Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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BemPPOX
CAS :<p>BemPPOX is a potent inhibitor of DGL.</p>Formule :C23H20N2O5Couleur et forme :SolidMasse moléculaire :404.42BW-1370U87
CAS :BW-1370U87 is an MAO-A inhibitor increasing brain amines, showing promise in depression models.Formule :C14H12O3SDegré de pureté :99.82% - 99.89%Couleur et forme :SolidMasse moléculaire :260.31JNJ-40355003
CAS :<p>JNJ-40355003 is a FAAH inhibitor that increases plasma levels of fatty acid amides in rats, dogs, and crabs.</p>Formule :C23H23ClN4O2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :422.91Ladostigil
CAS :<p>Ladostigil is an oral cholinesterase & MAO-B inhibitor used for depression and Alzheimer's studies.</p>Formule :C16H20N2O2Degré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :272.34Lonapalene
CAS :<p>Lonapalene is a topically effective inhibitor of 5-lipoxygenase.</p>Formule :C16H15ClO6Degré de pureté :98.67% - 99.33%Couleur et forme :SolidMasse moléculaire :338.74KT203
CAS :<p>KT203 is an α/β hydrolase structural domain 6 (ABHD6) inhibitor with potential antiviral and anti-inflammatory activity for the study of pneumonia.</p>Formule :C28H26N4O3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :466.53A-69412
CAS :<p>A-69412 is a reversible 5-lipoxygenase inhibitor, potentially treating ulcerative colitis and asthma.</p>Formule :C7H10N2O3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :170.17SR2211
CAS :<p>SR2211 is a specific modulator and an inverse agonist of RORγ(IC50 = 320 nM, Ki = 105 nM).</p>Formule :C26H24F7N3ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :527.48Isomazole
CAS :<p>Isomazole is a novel orally available phosphodiesterase (PDE) inhibitor with calcium-sensitizing properties that inhibits PDE3 and PDE4.</p>Formule :C14H13N3O2SDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :287.34C75
CAS :<p>C75 is an inhibitor synthetic fatty-acid synthase (FASN) and inhibits prostate cancer cells PC3 (IC50: 35 μM).</p>Formule :C14H22O4Degré de pureté :98.84% - >99.99%Couleur et forme :SolidMasse moléculaire :254.32PDE IV-IN-1
CAS :PDE IV-IN-1 is a potent phosphodiesterase 4 (PDE4) inhibitor with anti-inflammatory activity for the treatment of asthma, chronic obstructive pulmonary diseaseFormule :C20H23ClN4O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :386.88IDH2R140Q-IN-2
CAS :IDH2R140Q-IN-2 is an IDH2R140Q inhibitor indicated for the study of acute myeloid leukaemia (AML).Formule :C21H18F6N6ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :484.4JNJ-DGAT2-A
CAS :<p>JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.</p>Formule :C24H16BrFN4O2SDegré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :523.3811-cis-Vaccenyl acetate
CAS :<p>11-cis-Vaccenyl acetate ((Z)-Octadec-11-enyl acetate) activates olfactory neurons located in the T1 sensilla on the antenna and mediates aggregation behavior in</p>Formule :C20H38O2Degré de pureté :96.53% - 99.95%Couleur et forme :LiquidMasse moléculaire :310.51PKUMDL-WQ-2101
CAS :<p>PKUMDL-WQ-2101 is a selective allosteric inhibitor of phosphoglycerate dehydrogenase with anti-tumor activity.</p>Formule :C14H11N3O6Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :317.25Edoxaban
CAS :<p>Edoxaban: potent, selective FXa inhibitor; Ki 0.561 nM. Used as an oral anticoagulant for stroke prevention, also inhibits thrombin and FIXa.</p>Formule :C24H30ClN7O4SDegré de pureté :97.67% - 99.71%Couleur et forme :SolidMasse moléculaire :548.06Olorofim
CAS :<p>Olorofim（F-901318）is a new selective antifungal compound that inhibits Aspergillus fumigatus DHODH (IC50: 44 nM). Cost-effective and quality-assured.</p>Formule :C28H27FN6O2Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :498.55Fidexaban
CAS :<p>Fidexaban (CI1031) is a novel, potent, selective and orally active factor Xa inhibitor that has demonstrated antithrombotic activity in a variety of assays</p>Formule :C25H24F2N6O5Degré de pureté :98.64% - 99.43%Couleur et forme :SolidMasse moléculaire :526.49Crobenetine
CAS :<p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>Formule :C25H33NO2Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :379.54Mopidamol
CAS :<p>Mopidamol (RA 233) is a phosphodiesterase inhibitor, a dipyridamole derivative, with anticancer activity that prevents retinal vascular defects in experimental</p>Formule :C19H31N7O4Degré de pureté :99.05% - 99.78%Couleur et forme :SolidMasse moléculaire :421.49Fluorobexarotene
CAS :<p>Fluorobexarotene, a potent RXR agonist, has 75% higher affinity than Bexarotene with Ki of 12 nM and EC50 of 43 nM for RXRα.</p>Formule :C24H27FO2Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :366.47AA 2379
CAS :<p>N6-Allyladenosine (N Allyladenosine) is a nucleoside analog with antimicrobial activity and anticancer activity.</p>Formule :C15H23N5O4Degré de pureté :97.78% - 98.87%Couleur et forme :SolidMasse moléculaire :337.37Autotaxin-IN-3
CAS :<p>Autotaxin-IN-3 is an inhibitor of Autotaxin (IC50 = 2.4 nM) which is responsible for the increase in lysophosphatidic acid in ascites and plasma.</p>Formule :C22H21N9O2Degré de pureté :99.54% - 99.79%Couleur et forme :SolidMasse moléculaire :443.46L-Threonine derivative-1
CAS :L-Threonine derivative-1 is acetylsalicylic acid-L-threonine ester with potential analgesic activity.Formule :C13H15NO6Degré de pureté :97.03% - 98.91%Couleur et forme :SolidMasse moléculaire :281.26K-111
CAS :<p>K-111 is a PPAR alpha agonist. K-111 improves insulin resistance, reducing bodyweight, and ameliorating atherogenic dyslipidemia.</p>Formule :C18H25Cl3O2Degré de pureté :99.64% - 99.88%Couleur et forme :SolidMasse moléculaire :379.75HSD-016
