Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Phenylpyropene A
CAS :<p>Phenylpyropene A, a P. griseofulvum fungus product, blocks ACAT (IC50=0.8μM) and DGAT, kills M. persicae at 5ppm.</p>Formule :C32H38O10Couleur et forme :SolidMasse moléculaire :582.64hCAI/II/IV-IN-28
CAS :<p>hCAI/II/IV-IN-28(WAY-638358) is a potent carbonic anhydrase inhibitor with potential anticonvulsant activity.</p>Formule :C14H15N3O3SDegré de pureté :96.48%Couleur et forme :SolidMasse moléculaire :305.35Antiproliferative agent-12
<p>Antiproliferative agent-10, a ruthenium(II) complex, inhibits cancer by blocking mitochondrial calcium uptake.</p>Formule :C46H40Cl2N6P2RuCouleur et forme :SolidMasse moléculaire :910.79Zabicipril HCl
CAS :<p>Zabicipril HCl（S 9650） is a potent angiotensin-converting enzyme inhibitor.</p>Formule :C23H33ClN2O5Degré de pureté :99.66%Couleur et forme :SoildMasse moléculaire :452.971-β-D-Glucosylsphingadienine (d18:2 (4E,8E))
CAS :<p>1-β-D-Glucosylsphingadienine is a glucosylsphingosine, which are deacetylated lysolipid derivatives of glucosylcerebrosides .</p>Formule :C24H45NO7Couleur et forme :SolidMasse moléculaire :459.6244,7,10,13,16-Docosapentaenoic acid
CAS :<p>4,7,10,13,16-Docosapentaenoic acid is an endogenous metabolite.</p>Formule :C22H34O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.51AV22-149
<p>AV22-149 (compound 22) is an inhibitor of Carbonic Anhydrase .</p>Formule :C23H28F3N3O6S2Couleur et forme :SolidMasse moléculaire :563.612-Chlorophenylboronic acid
CAS :<p>2-Chlorophenylboronic acid: A monohalogenated phenylboronic acid used in drug synthesis and as a fatty acid amidase inhibitor.</p>Formule :C6H6BClO2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :156.375-(3'-Hydroxyphenyl)-γ-Valerolactone
CAS :<p>5-(3'-Hydroxyphenyl)-γ-valerolactone, a metabolite resulting from the transformation of polyphenols such as (+)-catechin and (−)-epicatechin by gut microbiota,</p>Formule :C11H12O3Couleur et forme :SolidMasse moléculaire :192.21ARL67156 triethylamine
<p>ARL67156, a selective ecto-ATPase inhibitor, blocks NTPDase1, 3, and NPP1; used in calcific valve, asthma research. Ki: 11-18 μM.</p>Formule :C15H24Br2N5O12P3·3C6H15N)Couleur et forme :SolidMasse moléculaire :1154.23Secaubryenol
CAS :<p>Secaubryenol is a 3,4-secocycloartane triterpenes isolated from Coussarea macrophylla.</p>Formule :C30H48O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.7NAMPT degrader-3
<p>NAMPT Degrader-3 (compound C5) is a NAMPT degrader that functions through a VHL- and proteasome-dependent mechanism.</p>Formule :C56H74N8O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1003.3Mebeverine acid
CAS :<p>Mebeverine acid (Mebeverine metabolite Mebeverine acid) is a secondary metabolite of Mebeverine and can be used as a marker of oral exposure to Mebeverine.</p>Formule :C16H25NO3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :279.37SHP2-IN-37
<p>SHP2-IN-37 (compound C5) is a potent allosteric inhibitor selective for SHP2, with an IC50 of 0.023 μM. It exhibits antiproliferative effects on KYSE-520 and MV-411 cells, with IC50 values of 6.97 μM and 0.67 μM, respectively.</p>Formule :C19H22Cl2N4O2SCouleur et forme :SolidMasse moléculaire :440.08405PDK-IN-2
<p>PDK-IN-2 (Compound 1F), with an IC50 of 68 nM, is a potent PDK inhibitor that downregulates the expression of PDK1 and PDK4 in cells.</p>Formule :C17H23AsCl2N2O2S2Couleur et forme :SolidMasse moléculaire :497.33DP-1 hydrochloride
