Métabolisme

Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.

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MJ33-OH lithium
CAS :
- 1135306-36-3
MJ33-OH lithium is a metabolite of MJ33.
Formule :C₂₂H₄₃F₃LiO₇P
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :514.48
Ref: TM-T12053
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Monoisobutyl phthalic acid
CAS :
- 30833-53-5
Monoisobutyl phthalic acid is a metabolite of phthalate that is in human semen and in meconium.
Formule :C₁₂H₁₄O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :222.24
Ref: TM-T13778
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PTP1B-IN-13
CAS :
- 650621-20-8
PTP1B-IN-13 inhibits PTP1B at an allosteric site with 1.59 μM IC50.
Formule :C₂₄H₂₅N₃O₃S₂
Couleur et forme :Solid
Masse moléculaire :467.6
Ref: TM-T40745
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3α,7α-Dihydroxycoprostanic acid
CAS :
- 17974-66-2
3α,7α-Dihydroxycoprostanic acid, an endogenous metabolite and bile acid, serves as the precursor to chenodeoxycholic acid [1].
Formule :C₂₇H₄₆O₄
Masse moléculaire :434.65
Ref: TM-TN7609
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5(S)-HPETE
CAS :
- 71774-08-8
5(S)-HpETE is a PUFA made by 5-LO from arachidonic acid, metabolized into LTA4, a key leukotriene precursor.
Formule :C₂₀H₃₂O₄
Couleur et forme :Solid
Masse moléculaire :336.472
Ref: TM-T40826
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α-Glucosidase-IN-39
α-Glucosidase-IN-39 is a potent α-glucosidase enzyme inhibitor, exhibiting an IC50 value of 869.06 ppm. It is applicable for use in antidiabetic studies [1].
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T80711
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Validamine
CAS :
- 32780-32-8
Validamine is a natural pseudo-aminosugar.
Formule :C₇H₁₅NO₄
Degré de pureté :98%
Couleur et forme :White Powder
Masse moléculaire :177.2
Ref: TM-T7731
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(Z)-7-Dodecen-1-ol
CAS :
- 20056-92-2
(Z)-7-Dodecen-1-ol counteracts the attractive properties of Z-7-dodecen-1-yl acetate.
Formule :C₁₂H₂₄O
Masse moléculaire :184.32
Ref: TM-TN7982
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N,N'-Diacetyl-L-cystine
CAS :
- 5545-17-5
DiNAC is a disulphide dimer with immune-modulating effects and reduces atherosclerosis in WHHL rabbits; also modulates rodent sensitivity reactions.
Formule :C₁₀H₁₆N₂O₆S₂
Degré de pureté :98.76%
Couleur et forme :White Powder
Masse moléculaire :324.37
Ref: TM-T16240
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Plipastatin A1
CAS :
- 103651-09-8
Plipastatin A1, a lipopeptide isolated from B.
Formule :C₇₂H₁₁₀N₁₂O₂₀
Couleur et forme :Solid
Masse moléculaire :1463.71
Ref: TM-T83864
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11(R)-HETE
CAS :
- 73347-43-0
11(R)-HETE aids in oocyte maturation in sea urchins and tentacle regeneration in hydras; it is also made by aspirin-influenced COX-2 and arachidonic acid.
Formule :C₂₀H₃₂O₃
Couleur et forme :Solid
Masse moléculaire :320.473
Ref: TM-T37490
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KT-362 free base
CAS :
- 93392-97-3
KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.
Formule :C₂₂H₂₈N₂O₃S
Degré de pureté :99.76%
Couleur et forme :Soild
Masse moléculaire :400.53
Ref: TM-T73587
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Atagabalin HCl
CAS :
- 223445-67-8
Atagabalin HCl is a novel voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) ligand that affects slow-wave sleep and can be used to treat insomnia.
Formule :C₁₀H₂₀ClNO₂
Degré de pureté :99.96% - ≥98%
Couleur et forme :Soild
Masse moléculaire :221.72
Ref: TM-T30188L
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DSPE-PEG5000-APRPG
DSPE-PEG5000-APRPG is a PEG compound composed of DSPE and the APRPG peptide, utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01195
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Previridicatumtoxin
CAS :
- 1379585-81-5
Previridicatumtoxin, found in P. aethiopicum, fights MRSA, VRE, C. albicans, S. cerevisiae, and kills NCI H460, KB-3-1, SW620 cancer cells.
Formule :C₃₀H₃₃NO₁₀
Couleur et forme :Solid
Masse moléculaire :567.58
Ref: TM-T37006
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Clocortolone
CAS :
- 4828-27-7
Clocortolone, a medium-strength corticosteroid, treats dermatitis as a cream ester called clocortolone pivalate.
Formule :C₂₂H₂₈ClFO₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :410.91
Ref: TM-T21374
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PNGase F
CAS :
- 83534-39-8
PNGase F is an endoglycosidase and amide hydrolase that catalyses the cleavage of internal glycosidic bonds in oligosaccharides.
Couleur et forme :Solid
Ref: TM-T76153
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SPL-334
CAS :
- 688347-51-5
SPL-334 is an inhibitor of S-nitrosoglutathione reductase.
Formule :C₂₂H₁₅N₃O₃S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :433.50
Ref: TM-T28837
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Bicyclic UK18
CAS :
- 1393680-45-9
Bicyclic UK18 is a competitive inhibitor of human urokinase-type plasminogen activator (uPA) with a Ki value of 53 nM.
Formule :C₇₇H₁₁₈N₂₆O₂₅S₃
Couleur et forme :Solid
Masse moléculaire :1904.11
Ref: TM-TP3037
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LOX-IN-5
CAS :
- 2125665-47-4
LOX-IN-5 (compound 22) is a non-selective LOX inhibitor.
Formule :C₂₁H₂₅FN₄O₂S
Couleur et forme :Solid
Masse moléculaire :416.51
Ref: TM-T203241
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Leucine dehydrogenase
CAS :
- 9082-71-7
Leucine dehydrogenase from Bacillus spheroides oxidizes/reduces branched-chain amino acids and their keto analogs.
Couleur et forme :Solid
Ref: TM-T76108
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PDK-IN-2
PDK-IN-2 (Compound 1F), with an IC50 of 68 nM, is a potent PDK inhibitor that downregulates the expression of PDK1 and PDK4 in cells.
Formule :C₁₇H₂₃AsCl₂N₂O₂S₂
Couleur et forme :Solid
Masse moléculaire :497.33
Ref: TM-T79723
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DSPE-PEG-Maleimide (MW 3400) ammonium
DSPE-PEG-Maleimide (MW 3400) ammonium combines DSPE phospholipids with maleimide for the preparation of nanostructured lipid carriers. It is applicable in drug delivery research.
Couleur et forme :Odour Solid
Ref: TM-TCL-01067
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Lumisterol
CAS :
- 474-69-1
Lumisterol, a steroid, is anti-UVB and inhibits cell growth; it's a (9β,10α)-stereoisomer of Ergosterol.
Formule :C₂₈H₄₄O
Couleur et forme :Solid
Masse moléculaire :396.659
Ref: TM-T38036
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TSPO/Carbonic Anhydrase Modulator 1
TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.
Formule :C₃₅H₅₁N₃O₃
Couleur et forme :Solid
Masse moléculaire :561.798
Ref: TM-T204394
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hCAI/II-IN-10
hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.
Formule :C₂₄H₁₇Cl₂N₃O₃S₂
Couleur et forme :Solid
Masse moléculaire :530.446
Ref: TM-T204359
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DG013A formate
DG013A (formate) is a tripeptide-mimicking inhibitor of hypophosphorous acid. It exhibits IC50 values of 33 nM for ERAP1 and 11 nM for ERAP2. This compound can be utilized in research related to autoimmune diseases and cancer.
Formule :C₂₇H₃₇N₄O₄PCH₂O₂
Couleur et forme :Solid
Masse moléculaire :530.99
Ref: TM-T205046
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Citrulline malate
CAS :
- 70796-17-7
Citrulline malate is a cpd of anti-fatigue.
Formule :C₁₀H₁₉N₃O₈
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :309.27
Ref: TM-T20200
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12α-Hydroxysteroid dehydrogenase
CAS :
- 61642-40-8
12α-Hydroxysteroid dehydrogenase, an NAD-dependent enzyme expressed in Bacillus sphaericus, actively processes both free and conjugated bile salts. It is utilized to determine the levels of 12α-hydroxy bile acids in serum.