CAS :HSD-016: Oral 11β-HSD1 inhibitor, active in humans, mice, rats (IC50: 11, 1, 8 nM), potential for type 2 diabetes research.Formule :C21H21F7N2O3SDegré de pureté :99.40% - >99.99%Couleur et forme :SolidMasse moléculaire :514.46Tamolarizine
CAS :<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Formule :C27H32N2O3Degré de pureté :98.17%Couleur et forme :SoildMasse moléculaire :432.55SAK3
CAS :<p>SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.</p>Formule :C20H23N3O4Degré de pureté :98.37% - 99.43%Couleur et forme :SolidMasse moléculaire :369.41EMD-503982
CAS :<p>EMD-503982 is a potential Factor Xa and Factor VIIa inhibitor with anticancer activity for the study of thromboembolic and neurologic diseases.</p>Formule :C22H23ClN4O5Degré de pureté :97.09% - 99.81%Couleur et forme :SolidMasse moléculaire :458.90AC-261066
CAS :<p>AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.</p>Formule :C17H20FNO4SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :353.41Fumarate hydratase-IN-1
CAS :Fumarate hydratase-IN-1 is a cell-permeable fumarate hydratase inhibitor with antiproliferative activity and can be used to study cellular activity.Formule :C27H30N2O4Degré de pureté :98.96% - 99.49%Couleur et forme :SolidMasse moléculaire :446.54BRD7389
CAS :<p>BRD7389 is an inhibitor of RSK family kinase with IC50s of 1.5 μM, 2.4 μM, and 1.2 μM for RSK1, RSK2, and RSK3, respectively.</p>Formule :C24H18N2O2Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :366.41IMPDH2-IN-2
CAS :<p>IMPDH2-IN-2 is an IMPDH inhibitor with antimicrobial activity and potential anti-tuberculosis activity for the study of inflammation and immune dysfunction.</p>Formule :C21H15Cl2N3O3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :428.27ARRY-403
CAS :<p>ARRY-403 is a novel glucokinase activator that reduces fasting and postprandial blood glucose in patients with type 2 diabetes.</p>Formule :C20H18N6O3S2Degré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :454.52CYP1B1-IN-5
CAS :<p>CYP1B1-IN-5: selective CYP1B1 inhibitor, IC50 = 4.7 nM, useful for metabolism disease research.</p>Formule :C14H8INO2Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :349.12Nampt activator-2
CAS :<p>Nampt activator-2: Potent NAMPT activator (EC50: 0.023 μM), binds CYP2C9 (0.060 μM), 2D6 (0.41 μM), 2C19 (0.59 μM); useful in metabolic disease research.</p>Formule :C17H15ClN4O3SDegré de pureté :98.30% - 98.33%Couleur et forme :SolidMasse moléculaire :390.84NNC 05-2090 hydrochloride
CAS :<p>NNC 05-2090 HCl: BGT-1 inhibitor, IC50 = 10.6 μM, potential for epilepsy, neurological research.</p>Formule :C27H31ClN2O2Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :451IPN60090
CAS :<p>IPN60090: potent oral GLS1 inhibitor, IC50 of 31 nM, potential for anticancer and immunomodulation.</p>Formule :C24H27F3N8O3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :532.524-Hydroxymephenytoin
CAS :<p>4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.</p>Formule :C12H14N2O3Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :234.25Utreloxastat
CAS :<p>Utreloxastat (PTC857) is a novel 15-lipoxygenase inhibitor that can be used to study amyotrophic lateral sclerosis<br>.</p>Formule :C18H28O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :276.41CERM-11956
CAS :<p>Pelretin (BASF 43915) is a potential protein inhibitor for the study of dermatologic diseases.</p>Formule :C29H38N2O7Degré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :526.62Allopurinol riboside
CAS :<p>Allopurinol riboside, an allopurinol metabolite, inhibits purine nucleoside phosphorylase in parasites with a Ki of 277 μM.</p>Formule :C10H12N4O5Degré de pureté :99.46% - 99.73%Couleur et forme :SolidMasse moléculaire :268.235-ALA benzyl ester hydrochloride
CAS :<p>5-ALA benzyl ester hydrochloride: a photodetection agent that promotes PPIX in colon cancer cells.</p>Formule :C12H16ClNO3Degré de pureté :98.39% - 99.38%Couleur et forme :SolidMasse moléculaire :257.71AZ3976
CAS :<p>AZ3976 is an inhibitor of PAI-1 with an IC50 of 16 μM in a plasma clot lysis assay. AZ3976 displays profibrinolytic activities.</p>Formule :C15H19N5O3Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :317.34Carbonic anhydrase inhibitor 6
CAS :<p>Carbonic anhydrase inhibitor 6 is an hCA inhibitor that inhibits hCA IX, hCA II, hCA XII, and hCA I. It is used in the study of lupus erythematosus.</p>Formule :C26H25N3O5SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :491.56Cholesterol 24-hydroxylase-IN-1
CAS :<p>Cholesterol 24-hydroxylase-IN-1 is a cholesterol 24-hydroxylase (CH24H or CYP46A1) inhibitor used in the study of neurological disorders such as epilepsy.</p>Formule :C17H23N5ODegré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :313.40Bupicomide
CAS :<p>Bupicomide is a dopamine β-hydroxylase inhibitor with antihypertensive and vasodilatory activity and may be used in the study of hypertension.</p>Formule :C10H14N2ODegré de pureté :99.84% - >99.99%Couleur et forme :SolidMasse moléculaire :178.23Tigulixostat
CAS :<p>Tigulixostat (LC350189) is a novel xanthine oxidase inhibitor (XOI) that reduces uric acid production and may be used to study gout-related diseases.</p>Formule :C16H14N4O2Degré de pureté :98.22% - 99.71%Couleur et forme :SolidMasse moléculaire :294.31Dovramilast
CAS :<p>Dovramilast (CC-11050) is a PDE4 inhibitor that reduces the production of pro-inflammatory mediators in lupus erythematosus.</p>Formule :C24H28N2O6SDegré de pureté :98.75% - 99.62%Couleur et forme :SolidMasse moléculaire :472.55BMS-823778
