Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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Ro 41-0960
CAS :<p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>Formule :C13H8FNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.2Endothelial lipase inhibitor-1
CAS :<p>Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.</p>Formule :C22H22N4O4Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :406.43Deltasonamide 2
CAS :<p>Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>Formule :C30H39ClN6O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :647.25IHVR-11029
CAS :<p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>Formule :C18H27F2NO5Couleur et forme :SolidMasse moléculaire :375.41CP-532623
CAS :<p>CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.</p>Formule :C27H27F9N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :598.5IDO-IN-3
CAS :IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).Formule :C11H12BrFN6O2Couleur et forme :SolidMasse moléculaire :359.15Rovazolac
CAS :<p>Rovazolac (ALX-101) is a liver x receptor (LXR) modulator used in the study of immune system disorders and atopic dermatitis.</p>Formule :C21H19F3N2O4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :452.45ALDH1A1-IN-2
CAS :<p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>Formule :C25H23ClN4O3SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :494.99BAY 73-6691
CAS :<p>BAY 73-6691 is an inhibitor of brain penetrant PDE9A.</p>Formule :C15H12ClF3N4OCouleur et forme :SolidMasse moléculaire :356.73β-Amino Acid Imagabalin Hydrochloride
CAS :β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.Formule :C9H20ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :209.7114-dehydro Zymostenol
CAS :<p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>Formule :C27H44OCouleur et forme :SolidMasse moléculaire :384.64TAK 21d
CAS :<p>Potent FAAH inhibitor</p>Formule :C19H17F2N7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.38GSK376501A
CAS :<p>GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.</p>Formule :C32H37NO6Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :531.64PF 04671536 hydrochloride
CAS :<p>Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.</p>Formule :C14H19ClN8OSCouleur et forme :SolidMasse moléculaire :382.87Mesopram
CAS :<p>PDE4 inhibitor, orally active</p>Formule :C14H19NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.3hCAI/II-IN-2
CAS :<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Formule :C12H12N4O5S2Couleur et forme :SolidMasse moléculaire :356.38103D5R
CAS :<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4Cgp 8065
CAS :<p>Cgp 8065 is a filaricidal compound, a dithiocarbamate-derivative of amoscanate.</p>Formule :C16H15N3O4S2Couleur et forme :SolidMasse moléculaire :377.44Prolyl Endopeptidase Inhibitor 1
CAS :Prolyl Endopeptidase Inhibitor 1 is a potent inhibitor of prolyl endopeptidase (PEP; PE)(Ki : 15 nM) , has anti-amnesic effect.Formule :C15H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.36Enazadrem
CAS :<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Formule :C18H25N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.41Acetaldophosphamide
CAS :<p>Acetaldophosphamide is a novel stable aldophosphamide analog.</p>Formule :C11H21Cl2N2O6PCouleur et forme :SolidMasse moléculaire :379.17SAR629
CAS :<p>SAR-629 is an MGL inhibitor or 2-AG degradation inhibitor.</p>Formule :C20H19F2N5OCouleur et forme :SolidMasse moléculaire :383.39SDZ-MKS 492
CAS :SDZ-MKS 492 is a selective type III isozyme cyclic nucleotide phosphodiesterase inhibitor.Formule :C20H27N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.46SHP836
CAS :<p>SHP836 is an inhibitor of SHP2 allosteric (IC50: 12 μM for the full-length SHP2).</p>Formule :C16H19Cl2N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.26Dapaconazole
CAS :<p>Dapaconazole is used as a drug candidate for antifungals.</p>Formule :C19H15Cl2F3N2OCouleur et forme :SolidMasse moléculaire :415.24Quinalizarin
CAS :Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.Formule :C14H8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :272.214-Desmethyl Istradefylline
CAS :<p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>Formule :C19H22N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :370.407-Biopterin
