Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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C22 Phytoceramide (t18:0/22:0)
CAS :<p>C22 Phytoceramide (t18:0/22:0) is a lipid molecule that can be used in life science related research. The CAS number of C22 Phytoceramide (t18:0/22:0) is 164576-03-8.</p>Formule :C40H81NO4Couleur et forme :SolidMasse moléculaire :640.1BBT
CAS :<p>BBT has anti-hyperglycemic activity, protecting beta cells from cytokine or streptozotocin-induced cell death, and restoring beta cell function.</p>Formule :C18H12BrNO2SDegré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :386.26Sch59498
CAS :<p>Sch59498 is a potent phosphodiesterase 1c (Pde1c) inhibitor.</p>Formule :C17H25N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.41Hypusine
CAS :<p>Hypusine is an N-terminal amino alcohol derivative of Lys occurring in bovine brain &</p>Formule :C10H23N3O3Couleur et forme :SolidMasse moléculaire :233.31KCA-1490
CAS :KCA-1490 is an inhibitor of dual PDE3/4.Formule :C14H13F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.27Antiviral agent 46
CAS :<p>Antiviral agent 46, also known as compound 4, is a cannabidiol (CBD) derivative exhibiting anti-SARS-CoV-2 activity (IC50: 1.90 μM) and ACE2 inhibition (IC50: 1.37 μM) [1].</p>Formule :C21H32O2Couleur et forme :SolidMasse moléculaire :316.482-Myristyldistearin
CAS :<p>2-Myristyldistearin (SMS), a triacylglycerol comprising myristic acid and stearic acid [1], showcases its intricate structural composition.</p>Formule :C53H102O6Couleur et forme :SolidMasse moléculaire :835.37Diethyl-pythiDC
CAS :<p>Diethyl-pythiDC is an collagen prolyl 4-hydroxylase inhibitor.</p>Formule :C14H14N2O4SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :306.34AS1468240
CAS :<p>AS1468240 is a factor Xa inhibitor. It has significant oral anticoagulant activity.</p>Formule :C25H25Cl2N5O3Couleur et forme :SolidMasse moléculaire :514.4TMDJ-035
CAS :<p>TMDJ-035 is a selective inhibitor of the RyR2 (ryanodine receptor 2).</p>Formule :C16H12F3N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.29ICMT-IN-19
CAS :<p>ICMT-IN-19 (compound 53) serves as a potent inhibitor of ICMT, demonstrating an IC50 value of 0.026 μM [1].</p>Formule :C21H26N2O3Couleur et forme :SolidMasse moléculaire :354.44BMS-986172
CAS :<p>BMS-986172 is an orally active, highly selective inhibitor of MGAT2, demonstrating inhibitory concentrations (IC50) of 4.6 nM for human MGAT2 (hMGAT2) and 20 nM</p>Formule :C24H22F7N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.471a,1b-dihomo Prostaglandin F2α
CAS :<p>1a,1b-Dihomo Prostaglandin F2α (1a,1b-dihomo PGF2α), a hypothetical product of adrenic acid in the COX pathway, is predominantly synthesized in the renal medulla, reflecting the selective distribution of adrenic acid in this region.</p>Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.541T-0156 hydrochloride
CAS :<p>inhibitor of phosphodiesterase type 5 (PDE5)</p>Formule :C31H30ClN5O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :620.05Implitapide Racemate
CAS :<p>Implitapide Racemate is the racemate of Implitapide. Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).</p>Formule :C35H37N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.69Quizalofop
CAS :Quizalofop (Xylafop) is a reagent of biochemical.Formule :C17H13ClN2O4Degré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :344.75Dendrogenin A
CAS :<p>Dendrogenin A (DDA) is a compound acting as a selective liver X receptor (LXR) modulator, cholesterol epoxide hydrolase inhibitor (Ki = 120 nM), and a metabolic</p>Formule :C32H55N3O2Couleur et forme :SolidMasse moléculaire :513.80II-B08
CAS :<p>II-B08 is a cell-permeable SHP2 inhibitor (IC50 = 5.5 µM). II-B08 blocks growth factor stimulated ERK1/2 activation and hematopoietic progenitor proliferation.</p>Formule :C33H27N5O4Couleur et forme :SolidMasse moléculaire :557.6Kelatorphan
CAS :<p>Kelatorphan is an enkephalin degrading enzyme full inhibitor.</p>Formule :C14H18N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.3Glycosidase-IN-1
CAS :<p>Glycosidase-IN-1, a D-mannose-derived inhibitor, has hypoglycemic effects and aids in creating immunosuppressants and β-glucosidase blockers.</p>Formule :C13H23NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :273.33PF-04937319
