Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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Ninopterin
CAS :<p>Ninopterin is an experimental antineoplastic and folic acid analog.</p>Formule :C20H21N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.42NPE-caged-proton
CAS :<p>Generates rapid acidifications down to pH 2</p>Formule :C8H9NNaO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.225,7-Dichloropyrazolo[1,5-a]pyrimidine
CAS :<p>5,7-Dichloropyrazolo[1,5-a]pyrimidine (fragment 5) is an inhibitor of the enzyme phosphodiesterase 10A (PDE10A) with a Ki value of 24 μM. This compound can be employed in research related to schizophrenia.</p>Formule :C6H3Cl2N3Couleur et forme :SolidMasse moléculaire :188.01Fibrostatin C
CAS :<p>Fibrostatin C is an inhibitor of prolyl 4-hydroxylase. It is produced by Streptomyces catenulae subsp.</p>Formule :C18H19NO8SCouleur et forme :SolidMasse moléculaire :409.41Muvalaplin tetrahydrochloride
CAS :<p>Muvalaplin tetrahydrochloride (LY3473329) is an orally active lipoprotein (a)Lp(a) agent currently under investigation. Research on the oral formulation of Muvalaplin tetrahydrochloride is ongoing.</p>Formule :C42H58Cl4N4O6Couleur et forme :SolidMasse moléculaire :856.75Dactylocycline A
CAS :<p>Dactylocyclines A: novel antibiotic from Dactylosporangium, effective against tetracycline-resistant microbes.</p>Formule :C31H40ClN3O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :698.11SHP2-IN-34
CAS :<p>SHP2-IN-34 (compound A8) is a phenylurea SHP2 inhibitor with anti-cancer properties. It significantly suppresses tumor growth in CT26 mouse models.</p>Formule :C23H25Cl2N7OSCouleur et forme :SolidMasse moléculaire :518.46Rubratoxin B
CAS :<p>Rubratoxin B is a mycotoxin that causes hypoglycemia and fatty liver and has exhibited anticancer activity.</p>Formule :C26H30O11Degré de pureté :98%Couleur et forme :Long Lathes; Hexagonal Plates From Amyl Acetate SolidMasse moléculaire :518.511,3-Dipalmitoleoyl-rac-glycerol
CAS :<p>1,3-Dipalmitoleoyl-rac-glycerol: a diacylglycerol inhibiting yeast α-glucosidase over rat's (IC50s: 4.45 vs 9326.5 μM). Used to study membrane potentials.</p>Formule :C35H64O5Couleur et forme :SolidMasse moléculaire :564.892Methylbenzethonium chloride hydrate
CAS :<p>Methylbenzethonium chloride hydrate exhibits broad-spectrum antimicrobial activity against bacteria, viruses, and fungi. Additionally, it is utilized as a preservative in cosmetics and pharmaceutical formulations to inhibit microbial growth.</p>Formule :C28H46ClNO3Couleur et forme :SolidMasse moléculaire :480.12Etodolac Acyl Glucuronide
CAS :<p>Etodolac acyl glucuronide is an NSAID metabolite formed by UGT1A9, UGT1A10, and UGT2B7 glucuronidation.</p>Formule :C23H29NO9Couleur et forme :SolidMasse moléculaire :463.483Edoxaban impurity 6
CAS :<p>Edoxaban impurity 6 is a byproduct of the anticoagulant Edoxaban, a potent oral factor Xa inhibitor with Kis of 0.561 nM. Used to prevent stroke.</p>Formule :C16H22ClN5O3Couleur et forme :SolidMasse moléculaire :367.83Acrihellin
CAS :<p>Acrihellin is a cardioactive steroid, a cardiotonic drug.</p>Formule :C29H38O7Couleur et forme :SolidMasse moléculaire :498.61Aspergillomarasmine A
CAS :<p>Aspergillomarasmine A is a polyamine acid naturally produced by the mold Aspergillus Versicolor.</p>Formule :C10H17N3O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.262,3-Indolobetulonic Acid