CAS :<p>DP-1 hydrochloride is a degradation product of SDC-TRAP-0063, a fragment of Ganetespib, a heat shock protein 90 (HSP90) inhibitor with antitumor activity.</p>Formule :C26H32ClN5O3Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :498.02Raloxifene 6,4'-Bis-β-D-glucuronide
CAS :<p>Raloxifene 6,4'-Bis-β-D-glucuronide is a Raloxifene metabolite. Raloxifene is a selective antagonist of estrogen receptor for the prevention of osteoporosis.</p>Formule :C40H43NO16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :825.8312α-Hydroxysteroid dehydrogenase
CAS :<p>12α-Hydroxysteroid dehydrogenase, an NAD-dependent enzyme expressed in Bacillus sphaericus, actively processes both free and conjugated bile salts. It is utilized to determine the levels of 12α-hydroxy bile acids in serum.</p>Couleur et forme :Solid21-Deoxy Cortisone
CAS :<p>21-Deoxy Cortisone (21-Desoxycortisone; NSC 38722) is a corticosteroid metabolite of 11-ketoprogesterone. It is generated from 11-ketoprogesterone by the cytochrome P450 (CYP) isoform CYP17A1, and can also be produced by oxidation via 11β-hydroxysteroid dehydrogenase type 2 (11β-HSD2) from 21-deoxycorticosterone. In patients with congenital adrenal hyperplasia, a metabolic disorder characterized by a deficiency of 21-hydroxylase, levels of 21-Deoxy Cortisone are elevated.</p>Formule :C21H28O4Couleur et forme :SolidMasse moléculaire :344.4413-cis Acitretin D3
CAS :<p>13-cis Acitretin D3, a deuterium-labeled metabolite of Acitretin, is a second-gen systemic retinoid.</p>Formule :C21H26O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.454Doxorubicinol
CAS :<p>Doxorubicinol is the major circulating metabolite of doxorubicin with antineoplastic acitivity.</p>Formule :C27H31NO11Couleur et forme :SolidMasse moléculaire :545.54BBOX-IN-1
<p>BBOX-IN-1 (compound 58) is a potent BBOX inhibitor with an IC50 of 0.02 μM, and it is applicable in research related to triple-negative breast cancer (TNBC).</p>Formule :C18H17N3O6SCouleur et forme :SolidMasse moléculaire :403.41(3S,5R)-Fluvastatin D6 sodium
CAS :<p>(3S,5R)-Fluvastatin D6 sodium: deuterium-labeled synthetic HMG-CoA reductase inhibitor with 8 nM IC50.</p>Formule :C24H25FNNaO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.49(S)-3,4-Dihydroxybutyric acid
CAS :<p>(S)-3,4-Dihydroxybutyric acid is a human urinary metabolite.</p>Formule :C4H8O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :120.1DSPE-PEG2000-LTLRWVGLMS
<p>DSPE-PEG2000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 is the receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG2000-LTLRWVGLMS can be utilized for drug delivery.</p>Couleur et forme :Odour SolidSuberylglycine
CAS :<p>Suberylglycine is an acyl glycine that is a normally minor metabolite of fatty acid.</p>Formule :C10H17NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.25CP-610431
CAS :<p>CP-610431 inhibits ACC1/ACC2 (nonselective) with ~50 nM IC50, potentially aiding metabolic syndrome research.</p>Formule :C30H37N3O2Couleur et forme :SolidMasse moléculaire :471.6459(S)-HpOTrE
CAS :<p>9(S)-HpOTrE, a product of 5-LO on α-linolenic acid, transforms into colnelenic acid and 9,16-dihydroperoxy acid; it inactivates LOs through epoxide formation.</p>Formule :C18H30O4Couleur et forme :SolidMasse moléculaire :310.434THX6
<p>THX6 is an activator of human mitochondrial protease ClpP, with an EC50 of 1.18 μM. It displays cytotoxicity in ONC201-resistant SU-DIPG-VI cells, with an IC50 of 0.13 μM. THX6 inhibits the expression of mitochondria-related proteins (such as parkin, TFAM, NRF1, SDHA), leading to impaired mitochondrial function. Additionally, THX6 affects cell membrane lipid metabolism and exhibits antitumor potential.</p>Formule :C22H18Cl2N4O2Couleur et forme :SolidMasse moléculaire :441.31Aromatase-IN-2