CAS :<p>BMS-823778 is a potent inhibitor of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1) for the study of type 2 diabetes.</p>Formule :C18H18ClN3ODegré de pureté :99.39% - 99.75%Couleur et forme :SolidMasse moléculaire :327.81Indeglitazar
CAS :<p>Indeglitazar (PPM 204) is orally available pan-agonist of PPAR (PPAR subtypes alpha (α), delta (δ), and gamma (γ)).</p>Formule :C19H19NO6SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :389.42IHVR-17028
CAS :<p>IHVR-17028 is a potent broad-spectrum ERα-glucosidase I (α-glucosidase? I) inhibitor with IC50 of 0.24 μM and antiviral activity.</p>Formule :C23H44N2O5Degré de pureté :97.90%Couleur et forme :SolidMasse moléculaire :428.61MM 11253
CAS :<p>MM 11253 is a RARγ antagonist with IC50 of 44nM.</p>Formule :C28H30O2S2Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :462.67PC945
CAS :<p>PC945 (Opelconazole) is an antifungal compound that inhibits CYP51A/CYP51B and can be used to study fungal infections of the lungs.</p>Formule :C38H37F3N6O3Degré de pureté :98.89% - 99.37%Couleur et forme :SolidMasse moléculaire :682.73JJKK 048
CAS :<p>JJKK 048 is a potent and selective MAGL inhibitor.</p>Formule :C23H22N4O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :434.44Sultiame
CAS :<p>Sultiame is an inhibitor of carbonic anhydrase. Sultiame can be used in antiepileptic research.</p>Formule :C10H14N2O4S2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :290.365-LOX-IN-1
CAS :<p>5-LOX-IN-1 is a 5-Lipoxygenase (5-LOX) inhibitor (IC50: 2.3 μM).5-LOX-IN-1 can be used for cancer research.</p>Formule :C20H18N2O2SDegré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :350.43Giripladib
CAS :<p>Giripladib (PLA695/PLX-695) blocks radiation-boosted phosphorylation of ERK and Akt in endothelial cells.</p>Formule :C41H36ClF3N2O4SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :745.25sEH inhibitor-7
CAS :<p>sEH inhibitor-7 is a soluble epoxide hydrolase (sEH) inhibitor that inhibits sEH in human and mouse with IC 50 s of 6.2 μM and 0.15 μM, respectively.</p>Formule :C15H21NO2Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :247.33Xanthine oxidoreductase-IN-3
CAS :<p>Xanthine oxidoreductase-IN-3, an oral XOR inhibitor with IC50 of 26.3 nM, is useful for acute hyperuricemia research.</p>Formule :C14H10ClN5ODegré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :299.72S-2474
CAS :<p>S-2474, an inhibitor of COX-2 and 5-lipoxygenase, has anti-inflammatory and neuroprotective activities, and inhibits cell death.</p>Formule :C20H31NO3SDegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :365.53Troriluzole
CAS :<p>Troriluzole is a glutamate modulator with anticancer activity and is used in the study of spinocerebellar ataxia.</p>Formule :C15H16F3N5O4SDegré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :419.38Imanixil
CAS :<p>Imanixil boosts LDLR, cuts cholesterol and VLDL production, reducing atherosclerosis.</p>Formule :C17H17F3N6O2Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :394.35AMG-1694
CAS :<p>AMG-1694 disrupts GK-GKRP complex, enhancing GK activity with 7 nM IC50; normalizes glucose in diabetic rodents without affecting normoglycemic animals.</p>Formule :C23H30F3N3O4S2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :533.63Chloramphenicol succinate
CAS :<p>Chloramphenicol succinate is a bacteriostatic antibiotic. CPSA is a competitive substrate and inhibitor of succinate dehydrogenase (SDH),can be oxidized by.</p>Formule :C15H16Cl2N2O8Degré de pureté :95.32%Couleur et forme :Physical Description White Powder (Ntp 1992)Masse moléculaire :423.2Pradefovir
CAS :<p>Pradefovir (Remofovir) is a prodrug for chronic HBV, converting to PMEA in the liver with a Km of 60 μM and clearance of 359 ml/min.</p>Formule :C17H19ClN5O4PDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :423.79BPDA2
CAS :BPDA2 selectively inhibits SHP2 (IC50=92nM) over SHP1/1B (33.39/40.71μM), curbs RTKs, and hampers SHP2-driven breast cancer cell traits.Formule :C24H30O5Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :398.49MFI8
CAS :MFI8 is a compound that regulates mitochondrial fission and can be used to study aging.Formule :C16H18ClNODegré de pureté :99.08% - 99.78%Couleur et forme :SolidMasse moléculaire :275.77IGP-1
CAS :<p>iGP-1 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>Formule :C17H15N3O3Degré de pureté :99.12% - 99.15%Couleur et forme :SolidMasse moléculaire :309.32Cronidipine
CAS :<p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>Formule :C30H32ClN3O8Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :598.04hCAI/II-IN-6
CAS :<p>hCAI/II-IN-6 is a selective and orally active inhibitor of human carbonic anhydrase (CA).</p>Formule :C19H24N4O3SDegré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :388.48hCAII-IN-9
CAS :<p>hCAII-IN-9 inhibits hCA II/IX/XII with IC50s of 1.18, 0.17, 2.99 μM; not BBB permeable.</p>Formule :C15H16ClN3O5S2Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :417.89Dasantafil
CAS :Dasantafil (SCH446132) is a small molecule phosphodiesterase-5A (PDE5A) inhibitor used to treat genitourinary disorders and study erectile dysfunction.Formule :C22H28BrN5O5Degré de pureté :99.4% - 99.50%Couleur et forme :SolidMasse moléculaire :522.39Lifarizine
CAS :<p>Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.</p>Formule :C29H32N4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :436.59Tofimilast
CAS :<p>Tofimilast (CP-325366), a PDE4 inhibitor, is used potentially for the treatment of asthma and chronic obstructive pulmonary disease.</p>Formule :C18H21N5SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :339.46PKM2 activator 2
CAS :<p>PKM2 activator 2 is a pyruvate kinase M2 (PKM2) activator with an AC 50 value of 66 nM.PKM2 activator 2 has anti-tumor proliferative properties and attenuates</p>Formule :C20H18F2N2O4S2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :452.49G6PD activator AG1