CAS :<p>7-Biopterin, a 7-substituted pterin, forms non-enzymatically and elevates in urine of hyperphenylalaninemics with PCBD mutations.</p>Formule :C9H11N5O3Couleur et forme :SolidMasse moléculaire :237.22GS 389
CAS :<p>GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.</p>Formule :C19H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.39Transketolase-IN-2
CAS :<p>Transketolase-IN-2, potent herbicidal agent, inhibits weeds like Digitaria sanguinalis and Amaranthus retroflexus.</p>Formule :C18H9F3N2O3SCouleur et forme :SolidMasse moléculaire :390.34IQA
CAS :<p>IQA is a casein kinase 2 (CK2) inhibitor.</p>Formule :C17H12N2O3Couleur et forme :SolidMasse moléculaire :292.29Dibefurin
CAS :<p>Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.</p>Formule :C18H16O8Couleur et forme :SolidMasse moléculaire :360.3111β-HSD1-IN-10
CAS :<p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>Formule :C16H10F3NO2Couleur et forme :SolidMasse moléculaire :305.25Enpp-1-IN-9
CAS :<p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>Formule :C17H24N4O5SCouleur et forme :SolidMasse moléculaire :396.46AMP-Deoxynojirimycin
CAS :<p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>Formule :C22H39NO5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :397.55BMS-351
CAS :<p>BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.</p>Formule :C15H12F3N3Couleur et forme :SolidMasse moléculaire :291.27Epostane
CAS :<p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>Formule :C22H31NO3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :357.49SCD1 Inhibitor
CAS :<p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>Formule :C21H20F3N3O3Couleur et forme :SolidMasse moléculaire :419.4BMS 961
CAS :BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).Formule :C23H26FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.46Choline theophyllinate
CAS :<p>Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and</p>Formule :C12H21N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.33RORγt inverse agonist 28
CAS :<p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>Formule :C23H18Cl2F3NO5SCouleur et forme :SolidMasse moléculaire :548.36SHP844
CAS :<p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>Formule :C29H24ClN5O6Couleur et forme :SolidMasse moléculaire :573.98Factor VII-IN-1
CAS :<p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>Formule :C15H10BrNO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :332.15hCAIX-IN-10
CAS :<p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>Formule :C28H21N3O3SCouleur et forme :SolidMasse moléculaire :479.55FR-221647
CAS :<p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>Formule :C14H17N3O2Couleur et forme :SolidMasse moléculaire :259.3CAY10761
CAS :<p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).</p>Formule :C7H8N4O2S2Couleur et forme :SolidMasse moléculaire :244.29Y-29794 oxalate
CAS :<p>Inhibitor of prolyl endopeptidase</p>Formule :C25H36N2O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.69S07-2010
CAS :<p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>Formule :C19H21N3O3SDegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :371.45Sp-Cyclic AMPS (sodium salt)
CAS :<p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>Formule :C10H12N5NaO5PSCouleur et forme :SolidMasse moléculaire :367.254,5,6,7-Tetrabromobenzimidazole
CAS :<p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>Formule :C7H2Br4N2Couleur et forme :SolidMasse moléculaire :433.72Atreleuton
CAS :<p>Atreleuton (ABT-761), reversible oral 5-LO inhibitor, selectively blocks leukotriene formation.</p>Formule :C16H15FN2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.37Argininic acid
CAS :<p>Argininic acid is an α-amino acid used in the biosynthesis of proteins.</p>Formule :C6H13N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :175.19Sp-cAMPS
CAS :<p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>Formule :C10H12N5O5PSCouleur et forme :SolidMasse moléculaire :345.27hCAI/II-IN-3
CAS :<p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>Formule :C16H18N4O4S2Couleur et forme :SolidMasse moléculaire :394.47GOAT-IN-1
CAS :<p>GOAT-IN-1 blocks GOAT, potentially treating diabetes, hyperlipidemia, and various brain disorders.</p>Formule :C18H13ClF3NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.81Xanthine oxidase-IN-7