Couleur et forme :Solid
Ref: TM-T200077
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2-Methylnicotinamide
CAS :
- 58539-65-4
2-Methylnicotinamide is an endogenous metabolite of nicotinamide and can be used for related research in the life sciences.
Formule :C₇H₈N₂O
Degré de pureté :99.84%
Couleur et forme :Solid
Masse moléculaire :136.15
Ref: TM-TN9444
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GSK-3β/CK-1δ-IN-1
GSK-3β/CK-1δ-IN-1 (8d) is a dual inhibitor of GSK-3β and CK-1δ that can cross the blood-brain barrier, with IC50 values of 0.77 μM and 0.57 μM, respectively. GSK-3β/CK-1δ-IN-1 (8d) is applicable in neuroblastoma research.
Formule :C₂₂H₁₇F₃N₄O
Couleur et forme :Solid
Masse moléculaire :410.39
Ref: TM-T207691
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GPX4-IN-16
GPX4-IN-16 ((R)-9i) is a potent inhibitor of GPX4 with a KD value of 20.4 nM, exhibiting cytotoxic properties and anticancer activity.
Formule :C₂₉H₂₄N₄O₃S₂
Couleur et forme :Solid
Masse moléculaire :540.656
Ref: TM-T204889
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Ppack trifluoroacetate
CAS :
- 157379-44-7
Ppack trifluoroacetate: Peptide, inhibits thrombin, prevents clotting (Ki: 0.24 nM), used in anticoagulation & thrombin research.
Formule :C₂₃H₃₂ClF₃N₆O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :564.99
Ref: TM-T25977
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Trihydroxycholestanoic Acid
CAS :
- 547-98-8
Trihydroxycholestanoic acid aids cholic acid creation; high levels indicate Zellweger syndrome due to faulty PEX genes.
Formule :C₂₇H₄₆O₅
Couleur et forme :Solid
Masse moléculaire :450.66
Ref: TM-T37666
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Largazole
CAS :
- 1009815-87-5
Largazole is a potent and selective histone deacetylase (HDAC) inhibitor and antiproliferative agent from Symploca.
Formule :C₂₉H₄₂N₄O₅S₃
Couleur et forme :Solid
Masse moléculaire :622.86
Ref: TM-T25630
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DSPE-PEG5000-M2pep
DSPE-PEG5000-M2pep is a PEG compound composed of DSPE and the M2 macrophage-targeting peptide (M2pep). Serving either as a monovalent or multivalent ligand, M2pep is conjugated with pro-apoptotic peptides to direct toxicity specifically toward M2 macrophages. DSPE-PEG5000-M2pep is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01080
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Aminopeptidase N inhibitor 2
AminopeptidaseN inhibitor 2 is an APN inhibitor (IC50: 4.3 μM) with antitumor properties.
Formule :C₁₂H₁₆F₂N₂O₄S
Couleur et forme :Solid
Masse moléculaire :322.07988
Ref: TM-T207518
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14,15-Leukotriene D4
CAS :
- 75290-64-1
14,15-LTD4, an eoxin synthesized by eosinophils, mast cells, and nasal polyps, has modest contractile activity but can increase vascular permeability.
Formule :C₂₅H₄₀N₂O₆S
Couleur et forme :Solid
Masse moléculaire :496.66
Ref: TM-T37261
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GlcNAc kinase (EcNagK)
GlcNAc kinase (EcNagK), ATP-dependent, phosphorylates C-6 hydroxyl on GlcNAc, producing GlcNAc-6-P.
Couleur et forme :Solid
Ref: TM-T75405
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SHO1122147
SHO1122147 (Compound 7m) disrupts the mitochondrial electron transport chain, demonstrating mitochondrial uncoupling activity (EC50=3.6 μM). It increases the cellular oxygen consumption rate (OCR=69%) and enhances cellular respiration. Additionally, SHO1122147 is orally active and can be utilized in research related to obesity and metabolic dysfunction-associated steatohepatitis (MASH).
Formule :C₁₇H₁₁ClN₄O₂
Couleur et forme :Solid
Masse moléculaire :338.748
Ref: TM-T204360
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Zaragozic acid D
CAS :
- 155179-14-9
Zaragozic acid D inhibits squalene synthase and ras farnesyl-protein transferase isolated from the keratinophilic fungus Amauroascus niger.
Formule :C₃₄H₄₆O₁₄
Couleur et forme :Solid
Masse moléculaire :678.72
Ref: TM-T26347
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Lodenafil carbonate
CAS :
- 398507-55-6
Lodenafil carbonate is a prodrug, orally used as a PDE5 inhibitor for ED treatment.
Formule :C₄₇H₆₂N₁₂O₁₁S₂
Couleur et forme :Solid
Masse moléculaire :1035.21
Ref: TM-T37325
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Resveratrol-3-O-sulfate sodium
CAS :
- 858127-11-4
Resveratrol-3-O-sulfate reduces IL-1α/β, IL-6, TNF-α in LPS-stimulated U-937 cells, inhibits Caco-2 cell growth, induces apoptosis, and binds mitoNEET.
Formule :C₁₄H₁₁NaO₆S
Couleur et forme :Solid
Masse moléculaire :330.29
Ref: TM-T36517
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1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol
CAS :
- 80840-09-1
1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is a quinoxaline derivative and endogenous metabolite applicable to biochemical experiments and drug synthesis research.
Formule :C₁₂H₁₄N₂O₄
Degré de pureté :99.49%
Couleur et forme :Solid
Masse moléculaire :250.25
Ref: TM-T10010
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BMT-297376
CAS :
- 2251031-81-7
BMT-297376, the optimized Linrodostat, is a potent IDO1 inhibitor.
Formule :C₂₃H₂₉F₂N₃O₃
Couleur et forme :Solid
Masse moléculaire :433.5
Ref: TM-T39779
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DSPE-PEG2000-TAT
DSPE-PEG2000-TAT is a PEG compound consisting of DSPE and the cell-penetrating peptide (TAT) peptide. It can be used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01111
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(±)-CBCQ
CAS :
- 2415352-36-0
(±)-CBCQ, an oxidation product of cannabidiol, exhibits an EC50 value of 14.7 μM for the activation of peroxisome proliferator-activated receptor γ (PPAR-γ).
Formule :C₂₁H₂₈O₃
Couleur et forme :Solid
Masse moléculaire :328.45
Ref: TM-T203263
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7-Methylguanosine 5'-diphosphate sodium
CAS :
- 104809-16-7
7-Methylguanosine 5’-diphosphate (7-Methyl-GDP) sodium, a cap analog, is utilized in the synthesis of mRNA cap analogues[1].
Formule :C₁₁H₁₆N₅NaO₁₁P₂
Couleur et forme :Solid
Masse moléculaire :479.21
Ref: TM-T37154
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(24R)-MC 976
CAS :
- 112828-09-8
(24R)-MC 976 is a derivative of Vitamin D3.
Formule :C₂₇H₄₂O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :414.62
Ref: TM-T16023L
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LYP-8
LYP-8 is a potent NAMPT degrader that achieves a maximum degradation rate of 97% in NAMPT within SKOV-3 cells at a concentration of 0.5 μM. LYP-8 also demonstrates anticancer activity both in vitro and in vivo.
Formule :C₅₆H₇₄N₈O₁₀S
Masse moléculaire :1050.52486
Ref: TM-T209938
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(3S,5R)-Fluvastatin D6 sodium
CAS :
- 2249799-35-5
(3S,5R)-Fluvastatin D6 sodium: deuterium-labeled synthetic HMG-CoA reductase inhibitor with 8 nM IC50.
Formule :C₂₄H₂₅FNNaO₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :439.49
Ref: TM-T10128
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Methyl gerfelin
CAS :
- 700870-56-0
Methyl gerfelin, a flavonoid, hinders osteoclast formation by targeting GLO1, SCP2, and SGTA proteins.
Formule :C₁₆H₁₆O₆
Couleur et forme :Solid
Masse moléculaire :304.29
Ref: TM-T73885
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DMPS-Na
CAS :
- 105405-50-3
DMPS-Na is an arsenicolytic agent with toxicity that can be used to study cell membranes.