CAS :<p>G6PD activator AG1 is a G6PD agonist that promotes G6PD oligomerization to a catalytically competent form.</p>Formule :C24H30N4S2Degré de pureté :98.38% - 99.51%Couleur et forme :SolidMasse moléculaire :438.65Diproteverine HCl
CAS :<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Formule :C26H36ClNO4Degré de pureté :98.55% - 99.84%Couleur et forme :SolidMasse moléculaire :462.02GSK205
CAS :GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.Formule :C24H25BrN4SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :481.45Opc 8490
CAS :<p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>Formule :C30H35N3O10Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :597.61Isolithocholic Acid
CAS :<p>Isolithocholic Acid, a bile acid isomer, forms through microbial metabolism of Lithocholic acid or its 3α-sulfate.</p>Formule :C24H40O3Degré de pureté :99.56% - 99.84%Couleur et forme :SolidMasse moléculaire :376.57PBRM
CAS :<p>PBRM (17β-HSD1-IN-2) is a selective covalent inhibitor of 17β-HSD1, used in breast cancer and endometriosis research.</p>Formule :C28H34BrNO2Degré de pureté :99.56% - 99.59%Couleur et forme :SolidMasse moléculaire :496.48Xanthine oxidoreductase-IN-5
CAS :<p>Xanthine oxidoreductase-IN-5: oral XOR inhibitor; IC50 55 nM; for acute hyperuricemia research.</p>Formule :C17H17N5O2Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :323.35CYP1B1-IN-1
CAS :<p>CYP1B1-IN-1 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with potential anticancer and antitumor activity for breast cancer research.</p>Formule :C19H11ClO2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :306.74MAO-B-IN-8
CAS :<p>MAO-B-IN-8 is a highly potent and reversible inhibitor of monoamine oxidase-B (MAO-B), which also exhibits inhibitory effects on the microglial production of</p>Formule :C18H16O6Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :328.32BMS 753
CAS :<p>BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).</p>Formule :C21H21NO4Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :351.4CYP4A11/CYP4F2-IN-1
CAS :<p>CYP4A11/CYP4F2-IN-1 is a cytochrome P450 (CYP) 4A11 and CYP4F2 inhibitor for the study of kidney disease and cardiovascular disease.</p>Formule :C15H15N3OSDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :285.36MM-433593
CAS :<p>MM-433593 is a selective fatty acid amide hydrolase (FAAH-1) inhibitor for the treatment of pain, inflammation, and other disorders.</p>Formule :C25H22ClN3O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :447.91KRH102140
CAS :<p>KRH102140 is a PHD2 activator that reduces angiogenesis by inhibiting HIF-1alpha, used in cardiovascular disease research.</p>Formule :C25H24FNODegré de pureté :98.31% - 99.61%Couleur et forme :SolidMasse moléculaire :373.46MK-0873
CAS :<p>MK-0873 is a novel and potent selective phosphodiesterase 4 (PDE4) inhibitor.</p>Formule :C25H18N4O3Degré de pureté :98.40%Couleur et forme :SolidMasse moléculaire :422.44JNJ-42226314
CAS :<p>JNJ-42226314 is a MAGL inhibitor with anti-injury effects and has shown efficacy in neuropathic pain and inflammatory pain models.</p>Formule :C26H24FN5O2SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :489.56MY10
CAS :<p>MY10, a potent and orally active inhibitor of the receptor protein tyrosine phosphatase (RPTPβ/ζ), effectively reduces binge-like ethanol consumption and</p>Formule :C15H10F6OS2Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :384.36Ulodesine
CAS :<p>Ulodesine (BCX4208), a PNP inhibitor, has an IC50 of 2.293 nM/L, potentially useful for hyperuricaemia research.</p>Formule :C12H16N4O3Degré de pureté :99.68%Couleur et forme :SoildMasse moléculaire :264.28Esuprone
CAS :<p>Esuprone (LU-43839) is a novel reversible and highly selective MAO-A inhibitor with anticonvulsant activity for the treatment of depression.</p>Formule :C13H14O5SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :282.31Clopimozide
CAS :<p>Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.</p>Formule :C28H28ClF2N3ODegré de pureté :98.19% - >99.99%Couleur et forme :SolidMasse moléculaire :495.99MLS000544460
CAS :<p>MLS000544460 is a highly selective and reversible Eya2 phosphatase inhibitor (Kd: 2.0 μM, IC50: 4 μM).MLS000544460 exhibits inhibitory effects on Eya2</p>Formule :C17H12FN3O2SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :341.36PF-04447943
CAS :<p>PF-04447943, a selective PDE9A inhibitor (IC50=12nM), may aid sickle cell anemia research with its anti-inflammatory properties.</p>Formule :C20H25N7O2Degré de pureté :99.36% - 99.59%Couleur et forme :SolidMasse moléculaire :395.46Rbin-2
CAS :Rbin-2: Potent, selective Midasin inhibitor; reversible, cell-permeable; halts eukaryotic ribosome assembly.Formule :C13H11BrN4SDegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :335.22Fenoverine
CAS :<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Formule :C26H25N3O3SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :459.56BAY-0069
CAS :<p>BAY-0069 is a potent and selective PPARγ transactivator that inhibits human PPARγ and murine PPARγ with IC50s of 6.3 nM and 24 nM, respectively.BAY-0069 can be</p>Formule :C22H16BrN3O4Degré de pureté :99.41%Couleur et forme :SoildMasse moléculaire :466.28Xanthine oxidoreductase-IN-4
CAS :<p>Xanthine oxidoreductase-IN-4: oral XOR inhibitor, IC50 of 29.3 nM, potential for hyperuricemia research.</p>Formule :C16H15N5O2Degré de pureté :98.25%Couleur et forme :SoildMasse moléculaire :309.32Tanimilast
CAS :<p>Tanimilast (CHF-6001) is a potent PDE4 inhibitor with IC50 of 0.026 nM, used topically for obstructive lung disease.</p>Formule :C30H30Cl2F2N2O8SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :687.54Tiapamil hydrochloride