CAS :<p>Aromatase-IN-2 has anti-inflammatory, antitumor and antiasthmatic effects.</p>Formule :C17H22N2ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :270.37Adenosine 3',5'-diphosphate sodium salt
CAS :<p>Adenosine 3',5'-diphosphate sodium inhibits hydroxysteroid sulfotransferases and studies SULT kinetics/structure.</p>Formule :C10H15N5NaO10P2Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :450.192,3,4,6,7,8-Hexachlorodibenzofuran
CAS :<p>2,3,4,6,7,8-Hexachlorodibenzofuran (2,3,4,6,7,8-HxCDF) is a type of polychlorinated dibenzofuran (PCDF). It induces the expression of aryl hydrocarbon hydroxylase (AHH) and ethoxyresorufin-o-deethylase (EROD) genes in H-4-II-E rat hepatoma cells, with EC50 values of 0.687 and 0.575 nM, respectively.</p>Formule :C12H2Cl6OCouleur et forme :SolidMasse moléculaire :374.86E0924G
CAS :<p>E0924G is an orally active PPARδ agonist with an EC50 of 2.82 μM. It enhances the upregulation of osteoprotegerin (OPG) expression, with an EC50 of 0.29 μM. E0924G reduces RANKL-induced osteoclast differentiation and inhibits F-actin ring formation in RAW264.7 macrophages. Additionally, E0924G modulates bone density and bone loss in models of ovariectomy (OVX) and age-related osteoporosis.</p>Formule :C12H12N2O3Couleur et forme :SolidMasse moléculaire :232.24Vitamin K1 2,3-epoxide
CAS :<p>Vitamin K1 2,3-epoxide (Phylloquinone oxide) is reduced to vitamin k and is involved in the vitamin k cycle.</p>Formule :C31H46O3Degré de pureté :98% - 98.05%Couleur et forme :SolidMasse moléculaire :466.7Pregnant mare serum gonadotropin
CAS :<p>Pregnant mare serum gonadotropin (PMSG) functions as a gonadotropin that enhances follicular development and ovulation in animals. This compound operates by modulating blood hormones, gonadotropins, and cytoplasmic estradiol receptors in the anterior pituitary and hypothalamus. Commonly employed in livestock to boost reproductive efficiency, PMSG is also valuable for research focused on estrous cycle regulation.</p>Couleur et forme :SolidIGUANA-1
CAS :<p>IGUANA-1 is a highly efficient and selective ALDH1B1 inhibitor that inhibits the growth of colorectal cancer cells and colorectal cancer cell-derived organoids.</p>Formule :C27H26ClN3O4Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :491.97β-Apooxytetracycline
CAS :<p>β-Apooxytetracycline is a potential impurity found in commercial preparations of oxytetracycline.</p>Formule :C22H22N2O8Couleur et forme :SolidMasse moléculaire :442.424Adenylosuccinic acid tetraammonium
<p>Adenylosuccinic acid, orally active, is a purine ribonucleotide involved in nucleotide metabolism, may aid in DMD studies.</p>Formule :C14H30N9O11PCouleur et forme :SolidMasse moléculaire :531.42LXQ-87
CAS :<p>LXQ-87 is an orally administered, non-competitive inhibitor of PTP1B with an IC50 of 1.061 μM, demonstrating hypoglycemic activity. It alleviates insulin resistance and enhances cellular glucose uptake, making it useful for type 2 diabetes research.</p>Formule :C23H18Br2O5Couleur et forme :SolidMasse moléculaire :534.195-(3',4'-Dihydroxyphenyl)-γ-valerolactone
CAS :<p>5-(3',4'-Dihydroxyphenyl)-γ-valerolactone is a metabolic byproduct of gut microbiota processing of (-)-Epicatechin. [5-(3',4'-Dihydroxyphenyl)-γ-valerolactone] exhibits antioxidant properties.</p>Formule :C11H12O4Couleur et forme :SolidMasse moléculaire :208.21Mono(5-carboxy-2-ethylpentyl) phthalate
