Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
RPR132595A
CAS :RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).Formule :C28H30N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.56Betrixaban
CAS :Betrixaban is a non-VKORC1 anticoagulant targeting factor Xa, with low hERG affinity, used to prevent VTE in adults with mobility issues.Formule :C23H22ClN5O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :451.91JZP-MA-11
CAS :<p>"JZP-MA-11 is a PET ligand that selectively targets ABHD6, inhibits with 126 nM IC50, and crosses the BBB for preclinical brain studies."</p>Formule :C15H17FN4O2SCouleur et forme :SolidMasse moléculaire :336.381,2-Dipalmitoyl-sn-glycerol 3-phosphate
CAS :<p>1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.</p>Formule :C35H69O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.89Z-Arg(Z)2-OH
CAS :<p>Z-Arg(Z)2-OH can be used in the assay to screen proteolytic activities in mite homogenates.</p>Formule :C30H32N4O8Degré de pureté :99.1400%Couleur et forme :SolidMasse moléculaire :576.6Buthidazole
CAS :<p>Buthidazole is a herbicide for selective weed control in corn.</p>Formule :C10H16N4O2SCouleur et forme :SolidMasse moléculaire :256.33PTC-510 TFA salt
CAS :<p>PTC-510 TFA salt inhibits hypoxia-induced VEGF expression.</p>Formule :C26H26BrN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.48Tetrachlorvinphos
CAS :Tetrachlorvinphos, an organophosphate cholinesterase inhibitor, is used as an insecticide. It has low toxicity to mammals.Formule :C10H9Cl4O4PDegré de pureté :98%Couleur et forme :Less Crystals Or White Powder Colorless Crystals Or White PowderMasse moléculaire :365.96Difluoro atorvastatin
CAS :<p>Difluoro atorvastatin: an atorvastatin impurity reducing blood lipids, inhibits SV-SMC proliferation/invasion (IC50: 0.39/2.39 μM).</p>Formule :C33H34F2N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.63Roflumilast Impurity E
CAS :Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast acts as a selective and long-acting the enzyme PDE-4 inhibitor(IC50 value of 0.8 nM).Formule :C13H8Cl2F2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.121-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine
CAS :1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.Formule :C44H84NO8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :786.11H-Arg-Lys-OH
CAS :<p>H-Arg-Lys-OH is a dipeptide formed from L-lysine residues and L-arginyl.</p>Formule :C12H26N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.37PAT-494
CAS :<p>PAT-494 is an inhibitor of type II Autotaxin.</p>Formule :C20H16FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.36Proadifen
CAS :<p>Proadifen is a non-selective cytochrome P450 enzymes inhibitor, preventing some types of drug metabolism.</p>Formule :C23H31NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :353.5Transketolase-IN-3
CAS :<p>Transketolase-IN-3: potent TK inhibitor with herbicidal effects on DS and AR, useful for herbicide research.</p>Formule :C20H9ClF3NO3Couleur et forme :SolidMasse moléculaire :403.74LAPAO
CAS :<p>Lauramide propyl amine oxide is an amphoteric surfactant</p>Formule :C17H36N2O2Couleur et forme :SolidMasse moléculaire :300.48(+)-Xylariamide A
CAS :<p>(+)-Xylariamide A is a probe used for mycobacterial and fungal carbonic anhydrase.</p>Formule :C14H14ClNO6Couleur et forme :SolidMasse moléculaire :327.72Ethyl phenylglyoxylate
CAS :<p>Ethyl phenylglyoxylate (AI3 10033) is a simultaneous inhibitor and substrate of chicken liver carboxylesterase.</p>Formule :C10H10O3Degré de pureté :98.46%Couleur et forme :Yellow LiquidMasse moléculaire :178.18BAY-721973
CAS :<p>BAY-721973 is a bio-active chemical.</p>Formule :C21H16ClF3N4O4Couleur et forme :SolidMasse moléculaire :480.82Fmoc-Asp(OtBu)-Thr(psi(Me,Me)pro)-OH
CAS :<p>Fmoc-Asp(OtBu)-Thr(psi(Me,Me)pro)-OH is a dipeptide.</p>Formule :C30H36N2O8Couleur et forme :SolidMasse moléculaire :552.62AKU-005
CAS :<p>AKU-005 is a dual inhibitor of FAAH and MAGL, exhibiting IC50 values of 63 nM and 389 nM against rat and human FAAH, respectively. This compound has potential for researching trigeminal nociceptive hypersensitivity.</p>Formule :C20H21N5OCouleur et forme :SolidMasse moléculaire :347.41Dimepiperate
CAS :<p>Dimepiperate is an agent of biochemical.</p>Formule :C15H21NOSCouleur et forme :SolidMasse moléculaire :263.40Milvexian
CAS :<p>Milvexian (BMS-986177) is an oral antithrombotic, reversibly inhibiting human/rabbit FXIa with K i of 0.11/0.38 nM.</p>Formule :C28H23Cl2F2N9O2Couleur et forme :SolidMasse moléculaire :626.45Desmethylnortriptyline