CAS :<p>Xanthine oxidase-IN-7: Potent oral XO inhibitor (IC50=0.36μM), lowers serum uric acid, promising for hyperuricemia/gout research.</p>Formule :C16H14N4O2Couleur et forme :SolidMasse moléculaire :294.31Glyoxalase I inhibitor
CAS :<p>Glyoxalase I inhibitor, a candidate for anticancer agents, is a potent Glyoxalase I (GLO1) inhibitor.</p>Formule :C21H30BrClN4O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :613.919(R)-HODE
CAS :9(R)-HODE, a linoleic acid product, is made by some human/bovine endothelial cells, but its function and forming enzyme are unknown.Formule :C18H32O3Couleur et forme :SolidMasse moléculaire :296.44TP-004
CAS :<p>TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).</p>Formule :C17H16F3N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.34L-(-)-threo-3-Hydroxyaspartic acid
CAS :L-(-)-threo-3-Hydroxyaspartic acid is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.Formule :C4H7NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :149.1Riboflavine phosphate
CAS :<p>Riboflavine phosphate (Flavin mononucleotide) is a derivative of Riboflavin.</p>Formule :C17H21N4O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.34ATX inhibitor 14
CAS :<p>ATX inhibitor 14, an indole carbamate, potently blocks self-adhesive proteins (IC50: 0.41 nM), aiding fibrosis research.</p>Formule :C26H26Cl2N4O3SCouleur et forme :SolidMasse moléculaire :545.48hCAIX/XII-IN-6
<p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>Formule :C26H23N3O6S4Couleur et forme :SolidMasse moléculaire :601.74Kurasoin B
CAS :<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Formule :C18H17NO2Couleur et forme :SolidMasse moléculaire :279.33ATX inhibitor 5
CAS :ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.Formule :C22H18ClF3N6ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :474.87PX20606
CAS :<p>PX20606 is an orally active farnesoid X receptor (FXR) agonist, demonstrating EC50 values of 220 nM (mFXR) and 50 nM (hFXR) in Gal4-FXR assays. It induces the expression of the tumor suppressor gene NDRG2 and inhibits tumor growth and metastasis in a mouse HCC model. Additionally, PX20606 exhibits hepatoprotective properties.</p>Formule :C29H22Cl3NO4Couleur et forme :SolidMasse moléculaire :554.85YCT529 free acid
CAS :<p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>Formule :C29H25NO3Couleur et forme :SolidMasse moléculaire :435.51JBP485
CAS :<p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>Formule :C8H12N2O4Couleur et forme :SolidMasse moléculaire :200.19Lipoxygenin
CAS :<p>Lipoxygenin: IC50 of 5 μM inhibits 5-LO, hedgehog, TGF-β, activin A, BMP, Wnt signaling, and boosts cardiac marker TnnT in iPSCs.</p>Formule :C24H22N2O4Couleur et forme :SolidMasse moléculaire :402.44Antitumor agent-87
CAS :<p>Antitumor agent-87: potent, high CYP1A1 affinity (Ki 0.23µM), antiproliferative, arrests G2/M cell cycle.</p>Formule :C22H28N2O6SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :448.53Quinapril-d5
CAS :<p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>Formule :C25H25D5N2O5Couleur et forme :SolidMasse moléculaire :443.55Anserinone B
CAS :<p>Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).</p>Formule :C11H14O4Couleur et forme :SolidMasse moléculaire :210.23EDP-305
CAS :<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Formule :C36H58N2O5SCouleur et forme :SolidMasse moléculaire :630.92Ciraparantag
CAS :<p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>Formule :C22H48N12O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.7Safusidenib
CAS :<p>Safusidenib, oral mutant IDH1 inhibitor, selectively targets IDH1R132H/C mutations with IC50 of 15/130 nM; impairs chondrosarcoma growth.</p>Formule :C25H18Cl3FN2O4Couleur et forme :SolidMasse moléculaire :535.78IHMT-PI3Kδ-372
CAS :<p>IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.</p>Formule :C26H23F2N7O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :503.5hCAII-IN-1
CAS :<p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>Formule :C21H21BrN6O4SCouleur et forme :SolidMasse moléculaire :533.4Methazolamide-d6
CAS :<p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>Formule :C5H2D6N4O3S2Couleur et forme :SolidMasse moléculaire :242.31Quazodine
CAS :<p>Quazodine is a phosphodiesterase inhibitor.</p>Formule :C12H14N2O2Couleur et forme :SolidMasse moléculaire :218.25Izumerogant
CAS :<p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>Formule :C22H18ClF4N5O2Couleur et forme :SolidMasse moléculaire :495.86ONO-6126