CAS :<p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>Formule :C26H38ClNO8S2Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :592.16Phosphatase-IN-1
CAS :<p>Phosphatase-IN-1 is a phosphatidic acid phosphatase (Pah) inhibitor with antifungal activity for the study of rice blast and ruderalia.</p>Formule :C16H16Cl2FNO2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :344.21SBI-425
CAS :<p>SBI-425: orally available TNAP inhibitor, enhances cardiovascular health & survival, no bone impact.</p>Formule :C13H12ClN3O4SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :341.77alphaSYN-IN-NAB2
CAS :<p>alphaSYN-IN-NAB2: a NAB2 gene protein guarding neurons against alpha-SYN harm; aids endosomal transport, cell processes, and can study various diseases.</p>Formule :C23H20ClN3ODegré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :389.88Izonsteride
CAS :<p>Izonsteride (LY320236) is a selective and potent 5alpha reductase inhibitor with dual action on the type I and type II isoforms of the enzyme.Izonsteride is</p>Formule :C24H26N2OS2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :422.61HTS07545
CAS :<p>HTS07545, an SQOR inhibitor (IC50: 30nM), slows H2S breakdown, researched for heart failure.</p>Formule :C22H18N2O3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :358.39Zifaxaban
CAS :<p>Zifaxaban (TY-602) is an oral selective factor Xa inhibitor with an IC50 of 11.1 nM, highly specific over other serine proteases, used in thrombosis studies.</p>Formule :C20H16ClN3O4SDegré de pureté :97.46% - 99.82%Couleur et forme :SolidMasse moléculaire :429.88Acetyl-L-carnitine
CAS :<p>Acetyl-L-carnitine, an amino-acid supplement, crosses the blood-brain barrier to aid in neuroinflammation and Alzheimer's.</p>Formule :C9H17NO4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :203.24YM 511
CAS :<p>YM 511 is a specific non-steroidal aromatase inhibitor with IC50s of 0.4 and 0.12 nM, minimally affecting other steroids.</p>Formule :C16H12BrN5Degré de pureté :99.965%Couleur et forme :SolidMasse moléculaire :354.2ML 209
CAS :<p>ML-209 is an antagonist of retinoic acid receptor-related orphan receptor γt (RORγt; IC50= 1.1 μM in a reporter assay).1It inhibits RORγt-induced transcription</p>Formule :C25H31NO6Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :441.52Ch55
CAS :<p>Ch55, a potent HL60 cell differentiator (EC50=200nM), binds well to RAR-α/β, useful for cancer research.</p>Formule :C24H28O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :364.48NecroX-5
CAS :<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Formule :C27H39N3O9S3Degré de pureté :99.944%Couleur et forme :SolidMasse moléculaire :645.81Aleplasinin
CAS :<p>Aleplasinin (PAZ 417) is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic</p>Formule :C28H27NO3Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :425.52NAAD sodium salt
CAS :<p>NAAD sodium salt (NAAD Na salt) is a substrate of nicotinamide adenine dinucleotide synthase and can be used in studies about the specificity and kinetics of</p>Formule :C21H25N6NaO15P2Degré de pureté :98.6% - 99.87%Couleur et forme :SolidMasse moléculaire :686.4LY 517717
CAS :<p>LY 517717 is an orally active inhibitor of coagulation factor Xa with antithrombotic activity for the study of venous thromboembolism (VTE).</p>Formule :C27H33N5O2Degré de pureté :99.77% - 99.88%Couleur et forme :SolidMasse moléculaire :459.58Carbazeran
CAS :<p>Carbazeran (UK-31,557) is an inhibitor of PDE2 and PDE3 and can be used for studies about metabolic diseases.</p>Formule :C18H24N4O4Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :360.41DS16570511
CAS :<p>DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.</p>Formule :C30H25Cl2N3O4Degré de pureté :98.34% - 98.45%Couleur et forme :SolidMasse moléculaire :562.44Orellanine
CAS :<p>Orellanine, from Cortinarius orellanus, is nephrotoxic and hinders macromolecule synthesis in kidney cells and liver mitochondria.</p>Formule :C10H8N2O6Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :252.18Vatanidipine
CAS :<p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>Formule :C41H42N4O6Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :686.8KT182
CAS :<p>KT182 is a selective and potent inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells.</p>Formule :C27H26N4O2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :438.52uk-50001
CAS :<p>UK-50001 is a PDE4 inhibitor for treating inflammation, allergies, respiratory issues, and wounds.</p>Formule :C26H24F3N3O4Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :499.48UCM05
CAS :<p>UCM05 is a potent FASN and FtsZ inhibitor active against HER2+ breast cancer and B. subtilis (MIC 100 μM), but not E. coli.</p>Formule :C24H16O10Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :464.38KLH45
CAS :<p>KLH45 is an effective and selective inhibitor of Spastic Paraplegia-Related Triglyceride Hydrolase DDHD2(IC50 = 1.3 nM).</p>Formule :C24H25F3N4O2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :458.48Qc1
CAS :<p>Qc1 is an inhibitor of threonine dehydrogenase (TDH) inhibitor and can be used in studies about metabolic diseases.</p>Formule :C23H16F3N3O2SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :455.45Filaminast
CAS :<p>Filaminast (UNII-CDD69JC61J) is an analog of a phosphodiesterase 4 inhibitor (PDE4 inhibitor) and roliplam, which is used as an anti-asthma drug.</p>Formule :C15H20N2O4Degré de pureté :98.53% - 98.93%Couleur et forme :SolidMasse moléculaire :292.33Farglitazar