CAS :<p>Desmethylnortriptyline, a tricyclic antidepressant metabolite of nortriptyline and amitriptyline, treats depression.</p>Formule :C18H19NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.351,2-Dibehenoyl-sn-glycero-3-phosphocholine
CAS :<p>1,2-Dibehenoyl-sn-glycero-3-phosphocholine (DBPC), a phospholipid integral to cell membranes, facilitates the formation of micelles, liposomes, and various artificial membranes [1].</p>Formule :C48H80NO8PCouleur et forme :SolidMasse moléculaire :830.141GPAT-IN-1
CAS :<p>GPAT-IN-1 is a glycerol 3-phosphate acyltransferase (GPAT) inhibitor, which can be used to study obesity and diabetes.</p>Formule :C21H26ClNO4SDegré de pureté :99.60% - 99.60%Couleur et forme :SolidMasse moléculaire :423.95Prasugrel chloride impurity
CAS :Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.Formule :C20H21ClFNO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :409.9Nitrophenide
CAS :Nitrophenide, a 3,3'-Dinitrodiphenyl disulfide, blocks M1PDH in the mannitol cycle, serving as an anticoccidial.Formule :C12H8N2O4S2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :308.33Leucylarginine
CAS :<p>Leucylarginine hinders antinociception induced by L-arginine.</p>Formule :C12H25N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.368-Azaadenine
CAS :<p>8-Azaadenine (NSC-32797) is an inhibitor of xanthine oxidase with IC50 of 0.54 μM and Ki of 0.66 μM.</p>Formule :C4H4N6Degré de pureté :99.68%Couleur et forme :White PowderMasse moléculaire :136.11Acetaminophen mercapturate
CAS :<p>Paracetamol Mercapturate is a metabolite of Acetaminophen. It can also be used in the biological study of urinary antihypertensive drugs.</p>Formule :C13H16N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.34Prothioconazole
CAS :<p>Prothioconazole (Proline 480 SC Fungicide) is a chiral triazole fungicide in plant pathogen control.</p>Formule :C14H15Cl2N3OSDegré de pureté :99.77%Couleur et forme :Un3077 9/Pg 3Masse moléculaire :344.26Tolrestat
CAS :<p>Tolrestat (AY-27773) is a potent inhibitor of aldose reductase (IC50 = 35 nM).</p>Formule :C16H14F3NO3SDegré de pureté :98.89% - >99.99%Couleur et forme :SolidMasse moléculaire :357.35BIBB 515
CAS :<p>BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.</p>Formule :C22H21ClN2O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :380.87E3330
CAS :<p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>Formule :C21H30O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :378.46L-m-Tyrosine
CAS :<p>L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.</p>Formule :C9H11NO3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :181.191-Decanesulfonic acid
CAS :<p>1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.</p>Formule :C10H22O3SCouleur et forme :SolidMasse moléculaire :222.35Calcipotriol monohydrate
CAS :<p>Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.</p>Formule :C27H42O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :430.62Tesaglitazar
CAS :<p>Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα</p>Formule :C20H24O7SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :408.47PF-05175157
CAS :<p>PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,</p>Formule :C23H27N5O2Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :405.49PCI-27483
CAS :<p>PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.</p>Formule :C26H24N6O9SDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :596.574-POBN
CAS :<p>4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).</p>Formule :C7H9N3ODegré de pureté :99.60%Couleur et forme :White Crystalline PowderMasse moléculaire :151.173-Phenylbutyric acid
CAS :<p>3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.</p>Formule :C10H12O2Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :164.2Nafenopin
CAS :<p>Nafenopin is a peroxisome proliferator, it is used to promote liver tumors and has been used as an antihyperlipoproteinemic agent.</p>Formule :C20H22O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.39Peliglitazar racemate
CAS :<p>Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity</p>Formule :C30H30N2O7Degré de pureté :97.75%Couleur et forme :SolidMasse moléculaire :530.57JNJ-DGAT1-A
CAS :<p>JNJ-DGAT1-A is a DGAT1-selective inhibitor.</p>Formule :C31H35Cl2N5O3Couleur et forme :SolidMasse moléculaire :596.55TRC210258
