaire :447.53Enpp-1-IN-8
CAS :Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.Formule :C19H26N6O4SCouleur et forme :SolidMasse moléculaire :434.51MDK-4823
CAS :MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.Formule :C28H36N4OCouleur et forme :SolidMasse moléculaire :444.61Umbralisib tosylate
CAS :Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.Formule :C38H32F3N5O6SCouleur et forme :SolidMasse moléculaire :743.75JNJ-61803534
CAS :JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.Formule :C23H23Cl2F6N3O4SCouleur et forme :SolidMasse moléculaire :622.41GKA-71
CAS :GKA-71 is an effective glucokinase activator (GKA).Formule :C21H23N3O6S2Couleur et forme :SolidMasse moléculaire :477.55Umbralisib sulfate
CAS :Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.Formule :C31H26F3N5O7SCouleur et forme :SolidMasse moléculaire :669.63Liarozole HCl
CAS :Liarozole HCl: antineoplastic, boosts ATRA levels, impedes cell growth, promotes differentiation, aromatase inhibitor.Formule :C17H14Cl2N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.23Delapril
CAS :Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.Formule :C26H32N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.54Metyltetraprole
CAS :Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.Formule :C19H17ClN6O2Couleur et forme :SolidMasse moléculaire :396.83α-Glucosidase-IN-9
CAS :α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].Formule :C19H12N4OSCouleur et forme :SolidMasse moléculaire :344.39HIF-1α-IN-3
CAS :HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].Formule :C19H17N5O2Couleur et forme :SolidMasse moléculaire :347.37GNX-865
CAS :GNX-865 is an inhibitor of mitochondrial permeability transition pore (mtPTP).Formule :C16H14ClNO3Couleur et forme :SolidMasse moléculaire :303.74Agn 190727
CAS :Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.Formule :C20H22O2Couleur et forme :SolidMasse moléculaire :294.39α-Glycosidase-IN-1
CAS :α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).Formule :C21H19N9O6S2Couleur et forme :SolidMasse moléculaire :557.56Glucosylceramide synthase-IN-1
CAS :Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.Formule :C24H20F4N2O3Couleur et forme :SolidMasse moléculaire :460.42α-Amylase-IN-2
CAS :α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =Formule :C39H52BrNO4Couleur et forme :SolidMasse moléculaire :678.74HIF-PHD-IN-2
CAS :HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].Formule :C17H15N5O3SCouleur et forme :SolidMasse moléculaire :369.4LEO-29102
CAS :LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.Formule :C20H22Cl2N2O5Couleur et forme :SolidMasse moléculaire :441.31DHODH-IN-21
CAS :DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.Formule :C20H19ClF4N6O4Couleur et forme :SolidMasse moléculaire :518.85Chaetomellic acid A
CAS :Chaetomellic acid A inhibits farnesyltransferase (IC50=55nM), not active in cells, and selective over geranylgeranyltransferases (IC50: 92µM, 34µM).Formule :C19H34O4Couleur et forme :SolidMasse moléculaire :326.47Lp-PLA2-IN-11
CAS :Lp-PLA2-IN-11, a potent Lp-PLA2 inhibitor, may be explored for atherosclerosis and Alzheimer's (WO2014114249A1, E145).Formule :C22H20F4N4O3Couleur et forme :SolidMasse moléculaire :464.41α-Glucosidase-IN-20
CAS :α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.Formule :C23H21NOSCouleur et forme :SolidMasse moléculaire :359.48TMCB
CAS :CK2 and ERK8 inhibitorFormule :C11H9Br4N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.82BMS 740808
CAS :BMS-740808 is a highly effective and selective factor X inhibitor.Formule :C31H27F3N6O3Couleur et forme :SolidMasse moléculaire :588.58(Rac)-3′-Hydroxy simvastatin
