Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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N-Methylmoranoline
CAS :N-Methylmoranoline is an inhibitor of α-glucosidase.Formule :C7H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :177.2IDO-IN-16
CAS :<p>IDO-IN-16 (compound 5) is an IDO inhibitor (IC50: 36 nM).</p>Formule :C22H21F3N4OCouleur et forme :SolidMasse moléculaire :414.42RORγt/DHODH-IN-2
CAS :<p>RORγt/DHODH-IN-2 (compound 1) is a potent dual RORγt/DHODH inhibitor that can be used in the study of inflammatory bowel disease (IBD).</p>Formule :C25H30N4OSCouleur et forme :SolidMasse moléculaire :434.6Glyoxalase I inhibitor 1
CAS :<p>Glyoxalase I inhibitor 1 is a potent inhibitor of glyoxalase I (GLO1) (IC50: 26 nM).</p>Formule :C30H27FN6O4SCouleur et forme :SolidMasse moléculaire :586.64(+)-Cembrene A
CAS :<p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>Formule :C20H32Couleur et forme :SolidMasse moléculaire :272.47UK-371804 HCl
CAS :<p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>Formule :C14H17Cl2N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :422.29IDO/TDO-IN-1
CAS :<p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>Formule :C25H24FN5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.49SCD1 inhibitor-1
CAS :SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).Formule :C21H23N3NaO3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.54BMS 961
CAS :BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).Formule :C23H26FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.46A-1293201
CAS :<p>A-1293201 is a potent and selective NAMPT inhibitor.</p>Formule :C21H23N3O3Couleur et forme :SolidMasse moléculaire :365.43BBMP
CAS :<p>BBMP is an inhibitor of mitochondrial permeability transition pore.</p>Formule :C12H11BrN2O3SCouleur et forme :SolidMasse moléculaire :343.2Senazodan
CAS :Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.Formule :C15H14N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.3CFG920
CAS :<p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>Formule :C14H13ClN4OCouleur et forme :SolidMasse moléculaire :288.73L-5-BromoTryptophan
CAS :<p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>Formule :C11H11BrN2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :283.12DA 3003-2
CAS :<p>DA 3003-2: Potent Cdc25 inhibitor, halts cell division, may aid prostate cancer research.</p>Formule :C15H16ClN3O3Couleur et forme :SolidMasse moléculaire :321.76Entacapone sodium salt
CAS :<p>Entacapone sodium salt, a potent peripheral COMT inhibitor (IC50=151 nM), hinders α-syn/β-amyloid aggregation and protects PC12 cells.</p>Formule :C14H15N3NaO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.28TM6008
CAS :<p>TM6008 is an inhibitor of prolyl hydroxylase that protects against cell death after hypoxia.</p>Formule :C21H17N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.39Allylglycine
CAS :<p>Allylglycine is a glutamate decarboxylase inhibitor and a GAMMA-AMINOBUTYRIC ACID antagonist. It is used to induce convulsions in experimental animals.</p>Formule :C5H9NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :115.13Tibenelast sodium
CAS :Tibenelast sodium is an inhibitor of phosphodiesterase.Formule :C13H14NaO4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :289.3p-Synephrine
CAS :p-Synephrine is a natural product for research related to life sciences. The catalog number is T8265 and the CAS number is 614-35-7.Formule :C9H13NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :167.21Pulixin
CAS :Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).Formule :C14H11NO4Couleur et forme :SolidMasse moléculaire :257.24Incadronate Disodium
CAS :Incadronate Disodium: halts bone loss, limits macrophage migration and inflammation, and induces cancer cell apoptosis in vitro.Formule :C8H19NNaO6P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.178(RS)-Eflucimibe
CAS :<p>Eflucimibe is an ACAT inhibitor.</p>Formule :C29H43NO2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.72GSK2945