CAS :<p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>Formule :C20H27N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :373.45Trandolaprilate hydrate
CAS :<p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>Formule :C22H32N2O6Couleur et forme :SolidMasse moléculaire :420.5A-1293201
CAS :<p>A-1293201 is a potent and selective NAMPT inhibitor.</p>Formule :C21H23N3O3Couleur et forme :SolidMasse moléculaire :365.43ASP3662
CAS :<p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>Formule :C19H16ClF3N4O2Couleur et forme :SolidMasse moléculaire :424.8LCL521
CAS :<p>LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.</p>Formule :C31H52N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :592.77TM-1
CAS :<p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>Formule :C26H32N2O6Couleur et forme :SolidMasse moléculaire :468.54Ro-15-2041
CAS :Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.Formule :C12H12BrN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.15IACS-8968 S-enantiomer
CAS :<p>IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Formule :C17H18F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.35RORγt/DHODH-IN-2
CAS :<p>RORγt/DHODH-IN-2 (compound 1) is a potent dual RORγt/DHODH inhibitor that can be used in the study of inflammatory bowel disease (IBD).</p>Formule :C25H30N4OSCouleur et forme :SolidMasse moléculaire :434.6TF-S14
CAS :<p>TF-S14 is an inverse agonist of RORγt. It functions by binding to RORγt and inhibiting its activity, leading to a reduction in Th17 cell-associated cytokine production, including IL-17A, IL-21, and IL-22. TF-S14 is applicable in research related to autoimmune diseases and allogeneic transplant rejection.</p>Formule :C22H27N3O2SCouleur et forme :SolidMasse moléculaire :397.53Transketolase-IN-4
CAS :<p>Transketolase-IN-4: IC50 3.9 μM; targets M. tuberculosis DXS (IC50 114.1 μM) & hinders SW620, LS174T, MIA PaCa-2 tumor cell growth.</p>Formule :C19H14ClN3ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :335.79AVX-001
CAS :<p>AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.</p>Formule :C21H29F3OSCouleur et forme :SolidMasse moléculaire :386.51NCX899
CAS :<p>NCX899 shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.</p>Formule :C23H33N3O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.52CAY10762
CAS :<p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>Formule :C15H13NOSCouleur et forme :SolidMasse moléculaire :255.33Afegostat HCl
CAS :<p>Afegostat: GCase inhibitor, Ki ~30 nM for wild-type/mutant, experimental Gaucher's disease drug.</p>Formule :C6H14ClNO3Couleur et forme :SolidMasse moléculaire :183.63BAY 59-9435
CAS :<p>HSL-IN-2 is a selective inhibitor of Hormone Sensitive Lipase (HSL; IC50: 0.023 μM).</p>Formule :C14H22N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.34Lu AF58801
CAS :<p>Lu AF58801 is a brain penetrant positive allosteric and selective modulator of alpha-7 nicotinic acetylcholine receptors.</p>Formule :C20H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :325.44′-Deoxyphlorizin
CAS :<p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>Formule :C21H24O9Couleur et forme :SolidMasse moléculaire :420.41KB 5666
CAS :<p>KB 5666, a quinazoline derivative, is a lipid peroxidation inhibitor. It protects the brain from both cellular and functional consequences of ischemia.</p>Formule :C24H32N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.54Levophencynonate HCl
CAS :<p>Levophencynonate HCl is a muscarinic receptor antagonist.</p>Formule :C22H32ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.95GSK 264220A
CAS :<p>endothelial lipase and lipoprotein lipase inhibitor</p>Formule :C17H21N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.43HT-0712
CAS :<p>HT-0712 is a phosphodiesterase 4 (PDE4) inhibitor.</p>Formule :C25H31NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.52iGP-5
CAS :<p>iGP-5 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>Formule :C21H17N3O3Couleur et forme :SolidMasse moléculaire :359.38Benanserin HCl
CAS :<p>Benanserin HCl is a serotonin antagonist. It causes psychotropic effects in humans.</p>Formule :C19H23ClN2OCouleur et forme :SolidMasse moléculaire :330.85K103 Hydrochloride
CAS :<p>K103 Hydrochloride, an inhibitor of peptidoglycan synthesis, targets the lipid II precursor.</p>Formule :C19H22Cl2N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.36Benzpiperylone