CAS :<p>TRC210258 is a TGR5 agonist that acts by decreasing glycemic and dyslipidemic cardiovascular risk in animal models of diabesity.</p>Formule :C20H14ClFN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.8Statine
CAS :<p>Statine is a protease inhibitor that is active against pepsin and other acid proteases.</p>Formule :C8H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :175.23Mixanpril
CAS :Mixanpril is an RB 105 lipophilic prodrug.Formule :C21H23NO4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.48BAY 59-9435
CAS :<p>HSL-IN-2 is a selective inhibitor of Hormone Sensitive Lipase (HSL; IC50: 0.023 μM).</p>Formule :C14H22N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.34DBC
CAS :<p>DBC is a halogenated hydrocarbon, widely used in biochemical experiments and drug synthesis research.</p>Formule :C20H13NDegré de pureté :99.76%Couleur et forme :Needles From Ethanol 7H-Dibenzo(C G)Carbazole Is A Crystalline SolidMasse moléculaire :267.32Chlorisondamine diiodide
CAS :Chlorisondamine diiodide is a selective nAChR antagonist and ganglionic blocker that persistently antagonizes partial central effects of nicotine.Formule :C14H20Cl4I2N2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :611.94PTP1B-IN-15
CAS :<p>PTP1B-IN-15 is a potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor that has shown research potential in type II diabetes and obesity.</p>Formule :C19H17Br2NO5SCouleur et forme :SolidMasse moléculaire :531.22Ornithine-α-ketoglutarate
CAS :<p>Ornithine-α-ketoglutarate (L-Ornithine-α-ketoglutarate) is a salt formed of 2 molecules of ornithine and 1 alpha-ketoglutarate.</p>Formule :C10H18N2O7Degré de pureté :≥98%Couleur et forme :White PowderMasse moléculaire :278.26Letimide HCl
CAS :<p>Letimide HCl is an analgesic agent.</p>Formule :C14H19ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.77MDK-4683
CAS :<p>MDK-4683, also known as CA IX/XII Inhibitor, is a hCA IX and hCA XII inhibitor.</p>Formule :C13H12N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.32CGP-28014
CAS :<p>CGP-28014 inhibits COMT, boosts renal dopamine & DOPAC excretion, lowers HVA, no effect on renal sodium.</p>Formule :C12H19N3OCouleur et forme :SolidMasse moléculaire :221.3DU717
CAS :<p>DU717 is an antihypertensive agent.</p>Formule :C12H15ClN4O2SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :314.79Z-321
CAS :<p>Z-321 is an inhibitor of prolyl endopeptidase.</p>Formule :C19H24N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.47Moperone Hydrochloride
CAS :<p>Moperone Hydrochloride, a dopamine D2-receptor antagonist, is used for the treatment of psychiatric disorders.</p>Formule :C22H27ClFNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.91L 652343
CAS :<p>L 652343 is an inhibitor of cyclooxygenase and 5-lipoxygenase in vitro. It also inhibits the synthesis of the products of both these pathways in whole cells.</p>Formule :C22H14F3NO2S2Couleur et forme :SolidMasse moléculaire :445.48Chlorambucyl-proline
CAS :<p>Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.</p>Formule :C19H26Cl2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.33GA11
CAS :<p>GA11is an inhibitor of ALDH1. It also displays anti-GBM effects in vitro and in vivo.</p>Formule :C19H14N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.33UCM 765
CAS :<p>UCM 765 is a partial agonist of melatonin MT(2) receptor.</p>Formule :C17H20N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.352-Methyldecanenitrile
CAS :<p>2-Methyldecanenitrile, intense peach scent with lactone notes, stable in all pH, effective at low concentration.</p>Formule :C11H21NDegré de pureté :98%Couleur et forme :Colourless Liquid LiquidMasse moléculaire :167.29ML350
CAS :<p>ML350 (CYM-50202) is a potent KOR antagonist (IC50: 12.6 nM), selective over DOR/MOR, with high solubility and CNS penetration, lacking long-term effects.</p>Formule :C18H26BrN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.32LY 79771
CAS :<p>LY-79771, a phenethanolamine antiobesity agent, can be effective in preventing fat regain following energy deprivation.</p>Formule :C18H24ClNO2Couleur et forme :SolidMasse moléculaire :321.84AHR-activator-1023
CAS :<p>AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.</p>Formule :C14H8Cl2N2OCouleur et forme :SolidMasse moléculaire :291.13Albifylline
CAS :<p>Albifylline: a xanthine derivative, anti-asthmatic, reduces leukocyte adhesion, enhances liver microcirculation post-hemorrhagic shock.</p>Formule :C13H20N4O3Couleur et forme :SolidMasse moléculaire :280.32AJS1669