Formule :C₃₄H₆₅NNaO₁₀P
Degré de pureté :98%
Couleur et forme :Soild
Masse moléculaire :701.84
Ref: TM-TN7245
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CMP-Sialic acid
CAS :
- 3063-71-6
CMP-Sialic acid inhibits UDP-GlcNAc 2-epimerase and is a key substrate for sialic acid biosynthesis.
Formule :C₂₀H₃₁N₄O₁₆P
Couleur et forme :Solid
Masse moléculaire :614.45
Ref: TM-T73747
+ Info
Anticancer agent 232
Anticanceragent 232 (compound 12f) is a sugar hybrid designed from 1-azide glycosides derived from d-glucose, d-galactose, and d-mannose. The IC50 values for this compound are 1.05 μM against MCF-7 cells and 18.03 μM for MDA-MB231 cells.
Formule :C₃₂H₃₁BrN₄O₁₁
Masse moléculaire :726.11727
Ref: TM-T210293
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Fluazifop-P-butyl
CAS :
- 79241-46-6
Fluazifop-P-butyl is an arylophenoxypropionate group graminicide that functions as an inhibitor of acetyl-CoA carboxylase (ACCase)[1].
Formule :C₁₉H₂₀F₃NO₄
Couleur et forme :Light Yellow Liquid
Masse moléculaire :383.36
Ref: TM-T36785
+ Info
α-Glucosidase-IN-58
α-Glucosidase-IN-58 (Compound 6d) is an α-glucosidase inhibitor with an IC50 of 1.47 μM.
Formule :C₂₂H₁₃F₃N₂OS
Masse moléculaire :410.07007
Ref: TM-T209494
+ Info
13,14-dihydro Prostaglandin E1
CAS :
- 19313-28-1
13,14-dihydro PGE1, a metabolite of PGE1, inhibits platelet aggregation and activates adenylate cyclase with IC50 of 31/21 nM and Kact 668 nM.
Formule :C₂₀H₃₆O₅
Couleur et forme :Solid
Masse moléculaire :356.503
Ref: TM-T36775
+ Info
2,3,4,6,7,8-Hexachlorodibenzofuran
CAS :
- 60851-34-5
2,3,4,6,7,8-Hexachlorodibenzofuran (2,3,4,6,7,8-HxCDF) is a type of polychlorinated dibenzofuran (PCDF). It induces the expression of aryl hydrocarbon hydroxylase (AHH) and ethoxyresorufin-o-deethylase (EROD) genes in H-4-II-E rat hepatoma cells, with EC50 values of 0.687 and 0.575 nM, respectively.
Formule :C₁₂H₂Cl₆O
Couleur et forme :Solid
Masse moléculaire :374.86
Ref: TM-T203593
+ Info
Adenosylhomocysteinase
CAS :
- 9025-54-1
SAHH, an enzyme, reversibly converts SAH into adenosine and L-homocysteine, and may predict HBV-LC outcomes.
Formule :C₁₄H₁₃N₃O₂S₂
Couleur et forme :Solid
Masse moléculaire :319.04492
Ref: TM-T74764
+ Info
Norpropranolol hydrochloride
CAS :
- 62618-09-1
Norpropranolol hydrochloride is the active metabolite of Propranolol.
Formule :C₁₃H₁₆ClNO₂
Couleur et forme :Solid
Masse moléculaire :253.73
Ref: TM-T203546
+ Info
Cy3-PEG-DSPE (MW 3400)
Cy3-PEG-DSPE (MW 3400) is a PEG phospholipid that incorporates Cy3 dye, utilized for labeling proteins/nucleic acids and in fluorescence microscopy. It can self-assemble in aqueous solutions to form micelles/lipid bilayers, and is employed in the creation of liposomes or nanoparticles for delivering nutrients such as mRNA or DNA vaccines.
Couleur et forme :Solid
Masse moléculaire :3400 (Average)
Ref: TM-T204869
+ Info
ABC34
CAS :
- 1831135-56-8
ABC34, an inactive JJH260 control, poorly inhibits AIG1 enzyme at IC50 >25 μM; potently blocks off-target hydrolases ABHD6 and PPT1.
Formule :C₃₁H₃₃N₅O₆
Couleur et forme :Solid
Masse moléculaire :571.634
Ref: TM-T38316
+ Info
Alcohol oxidase
CAS :
- 9073-63-6
Alcohol oxidase, a key enzyme in the methanol utilization pathway, is derived from yeast peroxisomes.
Couleur et forme :Solid
Ref: TM-T76105
+ Info
Inostamycin A
CAS :
- 129905-10-8
Inostamycin A, a anticancer bacterial metabolite isolated from Streptomyces, is a selective inhibitor of CDP-diacylglycerol:inositol 3-phosphatidyltransferase.
Formule :C₃₈H₆₈O₁₁
Couleur et forme :Solid
Masse moléculaire :700.94
Ref: TM-T36844
+ Info
Desbutyl Lumefantrine D9
CAS :
- 1346606-35-6
Desbutyl Lumefantrine D9, a deuterium-labeled metabolite of Lumefantrine, exhibits the incorporation of deuterium atoms.
Formule :C₂₆H₂₄Cl₃NO
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :481.89
Ref: TM-T19275
+ Info
ACAT-IN-5
CAS :
- 199983-93-2
ACAT-IN-5 inhibits ACAT, suppressing NF-κB-mediated transcription.
Formule :C₃₂H₄₉N₃O₅S
Couleur et forme :Solid
Masse moléculaire :587.82
Ref: TM-T39412
+ Info
Ophiobolin A
CAS :
- 4611-05-6
Ophiobolin A: Fungal metabolite, phytotoxin, inhibits calmodulin-activated phosphodiesterase (IC50: 9μM), with antimicrobial and anticancer properties.
Formule :C₂₅H₃₆O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :400.559
Ref: TM-T16397
+ Info
β-Apooxytetracycline
CAS :
- 18751-99-0
β-Apooxytetracycline is a potential impurity found in commercial preparations of oxytetracycline.
Formule :C₂₂H₂₂N₂O₈
Couleur et forme :Solid
Masse moléculaire :442.424
Ref: TM-T35425
+ Info
PROTAC SGK3 degrader-1
CAS :
- 2381320-35-8
PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC coupler that targets SGK3 and binds ligands to VH032 VHL to induce endogenous SGK3 degradation.
Formule :C₅₇H₇₃FN₁₀O₁₁S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1157.38
Ref: TM-T13847
+ Info
ML266
CAS :
- 1462267-08-8
ML266: GCase chaperone, non-inhibiting, IC50=2.5 µM, aids mutant protein transport, may help in Gaucher disease study.
Formule :C₂₄H₂₂BrN₃O₄
Degré de pureté :99.58%
Couleur et forme :Solid
Masse moléculaire :496.35
Ref: TM-T8990
+ Info
Adenosine deaminase
CAS :
- 9026-93-1
Adenosine deaminase is an enzyme that catalyzes the irreversible deamination of 2'-deoxyadenosine and adenosine to 2'-deoxyinosine and inosine, respectively.
Degré de pureté :98%
Couleur et forme :Solid
Ref: TM-T19179
+ Info
DCG04
CAS :
- 314263-42-8
DCG04: a mannose-6-phosphate receptor ligand, fluorescent cysteine cathepsin probe for endolysosomal targeting.
Formule :C₄₃H₆₆N₈O₁₁S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :903.11
Ref: TM-T27131
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Daclatasvir Impurity B
CAS :
- 2226541-13-3
Daclatasvir Impurity B, a noted impurity of the antiviral agent Daclatasvir, acts as a potent inhibitor of the HCV NS5A protein [1].
Formule :C₃₅H₄₁N₇O₄
Couleur et forme :Solid
Masse moléculaire :623.74
Ref: TM-T74006
+ Info
Vitamin K1 2,3-epoxide
CAS :
- 25486-55-9
Vitamin K1 2,3-epoxide (Phylloquinone oxide) is reduced to vitamin k and is involved in the vitamin k cycle.
Formule :C₃₁H₄₆O₃
Degré de pureté :98% - 98.05%
Couleur et forme :Solid
Masse moléculaire :466.7
Ref: TM-T36730
+ Info
Herbicidal agent 6
Herbicidal agent 6 (D15) functions as a Transketolase (TKL) inhibitor and exhibits herbicidal activity.