CAS :<p>Benzpiperylone is a synthetic anti-inflammatory drug. It also has anti-inflammatory activity.</p>Formule :C22H25N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.45SMP-028
CAS :<p>SMP-028 is a neutral cholesterol esterase (CEase) inhibitor(IC50 : 1.01 μM).</p>Formule :C23H26FN5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.55Noreximide
CAS :<p>Noreximide is an agent of sedative.</p>Formule :C9H9NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :163.17DBC
CAS :<p>DBC is a halogenated hydrocarbon, widely used in biochemical experiments and drug synthesis research.</p>Formule :C20H13NDegré de pureté :99.76%Couleur et forme :Needles From Ethanol 7H-Dibenzo(C G)Carbazole Is A Crystalline SolidMasse moléculaire :267.32Besigliptin Tosylate
CAS :<p>Besigliptin Tosylate, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Formule :C25H36FN5O5SCouleur et forme :SolidMasse moléculaire :537.65A 924
CAS :<p>A 924 is an amino acid derivative with antineoplastic activity.</p>Formule :C30H57N7O11Couleur et forme :SolidMasse moléculaire :691.81Renytoline
CAS :<p>Renytoline is a new anti-inflammatory of arthritis.</p>Formule :C21H16N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.37PF04471141 HCl
CAS :<p>PF-04471141 is an effective and selective inhibitor of the calcium-activated phosphodiesterase PDE1 (IC50 = 35 nM).</p>Formule :C16H24ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.83MDK-0738
CAS :<p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>Formule :C15H16O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :244.29Pparδ agonist 2
CAS :<p>Pparδ agonist 2 is an agonist of PPARδ.</p>Formule :C20H18F3N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :437.44AF267
CAS :<p>AF267 is a M1 muscarinic agonist that works by restoring cognitive impairments.</p>Formule :C10H18N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :214.33Safrazine Hydrochloride
CAS :<p>Safrazine Hydrochloride is a monoamine oxidase inhibitor (MOI) that is irreversible.</p>Formule :C11H17ClN2O2Couleur et forme :SolidMasse moléculaire :244.718ABT-418
CAS :<p>ABT-418, a nicotinic acetylcholine receptor (nAchR) agonist, is used potentially for the treatment of attention deficit disorder.</p>Formule :C9H14N2OCouleur et forme :SolidMasse moléculaire :166.22CM026
CAS :<p>CM026 inhibits ALDH1A1 selectively, binds to its aldehyde pocket uncompetitively.</p>Formule :C22H30N6O4Couleur et forme :SolidMasse moléculaire :442.51Nafenopin
CAS :<p>Nafenopin is a peroxisome proliferator, it is used to promote liver tumors and has been used as an antihyperlipoproteinemic agent.</p>Formule :C20H22O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.39Bucricaine
CAS :<p>Bucricaine is an anesthetic drug.</p>Formule :C17H22N2Couleur et forme :SolidMasse moléculaire :254.37Dehydro-ZINC39395747
CAS :Dehydro-ZINC39395747 enhances NO in cells and inhibits cytochrome b5 reductase 3 (IC50: 9.14μM, Kd: 1.11μM).Formule :C12H9N3O2S2Couleur et forme :SolidMasse moléculaire :291.35WES-1
CAS :<p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>Formule :C20H20N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.46Clinolamide
CAS :<p>Clinolamide is an antilipidemic agent.</p>Formule :C24H43NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.6Tritoqualine
CAS :<p>Tritoqualine is used as an inhibitor of histidine decarboxylase.</p>Formule :C26H32N2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.5417β-HSD10-IN-2
CAS :<p>17β-HSD10-IN-2 (compound 11), a benzothiazolylurea-based inhibitor, specifically targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), avoiding</p>Formule :C15H10ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.78BI-135585
CAS :<p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>Formule :C28H32N2O4Degré de pureté :99.45% - 99.57%Couleur et forme :SolidMasse moléculaire :460.576-Hydroxyluteolin
CAS :<p>6-Hydroxyluteolin, a flavonoid compound extracted from Salvia amarissima Ortega, inhibits aldose reductase (AR) and has antimicrobial activity.</p>Formule :C15H10O7Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :302.24MAGL-IN-1
CAS :<p>MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.</p>Formule :C22H24FNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.43ML404
CAS :<p>ML404 is the mitochondrial permeability transition pore inhibitor.</p>Formule :C17H13ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.75Tilivapram