CAS :<p>PF-04937319 activates glucokinase (EC50=154.4μM) with low hypoglycemia risk, researched for type 2 diabetes treatment.</p>Formule :C22H20N6O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :432.43S-Benzylglutathione
CAS :<p>S-Benzylglutathione acts as a competitive inhibitor of glutathionase and undergoes conversion by rat kidney microsomes into its cysteine derivatives.</p>Formule :C17H23N3O6SCouleur et forme :SolidMasse moléculaire :397.45OSMI-1
CAS :OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Formule :C28H25N3O6S2Degré de pureté :96.79% - 99.39%Couleur et forme :SolidMasse moléculaire :563.641-Oleoyl-2-hydroxy-sn-glycero-3-PG sodium
CAS :<p>1-Oleoyl-2-hydroxy-sn-glycero-3-PG (sodium salt), a lysophospholipid with oleic acid (18:1) at the sn-1 position, finds application in creating micelles, liposomes, and various artificial membranes, notably in lipid-based drug delivery systems.</p>Formule :C24H46NaO9PCouleur et forme :SolidMasse moléculaire :532.587ER 50891
CAS :<p>ER-50891 is a potent RARα antagonist, countering retinoic acid inhibition and aiding BMP2-induced osteoblast differentiation.</p>Formule :C29H24N2O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :432.51Xanthine oxidase-IN-1
CAS :<p>Xanthine oxidase-IN-1 is an effective inhibitor of xanthine oxidase with an IC50 value of 6.5 nM.</p>Formule :C16H8F2N2O3Degré de pureté :97.36% - 99.22%Couleur et forme :SolidMasse moléculaire :314.24Calcium channel-modulator-1
CAS :<p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>Formule :C26H24Cl2N2O7SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :579.45p-Ethynylphenylalanine
CAS :<p>p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a tryptophan hydroxylase (TPH) inhibitor, is competitive, effective, selective, and reversible, with a Ki of</p>Formule :C11H11NO2Degré de pureté :97.57%Couleur et forme :SolidMasse moléculaire :189.214A3-SC8
CAS :<p>4A3-SC8 is a modular, degradable dendrimer facilitating the extension of survival in aggressive liver cancer models through the delivery of small RNAs [1].</p>Formule :C75H139N3O16S4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :1467.18CCT365623
CAS :<p>CCT365623: oral Lysyl Oxidase inhibitor, potent, selective, good pharmacokinetics, anti-metastatic.</p>Formule :C18H17NO4S3Degré de pureté :97.299% - 99.49%Couleur et forme :SolidMasse moléculaire :407.53PA452
CAS :<p>PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.</p>Formule :C26H37N3O3Degré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :439.59Cis-22a
CAS :<p>Cis-22a: selective TRPV6 inhibitor (IC50=0.32μM), halts T47D breast cancer cell growth.</p>Formule :C24H30F3N3O2Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :449.51AMG 579
CAS :<p>AMG 579 is an efficacious and selective inhibitor of PDE10A (IC50 = 0.1 nM).</p>Formule :C25H23N5O3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :441.48Rilapladib
CAS :Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormule :C40H38F5N3O3SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :735.8Varespladib methyl
CAS :<p>Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.</p>Formule :C22H22N2O5Degré de pureté :99.42% - 99.97%Couleur et forme :SolidMasse moléculaire :394.42HIF-2α agonist 2
CAS :HIF-2α agonist 2 is an HIF-2α agonist with an EC50 value of 1.68 μM for HIF-2α.Formule :C13H8Br2N2O2SDegré de pureté :98.87%Couleur et forme :SoildMasse moléculaire :416.09WAY-620147
CAS :<p>WAY-620147 inhibits Monoamine Oxidase and can be used for the study of neurological disorders.</p>Formule :C12H16BrN3O2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :314.18Setileuton
CAS :<p>Setileuton (MK0633) is a specific 5-LOX inhibitor and can be used in research on asthma and atherosclerosis.</p>Formule :C22H17F4N3O4Degré de pureté :98.85% - 99.35%Couleur et forme :SolidMasse moléculaire :463.38OGT 2115
CAS :<p>OGT 2115 blocks heparanase (IC50=0.4µM), cleaving heparan sulfate; antiangiogenic (IC50=1µM).</p>Formule :C24H16BrFN2O4Degré de pureté :97.17%Couleur et forme :SolidMasse moléculaire :495.3WAY-297848