Couleur et forme :Odour Solid
Ref: TM-T200613
+ Info
SY-640
CAS :
- 168705-70-2
SY-640, an acetamide derivative, strongly protects the liver and lessens Propionibacterium acnes and lipopolysaccharide-induced damage in mice.
Formule :C₁₁H₁₃NO₃
Degré de pureté :99.51% - 99.66%
Couleur et forme :Solid
Masse moléculaire :207.23
Ref: TM-T37859
+ Info
Nicotinic Acid Adenine Dinucleotide
CAS :
- 6450-77-7
Nicotinic Acid Adenine Dinucleotide is a precursor of NAD (Nicotinamide adenine dinucleotide) and a substrate for glutamine-dependent NAD+ synthase
Formule :C₂₁H₂₆N₆O₁₅P₂
Couleur et forme :Soild
Masse moléculaire :664.41
Ref: TM-T205954
+ Info
RORγt inhibitor 1
CAS :
- 1561770-72-6
RORγt inhibitor 1 is a RORγt allosteric inhibitor with an IC 50 value of 1 nM.
Formule :C₂₃H₂₁ClFN₃O₄
Couleur et forme :Solid
Masse moléculaire :457.89
Ref: TM-T39038
+ Info
NAADP sodium
NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.
Formule :C₂₁H₂₇N₆O₁₈P₃
Couleur et forme :Solid
Masse moléculaire :744.39
Ref: TM-T35922
+ Info
Endoglycoceramidase II (EGCase II)
CAS :
- 2763216-34-6
EGCase II is an enzyme breaking down the glycan-ceramide bond in glycosphingolipids.
Couleur et forme :Solid
Ref: TM-T75406
+ Info
ARL67156 trisodium hydrate
ARL67156 trisodium hydrate inhibits ecto-ATPase, NTPDase1, NTPDase3, NPP1 (Kis 11-18µM), for calcific valve disease, asthma research.
Formule :C₁₅H₂₃Br₂N₅Na₃O₁₃P₃
Couleur et forme :Solid
Masse moléculaire :834.61
Ref: TM-T73644
+ Info
Cytochrome P450 reductase
CAS :
- 9039-06-9
Cytochrome P450 reductase, a NADPH-cytochrome reductase, facilitates an optimal conformation of aromatase for substrate binding [1].
Couleur et forme :Solid
Ref: TM-T80057
+ Info
α-Glucosidase-IN-67
α-Glucosidase-IN-67 (compound 5k) is a potent inhibitor of α-glucosidase, exhibiting IC50 values of 0.31 µM for α-glucosidase and 4.51 µM for α-amylase. This compound shows potential for research in type 2 diabetes.
Formule :C₂₄H₂₂BrN₃O₃S
Masse moléculaire :511.05653
Ref: TM-T210381
+ Info
Ferulic acid acyl-β-D-glucoside
CAS :
- 7196-71-6
Ferulic acid acyl-β-D-glucoside, a metabolite of Ferulic Acid, is a novel inhibitor of fibroblast growth factor receptor 1 (FGFR1).
Formule :C₁₆H₂₀O₉
Couleur et forme :Solid
Masse moléculaire :356.327
Ref: TM-T40832
+ Info
P-orlandin
CAS :
- 1407546-21-7
P-orlandin, a fungal compound, blocks FREP1, halting P. falciparum's mosquito infection.
Formule :C₂₂H₁₈O₈
Couleur et forme :Solid
Masse moléculaire :410.37
Ref: TM-T75450
+ Info
AP219
CAS :
- 779282-36-9
AP39 boosts mitochondrial H2S with triphenylphosphonium and dithiolethione; AP219 lacks H2S-donating part.
Formule :C₂₈H₃₄O₂P
Couleur et forme :Solid
Masse moléculaire :433.551
Ref: TM-T36240
+ Info
Dilaurylglycerosulfate
CAS :
- 99387-94-7
Dilauryl glycerol sulfate is an auxiliary emulsifier for lipase determination.
Formule :C₂₇H₅₆O₆S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :508.8
Ref: TM-T19283
+ Info
Endoglycoceramidase I (EGCase I)
CAS :
- 2768502-40-3
EGCase I is a glycosidase used in biochemistry to transfer GSL sugars to 1-alkanols' primary hydroxyl groups.
Couleur et forme :Solid
Ref: TM-T75407
+ Info
BMS-770767
CAS :
- 1875067-34-7
BMS-770767 is a novel 11-betahydroxysteroid dehydrogenase type I (11ß-HSD1) inhibitor.
Formule :C₁₉H₁₈ClN₃O₂
Couleur et forme :Solid
Masse moléculaire :355.82
Ref: TM-T26858
+ Info
PP5-IN-2
PP5-IN-2, a selective and orally active inhibitor of protein phosphatase 5 (PP5), exhibits an IC 50 of 0.9 μM. This compound activates p53 and leads to the downregulation of cyclin D1 and MGMT, thereby inducing cell cycle arrest and reversing Temozolomide (TMZ) resistance in the U87 MG cell line. Additionally, PP5-IN-2 has demonstrated effective inhibition of tumor growth in the xenograft mouse model.
Formule :C₁₆H₁₅NO₄
Couleur et forme :Solid
Masse moléculaire :285.29
Ref: TM-T89967
+ Info
Paraherquamide E
CAS :
- 125600-53-5
Fungal-derived paraherquamide E kills C. elegans and O. fasciatus, reduces T. colubriformis eggs in gerbils.
Formule :C₂₈H₃₅N₃O₄
Couleur et forme :Solid
Masse moléculaire :477.605
Ref: TM-T35908
+ Info
hCAII-IN-6
"hCAII-IN-6 (S-13) inhibits hCA II (4.4 nM) and isoforms I, IV, IX (9.2, 480.2, 14.7 nM). For glaucoma research."
Formule :C₂₀H₂₅N₃O₄S
Couleur et forme :Solid
Masse moléculaire :403.5
Ref: TM-T74330
+ Info
F-14329
CAS :
- 942195-19-9
F-14329 is a tetramic acid fungal metabolite [1] .
Formule :C₂₁H₂₇NO₅
Couleur et forme :Solid
Masse moléculaire :373.44
Ref: TM-T75654
+ Info
CE(20:5(5Z,8Z,11Z,14Z,17Z)
CAS :
- 74892-97-0
CE(20:5(5Z,8Z,11Z,14Z,17Z) is an endogenous metabolite.
Formule :C₄₇H₇₄O₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :671.09
Ref: TM-T10748
+ Info
Simvastatin Acyl-β-D-glucuronide
CAS :
- 463962-56-3
Simvastatin Acyl-β-D-glucuronide, a metabolite formed from Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, showcasing a potent Ki of 0.2 nM.
Formule :C₃₁H₄₈O₁₂
Couleur et forme :Solid
Masse moléculaire :612.71
Ref: TM-T40557
+ Info
DSPE-PEG
CAS :
- 145035-96-7
DSPE-PEG: a phospholipid-polymer for stable, efficient drug delivery with longer circulation.
Formule :C₄₅H₉₀NO₁₀P
Couleur et forme :Solid
Masse moléculaire :835.63024
Ref: TM-T74245
+ Info
HMG-CoA Reductase-IN-1
HMG-CoA Reductase-IN-1 is an inhibitor of HMG-CoA reductase, demonstrating strong inhibitory activity on HMGR and affinity for OATP1B1, with pIC50 and pKm
Formule :C₂₇H₂₉N₃O₇
Couleur et forme :Solid
Masse moléculaire :507.54
Ref: TM-T79520
+ Info
MAGL-IN-8
MAGL-IN-8 (compound 13) serves as a reversible inhibitor of monoacylglycerol lipase (MAGL), exhibiting an inhibitory concentration half-maximal (IC50) value of
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T81879
+ Info
Retinyl glucoside
CAS :
- 136778-12-6
Retinyl-β-D-glucoside, a biologically active metabolite of vitamin A, naturally occurs in fish and mammals.
Formule :C₂₆H₄₀O₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :448.59
Ref: TM-T13866
+ Info
Tetomilast
CAS :
- 145739-56-6
Tetomilast (OPC-6535) is a phosphodiesterase-4 (PDE4) inhibitor, potentially effective in treating inflammatory bowel disease (IBD) and chronic obstructive
Formule :C₁₉H₁₈N₂O₄S
Couleur et forme :Solid
Masse moléculaire :370.42
Ref: TM-T38944
+ Info
m-Tyramine
CAS :
- 588-05-6
m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator.