CAS :<p>MECPP is a metabolite of DEHP, a major plasticizer used in flexible PVC.</p>Formule :C16H20O6Couleur et forme :SolidMasse moléculaire :308.33SKI2852
CAS :<p>SKI2852 is an 11β-HSD1 inhibitor that improves metabolic syndrome in diabetic mouse models.</p>Formule :C27H34FN5O4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :543.65Boc-Ile-Glu-Gly-Arg-AMC
CAS :<p>Boc-IEGR-AMC: fluorogenic substrate for factor Xa and Halocynthia roretzi acrosin.</p>Formule :C34H50N8O10Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :730.81Methylcardol triene
CAS :<p>Methylcardol triene, a phenolic compound present in cashew nut shell liquid, demonstrates α-glucosidase inhibition (IC50= 39.6 µM) and exhibits schistosomicidal properties by eliminating 100% of adult S. mansoni worms within 24 hours at 100 and 200 µM concentrations. Moreover, it serves as a precursor for synthesizing mono- and bis-benzoxazines.</p>Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.496Valinotricin
CAS :<p>Valinotricin is a minor fungal metabolite.</p>Formule :C12H22N2O4Couleur et forme :SolidMasse moléculaire :258.31BMT-297376
CAS :<p>BMT-297376, the optimized Linrodostat, is a potent IDO1 inhibitor.</p>Formule :C23H29F2N3O3Couleur et forme :SolidMasse moléculaire :433.5Lantanose A
CAS :<p>Lantanose A is a bioactive chemical from Lantana cumara roots.</p>Formule :C30H52O26Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :828.72DSPE-PEG2000-APRPG
<p>DSPE-PEG2000-APRPG is a PEG compound composed of DSPE and the APRPG peptide. It is utilized in drug delivery applications.</p>Couleur et forme :Odour SolidCA Ⅱ-IN-1
<p>CAⅡ-IN-1 (compound 2i) is an inhibitor of the CA Ⅱ isozyme, exhibiting an IC50 of 0.44 µM. This compound is utilized in metabolic research.</p>Formule :C18H19NO6SCouleur et forme :SolidMasse moléculaire :377.41hCYP3A4-IN-1
<p>hCYP3A4-IN-1 (compound C6) is a potent, orally active inhibitor of hCYP3A4, exhibiting IC50 values of 43.93 nM in human liver microsomes (HLMs) and 153.00 nM in</p>Couleur et forme :Odour Solid(±)-CBCQ
CAS :<p>(±)-CBCQ, an oxidation product of cannabidiol, exhibits an EC50 value of 14.7 μM for the activation of peroxisome proliferator-activated receptor γ (PPAR-γ).</p>Formule :C21H28O3Couleur et forme :SolidMasse moléculaire :328.45Galactose 1-phosphate
CAS :<p>Galactose 1-phosphate, an intermediate substance in both galactose metabolism and nucleotide sugar processes, plays a crucial role in the biochemical pathways</p>Formule :C6H13O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :260.14D-myo-Inositol-1,4,5-triphosphate tripotassium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate tripotassium is a second messenger in the intracellular signaling system that induces Ca2+ mobilization.</p>Formule :C6H12K3O15P3Couleur et forme :SolidMasse moléculaire :534.37O-Methyl Atorvastatin hemicalcium
CAS :<p>O-Methyl Atorvastatin, an Atorvastatin impurity, orally inhibits HMG-CoA reductase to lower blood lipids.</p>Formule :C68H76CaF2N4O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1187.449LYS006 hydrochloride
CAS :<p>LYS006 hydrochloride is a potent inhibitor of leukotriene A4 hydrolase (LTA4H) with an IC50 value of 2 nM. It is applicable in the study of inflammatory and autoimmune diseases. For further details, please refer to compound 29 in patent document WO2015092740A1.</p>Formule :C16H15Cl2FN6O3Couleur et forme :SolidMasse moléculaire :429.23Beauveriolide I