CAS :(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.Formule :C25H38O6Couleur et forme :SolidMasse moléculaire :434.57Trandolaprilat
CAS :Trandolaprilat is an inhibitor of non-sulfhydryl angiotensin-converting enzyme.Formule :C22H30N2O5Couleur et forme :Pale Yellow SolidMasse moléculaire :402.48HX-600
CAS :HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.Formule :C29H30N2O2Couleur et forme :SolidMasse moléculaire :438.56YM-75466
CAS :YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.Formule :C28H35N5O8S2Couleur et forme :SolidMasse moléculaire :633.74GNE-3500
CAS :GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.Formule :C24H30FN3O3SCouleur et forme :SolidMasse moléculaire :459.58SQ 28853
CAS :SQ 28853 is an inhibitor of ACE with diuretic properties.Formule :C19H25ClN4NaO6S3Couleur et forme :SolidMasse moléculaire :560.05SCD1-IN-1
CAS :SCD1-IN-1, a potent inhibitor of SCD1 (IC50: 5.8 nM), is valuable in dermatologic research [1].Formule :C20H20F3NO4Couleur et forme :SolidMasse moléculaire :395.37Xanthine oxidoreductase-IN-1
CAS :Xanthine oxidoreductase-IN-1 is a xanthine oxidoreductase (XOR) inhibitor with an IC 50 value of 7.0 nM.Formule :C18H20N4O2Couleur et forme :SolidMasse moléculaire :324.38ML202
CAS :ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.Formule :C18H17N3O3S2Couleur et forme :SolidMasse moléculaire :387.48JNJ-40413269
CAS :JNJ-40413269 inhibits FAAH, engages central targets, and is effective in rat neuropathic pain.Formule :C19H15ClF3N3OCouleur et forme :SolidMasse moléculaire :393.79hCAIX-IN-7
CAS :hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).Formule :C18H12FNO3Couleur et forme :SolidMasse moléculaire :309.29DMPAC-Chol
CAS :DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.Formule :C33H58N2O2Couleur et forme :SolidMasse moléculaire :514.83LAS-31180
CAS :LAS-31180 is a phosphodiesterase 3 inhibitor. It also has positive inotropic and vasodilator properties.Formule :C11H12N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :252.29Imidazoleacetic acid
CAS :Imidazoleacetic acid, an endogenous ligand, stimulates imidazole receptors.Formule :C5H6N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :126.11YM 26734
CAS :Competitive inhibitor of secretory phospholipase A2 (sPLA2)Formule :C45H62O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :730.97YC-001
CAS :YC-001: inverse agonist/antagonist for rod opsin, prevents light-induced retinal degeneration.Formule :C12H7ClO2S2Couleur et forme :SolidMasse moléculaire :282.77Y-29794
CAS :Y-29794, a covalent POP inhibitor with a Ki of 0.95 nM, holds research potential for neurodegenerative diseases and cancer.Formule :C22H32N2OS2Couleur et forme :SolidMasse moléculaire :404.63(E/Z)-Ensifentrine
CAS :RPL-554 (LS-193,855) is a dual PDE3/4 inhibitor with bronchodilator and anti-inflammatory properties, in trials for asthma and hay fever by Verona Pharma.Formule :C26H31N5O4Couleur et forme :SolidMasse moléculaire :477.56Glyoxalase I inhibitor 2
CAS :Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.Formule :C24H23N3O4SCouleur et forme :SolidMasse moléculaire :449.52Fluindione
CAS :Fluindione is a hematologic drug.Formule :C15H9FO2Couleur et forme :SolidMasse moléculaire :240.23URB532
CAS :URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.Formule :C18H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.36SAR127303
CAS :SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.Formule :C16H17ClF6N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.834,6-O-Ethylidene-α-D-glucose
CAS :4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucoseFormule :C8H14O6Couleur et forme :SolidMasse moléculaire :206.19ALDH3A1-IN-2