CAS :<p>AJS1669, an activator of muscle glycogen synthase, improves glucose metabolism and reduces body fat mass in mice.</p>Formule :C26H21F2NO6SCouleur et forme :SolidMasse moléculaire :513.51Arabinose 1,5-diphosphate
CAS :<p>Arabinose 1,5-diphosphate is a bisphosphatase inhibitor.</p>Formule :C5H12O11P2Couleur et forme :SolidMasse moléculaire :310.09LYPLAL1-IN-1
CAS :LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.Formule :C29H29N7O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :539.59MP-10 succinate
CAS :<p>MP-10 succinate is a potent and specific inhibitor of PDE10A.</p>Formule :C29H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.54CP-319340(free base)
CAS :<p>CP-319340 free base is a inhibitor of microsomal triglyceride transfer protein (MTP) .</p>Formule :C27H23F3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :476.494′-Deoxyphlorizin
CAS :<p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>Formule :C21H24O9Couleur et forme :SolidMasse moléculaire :420.41MDK-0738
CAS :<p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>Formule :C15H16O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :244.29Safrazine Hydrochloride
CAS :<p>Safrazine Hydrochloride is a monoamine oxidase inhibitor (MOI) that is irreversible.</p>Formule :C11H17ClN2O2Couleur et forme :SolidMasse moléculaire :244.718ABT-418
CAS :<p>ABT-418, a nicotinic acetylcholine receptor (nAchR) agonist, is used potentially for the treatment of attention deficit disorder.</p>Formule :C9H14N2OCouleur et forme :SolidMasse moléculaire :166.22CM026
CAS :<p>CM026 inhibits ALDH1A1 selectively, binds to its aldehyde pocket uncompetitively.</p>Formule :C22H30N6O4Couleur et forme :SolidMasse moléculaire :442.51Noreximide
CAS :<p>Noreximide is an agent of sedative.</p>Formule :C9H9NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :163.17Benzpiperylone
CAS :<p>Benzpiperylone is a synthetic anti-inflammatory drug. It also has anti-inflammatory activity.</p>Formule :C22H25N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.45Levophencynonate
CAS :<p>Levophencynonate is a muscarinic receptor antagonist.</p>Formule :C22H31NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.49ARI-3531
CAS :<p>ARI-3531 is a selective prolyl endopeptidase inhibitor.</p>Formule :C15H22BN3O4Couleur et forme :SolidMasse moléculaire :319.16Ipenoxazone
CAS :<p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>Formule :C22H34N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.52Choline theophyllinate
CAS :<p>Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and</p>Formule :C12H21N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.33MLS000536924
CAS :<p>MLS000536924 is a potent and selective competitive human epithelial 15-lipoxygenase-2 inhibitor.</p>Formule :C16H15N3SCouleur et forme :SolidMasse moléculaire :281.38MMV-667492
CAS :<p>MMV-667492 is an effective inhibitor of Ezrin.</p>Formule :C17H19N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.35L-651392
CAS :<p>L-651392 is an inhibitor of leukotriene.</p>Formule :C14H10BrNO3SCouleur et forme :SolidMasse moléculaire :352.2D-4418
CAS :<p>D-4418, a PDE4 inhibitor in development, targets asthma and COPD as an anti-inflammatory treatment.</p>Formule :C16H11Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.18Pegnivacogin
CAS :Pegnivacogin is a coagulation factor IXa RNA aptamer inhibitor.Formule :C20H40N3O11PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.52Pirbuterol hydrochloride
CAS :<p>Pirbuterol hydrochloride is a bronchodilator.</p>Formule :C12H21ClN2O3Couleur et forme :SolidMasse moléculaire :276.76Manninotrionate
CAS :<p>Manninotrionate, an antitumor agent, linked to BSA; rabbit antiserum made, doesn't agglutinate Ehrlich tumor cells with alpha-D-galactosyl groups.</p>Formule :C18H32KO17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.535PMPMEase-IN L-28
CAS :<p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>Formule :C17H29FO2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.54BFE-37
CAS :<p>BFE-37 is a partial agonist of beta-adrenergic.</p>Formule :C16H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.36TA-7552
CAS :<p>TA-7552 is a potent agent of cholesterol-lowering.</p>Formule :C25H26O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :486.47BI-135585
CAS :<p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>Formule :C28H32N2O4Degré de pureté :99.45% - 99.57%Couleur et forme :SolidMasse moléculaire :460.57IACS-8968 R-enantiomer
CAS :<p>IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Formule :C17H18F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.35AN3199