CAS :<p>Beauveriolide I, a cyclodepsipeptide from Beauveria, inhibits lipid droplet and cholesterol synthesis in mouse macrophages; IC50=0.78 μM.</p>Formule :C27H41N3O5Couleur et forme :SolidMasse moléculaire :487.63Avenacin A 1
CAS :<p>Avenacin A 1 is a biochemical.</p>Formule :C55H83NO21Couleur et forme :SolidMasse moléculaire :1094.255FXR agonist 5
CAS :<p>FXR agonist 5 is an FXR agonist used in the study of liver diseases or diseases mediated by metabolic inflammation.</p>Formule :C40H53N5O5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :683.88tetranor-PGAM
CAS :<p>PGE2 is a biomarker for inflammation and disease; its unstable urinary metabolite, tetranor-PGEM, and its byproduct, tetranor-PGAM, indicate biosynthesis.</p>Formule :C16H22O6Couleur et forme :SolidMasse moléculaire :310.346Tetracosanoyl-sulfatide
CAS :<p>C24 3'-sulfo Galactosylceramide is a key myelin sulfatide, high in leukodystrophy patients, non-immunogenic compared to C24:1 variant.</p>Formule :C48H93NO11SCouleur et forme :SolidMasse moléculaire :892.32C-Type Natriuretic Peptide (1-53), Porcine, Rat,mouse
CAS :<p>C-Type Natriuretic Peptide (1-53), from porcine, rat, and mouse sources, serves as an activator of particulate guanylate cyclase B (pGC-B), prominently found in endothelial cells, kidneys, and the heart. This peptide efficiently mediates a potent anti-fibrotic effect in human cardiac and renal fibroblasts through the production of the second messenger cGMP.</p>Couleur et forme :SolidFASN-IN-4 tosylate
CAS :<p>FASN-IN-4 tosylate: Fatty acid synthase inhibitor, IC50 10 nM; blocks SARS-CoV-2, EC50 18.6 nM.</p>Formule :C33H35N3O7S2Couleur et forme :SolidMasse moléculaire :649.78FXIa-IN-15
CAS :<p>FXIa-IN-15 (Compound (S)-10h) is an inhibitor of factor XIa (FXIa) and plasma kallikrein (PKa) with IC50 values of 0.38 nM and 59.2 nM, respectively. It exhibits anticoagulant properties by prolonging the 50% activated partial thromboplastin time (aPTT) with an EC1.5X of 0.55 μM.</p>Formule :C32H23ClF3N7O4Couleur et forme :SolidMasse moléculaire :662.02MU1742
<p>MU1742 is a probe for CK1δ and CK1ε protein kinases [1] .</p>Formule :C22H22F2N6Couleur et forme :SolidMasse moléculaire :408.45APL180
CAS :<p>APL180 (L-4F) is an apolipoprotein A-I mimetic peptide that enhances the anti-inflammatory activity of high-density lipoprotein (HDL). It is applicable for cardiovascular disease research.</p>Formule :C114H156N24O28Couleur et forme :SolidMasse moléculaire :2310.610(S),17(S)-DiHDHA
CAS :<p>Protectin D1, or neuroprotectin D1 in neurons, is anti-inflammatory. 10(S),17(S)-DiHDHA, also PDX, differs in structure and inhibits neutrophils and platelets.</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.494DSPE-PEG-Maleimide ammonium (MW 2000)
<p>DSPE-PEG-Maleimide (ammonium) (MW 2000) is a compound containing DSPE phospholipids and maleimide, designed for the preparation of nanoscale lipid carriers. It is applicable in the study of drug delivery systems.</p>Couleur et forme :Odour Solidω-Hexatoxin-Hv1a
CAS :<p>ω-Hexatoxin-Hv1a, a neurotoxin extracted from the venom of the spider Hadronyche versuta, inhibits voltage-gated calcium channels [1] [2].</p>Formule :C162H247N49O61S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4049.38Dextranase
CAS :<p>Dextranase, a glucan hydrolase, breaks down α-(1,6)-glucosidic bonds in dextran, useful in food, sugar modification, medicine, and more.</p>Couleur et forme :SolidSialyl-Lewis X
CAS :<p>sLeX: sialylated, fucosylated tetrasaccharide, ligand for selectins, inhibits neutrophil recruitment.</p>Formule :C31H52N2O23Couleur et forme :SolidMasse moléculaire :820.748Nedosiran sodium