CAS :<p>GSK2945, a specific Rev-erbα antagonist, boosts CYP7A1 and cholesterol metabolism. EC50: 21.5 μM (mouse), 20.8 μM (human).</p>Formule :C20H18Cl2N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.34hACC2-IN-1
CAS :<p>hACC2-IN-1 is a potent inhibitor of acetyl coenzyme A carboxylase 2 (ACC2) with an IC50 value of 2.5 μM for hACC2. hACC2-IN-1 has potential for obesity studies.</p>Formule :C23H32N2O4SCouleur et forme :SolidMasse moléculaire :432.58SCH-351591
CAS :<p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>Formule :C17H10Cl2F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.18Nebicapone
CAS :Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.Formule :C14H11NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :273.24CAY10487
CAS :<p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>Formule :C13H15NO5Couleur et forme :SolidMasse moléculaire :265.26Enpp-1-IN-13
CAS :<p>Enpp-1-IN-13 inhibits ENPP1 (IC50: 1.29 μM) & ENPP3 (IC50: 20.2 μM) with anticancer properties.</p>Formule :C28H22ClN5OSCouleur et forme :SolidMasse moléculaire :512.03Spiraprilat
CAS :<p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>Formule :C20H26N2O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.56sPLA2-X Inhibitor 31
CAS :sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).Formule :C19H15F3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.33AGN 191701
CAS :<p>AGN 191701 is an agonist of the Retinoid X receptor.</p>Formule :C23H28O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.5393-O17O
CAS :<p>93-O17O is a cationic lipidoid used in lipid nanoparticles for spleen-targeted delivery and genome editing in mice.</p>Formule :C44H83N3O6Couleur et forme :SolidMasse moléculaire :750.15Isospaglumate sodium
CAS :<p>Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.</p>Formule :C11H16N2NaO8Couleur et forme :SolidMasse moléculaire :327.245OSMI-3
CAS :OSMI-3 is a potent and cell-permeable inhibitor of O-GlcNAc transferase (OGT) for the study of cancer and cardiovascular disease.Formule :C32H35N3O9S2Degré de pureté :99.03% - 99.08%Couleur et forme :SolidMasse moléculaire :669.77NCT-506
CAS :<p>NCT-506 is an orally bioavailable inhibitors of aldehyde dehydrogenase 1A1 (ALDH1A1) (IC50 of 7 nM).</p>Formule :C25H23FN4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :478.54α-Glucosidase-IN-2
CAS :<p>α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an</p>Formule :C17H11N3O2S2Couleur et forme :SolidMasse moléculaire :353.42FTase-IN-1
CAS :<p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>Formule :C23H16N2O2SCouleur et forme :SolidMasse moléculaire :384.45ARN19874
CAS :<p>ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].</p>Formule :C19H14N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.4OL-135
CAS :<p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>Formule :C21H22N2O2Couleur et forme :SolidMasse moléculaire :334.41POP-IN-2
CAS :<p>Compound 7k (POP-IN-2) is a potent POP inhibitor with Ki of 6 nM, useful in neurodegenerative and cancer studies.</p>Formule :C24H33BN2O5Couleur et forme :SolidMasse moléculaire :440.34IDO1/TDO-IN-3
CAS :<p>IDO1/TDO-IN-3 inhibits IDO1 (IC50: 0.005 μM) and TDO (IC50: 0.004 μM) with strong anti-tumor activity and low toxicity.</p>Formule :C16H6ClF2N3O2Couleur et forme :SolidMasse moléculaire :345.69M8891
CAS :M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.Formule :C20H17F2N3O3Couleur et forme :SolidMasse moléculaire :385.36GW844520
CAS :<p>GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.</p>Formule :C20H15ClF3NO3Couleur et forme :SolidMasse moléculaire :409.79PF-06471553
CAS :<p>PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).</p>Formule :C23H25N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.54Oosponol
CAS :<p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>Formule :C11H8O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :220.18DPC-423
CAS :<p>DPC-423 is a factor Xa inhibitor potentially for the treatment of thrombosis.</p>Formule :C25H21ClF4N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :568.97T-1095A