CAS :<p>Tilivapram is a PDE4 (phosphodiesterase IV) inhibitor that can be used in the study of mental illness.</p>Formule :C16H15Cl2N3O4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :384.21FTX-6746
CAS :<p>FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.</p>Formule :C16H7ClF2N2ODegré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :316.69MR 16728 hydrochloride
CAS :<p>stimulates the release of acetylcholine from synaptosomes</p>Formule :C23H37ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.01Glycogen phosphorylase-IN-1
CAS :<p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>Formule :C17H15ClF2N4O4Degré de pureté :97.98% - 98.15%Couleur et forme :SolidMasse moléculaire :412.78Phytic acid dodecasodium salt hydrate
CAS :<p>Phytic acid salt hydrate: seed phosphorus compound, inhibits xanthine oxidase, IC50 6 mM, antioxidant, neuroprotective, anti-inflammatory.</p>Formule :C6H20NaO25P6Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :701.033AN3199
CAS :<p>AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.</p>Formule :C17H18BNO5Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :327.14ML387
CAS :<p>ML387 is an inhibitor of human NAD(+)- dependent 15- hydroxyprostaglandin dehydrogenase.</p>Formule :C20H21N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.4Manninotrionate
CAS :<p>Manninotrionate, an antitumor agent, linked to BSA; rabbit antiserum made, doesn't agglutinate Ehrlich tumor cells with alpha-D-galactosyl groups.</p>Formule :C18H32KO17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.535LYS006
CAS :<p>LYS006 is a highly efficient and selective LTA4H (leukotriene A4 hydrolase) inhibitor,for neutrophil-driven inflammatory diseases ulcerative colitis.</p>Formule :C16H14ClFN6O3Degré de pureté :99.33%Couleur et forme :SoildMasse moléculaire :392.77Pitstop1
CAS :<p>Clathrin-IN-1 selectively inhibits clathrin, potentially blocking virus entry and modulating cell signals.</p>Formule :C19H14N2NaO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.38LP8
CAS :<p>LP8 is a novel inhibitor of Trypanosoma cruzi CYP51.</p>Formule :C16H19N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.4KC-12615
CAS :<p>KC-12615 is an inhibitior of endopeptidase.</p>Formule :C29H34N2O6Couleur et forme :SolidMasse moléculaire :506.59hCAIX-IN-5
CAS :<p>hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.</p>Formule :C18H12FNO3Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :309.29Chlorisondamine diiodide
CAS :Chlorisondamine diiodide is a selective nAChR antagonist and ganglionic blocker that persistently antagonizes partial central effects of nicotine.Formule :C14H20Cl4I2N2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :611.94PKM2 activator 5
CAS :<p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>Formule :C18H19FN2O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.48Peliglitazar racemate
CAS :<p>Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity</p>Formule :C30H30N2O7Degré de pureté :97.75%Couleur et forme :SolidMasse moléculaire :530.57ACAT-IN-1 cis isomer
CAS :<p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>Formule :C29H25NO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :419.51Leucinal
CAS :<p>Leucinal inhibits the activity of brain aminopeptidase and potentiates analgesia induced by leu-enkephalen.</p>Formule :C6H13NOCouleur et forme :SolidMasse moléculaire :115.17BRD6897
CAS :BRD6897 is a mitochondrial content inducer that increases the cellular content of mitochondria.Formule :C25H21N3O2S2Degré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :459.58Texasin
CAS :<p>Texasin is a selective inhibitor of human leukocyte 5-lipoxygenase.</p>Formule :C16H12O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.26Lysine Orotate
CAS :<p>Lysine Orotate blocks Herpes virus replication, effective against HSV-1, HSV-2, CMV, EBV, and Varicella.</p>Formule :C11H18N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.28Thialysine HCl
CAS :<p>Thialysine HCl is a cytotoxic cysteine derivative that inhibits Escherichia coli, acting as a protein synthesis inhibitor and metabolite.</p>Formule :C5H13ClN2O2SCouleur et forme :SolidMasse moléculaire :200.69Benproperine
CAS :<p>Benproperine is a bioactive molecule with antineoplastic properties.</p>Formule :C21H27NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :309.45YM758 Phosphate