CAS :<p>Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer used in the study of diabetes.</p>Formule :C34H30N2O5Degré de pureté :99.4% - 99.52%Couleur et forme :SolidMasse moléculaire :546.61Dalvastatin
CAS :<p>Dalvastatin (RG-12561) is an orally available inhibitor of HMG-CoA reductase and cholesterol-lowering synthesis.Dalvastatin competitively inhibits rat hepatic</p>Formule :C24H31FO3Degré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :386.5AM 374
CAS :<p>AM 374 (HDSF), a fatty acid amide hydrolase (FAAH) inhibitor, demonstrates the capacity to inhibit amidase activity, boasting an IC50 value of 13 nM.</p>Formule :C16H33FO2SDegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :308.5Lidorestat
CAS :<p>Lidorestat (IDD-676) is an aldose reductase inhibitor (IC50: 5 nM) with effective, selective and oral activity.</p>Formule :C18H11F3N2O2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :376.35AGN 196996
CAS :<p>AGN 196996: strong RARα inhibitor (Ki: 2 nM), weak for RARβ/γ (Ki: 1087/8523 nM).</p>Formule :C24H20BrNO5Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :482.32CM037
CAS :<p>CM037 (A-37) is a selective ALDH1A1 (acetaldehyde dehydrogenase 1A1) inhibitor (IC50; 4.6 µM) with antitumor activity and may be used in studies to eliminate</p>Formule :C21H25N3O3S2Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :431.57CYP1B1-IN-4
CAS :<p>CYP1B1-IN-4: 2,4-diarylthiazole, selective CYP1B1 inhibitor (IC50=0.2 nM), low cytotoxicity, stable in liver microsomes.</p>Formule :C18H14N2O2SDegré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :322.38Atibeprone
CAS :Atibeprone is a MAO-B inhibitor with antidepressant activity for the study of Parkinson's disease.Formule :C17H18N2O3SDegré de pureté :99.18% - 99.86%Couleur et forme :SolidMasse moléculaire :330.4PHGDH-IN-3
CAS :<p>PHGDH-IN-3, an oral PHGDH blocker with 2.8 μM IC50, may help in cancer research.</p>Formule :C24H18FN3O4S2Degré de pureté :97.24% - 98.55%Couleur et forme :SolidMasse moléculaire :495.55EWP 815
CAS :<p>EWP 815, a disulfiram analog, inhibits Ins(1,4)P2, Ins(1,4,5)P3 phosphatases, and dopamine β-hydroxylase.</p>Formule :C12H22N4S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.59AChE/BChE/MAO-B-IN-1
CAS :<p>AChE/BChE/MAO-B-IN-1 is a reversible, non-time-dependent inhibitor of AChE, BChE and MAO-B that crosses the blood-brain barrier and exhibits inhibitory effects</p>Formule :C20H24N2O2Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :324.42PTP1B-IN-3
CAS :PTP1B-IN-3 是一种具有有选择性和高效性的 PTP1B 抑制剂，具有抗癌活性，抑制 PTP1B 和 TCPTP 。PTP1B-IN-3 可用于研究糖尿病。Formule :C12H7BrF2NO3PDegré de pureté :99.31% - 99.97%Couleur et forme :SolidMasse moléculaire :362.06SERCA2a activator 1
CAS :<p>SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.</p>Formule :C32H29N3O4SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :551.66AZD-0284
CAS :<p>AZD-0284 is an inverse agonist of the nuclear receptor RORγ. In development for the treatment of plaque psoriasis vulgaris and respiratory tract disorders[1].</p>Formule :C21H18F6N2O5SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :524.43RPR107393 free base
CAS :<p>NVP-BAG956 (BAG956) is a PI3K/PDK inhibitor that inhibits PI3Kδ, and can be used to study melanoma.</p>Formule :C22H22N2ODegré de pureté :99.13% - 99.57%Couleur et forme :SolidMasse moléculaire :330.42PKUMDL-LC-101-D04
CAS :<p>PKUMDL-LC-101-D04 enhances GPX4, curbs iron death, boosts enzyme activity 150% at 20 μM, effective in wild-type MEF, reduces lipid peroxide toxicity.</p>Formule :C14H23ClN4O2S2Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :378.94VU0155069
CAS :<p>VU0155069, a selective PLD1 inhibitor (IC50: 46 nM), halts cancer cell migration in transwell assays.</p>Formule :C26H27ClN4O2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :462.97BAY-4931
CAS :<p>BAY-4931 is a powerful, covalent, and selective inverse-agonist of PPARγ, exhibiting an IC50 value of 0.17 nM.</p>Formule :C22H16ClN3O4Degré de pureté :99.47%Couleur et forme :SoildMasse moléculaire :421.83Nanterinone
CAS :<p>Nanterinone: oral phosphodiesterase inhibitor, improves acute heart failure hemodynamics.</p>Formule :C15H15N3ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :253.3CX-157
CAS :CX-157 (KP 157) is a novel monoamine oxidase-A (MAO-A) inhibitor for the study of depression-like neurological disorders and cancer.Formule :C14H8F4O4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :348.27S19-1035
<p>S19-1035: potent AKR1C3 inhibitor with 3.04 nM IC50, useful for tumor research.</p>Formule :C19H17ClN2O3Degré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :356.80Luciferase-IN-1
CAS :<p>Luciferase-IN-1 is a luciferase inhibitor that can be used to study bacterial and fungal infections.</p>Formule :C15H14N2SDegré de pureté :97.84%Couleur et forme :SolidMasse moléculaire :254.35Verofylline
CAS :<p>Verofylline (Verofyllinum) is an orally available, long-acting, multiacting, methylxanthine-substituted bronchodilator with inhibitory effects on PDE4 for the</p>Formule :C12H18N4O2Degré de pureté :98.33% - 98.83%Couleur et forme :SolidMasse moléculaire :250.3ALDH1A3-IN-2
CAS :<p>ALDH1A3-IN-2 is a potent ALDH1A3 inhibitor with an IC50 of 0.30 μM.ALDH1A3-IN-2 has potential for cancer disease research.</p>Formule :C13H17NODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :203.28GAC0003A4
CAS :<p>GAC0003A4 is an LXR inverse agonist with antitumor activity for the study of advanced pancreatic cancer and other recalcitrant malignancies.</p>Formule :C20H24N2O3Degré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :340.42Didesethyl chloroquine
CAS :<p>Didesethyl chloroquine, a chloroquine metabolite, is an effective myocardial inhibitor and antimalarial.</p>Formule :C14H18ClN3Degré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :263.77DSM421