CAS :<p>AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.</p>Formule :C17H18BNO5Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :327.14BKIDC-1553
CAS :<p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>Formule :C22H23N5O2Couleur et forme :SolidMasse moléculaire :389.45AMP-Deoxynojirimycin
CAS :<p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>Formule :C22H39NO5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :397.55Epostane
CAS :<p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>Formule :C22H31NO3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :357.49Factor VII-IN-1
CAS :<p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>Formule :C15H10BrNO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :332.15Phytic acid dodecasodium salt hydrate
CAS :<p>Phytic acid salt hydrate: seed phosphorus compound, inhibits xanthine oxidase, IC50 6 mM, antioxidant, neuroprotective, anti-inflammatory.</p>Formule :C6H20NaO25P6Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :701.033ATX inhibitor 5
CAS :ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.Formule :C22H18ClF3N6ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :474.87Quinapril-d5
CAS :<p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>Formule :C25H25D5N2O5Couleur et forme :SolidMasse moléculaire :443.55TF-S14
CAS :<p>TF-S14 is an inverse agonist of RORγt. It functions by binding to RORγt and inhibiting its activity, leading to a reduction in Th17 cell-associated cytokine production, including IL-17A, IL-21, and IL-22. TF-S14 is applicable in research related to autoimmune diseases and allogeneic transplant rejection.</p>Formule :C22H27N3O2SCouleur et forme :SolidMasse moléculaire :397.53FTX-6746
CAS :<p>FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.</p>Formule :C16H7ClF2N2ODegré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :316.69Tilivapram
CAS :<p>Tilivapram is a PDE4 (phosphodiesterase IV) inhibitor that can be used in the study of mental illness.</p>Formule :C16H15Cl2N3O4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :384.21Tebuconazole-d9
CAS :<p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>Formule :C16H13ClD9N3OCouleur et forme :SolidMasse moléculaire :316.87SHP2-IN-5
CAS :<p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>Formule :C12H8O6Couleur et forme :SolidMasse moléculaire :248.19BTX161
CAS :<p>BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.</p>Formule :C15H16N2O3Couleur et forme :SolidMasse moléculaire :272.3Glyoxalase I inhibitor 7
CAS :<p>Glyoxalase I inhibitor 7 (Compound 6) is a potent inhibitor of glyoxalase I (Glo-I) with an IC50 of 3.65 μM. It exhibits potential as an anticancer agent [1].</p>Formule :C17H16N4O3SCouleur et forme :SolidMasse moléculaire :356.4Enpp-1-IN-17
CAS :<p>Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP</p>Formule :C18H24N4O2Couleur et forme :SolidMasse moléculaire :328.41IDO-IN-12
CAS :<p>IDO-IN-12 is an inhibitor of indoleamine 2,3-dioxygenase (IDO).</p>Formule :C13H11BrFN5O3SDegré de pureté :99.727%Couleur et forme :SolidMasse moléculaire :416.23hCA I-IN-2
CAS :<p>hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).</p>Formule :C26H20BrN5O3SCouleur et forme :SolidMasse moléculaire :562.44IACS-8968 S-enantiomer
CAS :<p>IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Formule :C17H18F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.35Thialysine HCl
CAS :<p>Thialysine HCl is a cytotoxic cysteine derivative that inhibits Escherichia coli, acting as a protein synthesis inhibitor and metabolite.</p>Formule :C5H13ClN2O2SCouleur et forme :SolidMasse moléculaire :200.697-Ketolithocholic acid
CAS :<p>7-Ketolithocholic acid absorbs and reduces endogenous bile acid and cholesterol secretion.</p>Formule :C24H38O4Degré de pureté :98.68% - 99.9%Couleur et forme :White - Almost White Solid PowderMasse moléculaire :390.56MK-0952
CAS :<p>MK-0952 treats memory loss and cognitive issues; it's a potent, selective PDE4 inhibitor with restricted blood activity.</p>Formule :C28H22FN3O4Couleur et forme :SolidMasse moléculaire :483.49PF-07208254
CAS :<p>PF-07208254, a potent BDK inhibitor, enhances cardiometabolic endpoints in mice [1].</p>Formule :C7H2ClFO2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :236.67SSI-4
CAS :<p>SSI-4 is a Stearoyl CoA desaturase 1 (SCD1) inhibitor that can be labeled with carbon-11 (11C) for use as a ligand in small animal in vivo PET/CT imaging</p>Formule :C19H21ClN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.853-Oxo-hop-22(29)-ene