CAS :ALDH3A1-IN-2 is a potent inhibitor targeting ALDH3A1 (IC50=1.29µM), potentially useful in cancer research.Formule :C11H14N2O3Couleur et forme :SolidMasse moléculaire :222.24(Z)-10-Hydroxynortriptyline
CAS :(Z)-10-Hydroxynortriptyline ((Z)-10-Hydroxy Nortriptyline) is a norepinephrine reuptake inhibitor with antidepressant activity.Formule :C19H21NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.38Kojibiose
CAS :Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.Formule :C12H22O11Degré de pureté :99.933%Couleur et forme :SolidMasse moléculaire :342.3Ref: TM-T20839
1mg90,00€5mg178,00€10mg295,00€25mg560,00€50mg859,00€100mg1.108,00€200mg1.513,00€500mg2.242,00€1mL*10mM (DMSO)215,00€1-Methyluric acid
CAS :1-Methyluric acid (1-Methylurate) acts on the bladder mucosa and increases the levels of insulin, triglycerides, cholesterol, and blood glucose.Formule :C6H6N4O3Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :182.14PDE7-IN-2
CAS :PDE7-IN-2 is an inhibitor of phosphodiesterase 7 (IC50 = 2.1 µM) and can be used in Parkinson's disease studies.Formule :C14H11ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.77Imazodan
CAS :Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.Formule :C13H12N4ODegré de pureté :98% - 98.31%Couleur et forme :SolidMasse moléculaire :240.26AChE/hCA I/II-IN-1
CAS :Compound 6: Potent inhibitor for AChE, Hca I & II with IC50s of 22.21, 60.79, 66.64 nM, useful in glaucoma, Alzheimer's, diabetes research.Formule :C15H13N3SCouleur et forme :SolidMasse moléculaire :267.35IDO inhibitor 1
CAS :IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 <100 nM).with potential immunomodulating and antineoplastic activities.Formule :C11H13BrFN7O4SDegré de pureté :99.805%Couleur et forme :SolidMasse moléculaire :438.23Ref: TM-T7660
1mg94,00€2mg138,00€5mg192,00€10mg294,00€25mg427,00€50mg625,00€100mg889,00€500mg1.783,00€1mL*10mM (DMSO)220,00€Propentofylline
CAS :Propentofylline (Hextol) has neuroprotective, antiproliferative and anti-inflammatory activities and can be used in the study of Alzheimer's disease.Formule :C15H22N4O3Degré de pureté :99.76% - 99.86%Couleur et forme :Off-White SolidMasse moléculaire :306.36Ref: TM-T19812
1mg65,00€5mg138,00€10mg200,00€25mg339,00€50mg500,00€100mg710,00€1mL*10mM (DMSO)148,00€α-Glucosidase-IN-16
CAS :α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM.Formule :C22H18FNSCouleur et forme :SolidMasse moléculaire :347.45Teglicar
CAS :Teglicar is a selective and reversible liver isoform of carnitine palmitoyl-transferase 1 (L-CPT1) inhibitor.Formule :C22H45N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.61HSL-IN-1
CAS :HSL-IN-1 is an HSL inhibitor that significantly reduces the reactive metabolite load and reduces the release of free fatty acids from stored fat.Formule :C19H13BClF3N2O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :436.58hCAXII-IN-2
CAS :hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.Formule :C21H18ClN3O4Couleur et forme :SolidMasse moléculaire :411.84LGE-899
CAS :LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.Formule :C15H11F3O3Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :296.2411β-HSD1-IN-1
CAS :11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM), and used for the treatment of pain.Formule :C18H14ClF4N3ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :399.77Ref: TM-T10160
1mg52,00€5mg111,00€10mg163,00€25mg235,00€50mg330,00€100mg452,00€1mL*10mM (DMSO)118,00€sEH inhibitor-6
CAS :sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].Formule :C21H14ClN3O2Couleur et forme :SolidMasse moléculaire :375.81OHM1
CAS :OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53Formule :C24H42N6O5Couleur et forme :SolidMasse moléculaire :494.63