CAS :<p>Nedosiran sodium, a GalNAc-dsRNA conjugate, is engineered to suppress the synthesis of the hepatic lactate dehydrogenase (LDH) enzyme.</p>Couleur et forme :SolidDapagliflozin-3-O-β-D-Glucuronide
CAS :<p>Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin .</p>Formule :C27H33ClO12Couleur et forme :SolidMasse moléculaire :585Orotidine
CAS :<p>Orotidine (Uridin-6-carboxylic acid) is a nucleoside found in bacteria, fungi, and plants. In humans, orotidine occurs as its 5'-phosphate (orotidylic acid).</p>Formule :C10H12N2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.21TXA707
CAS :<p>TXA707, the active metabolite of TXA-709, is an FtsZ inhibitor with antibacterial properties. It shows potential for use in research involving S. aureus.</p>Formule :C15H8F5N3O2SCouleur et forme :SolidMasse moléculaire :389.3h15-LOX-2 inhibitor 2
<p>Compound 10 (h15-LOX-2 inhibitor 2) suppresses h15-LOX activity, exhibiting IC 50 and K i values of 26.9 μM and 16.4 μM, respectively.</p>Formule :C22H30Cl2N6O3Couleur et forme :SolidMasse moléculaire :497.422-Methylpyrrolidine
CAS :<p>2-Methylpyrrolidine is an endogenous secondary metabolite that can be used for relevant research in the life sciences.</p>Formule :C5H11NCouleur et forme :SolidMasse moléculaire :85.15LOX-IN-5
CAS :<p>LOX-IN-5 (compound 22) is a non-selective LOX inhibitor.</p>Formule :C21H25FN4O2SCouleur et forme :SolidMasse moléculaire :416.51sEH inhibitor-20
<p>sEH inhibitor-20 is a metabolically stable, orally active sEH inhibitor with an IC50 of 0.2 nM. It exhibits significant analgesic and anti-inflammatory properties, making it a promising candidate for researching neuropathic pain.</p>Couleur et forme :Odour SolidSAICAR
CAS :<p>SAICAR is an intermediate of de novo purine nucleotide biosynthesis, activates pyruvate kinase isoform M2 (PKM2) in an isozyme-selective manner (EC50: 0.3 mM).</p>Formule :C13H19N4O12PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.28Naroparcil
CAS :<p>Naroparcil, an oral thioglycoside, has antithrombotic properties and alters thrombin complex formation.</p>Formule :C19H17NO4S2Degré de pureté :98.71% - 99.88%Couleur et forme :SolidMasse moléculaire :387.47Nampt degrader-2
<p>Nampt degrader-2: a fluorescent PROTAC that degrades NAMPT at IC50 41.9 nM, reducing NAD+ and having anti-tumor effects.</p>Formule :C59H73N9O7SCouleur et forme :SolidMasse moléculaire :1052.33N-Lactylvaline
CAS :<p>N-Lactylvaline is an endogenous metabolite detectable in patients with intermediate maple syrup urine disease.</p>Formule :C8H15NO4Couleur et forme :SolidMasse moléculaire :189.21NAD Synthetase
CAS :<p>NAD Synthetase is responsible for the final step in the synthesis of Nicotinamide Adenine Dinucleotide (NAD). The enzyme sourced from Escherichia coli exhibits Km values of 200 μM for NAD, 11 μM for ATP, and 0.65 μM for ammonia. Conversely, NAD Synthetase derived from yeast demonstrates Km values of 170 μM for NAD, 190 μM for ATP, and 64 μM for ammonia. This enzyme is applicable in enzymatic assays for ATP, ammonia, urea, or creatinine and can also be used in enzymatic recycling methods. Additionally, NAD Synthetase holds potential for research into metabolic diseases, cancer, aging, and neurodegenerative disorders.</p>Couleur et forme :SolidDSPE-PEG2000-CTT2
<p>DSPE-PEG2000-CTT2 is a PEG compound consisting of DSPE and the gelatinase inhibitor CTT2 (CTTHWGFTLC). It possesses the ability to specifically target tumors. DSPE-PEG2000-CTT2 is suitable for drug delivery applications.</p>Couleur et forme :Odour Solid5-Aminoisotonitazene