CAS :<p>WAY-297848 is a novel glucokinase activator for the prevention or treatment of hyperglycemia, diabetes mellitus, obesity, dyslipidemia, and metabolic syndrome.</p>Formule :C13H13ClN2O2SDegré de pureté :98.19%Couleur et forme :SolidMasse moléculaire :296.77TPN171
CAS :<p>TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6, which has the potential for the treatment of pulmonary</p>Formule :C24H35N5O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :441.57Ecopladib
CAS :<p>Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).</p>Formule :C39H33Cl3N2O5SDegré de pureté :95.15%Couleur et forme :SolidMasse moléculaire :748.11Cudetaxestat
CAS :<p>Cudetaxestat (BLD-0409) is a potent inhibitor of orally active autotaxin.</p>Formule :C21H15Cl2F2N3O2SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :482.33TP-10
CAS :<p>TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.</p>Formule :C26H19F3N4ODegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :460.45RS 8359
CAS :<p>RS 8359 is a selective MAO-A reversible inhibitor with a 2200:1 A:B ratio, exhibiting antidepressant effects.</p>Formule :C14H12N4ODegré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :252.27NPAS3-IN-1
CAS :<p>NPAS3-IN-1 is an NPAS3-ARNT heterodimerization inhibitor that regulates NPAS3 transcription by modulating the heterodimerization of NPAS3 with ARNT.</p>Formule :C10H5N3O2S3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :295.36Enpp-1-IN-16
CAS :<p>Enpp-1-IN-16 is an ENPP1 inhibitor, yo anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance and chondrocalcinosis.</p>Formule :C23H32N4O4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :428.52KB-74935
CAS :<p>KB-74935: enzyme inhibitor, mineralocorticoid blocker, treats cholesterol, hypolipidemia, neurological issues, Alzheimer's.</p>Formule :C19H18ClF4N3O3SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :479.88PXS-6302 hydrochloride
CAS :<p>PXS-6302 hydrochloride is a potent irreversible lysine oxidase (LOX) inhibitor, inhibiting Bovine LOX, rh LOXL1, rh LOXL2, rh LOXL3, and rh LOXL4 with IC50 of 3</p>Formule :C10H11ClF3NO2SDegré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :301.71BI-3231
CAS :<p>BI-3231 is a hydroxysteroid 17ß-dehydrogenase 13 HSD17B13 inhibitor that inhibits hHSD17B13 .BI-3231 can be used to study cirrhosis.</p>Formule :C16H14F2N4O3SDegré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :380.37Dechloro Rivaroxaban
CAS :<p>Dechloro Rivaroxaban is a Factor Xa inhibitor that inhibits free FXa and plasminogen and fibrin-associated FXa activity in humans.</p>Formule :C19H19N3O5SDegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :401.44CB29
CAS :<p>CB29 is a specific inhibitor of aldehyde dehydrogenase 3A1 (ALDH3A1).</p>Formule :C15H15N3O5SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :349.36ML400
CAS :<p>ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.</p>Formule :C24H29N3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :375.51Fluspirilene
CAS :<p>Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).</p>Formule :C29H31F2N3ODegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :475.57PDE9-IN-(S)-C33
CAS :<p>PDE9-IN-(S)-C33: potent PDE9 inhibitor with 11 nM IC50, for CNS diseases and diabetes study.</p>Formule :C18H20ClN5ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :357.84DGAT-1 inhibitor 2
CAS :<p>DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.</p>Formule :C24H28N4O3Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :420.5ALDH2 modulator 1
CAS :<p>ALDH2 modulator 1 is a potent and orally active modulator of acetaldehyde dehydrogenase-2 (ALDH2), which reduces blood alcohol levels in mice.</p>Formule :C18H18ClFN2O3Degré de pureté :99.68%Couleur et forme :SoildMasse moléculaire :364.87-BIA
CAS :<p>7-BIA is a receptor-type protein tyrosine phosphatase D (PTPRD) inhibitor with anti-addictive properties and can be used in the study of neuropathic pain.</p>Formule :C15H18O6Degré de pureté :≥98% - ≥98%Couleur et forme :SolidMasse moléculaire :294.3NEP-IN-1
CAS :<p>NEP-IN-1 is an inhibitor of neutral endopeptidase (NEP, IC50 = 2 nM) and can be used in studies about female sexual arousal disorders.</p>Formule :C21H30ClNO4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :395.92Mitiperstat