CAS :<p>T-1095A, a T-1095 metabolite, inhibits SGLTs, lowers blood glucose, improves glucose intolerance in mice, and prevents neuropathy in diabetic rats.</p>Formule :C24H26O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.46Crilvastatin
CAS :<p>Crilvastatin (PMD 387) is an HMGCR inhibitor with cholesterol-lowering activity that inhibits cholesterol uptake in rats with hereditary hypercholesterolemia.</p>Formule :C14H23NO3Degré de pureté :98.69% - 99.54%Couleur et forme :SolidMasse moléculaire :253.34ER21355
CAS :<p>ER21355, utilized for the treatment of prostatic diseases, acts as a phosphodiesterase 5 (PDE5) inhibitor.</p>Formule :C22H21ClN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.881E7-03
CAS :<p>1E7-03 is an inhibitor of HIV-1 transcription, by targeting host Protein Phosphatase-1 (PP1).</p>Formule :C28H29N3O6Couleur et forme :SolidMasse moléculaire :503.55ML299
CAS :<p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>Formule :C23H26BrFN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.38Aldophosphamide
CAS :<p>Aldophosphamide possesses apoptotic antitumor activity.</p>Formule :C7H15Cl2N2O3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.09NPD-001
CAS :<p>NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).</p>Formule :C33H40N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.71IDO1/TDO-IN-2
CAS :<p>IDO1/TDO-IN-2: IDO1/TDO inhibitor; IC50s: IDO1, 0.1μM; TDO, 0.07μM; potential for cancer research.</p>Formule :C16H9N3O2Couleur et forme :SolidMasse moléculaire :275.26L-Xylulose
CAS :<p>L-Xylulose: a rare sugar, key in metabolism, α-glucosidase inhibitor, lowers glucose, precursor to antiviral drug components.</p>Formule :C5H10O5Couleur et forme :SolidMasse moléculaire :150.13LAZABEMIDE
CAS :<p>Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).</p>Formule :C8H10ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :199.64Acetyltrialanine
CAS :<p>Acetyltrialanine is a dipeptide compound that binds at two sites on the Tb+3-pancreatic elastase complex and can be used as a nitrogen source.</p>Formule :C11H19N3O5Degré de pureté :99.53%Couleur et forme :White PowderMasse moléculaire :273.29Win-62005
CAS :<p>Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).</p>Formule :C12H10N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.23BN-82685
CAS :<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Formule :C12H15N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.33L 656224
CAS :L 656224 is a 5-LO inhibitor.Formule :C20H21ClO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.83Fenleuton
CAS :<p>Fenleuton is a 5-lipoxygenase inhibitor.</p>Formule :C17H15FN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :314.31Dimethyl-bisphenol A
CAS :<p>DMBPA inhibits HIF-1α, promotes its degradation by detaching Hsp90, and reduces Vegfa mRNA expression.</p>Formule :C17H20O2Couleur et forme :SolidMasse moléculaire :256.34Glucosylceramide synthase-IN-2
CAS :<p>T-690: Potent, BBB-permeable, oral GCS inhibitor; human IC50: 15 nM, mouse IC50: 190 nM; non-competitive with C8 ceramide/UDP glucose.</p>Formule :C22H20F3N3O4Couleur et forme :SolidMasse moléculaire :447.41GKA-22
CAS :<p>GKA-22 is a human glucokinase allosteric activator in the absence of glucose.</p>Formule :C22H22N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.49HCAIX-IN-2
CAS :HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).Formule :C19H16N8O4SCouleur et forme :SolidMasse moléculaire :452.45Mevalonic acid
CAS :<p>Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.</p>Formule :C6H12O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :148.16γ-Methylleucine
CAS :<p>Gamma-Methylleucine (2-Amino-3-tert-butylpropionic acid) is an auxiliary for copper-catalyzed asymmetric Michael reactions.</p>Formule :C7H15NO2Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :145.2Piragliatin
CAS :<p>Piragliatin (RO4389620) activates glucokinase, boosts insulin, and lowers glucose in type 2 diabetes.</p>Formule :C19H20ClN3O4SCouleur et forme :SolidMasse moléculaire :421.9Seviteronel racemate
CAS :Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase.Formule :C18H17F4N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.34Seviteronel R enantiomer