Formule :C₈H₁₁NO
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :137.18
Ref: TM-T11937
+ Info
N-Lactylleucine
CAS :
- 112757-17-2
N-Lactylleucine is an endogenous metabolite detectable in patients with intermediate maple syrup urine disease.
Formule :C₉H₁₇NO₄
Couleur et forme :Solid
Masse moléculaire :203.24
Ref: TM-TN8216
+ Info
Ferroleuton
Ferroleuton is a selective competitive inhibitor of 5-lipoxygenase with an IC50 of 0.21 μM. It demonstrates antioxidant properties, clearing 86% of DPPH at 50 μM and exhibiting activities in ABTS (EC50 = 19.42 μM) and FRAP (EC50 = 3.32 μM) assays.
Formule :C₁₃H₁₆FeN₂O₂
Couleur et forme :Solid
Masse moléculaire :288.12
Ref: TM-T205027
+ Info
Laurencin
CAS :
- 3442-58-8
Laurencin is a component of the sea hare, Aplysia dactylomela.
Formule :C₁₇H₂₃BrO₃
Couleur et forme :Solid
Masse moléculaire :355.27
Ref: TM-T32595
+ Info
α-Glucosidase-IN-38
α-Glucosidase-IN-38 (Compound 11j) is a potent α-glucosidase inhibitor, demonstrating an IC50 of 12.44±0.38 μM, and is significant in the context of Diabetes
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T80712
+ Info
1-Myristoyl-2-hydroxy-sn-glycero-3-PE
CAS :
- 123060-40-2
Naturally-occurring lysophospholipid raises intracellular calcium and is higher in breast cancer patients.
Formule :C₁₉H₄₀NO₇P
Couleur et forme :Solid
Masse moléculaire :425.50
Ref: TM-T36453
+ Info
R 80123
CAS :
- 133718-30-6
R 80123 is a highly selective inhibitor of phosphodiesterase,is the Z-isomer of R 79595
Formule :C₂₆H₂₉N₅O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :459.54
Ref: TM-T12611
+ Info
L-Lysine, sulfite (2:1)
CAS :
- 53411-64-6
L-Lysine, sulfite (2:1) is a drug/ therapeutic agent.
Formule :C₆H₁₄N₂O₂H₂O₃S
Couleur et forme :Solid
Masse moléculaire :187.23
Ref: TM-T32819
+ Info
ZINC77292789
CAS :
- 116783-35-8
ZINC77292789 (Fmoc-Thr[GalNAc(Ac)3-α-D]-OH) is a reagent for the preparation of a synthetic MUC1 Glycopeptide Bearing βGalNAc-Thr as a Tn antigen isomer which
Formule :C₃₃H₃₈N₂O₁₃
Degré de pureté :99.24%
Couleur et forme :Solid
Masse moléculaire :670.66
Ref: TM-TP1166
+ Info
Methionylserine
CAS :
- 14517-43-2
Methionylserine (H-MET-SER-OH), a dipeptide, binds hPEPT1 (Km 0.2 mM), inhibits ACE, used in hypertension research.
Formule :C₈H₁₆N₂O₄S
Couleur et forme :Solid
Masse moléculaire :236.29
Ref: TM-T77199
+ Info
6,8-Dihydroxy-1,2,7-trimethoxy-3-methylanthraquinone
CAS :
- 1622982-59-5
Compound 1, 6,8-Dihydroxy-1,2,7-trimethoxy-3-methylanthraquinone, is an anthraquinone α-glucosidase inhibitor with an IC50 of 185 μM, and it can be isolated
Formule :C₁₈H₁₆O₇
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :344.32
Ref: TM-T79964
+ Info
Tibenelast
CAS :
- 97852-72-7
Tibenelast is a cioactive chemical.
Formule :C₁₃H₁₄O₄S
Couleur et forme :Solid
Masse moléculaire :266.31
Ref: TM-T34874
+ Info
MTHFD2-IN-1
MTHFD2-IN-1 (compound 12) is a potent inhibitor of methylenetetrahydrofolate dehydrogenase (MTHFD2) [1].
Formule :C₂₄H₂₁NO₆
Couleur et forme :Solid
Masse moléculaire :419.43
Ref: TM-T74834
+ Info
Fmoc-Cys(Acm)-OH
CAS :
- 86060-81-3
Fmoc-Cys(Acm)-OH (Fmoc-S-acetamidomethyl-L-cysteine) is a cysteine derivative.
Formule :C₂₁H₂₂N₂O₅S
Degré de pureté :99.89%
Couleur et forme :Solid
Masse moléculaire :414.47
Ref: TM-T64327
+ Info
LQ-38
LQ-38 is an orally active, soluble epoxide hydrolase (sEH) inhibitor with an IC50 value of 5.2 nM. It has shown anti-inflammatory activity in rat foot edema models and in mouse models of acute pancreatitis, and exhibits analgesic effects in acetic acid-induced mouse writhing models.
Formule :C₄₂H₆₈N₂O₉
Couleur et forme :Solid
Masse moléculaire :745.00
Ref: TM-T200833
+ Info
Chaetosemin J
CAS :
- 2230052-47-6
Chaetosemin J, antifungal, inhibits Botrytis, Alternaria, Magnaporthe, Gibberella; MIC 12.5-25 μM.
Formule :C₁₄H₁₄O₄
Couleur et forme :Solid
Masse moléculaire :246.26
Ref: TM-T75475
+ Info
m-PEG8-DSPE
m-PEG8-DSPE is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.
Formule :C₅₉H₁₁₆NO₁₇P
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1142.52
Ref: TM-T18219
+ Info
1-Arachidonoyl Lysophosphatidic Acid (ammonium salt)
CAS :
- 799268-65-8
1-Arachidonoyl LPA: phospholipid with arachidonic acid, sn-1, LPA2 receptor binder, EC50 ~10 nM, modulates cytokine secretion, affects cell differentiation.
Formule :C₂₃H₄₂NO₇P
Couleur et forme :Solid
Masse moléculaire :475.563
Ref: TM-T36452
+ Info
11-epi-Chaetomugilin I
CAS :
- 1319729-88-8
11-epi-Chaetomugilin I, from Chaetomium globosum, has cytotoxic effects against P388, HL-60, L1210 leukemia, and KB carcinoma cells.
Formule :C₂₂H₂₇ClO₅
Couleur et forme :Solid
Masse moléculaire :406.9
Ref: TM-T75453
+ Info
N-Decanoyl p-Nitroaniline
CAS :
- 72298-63-6
DepNA, a nitroaniline fatty acid amide, measures FAAH activity by releasing yellow dye p-nitroaniline upon exposure, detectable via spectrophotometer.
Formule :C₁₆H₂₄N₂O₃
Couleur et forme :Solid
Masse moléculaire :292.379
Ref: TM-T37217
+ Info
2,7"-Phloroglucinol-6,6'-bieckol
CAS :
- 1621988-60-0
2,7"-Phloroglucinol-6,6'-bieckol serves as an effective oral dual α-amylase/α-glucosidase inhibitor, demonstrating IC 50 concentrations of 6.94 μM and 23.35 μM, respectively. This compound is beneficial in mitigating postprandial hyperglycemia among diabetic mice and is applicable in diabetes research [1].
Formule :C₄₈H₃₀O₂₃
Couleur et forme :Solid
Masse moléculaire :974.74
Ref: TM-TN7594
+ Info
Lofacimig
Lofacimig is a bispecific antibody of VH-VH-G1(h-CH2-CH3) dimer type that targets FXI/PTA.
Couleur et forme :Odour Liquid
Ref: TM-T9901A-464
+ Info
Chrysophanol triglucoside
CAS :
- 120181-07-9
Chrysophanol triglucoside from Cassia obtusifolia, blocks PTP1B (IC50 80.17μM) & α-glucosidase (IC50 197.06μM), may aid diabetes study.
Formule :C₃₃H₄₀O₁₉
Couleur et forme :Solid
Masse moléculaire :740.664
Ref: TM-T38587
+ Info
(25R)-12α-Hydroxyspirost-4-en-3-one
CAS :
- 50888-50-1
'(25R)-12α-Hydroxyspirost-4-en-3-one is a minor metabolite resulting from Nocardia globerula's metabolization of Hecogenin [1].'