CAS :<p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>Formule :C30H48OCouleur et forme :SolidMasse moléculaire :424.7ASM-IN-1
CAS :<p>ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.</p>Formule :C16H12BrN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :390.19LEO 39652
CAS :<p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>Formule :C23H23N3O5Couleur et forme :SolidMasse moléculaire :421.45hCAIX/XII-IN-4
CAS :<p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and >10000 nM (CAI/CAII).</p>Formule :C20H16N2O5Couleur et forme :SolidMasse moléculaire :364.35Carbonic anhydrase inhibitor 11
CAS :<p>Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.</p>Formule :C19H15F3N4O3S2Couleur et forme :SolidMasse moléculaire :468.47Calcium glycerophosphate
CAS :<p>CaGP inhibits intestinal alkaline phosphatase F3; used for calcium and phosphorus in parenteral nutrition.</p>Formule :C3H7CaO6PDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :210.14Nampt activator-3
CAS :<p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>Formule :C19H20N2O3Couleur et forme :SolidMasse moléculaire :324.37hDHODH-IN-11
CAS :<p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>Formule :C24H23N3O3Couleur et forme :SolidMasse moléculaire :401.46PF 4800567 hydrochloride
CAS :<p>casein kinase 1ε inhibitor</p>Formule :C17H19Cl2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.27Loxoprofenol-SRS
CAS :<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Formule :C15H20O3Couleur et forme :SolidMasse moléculaire :248.32PKM2 activator 3
CAS :<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Formule :C15H11ClF2N2O3SCouleur et forme :SolidMasse moléculaire :372.77SHP2 inhibitor LY6
CAS :<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Formule :C30H27Cl2N3O4Couleur et forme :SolidMasse moléculaire :564.46TFB-TBOA
CAS :<p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>Formule :C19H17F3N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.34hCAI/II-IN-5
CAS :<p>hCAI/II-IN-5 inhibits human carbonic anhydrase I & II, α-Glycosidase, and AChE, for diabetes, heart failure, Alzheimer's, ulcers, epilepsy research.</p>Formule :C21H18Cl2N8O4S2Couleur et forme :SolidMasse moléculaire :581.45Carbazomycin B
CAS :<p>Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).</p>Formule :C15H15NO2Couleur et forme :SolidMasse moléculaire :241.29Teglarinad chloride
CAS :<p>Teglarinad chloride (GMX-1777 chloride) is an inhibitor of NAMPT with antitumor activity that acts by interfering with DNA repair and inhibiting angiogenesis.</p>Formule :C30H43Cl2N5O8Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :672.6Darexaban glucuronide
CAS :<p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>Formule :C33H38N4O10Couleur et forme :SolidMasse moléculaire :650.68IDO1-IN-16
CAS :<p>IDO1-IN-16 (I-1) is an IDO1 inhibitor that targets holo-IDO1 (IC50: 127 nM).</p>Formule :C25H35BrFN5O2Couleur et forme :SolidMasse moléculaire :536.48ZSET-845
CAS :<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Formule :C21H18N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :314.38Dimethyl-bisphenol A
CAS :<p>DMBPA inhibits HIF-1α, promotes its degradation by detaching Hsp90, and reduces Vegfa mRNA expression.</p>Formule :C17H20O2Couleur et forme :SolidMasse moléculaire :256.34NPD-001
CAS :<p>NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).</p>Formule :C33H40N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.71Leniquinsin
CAS :Leniquinsin is an antihypertensive compound. It is a phosphodiesterase inhibitor and a potent vasodilator.Formule :C20H20N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.38ER21355
CAS :<p>ER21355, utilized for the treatment of prostatic diseases, acts as a phosphodiesterase 5 (PDE5) inhibitor.</p>Formule :C22H21ClN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.88IDO1/TDO-IN-3
CAS :<p>IDO1/TDO-IN-3 inhibits IDO1 (IC50: 0.005 μM) and TDO (IC50: 0.004 μM) with strong anti-tumor activity and low toxicity.</p>Formule :C16H6ClF2N3O2Couleur et forme :SolidMasse moléculaire :345.69POP-IN-2
CAS :<p>Compound 7k (POP-IN-2) is a potent POP inhibitor with Ki of 6 nM, useful in neurodegenerative and cancer studies.</p>Formule :C24H33BN2O5Couleur et forme :SolidMasse moléculaire :440.34AGN 191701
CAS :<p>AGN 191701 is an agonist of the Retinoid X receptor.</p>Formule :C23H28O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.53sPLA2-X Inhibitor 31