CAS :<p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>Formule :C18H17F4N3O3Degré de pureté :97.97% - >99.99%Couleur et forme :SolidMasse moléculaire :399.34ARL-67156 trisodium salt hydrate
CAS :ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.Formule :C15H24Br2N5O12P3Couleur et forme :SolidMasse moléculaire :719.11(Rac)-Etavopivat
CAS :<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Formule :C22H23N3O6SCouleur et forme :SolidMasse moléculaire :457.5Mufemilast
CAS :<p>Mufemilast is an inhibitor of phosphodiesterase 4 (PDE4).</p>Formule :C20H22N2O7S2Couleur et forme :SolidMasse moléculaire :466.53GS 389
CAS :<p>GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.</p>Formule :C19H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.39SAR629
CAS :<p>SAR-629 is an MGL inhibitor or 2-AG degradation inhibitor.</p>Formule :C20H19F2N5OCouleur et forme :SolidMasse moléculaire :383.39hCAIX-IN-11
CAS :<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Formule :C21H15ClN4O3Couleur et forme :SolidMasse moléculaire :406.82CD 2314
CAS :<p>CD2314 is a potent and subtype-selective RARβ receptor agonist with a Kd of 195 nM in S91 melanoma cells [1].</p>Formule :C23H24O2SCouleur et forme :SolidMasse moléculaire :364.5Carbazomycin B
CAS :<p>Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).</p>Formule :C15H15NO2Couleur et forme :SolidMasse moléculaire :241.29Anticancer agent 70
CAS :Compound 21 is a powerful anticancer agent with cytotoxicity against various cancers, causing cell cycle arrest and affecting p53/p21 levels and mitochondria.Formule :C13H9Cl2N3O2SCouleur et forme :SolidMasse moléculaire :342.2hCAI/II-IN-5
CAS :<p>hCAI/II-IN-5 inhibits human carbonic anhydrase I & II, α-Glycosidase, and AChE, for diabetes, heart failure, Alzheimer's, ulcers, epilepsy research.</p>Formule :C21H18Cl2N8O4S2Couleur et forme :SolidMasse moléculaire :581.45TFB-TBOA
CAS :<p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>Formule :C19H17F3N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.34LY 56110
CAS :<p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>Formule :C17H12Cl2N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.2LY367385
CAS :<p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>Formule :C10H11NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :209.2SHP2 inhibitor LY6
CAS :<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Formule :C30H27Cl2N3O4Couleur et forme :SolidMasse moléculaire :564.46PKM2 activator 3
CAS :<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Formule :C15H11ClF2N2O3SCouleur et forme :SolidMasse moléculaire :372.77LB42908
CAS :<p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>Formule :C32H31N5O3Couleur et forme :SolidMasse moléculaire :533.62N-Oleoyl Leucine
CAS :<p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>Formule :C24H45NO3Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :395.62MEDS433
CAS :<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Formule :C20H11F4N3O2Couleur et forme :SolidMasse moléculaire :401.31Loxoprofenol-SRS
CAS :<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Formule :C15H20O3Couleur et forme :SolidMasse moléculaire :248.32SR1555 HCl
CAS :<p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>Formule :C22H22F6N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.41TPN729MA
CAS :<p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>Formule :C29H40N6O8SCouleur et forme :SolidMasse moléculaire :632.73GlcN-6-P Synthase-IN-1
CAS :<p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase & CYP3A4. Has antimicrobial activity and CNS penetration.'</p>Formule :C20H21N7SCouleur et forme :SolidMasse moléculaire :391.49hCAI/II-IN-2
CAS :<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Formule :C12H12N4O5S2Couleur et forme :SolidMasse moléculaire :356.38103D5R
CAS :<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4SCD1 Inhibitor
CAS :<p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>Formule :C21H20F3N3O3Couleur et forme :SolidMasse moléculaire :419.4FR-221647