CAS :<p>YM758 Phosphate, a current channel inhibitor, selectively lowers a heart beat and decreases oxygen consumption of heart muscle.</p>Formule :C26H35FN3O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.54SQ-31765
CAS :<p>SQ-31765 is a blocker of benzazepine calcium channel.</p>Formule :C24H27F3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.48PG-9 maleate
CAS :<p>Increases release of acetylcholine</p>Formule :C21H26BrNO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.34STL1267
CAS :<p>STL1267 is a REV-ERB agonist that crosses the blood-brain barrier and inhibits BMAL1 gene expression.</p>Formule :C17H11ClN4ODegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :322.75CaV1.3 antagonist-1
CAS :<p>CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.</p>Formule :C17H19ClN2O3Couleur et forme :SolidMasse moléculaire :334.8Ipenoxazone
CAS :<p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>Formule :C22H34N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.52ARI-3531
CAS :<p>ARI-3531 is a selective prolyl endopeptidase inhibitor.</p>Formule :C15H22BN3O4Couleur et forme :SolidMasse moléculaire :319.16NC1153
CAS :<p>NC1153 blocks IL-2/JAK3/STAT5a/b, aids allograft survival, reduces toxicities.</p>Formule :C18H38Cl2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.42Risotilide
CAS :<p>Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.</p>Formule :C15H27N3O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.528-CSC
CAS :<p>8-CSC: hMAO-B inhibitor (Ki: 235 nM, baboon liver) & A2A receptor affinity (Ki: 36 nM, rat brain).</p>Formule :C16H15ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.77Camylofin Hydrochloride
CAS :<p>Camylofin HCl is an antispasmodic used in labor treatment and is also used to deliver drug therapy for ulcerative colinitis.</p>Formule :C19H33ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.94Ornithine-α-ketoglutarate
CAS :<p>Ornithine-α-ketoglutarate (L-Ornithine-α-ketoglutarate) is a salt formed of 2 molecules of ornithine and 1 alpha-ketoglutarate.</p>Formule :C10H18N2O7Degré de pureté :≥98%Couleur et forme :White PowderMasse moléculaire :278.26Letimide HCl
CAS :<p>Letimide HCl is an analgesic agent.</p>Formule :C14H19ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.77Oncrasin-72
CAS :Oncrasin-72 is an analog of oncrasin-1. It has antitumor activity mediated by JNK activation and STAT3 inhibition.Formule :C16H14ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :271.74sEH inhibitor-3
CAS :<p>sEH inhibitor-3 is an orally available, selective and potent inhibitor of sEH for cancer research.</p>Formule :C19H23F4N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.4Senazodan hydrochloride
CAS :<p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>Formule :C15H15ClN4ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :302.76(3S,5S)-Pitavastatin calcium
CAS :<p>(3S,5S)-Pitavastatin calcium is the 3-epimer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.</p>Formule :C25H26CaFNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.562EZ-482
CAS :<p>EZ-482 is an apolipoprotein (apoE) ligand used for Alzheimer's disease.</p>Formule :C23H19ClN4O5SDegré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :498.94Tenuazonic acid
CAS :<p>Tenuazonic acid, a nonhost-selective mycotoxin from Alternaria alternate, inhibits PSII by blocking electron transport at D1 protein.</p>Formule :C10H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :197.23Hydroxythiohomosildenafil
CAS :<p>Hydroxythiohomosildenafil, an analogue of sildenafil, is a phosphodiesterase-5 (PDE-5) inhibitor.</p>Formule :C23H32N6O4S2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :520.67(Z)-10-Hydroxynortriptyline
CAS :<p>(Z)-10-Hydroxynortriptyline ((Z)-10-Hydroxy Nortriptyline) is a norepinephrine reuptake inhibitor with antidepressant activity.</p>Formule :C19H21NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.38MRL-871
CAS :<p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>Formule :C22H12ClF3N2O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :444.79FABP4/5-IN-5
CAS :<p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>Formule :C23H14ClF2NO4SCouleur et forme :SolidMasse moléculaire :473.88Cholesteryl Palmitoleate