CAS :DSM421 (DSM-421) is a dihydrodehydrogenase inhibitor (DHODH) that is in preclinical development as a potential treatment option for malaria and has shownFormule :C14H11F5N6Degré de pureté :99.67% - 99.82%Couleur et forme :SolidMasse moléculaire :358.27Lecimibide
CAS :Lecimibide (DuP 128) is a potent and selective inhibitor of acyl coenzyme A: cholesterol acyltransferase (ACAT), which can be used to study diseases due to highFormule :C34H40F2N4OSDegré de pureté :98.1% - 99.54%Couleur et forme :SolidMasse moléculaire :590.77Lifibrol
CAS :<p>Lifibrol (U-83860) is an inhibitor of cholesterol synthesis.Lifibrol has anticholesterol and hypolipidemic properties and promotes the conversion of LDL Apo B-</p>Formule :C21H26O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :342.43PDE4B-IN-2
CAS :<p>PDE4B-IN-2 (A 33), an oral PDE4B inhibitor, IC50: 15 nM; less potent on PDE4D (IC50: 1.7 µM), has anti-inflammatory properties.</p>Formule :C19H18ClN3O2SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :387.88AICAR monophosphate
CAS :<p>AICAR monophosphate (Aica ribonucleotide) is a purine precursor with antineoplastic activity and can be used in studies about type 2 diabetes.</p>Formule :C9H15N4O8PDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :338.21PD173212
CAS :<p>PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).</p>Formule :C38H53N3O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :599.85IQB-782
CAS :<p>IQB-782 is a mucolytic agent with mucolytic expectorant activity for the study of obstructive lung disease.</p>Formule :C4H9N3O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :163.2Ibiglustat (L-Malic acid)
CAS :<p>Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.</p>Formule :C24H30FN3O7SDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :523.57NCGC 607
CAS :<p>NCGC 607 is a a noninhibitory chaperone of glucocerebrosidase (GCase).</p>Formule :C24H22IN3O4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :543.35AWD 12-281
CAS :<p>AWD 12-281 is a PDE4 inhibitor with anti-inflammatory activity and bronchodilator activity for the study of chronic obstructive pulmonary disease (COPD).</p>Formule :C22H14Cl2FN3O3Degré de pureté :99.25% - 99.85%Couleur et forme :SolidMasse moléculaire :458.27Salnacedin
CAS :<p>Salnacedin (G-201) treats immune, skin, and musculoskeletal issues, suitable for acne, dermatitis, and psoriasis research.</p>Formule :C12H13NO5SDegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :283.3Clozic
CAS :Clozic (ICI 55897) exhibits reversible anti-proliferative effects and can be used in studies about serving as a potential anti-arthritic agent.Formule :C17H17ClO3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :304.77Malic enzyme inhibitor ME1
CAS :Malic enzyme inhibitor ME1 (ME1) is a specific inhibitor of Malic enzyme (IC50 = 0.15 μM). Malic enzyme inhibitor ME1 reduces cell viability/metabolic activity.Formule :C20H21N3O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :351.4Lauroyl lysine
CAS :<p>Lauroyl lysine (N6-Lauroyl-L-lysine) functions as skin and hair conditioning agents and as surfactants-cleansing agents in personal care products.</p>Formule :C18H36N2O3Degré de pureté :99.18%Couleur et forme :White To Off-White Solid With Characteristic Faint OdorMasse moléculaire :328.49Imigliptin
CAS :<p>Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.</p>Formule :C21H24N6ODegré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :376.46NG-497
CAS :<p>NG-497, a selective inhibitor of human ATGL, blocks lipolysis in adipocytes and aids cancer research.</p>Formule :C18H21NO4Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :315.36Libenzapril
CAS :<p>Libenzapril (CGS 16617) is a potent angiotensin-converting enzyme inhibitor used to study myocardial injury.</p>Formule :C18H25N3O5Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :363.41LDL-IN-3
CAS :<p>LDL-IN-3 shows anti-atherosclerotic and antioxidant activities.</p>Formule :C24H36O3SiDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :400.63Dirlotapide
CAS :Dirlotapide (CP742033), an intestinal MTP inhibitor, cuts weight in diabetic dogs by lowering food intake and raising peptide YY.Formule :C40H33F3N4O3Degré de pureté :98.47% - 99.62%Couleur et forme :SolidMasse moléculaire :674.71TDO-IN-1
CAS :<p>TDO-IN-1 is a tryptophan 2,3-dioxygenase (TDO) inhibitor with antitumor activity that acts by reversing local immune tolerance in tumor tissues.</p>Formule :C16H13F3N4O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :350.3OSMI-4
CAS :<p>OSMI-4 is a low nanomolar O-GlcNAc transferase (OGT) inhibitor that can be used to study OGT inhibition in different human cell lines.Cost-effective and quality-assured.</p>Formule :C27H26ClN3O7S2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :604.09FASN-IN-1
CAS :<p>FASN-in-1 is an effective, specific inhibitor of fatty acid synthase (FASN), a compound specifically designed to target and inhibit the activity of the enzyme</p>Formule :C18H25N3O3S2Degré de pureté :99.92% - >99.99%Couleur et forme :SolidMasse moléculaire :395.54sPLA2 inhibitor 1
CAS :<p>KH064 is a sPLA2-IIA inhibitor of oral activity.</p>Formule :C31H37NO4Couleur et forme :SolidMasse moléculaire :487.63MK-0736
CAS :<p>MK-0736 is a potent and selective 11β-HSD-1 inhibitor.</p>Formule :C23H30F3N3O2SCouleur et forme :SolidMasse moléculaire :469.56BMS-986318
CAS :<p>BMS-986318: potent FXR agonist, EC50=53/350 nM, good ADME, effective in liver disease models, for nonalcoholic steatohepatitis research.</p>Formule :C30H23Cl2F3N4O3Couleur et forme :SolidMasse moléculaire :615.43M5N36