CAS :<p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>Formule :C14H17N3O2Couleur et forme :SolidMasse moléculaire :259.3CAY10761
CAS :<p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).</p>Formule :C7H8N4O2S2Couleur et forme :SolidMasse moléculaire :244.29Kurasoin B
CAS :<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Formule :C18H17NO2Couleur et forme :SolidMasse moléculaire :279.33YCT529 free acid
CAS :<p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>Formule :C29H25NO3Couleur et forme :SolidMasse moléculaire :435.51hCAII-IN-1
CAS :<p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>Formule :C21H21BrN6O4SCouleur et forme :SolidMasse moléculaire :533.4Quazodine
CAS :<p>Quazodine is a phosphodiesterase inhibitor.</p>Formule :C12H14N2O2Couleur et forme :SolidMasse moléculaire :218.25Izumerogant
CAS :<p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>Formule :C22H18ClF4N5O2Couleur et forme :SolidMasse moléculaire :495.86TM-1
CAS :<p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>Formule :C26H32N2O6Couleur et forme :SolidMasse moléculaire :468.54CAY10762
CAS :<p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>Formule :C15H13NOSCouleur et forme :SolidMasse moléculaire :255.33OHM1
CAS :<p>OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53</p>Formule :C24H42N6O5Couleur et forme :SolidMasse moléculaire :494.63sEH inhibitor-6
CAS :<p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>Formule :C21H14ClN3O2Couleur et forme :SolidMasse moléculaire :375.81hCAXII-IN-2
CAS :<p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>Formule :C21H18ClN3O4Couleur et forme :SolidMasse moléculaire :411.84Teglicar
CAS :<p>Teglicar is a selective and reversible liver isoform of carnitine palmitoyl-transferase 1 (L-CPT1) inhibitor.</p>Formule :C22H45N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.61α-Glucosidase-IN-16
CAS :<p>α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM.</p>Formule :C22H18FNSCouleur et forme :SolidMasse moléculaire :347.45Kojibiose
CAS :<p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>Formule :C12H22O11Degré de pureté :99.933%Couleur et forme :SolidMasse moléculaire :342.3SAR127303
CAS :<p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>Formule :C16H17ClF6N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.83(E/Z)-Ensifentrine
CAS :<p>RPL-554 (LS-193,855) is a dual PDE3/4 inhibitor with bronchodilator and anti-inflammatory properties, in trials for asthma and hay fever by Verona Pharma.</p>Formule :C26H31N5O4Couleur et forme :SolidMasse moléculaire :477.56Y-29794
CAS :<p>Y-29794, a covalent POP inhibitor with a Ki of 0.95 nM, holds research potential for neurodegenerative diseases and cancer.</p>Formule :C22H32N2OS2Couleur et forme :SolidMasse moléculaire :404.63YC-001
CAS :<p>YC-001: inverse agonist/antagonist for rod opsin, prevents light-induced retinal degeneration.</p>Formule :C12H7ClO2S2Couleur et forme :SolidMasse moléculaire :282.77YM 26734
CAS :<p>Competitive inhibitor of secretory phospholipase A2 (sPLA2)</p>Formule :C45H62O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :730.97Imidazoleacetic acid
CAS :<p>Imidazoleacetic acid, an endogenous ligand, stimulates imidazole receptors.</p>Formule :C5H6N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :126.11LAS-31180
CAS :<p>LAS-31180 is a phosphodiesterase 3 inhibitor. It also has positive inotropic and vasodilator properties.</p>Formule :C11H12N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :252.29ML202
CAS :<p>ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.</p>Formule :C18H17N3O3S2Couleur et forme :SolidMasse moléculaire :387.48Xanthine oxidoreductase-IN-1
CAS :<p>Xanthine oxidoreductase-IN-1 is a xanthine oxidoreductase (XOR) inhibitor with an IC 50 value of 7.0 nM.</p>Formule :C18H20N4O2Couleur et forme :SolidMasse moléculaire :324.38SCD1-IN-1
CAS :<p>SCD1-IN-1, a potent inhibitor of SCD1 (IC50: 5.8 nM), is valuable in dermatologic research [1].</p>Formule :C20H20F3NO4Couleur et forme :SolidMasse moléculaire :395.37SQ 28853
CAS :<p>SQ 28853 is an inhibitor of ACE with diuretic properties.</p>Formule :C19H25ClN4NaO6S3Couleur et forme :SolidMasse moléculaire :560.05HX-600