CAS :sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).Formule :C19H15F3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.33Enpp-1-IN-13
CAS :<p>Enpp-1-IN-13 inhibits ENPP1 (IC50: 1.29 μM) & ENPP3 (IC50: 20.2 μM) with anticancer properties.</p>Formule :C28H22ClN5OSCouleur et forme :SolidMasse moléculaire :512.03SQ28603
CAS :SQ28603 is a potent and selective neutral endopeptidase 3.4.24.11 (NEP) inhibitor.Formule :C13H17NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.34S32826 disodium
CAS :autotaxin inhibitorFormule :C21H36NNa2O4PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.47(-)-L-threo-PDMP (hydrochloride)
CAS :<p>(-)-L-threo-PDMP boosts ganglioside production, enhances neurite and synapse growth, and aids memory post-ischemia at 40 mg/kg/day.</p>Formule :C23H39ClN2O3Couleur et forme :SolidMasse moléculaire :427.03THR-0921
CAS :<p>THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study cardiovascular and metabolic diseases.</p>Formule :C28H25NO7SDegré de pureté :100% - 99.83%Couleur et forme :SolidMasse moléculaire :519.57Razaxaban hydrochloride
CAS :Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.Formule :C24H21ClF4N8O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :564.92MK-4409
CAS :MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.Formule :C22H17ClFN3O2SDegré de pureté :99.80% - 99.87%Couleur et forme :SolidMasse moléculaire :441.91Incadronate Disodium
CAS :Incadronate Disodium: halts bone loss, limits macrophage migration and inflammation, and induces cancer cell apoptosis in vitro.Formule :C8H19NNaO6P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.178Endothall
CAS :<p>Endothall is an effective protein phosphatase 2A (PP2A) inhibitor, exerting inhibitory effects on both PP2A and PP1, with IC50 values of 90 nM and 5 µM,</p>Formule :C8H10O5Degré de pureté :98.92% - ≥98%Couleur et forme :Cyrstalline White Solid The Monohydrate Is In The Form Of Colorless Crystals Non Corrosive Used As A Selective HerbicideMasse moléculaire :186.16Imazodan hydrochloride
CAS :<p>Imazodan hydrochloride (CI-914 HCl) is a potent and selective type III phosphodiesterase inhibitor used in the treatment of chronic congestive heart failure.</p>Formule :C13H13ClN4ODegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :276.72ML218
CAS :ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.Formule :C19H26Cl2N2ODegré de pureté :99.2% - 99.45%Couleur et forme :SolidMasse moléculaire :369.33Nampt-IN-9
CAS :<p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>Formule :C26H33N3O4Couleur et forme :SolidMasse moléculaire :451.56Imazodan
CAS :Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.Formule :C13H12N4ODegré de pureté :98% - 98.31%Couleur et forme :SolidMasse moléculaire :240.26Kurasoin B
CAS :<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Formule :C18H17NO2Couleur et forme :SolidMasse moléculaire :279.33Otamixaban
CAS :Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.Formule :C25H26N4O4Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :446.5ML-262
CAS :<p>ML-262 is an effective inhibitor of hepatic lipid droplet formation and is used in studies of non-alcoholic fatty liver disease.</p>Formule :C27H32N2O4SCouleur et forme :SolidMasse moléculaire :480.62Sp-cAMPS
CAS :<p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>Formule :C10H12N5O5PSCouleur et forme :SolidMasse moléculaire :345.27WAY127093B racemate
CAS :WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.Formule :C23H28N4O4Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :424.49(S)-Bromoenol lactone
CAS :<p>(S)-BEL, a chiral inhibitor of iPLA2β, blocks vasopressin-induced arachidonate release in A10 cells; IC50 = 2μM.</p>Formule :C16H13BrO2Couleur et forme :SolidMasse moléculaire :317.18SQ-31765
CAS :<p>SQ-31765 is a blocker of benzazepine calcium channel.</p>Formule :C24H27F3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.48Oxythiamine diphosphate
CAS :<p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>Formule :C12H17N3O8P2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.29CM39
CAS :<p>CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.</p>Formule :C19H15FN4OSCouleur et forme :SolidMasse moléculaire :366.41F-1394
CAS :<p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>Formule :C33H61N3O6Couleur et forme :SolidMasse moléculaire :595.85KCN1
CAS :<p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>Formule :C26H27NO5SCouleur et forme :SolidMasse moléculaire :465.56PKR activator 2