Formule :C₂₇H₄₀O₄
Couleur et forme :Solid
Masse moléculaire :428.6
Ref: TM-T75607
+ Info
5-(3-Hydroxyphenyl)-5-phenylhydantoin
CAS :
- 30074-03-4
5-(3-Hydroxyphenyl)-5-phenylhydantoin is a bioactive chemical.
Formule :C₁₅H₁₂N₂O₃
Couleur et forme :Solid
Masse moléculaire :268.27
Ref: TM-T29445
+ Info
ND-011992
CAS :
- 2446880-46-0
ND-011992: Quinazoline inhibitor of E. coli respiratory enzymes; IC50s: 0.12-2.47 μM; potential tuberculosis research.
Formule :C₂₁H₁₄F₃N₃O
Degré de pureté :99.7%
Couleur et forme :Soild
Masse moléculaire :381.35
Ref: TM-T77615
+ Info
Calcium gluconate monohydrate
CAS :
- 66905-23-5
Calcium gluconate monohydrate is a useful organic compound for research related to life sciences. The catalog number is T35350 and the CAS number is 66905-23-5.
Formule :C₆H₁₆CaO₈
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :256.264
Ref: TM-T35350
+ Info
Urate oxidase
CAS :
- 9002-12-4
Uricase catalyzes uric acid to allantoin in many mammals' peroxisomes, used in biochemistry.
Couleur et forme :Solid
Ref: TM-T73617
+ Info
Carboxypeptidase B
CAS :
- 9025-24-5
Carboxypeptidase B degrades peptides from C-terminal, freeing amino acids, and targets basic residues.
Couleur et forme :Solid
Ref: TM-T76102
+ Info
2-Methyl-1-naphthol
CAS :
- 7469-77-4
2-Methyl-1-naphthol is a prostaglandin G/H synthase and polyunsaturated fatty acid 5-lipoxygenase inhibitor, suitable for biochemical experiments.
Formule :C₁₁H₁₀O
Degré de pureté :98.33%
Couleur et forme :Solid
Masse moléculaire :158.2
Ref: TM-TN9522
+ Info
Amastatin hydrochloride
CAS :
- 100938-10-1
Amastatin HCl is an inhibitor of aminopeptidase. It also induces vasoconstriction.
Formule :C₂₁H₃₉ClN₄O₈
Couleur et forme :White To Off-White Powder
Masse moléculaire :511.01
Ref: TM-T19665
+ Info
ChAT IN-1
ChAT IN-1 is a selective inhibitor of Choline Acetyltransferase (ChAT) that is utilized in studying mechanisms related to non-neuronal ChAT overexpression in cancers such as colon cancer and lung cancer, as well as in research concerning Alzheimer's disease (AD).
Formule :C₂₁H₁₅N₃O₂
Couleur et forme :Solid
Masse moléculaire :341.36
Ref: TM-T203594
+ Info
HIV-IN-9
HIV-IN-9 (Compound 2b) is an HIV inhibitor with an IC50 value of 6.65 μg/mL, demonstrating high binding affinity for HIV-RT.
Couleur et forme :Odour Solid
Ref: TM-T82194
+ Info
CCR1/5/8 activator 1
CAS :
- 4771-50-0
CCR1/5/8 activator 1 is a cytoplasmic phospholipase A inhibitor with antifungal activity.
Formule :C₁₀H₉NO
Degré de pureté :>99.99%
Couleur et forme :Solid
Masse moléculaire :159.18
Ref: TM-T77349
+ Info
Carbazeran citrate
CAS :
- 153473-94-0
aldehyde oxidase (AO) substrate
Formule :C₂₄H₃₂N₄O₁₁
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :552.53
Ref: TM-T22622
+ Info
PROTAC MAGL degrader-1
PROTACMAGLdegrader-1 is an orally active PROTAC agent that simultaneously targets both monoacylglycerol lipase (MAGL) and the E3 ubiquitin ligase MDM2. It functions by degrading MAGL and inhibiting the interaction between MDM2 and p53. Additionally, PROTACMAGLdegrader-1 has partial blood-brain barrier (BBB) penetration and can induce apoptosis in glioblastoma stem cells (GSC).
Couleur et forme :Odour Solid
Ref: TM-T206750
+ Info
RORγt inverse agonist 31
RORγt inverse agonist 31 (14g) is a potent antagonist of the retinoic acid receptor-related orphan receptor γt (RORγt), exhibiting an inhibitory concentration (
Formule :C₂₃H₁₅Cl₂F₃N₄O₃S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :555.36
Ref: TM-T79470
+ Info
PKM2-IN-10
PKM2-IN-10 is a PKM2 inhibitor. It effectively suppresses the proliferation of A549 and HCC1833 cell lines with IC50 values of 3.36 μM and 9.20 μM, respectively. PKM2-IN-10 demonstrates antitumor activity in human non-small cell lung cancer (NSCLC) and mouse lung adenocarcinoma models. It is applicable for research in lung cancer.
Formule :C₂₁H₁₅F₄N₅
Couleur et forme :Solid
Masse moléculaire :413.12636
Ref: TM-T207198
+ Info
LDHA-IN-3
CAS :
- 227010-33-5
LDHA-IN-3 is a potent selenobenzene-based LDHA inhibitor with a 145.2 nM IC50, useful in cancer research.
Formule :C₁₃H₉F₃Se
Degré de pureté :99.71%
Couleur et forme :Solid
Masse moléculaire :301.17
Ref: TM-T39805
+ Info
LYP-IN-3
LYP-IN-3 (compound D34) is a selective Lymphoid-tyrosine phosphatase (LYP) inhibitor (Ki=0.93 μM) that modulates the T-cell receptor (TCR) signaling pathway
Formule :C₃₅H₂₇NO₆S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :589.66
Ref: TM-T79634
+ Info
2,3-Dehydrosilybin B
CAS :
- 142796-24-5
2,3-Dehydrosilybin B is a useful organic compound for research related to life sciences and the catalog number is T125883.
Formule :C₂₅H₂₀O₁₀
Couleur et forme :Solid
Masse moléculaire :480.42
Ref: TM-T125883
+ Info
Impurity of Doxercalciferol
CAS :
- 127516-23-8
Doxercalciferol impurity, synthetic ergocalciferol analog, treats secondary hyperparathyroidism, inhibits parathyroid.
Formule :C₂₈H₄₄O₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :412.65
Ref: TM-T19370
+ Info
Sulotroban potassium
Sulotroban potassium is a small molecule thromboxane A2 receptor (TXA2R) antagonist that can be used to study myocardial infarction and thrombosis.
Formule :C₁₆H₁₆KNO₅S
Degré de pureté :98.02%
Couleur et forme :Soild
Masse moléculaire :373.46
Ref: TM-T68022L
+ Info
Mono(5-carboxy-2-ethylpentyl) phthalate
CAS :
- 40809-41-4
MECPP is a metabolite of DEHP, a major plasticizer used in flexible PVC.
Formule :C₁₆H₂₀O₆
Couleur et forme :Solid
Masse moléculaire :308.33
Ref: TM-T74011
+ Info
Crotonyl-CoA tetrasodium
Crotonyl-CoA tetrasodium is the tetrasodium salt form of Crotonyl-CoA. It serves as an intermediate in butyrate fermentation and in the metabolism of lysine and tryptophan. This compound plays a crucial role in the metabolism of fatty acids and amino acids.
Formule :C₂₅H₃₆N₇Na₄O₁₇P₃S
Couleur et forme :Solid
Masse moléculaire :923.54
Ref: TM-T201796
+ Info
Naphthol AS-GR phosphate disodium
CAS :
- 100929-51-9
Naphthol AS-GR phosphate disodium: intense green fluorescent probe for phosphatases in histochemistry.
Formule :C₂₂H₁₆NNa₂O₅P
Couleur et forme :Solid
Masse moléculaire :451.32
Ref: TM-T75366
+ Info
Acetate kinase (ACK)
CAS :
- 9027-42-3
ACK, found in bacteria/archaea, phosphorylates acetate with ATP and cations, yielding acetyl-CoA; used in biochemistry.
Couleur et forme :Solid
Ref: TM-T76140
+ Info
Aculene D
CAS :
- 2043948-38-3
Aculene D, a fungal metabolite, inhibits quorum sensing in C. violaceum CV026, reducing violacein at low concentrations.