CAS :<p>5-Aminoisotonitazene is a metabolite of the synthetic opioid analgesic agent, Isotonitazene, found in urine.</p>Formule :C23H32N4OCouleur et forme :SolidMasse moléculaire :380.53Kallikrein
CAS :<p>Kallikrein is capable of forming the kallikrenase kalinin system (KKS) in plasma and tissues, producing bradykinin and kalin peptides , respectively [1] .</p>Couleur et forme :SolidHeptanoyl-L-carnitine (chloride)
CAS :<p>Heptanoyl-L-carnitine is a medium-chain acylcarnitine and derivative of L-carnitine .</p>Formule :C14H28ClNO4Couleur et forme :SolidMasse moléculaire :309.83Sorbitol-6-phosphate 2-dehydrogenase
CAS :<p>Sorbitol-6-phosphate 2-dehydrogenase, a dehydrogenase enzyme produced by Escherichia coli, catalyzes the interconversion of D-sorbitol 6-phosphate and D-fructose 6-phosphate. The enzyme oxidizes D-sorbitol 6-phosphate at a rate ten times faster than it reduces D-fructose 6-phosphate, playing a role in various cellular processes.</p>Couleur et forme :SolidDSPE-PEG5000-CREKA
<p>DSPE-PEG5000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide is utilized for targeting tumor cells and tumor vasculature, exhibiting anti-tumor activity. DSPE-PEG5000-CREKA is applicable in drug delivery systems.</p>Couleur et forme :Odour SolidAculene A
CAS :<p>Aculene A is a unique type of norsesquiterpene from Aspergillus aculeatus [1] .</p>Formule :C19H25NO3Couleur et forme :SolidMasse moléculaire :315.41N-Demethyl ivabradine hydrochloride
CAS :<p>N-Demethyl Ivabradine Hcl is a specific inhibitor of the funny channel.N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine.</p>Formule :C26H35ClN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :491.02Uridine 5'-triphosphate tris salt
CAS :<p>Uridine 5'-triphosphate tris salt is an endogenous metabolite .</p>Formule :C13H26N3O18P3Couleur et forme :SolidMasse moléculaire :605.28Fructosyl-lysine dihydrochloride
CAS :<p>Fructoselysine dihydrochloride, a Maillard reaction product and precursor to diabetes marker glucosepane.</p>Formule :C12H26Cl2N2O7Couleur et forme :SolidMasse moléculaire :381.258′-Hydroxy ABA
CAS :<p>8′-Hydroxy ABA (8'-OH-ABA), a key metabolite of abscisic acid (ABA), exhibits hormonal activity by promoting enhanced oil synthesis.</p>Formule :C15H20O5Couleur et forme :SolidMasse moléculaire :280.32Leuhistin
CAS :Leuhistin is an aminopeptidases N inhibitor isolated from Bacillus laterosporus BMI156-14F1.Formule :C11H19N3O3Degré de pureté :98%Couleur et forme :White To Off-White SolidMasse moléculaire :241.29Nucleocidin
CAS :<p>Nucleocidin, an antitrypanosomal antibiotic, inhibits the transfer of labeled amino acids from S-RNA to protein.</p>Formule :C10H13FN6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.31Clervonafusp alfa
CAS :<p>Clervonafusp alfa (VAL-1221) is a fusion protein for Pompe disease, targeting glycogen in cytosol and lysosomes.</p>Couleur et forme :LiquidGlycerol-3-phosphate oxidase
CAS :<p>Glycerol-3-phosphate oxidase, from E. coli, is crucial in glycerol metabolism and phospholipid formation, producing electrons via oxidation.</p>Couleur et forme :SolidHIV-1 inhibitor-58
<p>HIV-1 Inhibitor-58 (Compound 10c) is a non-nucleoside reverse transcriptase inhibitor with broad-spectrum antiviral properties, effective against both wild-type</p>Formule :C26H24N6O2Couleur et forme :SolidMasse moléculaire :452.51IDO1-IN-7
CAS :<p>IDO1-IN-7 is a potent IDO1 inhibitor with a 6.1 nM IC50 and immunomodulatory effects for cancer research.</p>Formule :C22H19ClFN3O3Couleur et forme :SolidMasse moléculaire :427.86