CAS :PKR activator 2 is a potent activator of pyruvate kinase-R (PKR).Formule :C18H16N8OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.44IDO-IN-14
CAS :<p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>Formule :C23H23ClN4O2Couleur et forme :SolidMasse moléculaire :422.91P-3FAX-Neu5Ac
CAS :<p>P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.</p>Formule :C22H30FNO14Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :551.47Glucokinase activator 3
CAS :<p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>Formule :C26H33N2O9PS2Couleur et forme :SolidMasse moléculaire :612.65UK-414,495
CAS :<p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>Formule :C16H25N3O3SCouleur et forme :SolidMasse moléculaire :339.45mIDH1-IN-1
CAS :<p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>Formule :C25H27N3O5Couleur et forme :SolidMasse moléculaire :449.5Enpp-1-IN-5
CAS :<p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>Formule :C17H26N6O4SCouleur et forme :SolidMasse moléculaire :410.49JTP-4819
CAS :<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Formule :C19H25N3O4Couleur et forme :SolidMasse moléculaire :359.42AMG-221
CAS :<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Formule :C14H22N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.4α-Amylase/α-Glucosidase-IN-2
CAS :α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μMFormule :C22H16ClN5Couleur et forme :SolidMasse moléculaire :385.85DP00477
CAS :<p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>Formule :C17H11ClF3N3OSCouleur et forme :SolidMasse moléculaire :397.8IDO1-IN-15
CAS :<p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>Formule :C13H14BrFN6O3Couleur et forme :SolidMasse moléculaire :401.19PF-06424439
CAS :<p>PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).</p>Formule :C22H26ClN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.94Antitumor agent-88
CAS :<p>Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).</p>Formule :C23H30N2O7SCouleur et forme :SolidMasse moléculaire :478.56CP 80633
CAS :<p>CP 80633 is a PDE4 inhibitor.</p>Formule :C18H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :316.39PDE11-IN-1
CAS :<p>PDE11-IN-1 is a PDE11 inhibitor and can be used for adrenal insufficiency research [1].</p>Formule :C16H10ClN3O3SCouleur et forme :SolidMasse moléculaire :359.79Transketolase-IN-4
CAS :<p>Transketolase-IN-4: IC50 3.9 μM; targets M. tuberculosis DXS (IC50 114.1 μM) & hinders SW620, LS174T, MIA PaCa-2 tumor cell growth.</p>Formule :C19H14ClN3ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :335.79SCD1 inhibitor-1
CAS :SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).Formule :C21H23N3NaO3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.54IMB-XMA0038
CAS :<p>IMB-XMA0038 is a Mycobacterium tuberculosis aspartate semialdehyde dehydrogenase inhibitor with antimicrobial activity for use in tuberculosis research.</p>Formule :C11H10N4O6Degré de pureté :98.94% - 99.96%Couleur et forme :SolidMasse moléculaire :294.22Metyltetraprole
CAS :<p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>Formule :C19H17ClN6O2Couleur et forme :SolidMasse moléculaire :396.83α-Glucosidase-IN-9
CAS :<p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>Formule :C19H12N4OSCouleur et forme :SolidMasse moléculaire :344.39GNX-865
CAS :<p>GNX-865 is an inhibitor of mitochondrial permeability transition pore (mtPTP).</p>Formule :C16H14ClNO3Couleur et forme :SolidMasse moléculaire :303.74Chaetomellic acid A
CAS :<p>Chaetomellic acid A inhibits farnesyltransferase (IC50=55nM), not active in cells, and selective over geranylgeranyltransferases (IC50: 92µM, 34µM).</p>Formule :C19H34O4Couleur et forme :SolidMasse moléculaire :326.47Trandolaprilat
CAS :<p>Trandolaprilat is an inhibitor of non-sulfhydryl angiotensin-converting enzyme.</p>Formule :C22H30N2O5Couleur et forme :Pale Yellow SolidMasse moléculaire :402.48hCAIX-IN-7
CAS :<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Formule :C18H12FNO3Couleur et forme :SolidMasse moléculaire :309.29DMPAC-Chol
CAS :<p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>Formule :C33H58N2O2Couleur et forme :SolidMasse moléculaire :514.83Glyoxalase I inhibitor 2
CAS :<p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>Formule :C24H23N3O4SCouleur et forme :SolidMasse moléculaire :449.52Fluindione
CAS :<p>Fluindione is a hematologic drug.</p>Formule :C15H9FO2Couleur et forme :SolidMasse moléculaire :240.23