Formule :C₁₄H₂₀O₂
Couleur et forme :Solid
Masse moléculaire :220.31
Ref: TM-T75448
+ Info
Clervonafusp alfa
CAS :
- 2145123-44-8
Clervonafusp alfa (VAL-1221) is a fusion protein for Pompe disease, targeting glycogen in cytosol and lysosomes.
Couleur et forme :Liquid
Ref: TM-T77131
+ Info
ACAT-IN-7
CAS :
- 199984-38-8
ACAT-IN-7 inhibits ACAT enzyme; blocks NF-κB mediated transcription.
Formule :C₃₂H₄₉N₃O₅S
Couleur et forme :Solid
Masse moléculaire :587.82
Ref: TM-T39414
+ Info
HIV-IN-7
Axl-IN-16 (Compound 4), an Axl inhibitor, not only suppresses Axl expression and HIF activity but also triggers fruiting body formation in Flammulina velutipes.
Formule :C₃₂H₆₁N₃O₁₀P₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :709.79
Ref: TM-T78834
+ Info
LYP-IN-4
LYP-IN-4 (compound D14), a reversible and selective lymphotyrosine phosphatase (LYP) inhibitor (Ki=1.34 μM, IC50=3.52μM), regulates TCR signaling, increases PD-
Formule :C₂₉H₂₁ClN₂O₈S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :593
Ref: TM-T79635
+ Info
Kahalalide A
CAS :
- 179733-11-0
Kahalalide A has antimycobacterial activity isolated from the mollusk Elysia rufescens.
Formule :C₄₆H₆₇N₇O₁₁
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :894.08
Ref: TM-T25565
+ Info
Sethoxydim
CAS :
- 74051-80-2
Sethoxydim is an effective herbicide.
Formule :C₁₇H₂₉NO₃S
Couleur et forme :Oily Liquid Sethoxydim Is An Oily Odorless Liquid Non Corrosive Used As An Herbicide
Masse moléculaire :327.48
Ref: TM-T21228
+ Info
1-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine
CAS :
- 76343-22-1
Endogenous metabolite: 1-myristoyl-2-stearoyl-sn-glycero-3-phosphocholine, a phosphatidylcholine example.
Formule :C₄₀H₈₀NO₈P
Degré de pureté :99.23%
Couleur et forme :Solid
Masse moléculaire :734.04
Ref: TM-T10022
+ Info
α-Glucosidase-IN-31
α-Glucosidase-IN-31 (compound R1) is a potent oral α-Glucosidase inhibitor with an IC50 of 10.1 μM, demonstrating significant blood glucose reduction and
Formule :C₁₈H₁₈N₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :290.36
Ref: TM-T78794
+ Info
Acivicin
CAS :
- 42228-92-2
Acivicin (AT-125) is a chlorinated amino acid antibiotic produced by Streptomyces porcineus, a GGT inhibitor with anticancer and antiparasitic activity.
Formule :C₅H₇ClN₂O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :178.57
Ref: TM-T14114
+ Info
HIF-1 α (556-574) (TFA)
HIF-1 alpha (556-574) TFA is a 19-residue fragment of hypoxia-inducible factor-1 (HIF-1), which serves as the master regulator of oxygen homeostasis [1].
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T82199
+ Info
Burnettramic Acid A aglycone
CAS :
- 2396676-46-1
Burnettramic acid A aglycone, from A. burnettii, has anticancer properties; cytotoxic to NS-1 cells (IC50 = 8.4 μg/ml), not to fibroblasts (>100 μg/ml).
Formule :C₃₅H₆₁NO₇
Couleur et forme :Solid
Masse moléculaire :607.873
Ref: TM-T36337
+ Info
1-Palmitoyl Lysophosphatidic Acid (sodium salt)
CAS :
- 17618-08-5
1-Palmitoyl LPA: a palmitic acid-containing LPA analog, targets GPCRs, affects cell responses, and boosts β-lactam antibiotics against Pseudomonas aeruginosa.
Formule :C₁₉H₃₈NaO₇P
Couleur et forme :Solid
Masse moléculaire :432.46
Ref: TM-T37283
+ Info
Bifenazate-diazene
CAS :
- 149878-40-0
Bifenazate-diazene, a significant degradation product of Bifenazate, is characterized as a selective carbazate acaricide and insecticide [1].
Formule :C₁₇H₁₈N₂O₃
Couleur et forme :Solid
Masse moléculaire :298.34
Ref: TM-T73723
+ Info
9-PAHSA
CAS :
- 1481636-31-0
FAHFAs, fats linked with insulin sensitivity, are altered by diet and fasting. Most common in AG4OX mice, 9-PAHSA is key, reduced in insulin-resistant humans.
Formule :C₃₄H₆₆O₄
Couleur et forme :Solid
Masse moléculaire :538.898
Ref: TM-T36590
+ Info
Mevalonic acid 5-pyrophosphate tetralithium
CAS :
- 108869-00-7
Mevalonic acid 5-pyrophosphate (also known as 5-Diphosphomevalonic acid) tetralithium is an endogenous metabolite involved in the mevalonate pathway.
Formule :C₆H₁₀Li₄O₁₀P₂
Couleur et forme :Solid
Masse moléculaire :331.85
Ref: TM-T38478
+ Info
HIF1-IN-3
CAS :
- 333314-79-7
HIF1-IN-3 (Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-) is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in
Formule :C₂₆H₂₄N₂O₃
Degré de pureté :99.59%
Couleur et forme :Solid
Masse moléculaire :412.48
Ref: TM-T9890
+ Info
Micafungin metabolite M1
CAS :
- 539823-80-8
Micafungin metabolite M1 is an active metabolite of Micafungin, generated through metabolism by arylsulfatase, and exhibits antifungal activity. It can be utilized in research on deep fungal infections caused by Candida species (Candidiasis) and Aspergillus species (Aspergillosis).
Formule :C₅₆H₇₁N₉O₂₀
Couleur et forme :Solid
Masse moléculaire :1190.21
Ref: TM-TP3139
+ Info
L-Isoleucyl-L-arginine
CAS :
- 55715-01-0
L-Isoleucyl-L-arginine, a dipeptide composed of L-isoleucine and L-arginine, acts as a potent angiotensin-converting enzyme (ACE) inhibitor and is utilized in
Formule :C₁₂H₂₅N₅O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :287.36
Ref: TM-T80096
+ Info
α-Glucosidase-IN-32
α-Glucosidase-IN-32 (compound f26) is a reversible, noncompetitive inhibitor of α-glucosidase that is orally active and exhibits an IC50 of 3.07 μM.
Formule :C₃₂H₂₂N₄OS
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :510.61
Ref: TM-T79700
+ Info
(S)-3-Thienylglycine
CAS :
- 1194-87-2
(S)-3-Thienylglycine is a thiophene derivative and can be used to investigate the genotoxicity of the similar structures with thiophene derivatives.
Formule :C₆H₇NO₂S
Degré de pureté :99.68%
Couleur et forme :Solid
Masse moléculaire :157.19
Ref: TM-T38311
+ Info
Angiotensin 1/2 (1-9)
CAS :
- 34273-12-6
Angiotensin 1/2 (1-9) is containing the amino acids 1-9 that are converted from Angiotensin I/II peptide.
Formule :C₅₆H₇₈N₁₆O₁₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1183.32
Ref: TM-T7663
+ Info
Forrestiacids K
CAS :
- 2920898-65-1
Forrestiacid K, a terpenoid derived from Pseudotsuga forrestii, functions as an inhibitor of ATP-citrate lyase (ACL) [1].
Formule :C₅₀H₇₄O₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :771.12
Ref: TM-T79936
+ Info
Hippadine
CAS :
- 52886-06-3
Hippadine is isolated from Crinum bulbs and has reproductive effect.
Formule :C₁₆H₉NO₃
Couleur et forme :Solid
Masse moléculaire :263.25
Ref: TM-T32076
+ Info
Xanthine oxidase-IN-16
Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.
Couleur et forme :Odour Solid
Ref: TM-T200654
+ Info
SB-435495 ditartrate
CAS :
- 304694-43-7
SB-435495 ditartrate is a potent, selective, reversible, non-covalent, and orally active inhibitor of Lp-PLA2, demonstrating an IC50 value of 0.06 nM [1] [3].