CAS :<p>HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.</p>Formule :C29H30N2O2Couleur et forme :SolidMasse moléculaire :438.56BMS 740808
CAS :<p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>Formule :C31H27F3N6O3Couleur et forme :SolidMasse moléculaire :588.58TMCB
CAS :<p>CK2 and ERK8 inhibitor</p>Formule :C11H9Br4N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.82Lp-PLA2-IN-11
CAS :<p>Lp-PLA2-IN-11, a potent Lp-PLA2 inhibitor, may be explored for atherosclerosis and Alzheimer's (WO2014114249A1, E145).</p>Formule :C22H20F4N4O3Couleur et forme :SolidMasse moléculaire :464.41Chaetomellic acid A
CAS :<p>Chaetomellic acid A inhibits farnesyltransferase (IC50=55nM), not active in cells, and selective over geranylgeranyltransferases (IC50: 92µM, 34µM).</p>Formule :C19H34O4Couleur et forme :SolidMasse moléculaire :326.47DHODH-IN-21
CAS :<p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>Formule :C20H19ClF4N6O4Couleur et forme :SolidMasse moléculaire :518.85LEO-29102
CAS :<p>LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.</p>Formule :C20H22Cl2N2O5Couleur et forme :SolidMasse moléculaire :441.31Glucosylceramide synthase-IN-1
CAS :<p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>Formule :C24H20F4N2O3Couleur et forme :SolidMasse moléculaire :460.42α-Glycosidase-IN-1
CAS :<p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>Formule :C21H19N9O6S2Couleur et forme :SolidMasse moléculaire :557.56Agn 190727
CAS :<p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>Formule :C20H22O2Couleur et forme :SolidMasse moléculaire :294.39RYL-552
CAS :<p>RYL-552 is a potent inhibitor of PfNDH2.</p>Formule :C24H17F4NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.39HIF-1α-IN-3
CAS :<p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>Formule :C19H17N5O2Couleur et forme :SolidMasse moléculaire :347.37Delapril
CAS :<p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>Formule :C26H32N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.54Liarozole HCl
CAS :<p>Liarozole HCl: antineoplastic, boosts ATRA levels, impedes cell growth, promotes differentiation, aromatase inhibitor.</p>Formule :C17H14Cl2N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.23Umbralisib sulfate
CAS :<p>Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.</p>Formule :C31H26F3N5O7SCouleur et forme :SolidMasse moléculaire :669.63MDK-4823
CAS :<p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>Formule :C28H36N4OCouleur et forme :SolidMasse moléculaire :444.61Enpp-1-IN-8
CAS :<p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>Formule :C19H26N6O4SCouleur et forme :SolidMasse moléculaire :434.51FAAH-IN-7
<p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>Formule :C26H29N3O4Couleur et forme :SolidMasse moléculaire :447.53hCAIX-IN-3
CAS :<p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>Formule :C21H21BrN6O4SCouleur et forme :SolidMasse moléculaire :533.4ATX inhibitor 8
CAS :<p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>Formule :C28H26N10OCouleur et forme :SolidMasse moléculaire :518.57hCAIX-IN-14
CAS :hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .Formule :C11H17ClN6O2SCouleur et forme :SolidMasse moléculaire :332.81PKM2 activator 4
CAS :<p>PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.</p>Formule :C16H16N2O4SCouleur et forme :SolidMasse moléculaire :332.37α-Glucosidase-IN-21
CAS :<p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>Formule :C24H23NO2SCouleur et forme :SolidMasse moléculaire :389.513,3-Dimethyl-1-butanol
CAS :<p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>Formule :C6H14OCouleur et forme :SolidMasse moléculaire :102.17Spirapril
CAS :<p>Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.</p>Formule :C22H30N2O5S2Couleur et forme :SolidMasse moléculaire :466.61hCA IX-IN-2
<p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>Formule :C23H24N2O4STeCouleur et forme :SolidMasse moléculaire :552.11Arasertaconazole
CAS :<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Formule :C20H15Cl3N2OSCouleur et forme :SolidMasse moléculaire :437.77A-908292