CAS :<p>M5N36: selective Cdc25C inhibitor, IC50: 0.15µM A, 0.19µM B, 0.06µM C; halts cell growth, boosts p-CDK1/2.</p>Formule :C20H16ClN5O3Couleur et forme :SolidMasse moléculaire :409.83HIF-2α-IN-6
CAS :<p>HIF-2α-IN-6 (117) is a HIF-2α inhibitor [1].</p>Formule :C15H13F4NO3SCouleur et forme :SolidMasse moléculaire :363.33Pactimibe sulfate
CAS :<p>Pactimibe sulfate is a dual ACAT1/2 inhibitor with anti-atherogenic potential, reducing plasma cholesterol.</p>Formule :C50H82N4O10SCouleur et forme :SolidMasse moléculaire :931.28LNP Lipid-8
CAS :<p>LNP Lipid-8 (11-A-M), an ionizable lipid, is utilized in lipid nanoparticles (LNP) for siRNA delivery to T cells without ligand targeting. When loaded with GFP siRNA (siGFP), it significantly silences the GFP gene in a mouse model [1].</p>Formule :C42H71NO7Couleur et forme :SolidMasse moléculaire :702.02DHODH-IN-22
CAS :<p>DHODH-IN-22: potent, selective DHODH inhibitor, orally active, IC50: 0.3 nM, for AML research.</p>Formule :C21H21ClF4N6O5Couleur et forme :SolidMasse moléculaire :548.88Mutant IDH1-IN-4
CAS :<p>Mutant IDH1-IN-4 is an mutant Isocitrate dehydrogenase 1 (IDH 1) inhibitor.</p>Formule :C25H34N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.56VT-1598 tosylate
CAS :<p>VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.</p>Formule :C38H28F4N6O5SCouleur et forme :SolidMasse moléculaire :756.72A 78773
CAS :<p>A 78773: potent reversible 5-lipoxygenase inhibitor; active in cells/tissues; targets inflammation, asthma, IBD.</p>Formule :C15H13FN2O4Couleur et forme :SolidMasse moléculaire :304.27sEH/AChE-IN-4
CAS :<p>sEH/AChE-IN-4-15 is a dual sEH and AChE inhibitor crossing the BBB, with IC50s: 3.1 nM (hsEH), 1660 nM (hAChE), 179 nM (hBChE), 14.5 nM (msEH), 102 nM (mAChE).</p>Formule :C35H39ClF3N5O3Couleur et forme :SolidMasse moléculaire :670.16(S,R)-WT IDH1 Inhibitor 2
CAS :<p>(S,R)-WT IDH1 Inhibitor 2: selectively targets mutant IDH1; IC50 - R132G: 2.9 nM, R132C: 3.8 nM, R132H: 4.6 nM, WT: 46 nM; potential for AML treatment.</p>Formule :C28H28FN5O3Couleur et forme :SolidMasse moléculaire :501.55RORγt inverse agonist 26
CAS :<p>RORγt inverse agonist 26, a potent reverse agonist of RORγt, effectively modulates Th17 cell differentiation and suppresses IL-17 production.</p>Formule :C27H21F7N2O5SCouleur et forme :SolidMasse moléculaire :618.52PTP1B-IN-20
PTP1B-IN-20: Selective PTP1B inhibitor, IC50=1.05μM; less effective on TCPTP (IC50=78μM), targets type 2 diabetes.Formule :C26H28O15Couleur et forme :SolidMasse moléculaire :580.499-SAHSA
CAS :<p>Branched fatty acid esters of hydroxy fatty acids (FAHFAs) are lipids that are modulated by dietary changes such as fasting and high-fat diets, and they play a role in insulin sensitivity. These compounds generally consist of a fatty acid chain of either 16 or 18 carbons (for example, palmitoleic, palmitic, oleic, or stearic acid) esterified to a similarly long hydroxy fatty acid. One specific FAHFA, 9-SAHSA, features stearic acid esterified at the 9th carbon of hydroxy stearic acid. The concentration of 9-SAHSA is notably increased in the serum of glucose-tolerant AG4OX mice, which specifically express the Glut4 glucose-transporting protein in adipose tissue.</p>Formule :C36H70O4Couleur et forme :SolidMasse moléculaire :566.9H2-003
CAS :<p>H2-003 is a selective inhibitor of diacylglycerol acyltransferase 2 (DGAT2).</p>Formule :C25H26N4O4Couleur et forme :SolidMasse moléculaire :446.5BMS-795311
CAS :<p>Potent CETP inhibitor, boosts HDL-C levels, orally active; IC50=4nM.</p>Formule :C33H23F10NO3Couleur et forme :SolidMasse moléculaire :671.52Mitochondria degrader-1
CAS :<p>Mitochondria degrader-1, a potent autophagy inducer, aids in neurodegenerative, cancer, and aging disease research.</p>Formule :C33H49ClFN7O8SCouleur et forme :SolidMasse moléculaire :758.3Benzoic acid lithium
CAS :<p>Lithium benzoate, an aromatic alcohol present in numerous plants, commonly serves as an additive in food, beverages, cosmetics, and various other products. This compound exhibits antibacterial and antifungal properties, functioning effectively as a preservative [1].</p>Formule :C7H5LiO2Couleur et forme :SolidMasse moléculaire :128.06GPX4-IN-2
CAS :<p>GPX4-IN-2 is a potent inhibitor of GPX4, exhibiting antiproliferative activity. It holds potential for cancer research applications.</p>Formule :C30H40N2OCouleur et forme :SolidMasse moléculaire :444.65NUCC-0223619
CAS :<p>NUCC-0223619 is an IDO1 inhibitor that induces the degradation of IDO protein and can be involved in the synthesis of PROTAC.</p>Formule :C24H24ClFN2O2Couleur et forme :SolidMasse moléculaire :426.91ATX inhibitor 15
CAS :<p>ATX inhibitor 15, an indole-based carbamate, has a 2.17 nM IC50 against ATX, suppresses pro-fibrotic genes, and protects against mouse lung fibrosis.</p>Formule :C27H32ClN5O4SCouleur et forme :SolidMasse moléculaire :558.095α-Androst-16-en-3-one
CAS :<p>5α-Androst-16-en-3-one, a mammalian pheromone present in boar saliva, plays a crucial role in facilitating social and sexual interactions by acting as a volatile chemical cue. It is utilized to prime sows in estrus for mating or artificial insemination, underscoring its significance in reproductive behavior. Additionally, this compound is detected in human sweat and urine, where it is involved in studies concerning receptor-mediated odorant detection and the genetic foundations of anosmias, thereby broadening its scope of relevance beyond the animal kingdom.</p>Formule :C19H28OCouleur et forme :SolidMasse moléculaire :272.432Clocortolone pivalate
CAS :<p>Clocortolone pivalate, a synthetic steroid, treats dermatitis and psoriasis.</p>Formule :C27H36ClFO5Couleur et forme :SolidMasse moléculaire :495.02