Formule :C₄₆H₅₂F₄N₆O₁₄S
Couleur et forme :Solid
Masse moléculaire :1020.99
Ref: TM-T75255L1
+ Info
Glutamate dehydrogenase (NAD(P))
CAS :
- 9029-12-3
GLDH, found in liver/kidney/brain/muscle/intestine, catalyzes glutamate to α-KG in urea cycle.
Couleur et forme :Solid
Ref: TM-T73616
+ Info
Plipastatin B 1
CAS :
- 103955-73-3
Plipastatin B 1 is a lipopeptide.
Formule :C₇₄H₁₁₄N₁₂O₂₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1491.79
Ref: TM-TP2467
+ Info
Pepsin A
CAS :
- 9001-75-6
Pepsin A is a protease and endopeptidase in the stomach, capable of breaking down proteins in food into small peptide fragments.
Couleur et forme :Solid
Ref: TM-T75993
+ Info
MK-8262
CAS :
- 1432054-03-9
MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.
Formule :C₃₅H₂₅F₉N₂O₅
Couleur et forme :Solid
Masse moléculaire :724.58
Ref: TM-T38908
+ Info
EDDA
CAS :
- 5657-17-0
Ethylenediaminediacetic acid is derived from two molecules of glycine linked by amines.
Formule :C₆H₁₂N₂O₄
Couleur et forme :Solid
Masse moléculaire :176.17
Ref: TM-T21207
+ Info
Glycogen phosphorylase-IN-2
Glycogen phosphorylase-IN-2 (compound 9C) is an inhibitor of glycogen phosphorylase, with a Ki value of 1.9 nM and an IC50 value of 4 nM.
Couleur et forme :Odour Solid
Ref: TM-T206787
+ Info
hCAIX/XII-IN-14
hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.
Formule :C₁₆H₁₄F₃N₃O₄S
Couleur et forme :Solid
Masse moléculaire :401.36
Ref: TM-T205536
+ Info
IOX2-NH2-1
CAS :
- 931400-77-0
IOX2-NH2-1 inhibits E. coli EGLN-3 (prolyl hydroxylase) with an IC50 of 0.02–1 μM.
Formule :C₁₉H₁₇N₃O₅
Degré de pureté :98.77% - 99.91%
Couleur et forme :Soild
Masse moléculaire :367.36
Ref: TM-T205895
+ Info
D-threo-PPMP
CAS :
- 139889-53-5
D-threo-PPMP, a powerful glucosylceramide (GlcCer) synthase inhibitor, effectively impedes karyokinesis and decreases cyst formation.
Formule :C₂₉H₅₀N₂O₃
Couleur et forme :Solid
Masse moléculaire :474.73
Ref: TM-T38822
+ Info
ER 50891 quarterhydrate
ER 50891 quarterhydrate is a potent RARα (retinoic acid receptor α) antagonist that markedly diminishes the inhibitory effects of ATRA (all-trans retinoic acid
Formule :C₂₉H₂₄N₂O₂H₂O
Couleur et forme :Solid
Masse moléculaire :437.02
Ref: TM-T78102
+ Info
MEY-003
MEY-003, an Autotaxin (ATX) inhibitor, exhibits EC50 values of 460 nM for hATX-β and 1.09 μM for hATX-ɣ (analysis with LPC18:1), demonstrating its potency
Couleur et forme :Odour Solid
Ref: TM-T81804
+ Info
N-Desmethyl imatinib mesylate
CAS :
- 404844-03-7
Norimatinib mesylate, N-Desmethyl imatinib metabolite, inhibits v-Abl, c-Kit, PDGFR.
Formule :C₂₉H₃₃N₇O₄S
Couleur et forme :Solid
Masse moléculaire :575.68
Ref: TM-T40504
+ Info
MU1742
MU1742 is a probe for CK1δ and CK1ε protein kinases [1] .
Formule :C₂₂H₂₂F₂N₆
Couleur et forme :Solid
Masse moléculaire :408.45
Ref: TM-T74661
+ Info
Inulobiose
CAS :
- 470-58-6
Inulobiose, a difructan disaccharide isolated from Pistacia vera L., demonstrates inhibitory effects on α-glycosidase (α-glycosidase) and α-amylase (α-amylase) activities, with IC50 values of 1.87 and 40.72 mg/mL respectively. It is utilized in research related to diabetes and glomerular filtration rate testing.
Formule :C₁₂H₂₂O₁₁
Couleur et forme :Solid
Masse moléculaire :342.3
Ref: TM-TN8319
+ Info
10'-Desmethoxystreptonigrin
CAS :
- 136803-89-9
'10'-Desmethoxystreptonigrin antibiotic derived from streptonigrin combats various bacteria and cancer cells, and inhibits p21ras farnesylation (IC50 = 21 nM).
Formule :C₂₄H₂₀N₄O₇
Couleur et forme :Solid
Masse moléculaire :476.445
Ref: TM-T35607
+ Info
Reticulol
CAS :
- 26246-41-3
Reticulol is an isocoumarin derivative produced by certain species of Streptomyces.
Formule :C₁₁H₁₀O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :222.19
Ref: TM-T28522
+ Info
6-Keto Cholestanol
CAS :
- 1175-06-0
6-Keto Cholestanol is a useful organic compound for research related to life sciences. The catalog number is T126283 and the CAS number is 1175-06-0.
Formule :C₂₇H₄₆O₂
Couleur et forme :Solid
Masse moléculaire :402.663
Ref: TM-T126283
+ Info
DSPE-PEG1000-M2pep
DSPE-PEG1000-M2pep is a PEG compound comprised of DSPE and the M2 macrophage-targeting peptide (M2pep). M2pep acts as a mono- or multivalent ligand conjugated with pro-apoptotic peptides to focus the peptides' toxic effects on M2 macrophages. DSPE-PEG1000-M2pep can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01148
+ Info
PDE4-IN-3
CAS :
- 2755687-49-9
PDE4-IN-3, a new oral drug, potently blocks PDE4 enzyme with 4.2 nM IC50.
Formule :C₃₅H₃₃FO₈
Couleur et forme :Solid
Masse moléculaire :600.639
Ref: TM-T40356
+ Info
Laccase-IN-1
Laccase-IN-1 (compound 4b) is an orally active laccase inhibitor, demonstrating an IC50 of 11.3 μM.
Formule :C₁₆H₁₉FN₂O₃
Couleur et forme :Solid
Masse moléculaire :306.33
Ref: TM-T78899
+ Info
Dactylocycline A
CAS :
- 125622-12-0
Dactylocyclines A: novel antibiotic from Dactylosporangium, effective against tetracycline-resistant microbes.
Formule :C₃₁H₄₀ClN₃O₁₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :698.11
Ref: TM-T23956
+ Info
1-Palmitoyl-2-Oleoyl-3-Arachidonoyl-rac-glycerol
CAS :
- 675876-04-7
Triacylglycerol with palmitic, oleic, arachidonic acids at sn-1, sn-2, sn-3; found in rat retina lipid extracts.
Formule :C₅₇H₁₀₀O₆
Couleur et forme :Solid
Masse moléculaire :881.421
Ref: TM-T38216
+ Info
TAK-778
CAS :
- 180185-61-9
TAK-778, a derivative of ipriflavone, demonstrates the ability to stimulate bone growth in both in vitro and in vivo models.
Formule :C₂₄H₂₈NO₇PS
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :505.52
Ref: TM-T13913
+ Info
Curcumin monoglucuronide
CAS :
- 2171091-50-0
Curcumin monoglucuronide, curcumin's in vivo metabolite, useful for metabolic research and cancer study.
Formule :C₂₇H₂₈O₁₂
Couleur et forme :Solid
Masse moléculaire :544.50
Ref: TM-T74279
+ Info
18:0,22:6 PS sodium
CAS :
- 474943-18-5
Sodium 18:0,22:6 phosphatidylserine (PS) is a lipid found within synaptic vesicles alongside cholesterol, utilized in metabolic research [1].
Formule :C₄₆H₇₇NNaO₁₀P
Couleur et forme :Solid
Masse moléculaire :858.07
Ref: TM-T74758
+ Info
Diadenosine pentaphosphate pentaammonium
CAS :
- 102783-61-9
Endogenous vasoactive dinucleotide isolated from thrombocytes; found in secretory vesicles across various cells.
Formule :C₂₀H₄₄N₁₅O₂₂P₅
Couleur et forme :Solid
Masse moléculaire :1001.524
Ref: TM-T37309