CAS :<p>A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.</p>Formule :C18H20N2O4SCouleur et forme :SolidMasse moléculaire :360.43FABP-IN-2
CAS :<p>FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.</p>Formule :C25H21ClN2O3Couleur et forme :SolidMasse moléculaire :432.9ENPP1 inhibitor 43
CAS :<p>ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.</p>Formule :C16H18N6O3SCouleur et forme :SolidMasse moléculaire :374.42PDE4-IN-11
CAS :<p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>Formule :C21H19FN2O2Couleur et forme :SolidMasse moléculaire :350.39Xanthine oxidase-IN-4
CAS :<p>Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.</p>Formule :C15H13N5O2Couleur et forme :SolidMasse moléculaire :295.3PRRSV/CD163-IN-1
CAS :<p>PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.</p>Formule :C25H24FN5O5S2Couleur et forme :SolidMasse moléculaire :557.62hCAIX-IN-8
CAS :<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Formule :C19H16N4O6Couleur et forme :SolidMasse moléculaire :396.35D-threo-PPMP hydrochloride
CAS :<p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>Formule :C29H51ClN2O3Couleur et forme :SolidMasse moléculaire :511.19NPD-1335
CAS :<p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>Formule :C28H29N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.55Sch 34826
CAS :<p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>Formule :C27H34N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.57Boc-Glu(OBzl)-OSu
CAS :<p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>Formule :C21H26N2O8Couleur et forme :SolidMasse moléculaire :434.44AMG-221
CAS :<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Formule :C14H22N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.4JTP-4819
CAS :<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Formule :C19H25N3O4Couleur et forme :SolidMasse moléculaire :359.42Andolast
CAS :<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Formule :C15H11N9OCouleur et forme :SolidMasse moléculaire :333.31sEH inhibitor-14
CAS :<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Formule :C16H12F3N3O4Couleur et forme :SoildMasse moléculaire :367.28Quinethazone
CAS :<p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>Formule :C10H12ClN3O3SCouleur et forme :Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)Masse moléculaire :289.74MitoTEMPO hydrate
CAS :<p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>Formule :C29H35N2O2P·Cl·H2OCouleur et forme :SolidMasse moléculaire :528.04SGK1 inhibitor
CAS :<p>SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.</p>Formule :C17H12Cl2N6O2SCouleur et forme :SolidMasse moléculaire :435.29CAY10485
CAS :<p>CAY10485 blocks human ACAT-1 & ACAT-2 (IC50: 95 & 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.</p>Formule :C27H27NO7Couleur et forme :SolidMasse moléculaire :477.51ATX inhibitor 11
CAS :<p>ATX inhibitor 11 blocks autotaxin (IC50: 2.7 nM), reduces fibrosis and α-SMA in mice. Useful for lung fibrosis studies.</p>Formule :C32H35N5O6Couleur et forme :SolidMasse moléculaire :585.65AMG-7980
CAS :<p>AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.</p>Formule :C19H22N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :338.4Xanthine oxidoreductase-IN-2
CAS :<p>Xanthine oxidoreductase-IN-2 inhibits XOR with 7.2 nM IC50 and shows hypouricemic effects in mice.</p>Formule :C21H19N3O2Couleur et forme :SolidMasse moléculaire :345.39α-Glucosidase-IN-8
CAS :<p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>Formule :C19H20FN3O2Couleur et forme :SolidMasse moléculaire :341.38Eggmanone
CAS :<p>EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.</p>Formule :C20H20N2O2S3Couleur et forme :SolidMasse moléculaire :416.58hCAIX-IN-6
CAS :<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Formule :C18H12N2O4SCouleur et forme :SolidMasse moléculaire :352.36Carbonic anhydrase inhibitor 13
CAS :<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Formule :C17H15N5O3S2Couleur et forme :SolidMasse moléculaire :401.46IDO1-IN-17