CAS :<p>Cholesteryl palmitoleate, a cholesterol ester, exhibits elevated plasma levels in ApoE-/- mice following exposure to cigarette smoke and in pediatric patients diagnosed with biliary atresia. It serves as a standard for identifying cholesterol esters in human meibomian gland secretions.</p>Formule :C43H74O2Couleur et forme :SolidMasse moléculaire :623.1Niraparib metabolite M1
CAS :<p>Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) is the carboxylic acid metabolite of niraparib.</p>Formule :C19H19N3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :321.37Tebuconazole-d9
CAS :<p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>Formule :C16H13ClD9N3OCouleur et forme :SolidMasse moléculaire :316.87IDO1-IN-2
CAS :<p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>Formule :C15H17FN6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.33SRPKIN-1
CAS :SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).Formule :C27H21FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.53MDPD
CAS :<p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>Formule :C21H19N3O3Couleur et forme :SolidMasse moléculaire :361.39AMPD2 inhibitor 2
<p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>Formule :C26H27F2N3O3Couleur et forme :SolidMasse moléculaire :467.51Propentofylline
CAS :<p>Propentofylline (Hextol) has neuroprotective, antiproliferative and anti-inflammatory activities and can be used in the study of Alzheimer's disease.</p>Formule :C15H22N4O3Degré de pureté :99.76% - 99.86%Couleur et forme :Off-White SolidMasse moléculaire :306.36N-(α-Linolenoyl) Tyrosine
CAS :<p>Certain chronic neurologic disorders, such as Parkinson's disease, are caused by an insufficiency of the neurotransmitter dopamine secondary to the degeneration</p>Formule :C27H39NO4Couleur et forme :SolidMasse moléculaire :441.6PF-04279405
CAS :<p>PF-04279405 is a potent and selective glucokinase activator.</p>Formule :C25H25FN4O4Couleur et forme :SolidMasse moléculaire :464.49YZ9
CAS :<p>Y29 is a potent PFKFB3 inhibitor with an IC50 of 0.183 µM, and acts as a competitive inhibitor against Fru-6-P with a Ki of 0.094 µM[1].</p>Formule :C12H10O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :234.2BI-L 357
CAS :<p>BI-L 357, a prodrug of BL-L 226, is a selective, orally active inhibitor of 5-lipoxygenase.</p>Formule :C18H18O4SCouleur et forme :SolidMasse moléculaire :330.4RO6806051
CAS :RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.Formule :C21H19ClN6Couleur et forme :SolidMasse moléculaire :390.87α-Glucosidase-IN-6
CAS :<p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>Formule :C24H17ClF3NO3SCouleur et forme :SolidMasse moléculaire :491.912-Hydroxy atorvastatin calcium salt
CAS :<p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>Formule :C33H34FN2O60·5CaDegré de pureté :97.06%Couleur et forme :SolidMasse moléculaire :593.6812(S)-HpETE
CAS :<p>12(S)-HpETE activates human blood leukocyte 5-LOE and mediates induction of c-fos and c-jun, activation of AP-1, and endothelium-dependent vasoconstriction.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47SHP2-IN-5
CAS :<p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>Formule :C12H8O6Couleur et forme :SolidMasse moléculaire :248.19JMS-053
CAS :<p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>Formule :C13H8N2O2SDegré de pureté :≥98.0%Couleur et forme :SolidMasse moléculaire :256.28CD 1530
CAS :<p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>Formule :C27H26O3Degré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :398.49trans-Ned 19
CAS :<p>trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.</p>Formule :C30H31FN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :514.59Teglarinad chloride
CAS :<p>Teglarinad chloride (GMX-1777 chloride) is an inhibitor of NAMPT with antitumor activity that acts by interfering with DNA repair and inhibiting angiogenesis.</p>Formule :C30H43Cl2N5O8Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :672.6Gcase activator 3
CAS :<p>Gcase activator 3 is a glucocerebrosidase (GCase) activator that enhances GBA1 mutant fibroblast lysosomal GCase activity.</p>Formule :C23H20N4O2Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :384.43LP-533401
CAS :<p>LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.</p>Formule :C27H22F4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :526.48PD0176078
CAS :PD0176078 () is a newly blocker of N-type Calcium channel.Formule :C23H30F2N2ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :388.49