CAS :<p>Mitiperstat, a strong MPO inhibitor, helps prevent heart failure and coronary artery disease.</p>Formule :C15H15ClN4OSDegré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :334.82Inolitazone
CAS :<p>Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.</p>Formule :C27H26N4O4SDegré de pureté :99.41% - 99.53%Couleur et forme :SolidMasse moléculaire :502.58h-NTPDase-IN-2
CAS :h-NTPDase-IN-2 is a broad-spectrum NTPDase inhibitor that inhibits multiple h-NTPDas isoforms.Formule :C19H16N4SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :332.42Mutant IDH1-IN-2
CAS :<p>Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of ＜22 nM in LS-</p>Formule :C24H31F2N5O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :459.53(R,R)-BMS-986397
CAS :<p>(R,R)-BMS-986397 is a CK1α degrader with a DC50 ranging from 0.1 to 0.5 pM. This compound is applicable in leukemia research.</p>Formule :C21H16ClF3N4O4Couleur et forme :SolidMasse moléculaire :480.82Monoamine oxidase/Aromatase-IN-1
Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.Formule :C19H19N3O3SCouleur et forme :SolidMasse moléculaire :369.44CYP1B1-IN-2
<p>CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].</p>Formule :C20H11F3O2Couleur et forme :SolidMasse moléculaire :340.3DLCI-1
CAS :<p>DLCI-1 is a potent and selective oral inhibitor of cytochrome P450 2A6 (CYP2A6), significantly reducing self-administered nicotine doses in both male and female mice.</p>Formule :C12H14N2SCouleur et forme :SolidMasse moléculaire :218.32Anticancer agent 142
CAS :<p>Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].</p>Formule :C13H14BrF2N2O7PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.26MAGL-IN-19
CAS :<p>MAGL-IN-19 (compound 7o) is a highly effective and selective inhibitor of MAGL.</p>Formule :C21H26F3N3O3Couleur et forme :SolidMasse moléculaire :425.45PDE4-IN-5
<p>PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.</p>Formule :C21H28N2O3Couleur et forme :SolidMasse moléculaire :356.46Mibefradil
CAS :<p>Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).</p>Formule :C29H38FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :495.63Hcyb1
<p>Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.</p>Formule :C24H20N4OCouleur et forme :SolidMasse moléculaire :380.44hDHODH-IN-10
<p>hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.</p>Formule :C21H15ClF4N2O4Couleur et forme :SolidMasse moléculaire :470.8Arphamenine A
CAS :<p>Arphamenine A is an inhibitor of aminopeptidase B (aminopeptidaseB) found in HMG361-CF4 of Actinomadura azurea. It exhibits inhibitory effects against Sarcoma 180 and invasive micropapillary carcinoma (IMC).</p>Formule :C16H24N4O3Couleur et forme :SolidMasse moléculaire :320.387hCAII-IN-4
CAS :hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Formule :C31H23NO9Couleur et forme :SolidMasse moléculaire :553.52(S)-CPP sodium
CAS :<p>(S)-CPP sodium serves as an inhibitor of the branched-chain α-keto acid dehydrogenase complex (BCKDC) kinase, commonly referred to as BDK or keto acid dehydrogenase kinase. As a negative regulator of BCKDC activity, (S)-CPP (IC50 of 6.3 μM) inhibits BDK, which activates the complex, leading to a significant reduction in the levels of leucine/isoleucine and valine in the plasma of wild-type mice.</p>Formule :C9H8ClNaO2Couleur et forme :SolidMasse moléculaire :206.60PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Formule :C30H35N3O4S2Couleur et forme :SolidMasse moléculaire :565.7511-Mercaptoundecanoate-NHS
CAS :<p>11-Mercaptoundecanoate-NHS is a lipid utilized in the synthesis of Linkers.</p>Formule :C15H25NO4SCouleur et forme :SolidMasse moléculaire :315.428Porphobilinogen
CAS :<p>Porphobilinogen act as a phytotoxin, a metabotoxin, and a neurotoxin.</p>Formule :C10H14N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.23hMAO-B/MB-COMT-IN-1
<p>Dual hMAO-B/MB-COMT inhibitor, IC50: 2.5 μΜ (hMAO-B), 3.84 μΜ (MB-COMT); potential in Parkinson's research.</p>Formule :C16H19NO3Couleur et forme :SolidMasse moléculaire :273.33AChE/PDE4-IN-1
<p>AChE/PDE4-IN-1, compound 12c, dual inhibitor; IC50: 0.28μM for AChE, 1.88μM for PDE4D, may reduce Alzheimer's neuroinflammation.</p>Formule :C23H28N2O3Couleur et forme :SolidMasse moléculaire :380.48Desmonomethylpromazine