CAS :<p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>Formule :C28H32BrClFN5O2Couleur et forme :SolidMasse moléculaire :604.94IDO-IN-14
CAS :<p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>Formule :C23H23ClN4O2Couleur et forme :SolidMasse moléculaire :422.91CYP3A4-IN-1
CAS :<p>CYP3A4-IN-1 is a potent inhibitor of cytochrome P450 3A4 (CYP3A4) (IC50: 0.085 μM).</p>Formule :C31H37N5O3SCouleur et forme :SolidMasse moléculaire :559.72FXR agonist 4
<p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>Formule :C21H28ClN3OCouleur et forme :SolidMasse moléculaire :373.92KCN1
CAS :<p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>Formule :C26H27NO5SCouleur et forme :SolidMasse moléculaire :465.56F-1394
CAS :<p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>Formule :C33H61N3O6Couleur et forme :SolidMasse moléculaire :595.85CYP1B1-IN-3
CAS :<p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>Formule :C20H16FN3O2S2Couleur et forme :SolidMasse moléculaire :413.49CM39
CAS :<p>CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.</p>Formule :C19H15FN4OSCouleur et forme :SolidMasse moléculaire :366.41Oxythiamine diphosphate
CAS :<p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>Formule :C12H17N3O8P2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.29DTP348
CAS :<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Formule :C6H11N5O4SCouleur et forme :SolidMasse moléculaire :249.25Nitrefazole
CAS :<p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>Formule :C10H8N4O4Couleur et forme :SolidMasse moléculaire :248.19URB-694
CAS :<p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>Formule :C19H21NO3Couleur et forme :SolidMasse moléculaire :311.3711β-HSD1-IN-6
CAS :<p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>Formule :C21H19ClN4OCouleur et forme :SolidMasse moléculaire :378.86Tyrphostin AG 1112
CAS :<p>Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.</p>Formule :C15H10N6Couleur et forme :SolidMasse moléculaire :274.28FASN-IN-4
CAS :<p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>Formule :C26H27N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.58Glucocerebrosidase-IN-1
CAS :<p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>Formule :C13H27NO3Couleur et forme :SolidMasse moléculaire :245.36MDPD
CAS :<p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>Formule :C21H19N3O3Couleur et forme :SolidMasse moléculaire :361.39Vorozole
CAS :<p>Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in</p>Formule :C16H13ClN6Degré de pureté :99.65% - 99.94%Couleur et forme :SolidMasse moléculaire :324.77Lombricine
CAS :<p>Lombricine, as a phosphodiester of 2-guanidinoethanol and D-serine in structure, is a phosphagen that is unique to earthworms.</p>Formule :C6H15N4O6PCouleur et forme :SolidMasse moléculaire :270.18Antiproliferative agent-10
<p>Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.</p>Formule :C35H36Cl2N7PRuCouleur et forme :SolidMasse moléculaire :757.66LY 113174
CAS :<p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>Formule :C17H10Cl2N2Couleur et forme :SolidMasse moléculaire :313.18FC11409B
CAS :<p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>Formule :C29H23BF4N2O3SCouleur et forme :SolidMasse moléculaire :566.38Cholesteryl Palmitoleate
CAS :<p>Cholesteryl palmitoleate, a cholesterol ester, exhibits elevated plasma levels in ApoE-/- mice following exposure to cigarette smoke and in pediatric patients diagnosed with biliary atresia. It serves as a standard for identifying cholesterol esters in human meibomian gland secretions.</p>Formule :C43H74O2Couleur et forme :SolidMasse moléculaire :623.1RORγt modulator 3
CAS :<p>RORγt modulator 3 is a modulator of retinol-related orphan receptor γt (RORγt) and can be used to study RORγt-mediated diseases such as pain, COPD, inflammation</p>Formule :C25H25ClFN3O4SCouleur et forme :SolidMasse moléculaire :518Zidovudine glucuronide
CAS :<p>Zidovudine glucuronide: an NRTI antiretroviral for HIV/AIDS treatment; blocks HIV reverse transcriptase, stops viral DNA formation.</p>Formule :C16H21N5O10Couleur et forme :SolidMasse moléculaire :443.37