CAS :<p>Desmonomethylpromazine is a demethylated metabolite of Promazine that can penetrate the brain. It enters red blood cells and tissues via passive diffusion and is distributed in organs such as the lungs, liver, and kidneys in rats.</p>Formule :C16H18N2SCouleur et forme :SolidMasse moléculaire :270.39m-APTA
CAS :<p>m-APTA (5'-S-(3-aminophenyl)-5'-thioadenosine) is a selective chemoprotective agent targeting methylthioadenosine phosphorylase (MTAP). It can be converted into adenine, which is a crucial step in shielding normal cells from the toxicity of nucleobase analogs (NBA). m-APTA holds potential for research in MTAP-deficient cancers.</p>Formule :C16H18N6O3SCouleur et forme :SolidMasse moléculaire :374.418PRL3-CNNM4 interaction-IN-1
CAS :<p>PRL3-CNNM4 interaction-IN-1 (Compound C28d52) is an inhibitor of the PRL3-CNNM4 interaction that also suppresses CNNM inhibition mediated by PRL. This compound exhibits favorable pharmacokinetic and drug metabolism properties.</p>Formule :C8H8O2SCouleur et forme :SolidMasse moléculaire :168.21Z57346765
CAS :<p>Z57346765 is a specific PGK1 inhibitor that inhibits PGK1-dependent cell proliferation by decreasing the metabolic enzyme activity of PGK1 during glycolysis.</p>Formule :C17H18N4ODegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :294.35Xanthosine-5'-monophosphate
CAS :<p>Xanthosine 5'-monophosphate is produced from inosine monophosphate (IMP) through the catalytic action of inosine monophosphate dehydrogenase (IMPDH).</p>Formule :C10H13N4O9PCouleur et forme :SolidMasse moléculaire :364.21TS010
<p>TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 μM. It holds significant promise for advancements in cancer research [1].</p>Formule :C16H12N4O4SCouleur et forme :SolidMasse moléculaire :356.36Oxythiamine diphosphate ammonium
<p>Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).</p>Couleur et forme :SolidIDO1-IN-14
<p>IDO1-IN-14 is an IDO1 enzyme inhibitor with an IC50 of 396.9 nM and suppresses HeLa cell activity with an EC50 of 3393 nM.</p>Formule :C18H12Cl2FN3O2Couleur et forme :SolidMasse moléculaire :392.21SAL-0010042
CAS :<p>SAL-0010042 is an inhibitor of Plasmodium phosphodiesterase β (PDEβ), effectively blocking the hydrolysis of cAMP and cGMP in gametocytes with an IC50 of 48.9 nM, thereby activating PKG and inhibiting the growth and development of Plasmodium (IC50s for 3D7 and Dd2 are 142 nM and 218 nM, respectively). It also inhibits hPDE5 and hPDE6 with IC50 values of 632 nM and 73 nM, respectively.</p>Formule :C15H15FN4OCouleur et forme :SolidMasse moléculaire :286.3043'-Hydroxy Repaglinide
CAS :<p>'3'-Hydroxy Repaglinide, a CYP2C8 metabolite of Repaglinide, treats type II diabetes.</p>Formule :C27H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.59α-Glucosidase-IN-13
<p>α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).</p>Formule :C25H28N4O3S2Couleur et forme :SolidMasse moléculaire :496.64(-)-Mesembrine
CAS :<p>Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).</p>Formule :C17H23NO3Couleur et forme :SolidMasse moléculaire :289.37OMDM169
CAS :<p>OMDM169: potent/selective MAGL inhibitor, raises 2-AG, analgesic via cannabinoid receptors, IC50: 0.13-0.41μM in rat/COS-7, inactive at CB1/CB2.</p>Formule :C25H45NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.63α-Glucosidase-IN-18
<p>α-Glucosidase-IN-18 (7B) is an orally active inhibitor of α-glucosidase, displaying an IC 50 value of 3.96 μM.</p>Formule :C23H19NO2SCouleur et forme :SolidMasse moléculaire :373.47HIF-1α-IN-4
<p>HIF-1α-IN-4 is an inhibitor of HIF-1α with IC50 of 24 nM in HEK293T cells which has potential antitumor effects.</p>Formule :C16H12N2O3Couleur et forme :SolidMasse moléculaire :280.28APOL1-IN-3
CAS :<p>APOL1-IN-3 is an APOL1 inhibitor used for kidney disease research.</p>Formule :C16H19F3N4O2SCouleur et forme :SolidMasse moléculaire :388.41CAII-IN-2
<p>CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.</p>Formule :C18H19BrN4SCouleur et forme :SolidMasse moléculaire :403.34SGK1-IN-3
<p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>Formule :C23H20Cl2N6O3SCouleur et forme :SolidMasse moléculaire :531.41EB-0156
<p>EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ <0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.</p>Formule :C21H32N6O7Couleur et forme :SolidMasse moléculaire :480.51