CAS :<p>2,3-Indolobetulonic acid is pentacyclic triterpenoid derivative of betulonic acid and an inhibitor of α-glucosidase (IC50= 1.8 μM).1</p>Formule :C36H49NO2Couleur et forme :SolidMasse moléculaire :527.793Liarozole fumarate
CAS :<p>Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.</p>Formule :C17H13ClN4C4H4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.88Dilaurylglycerosulfate
CAS :<p>Dilauryl glycerol sulfate is an auxiliary emulsifier for lipase determination.</p>Formule :C27H56O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.8(Iso)-Dehydroemetine
CAS :<p>(Iso)-Dehydroemetine (Dehydroisoemetine, (+/-)-) is a compound with antispasmolytic effect on smooth muscle.</p>Formule :C29H38N2O4Degré de pureté :98.26% - 98.31%Couleur et forme :SoildMasse moléculaire :478.62Meproscillarin
CAS :<p>Meproscillarin is a glycoside with high bioavailability (about 70%) and an elimination independent of renal function.</p>Formule :C31H44O8Couleur et forme :SolidMasse moléculaire :544.68(±)7(8)-EpDTE
CAS :<p>(±)7(8)-EpDTE is an oxylipin and an oxidative metabolite of docosapentaenoic acid .</p>Formule :C22H34O3Couleur et forme :SolidMasse moléculaire :346.511MeIQx
CAS :<p>MeIQx, a carcinogenic compound in cooked fish/meat, triggers DNA-reactive metabolites and rat tumors.</p>Formule :C11H11N5Couleur et forme :SolidMasse moléculaire :213.244TNAP-IN-1
CAS :<p>TNAP-IN-1 is a specific inhibitor of tissue-nonspecific alkaline phosphatase (TNAP) and is utilized in studying diseases related to soft tissue calcification.</p>Formule :C17H16N2O4SDegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :344.393'-sulfo Galactosylsphingosine (ammonium salt)
CAS :<p>Sulfatide derivative inhibits cell migration, adhesion, PKC, cytochrome c; accumulates in metachromatic leukodystrophy; used for LC-MS quantification.</p>Formule :C24H50N2O10SCouleur et forme :SolidMasse moléculaire :558.731-Pentadecanoyl-rac-glycerol
CAS :<p>1-Pentadecanoyl-rac-glycerol: a monoacylglycerol with sn-1 pentadecanoic acid, found in wheat bran, rises in fatty liver models.</p>Formule :C18H36O4Couleur et forme :SolidMasse moléculaire :316.482Mead acid
CAS :<p>Mead acid, a 5,8,11-Eicosatrienoic Omega-9 unsaturated fatty acid, signals essential fatty acid deficiency.</p>Formule :C20H34O2Couleur et forme :SolidMasse moléculaire :306.49Lead Ionophore IV
CAS :<p>Lead Ionophore IV, an ion carrier, actively facilitates the transport of metal ions. It is commonly utilized in biological research to investigate the biological effects of lead ions and their impact on cellular functions. Additionally, Lead Ionophore IV is employed in developing drug delivery systems to enhance the bioavailability of compounds.</p>Formule :C60H84N4O4S4Couleur et forme :SolidMasse moléculaire :1053.59O-Desethyl Sildenafil
CAS :<p>O-Desethyl sildenafil is a metabolite of the phosphodiesterase 5 (PDE5) inhibitor sildenafil .1</p>Formule :C20H26N6O4SCouleur et forme :SolidMasse moléculaire :446.53H-Tyr-Ala-OH
CAS :<p>Tyrosylalanine (H-Tyr-Ala-OH), a dipeptide comprising L-tyrosine and L-alanine, is referenced in studies [1] [2].</p>Formule :C12H16N2O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :252.27Prenisteine
CAS :<p>Prenisteine is a bioactive chemical.</p>Formule :C8H15NO2SCouleur et forme :SolidMasse moléculaire :189.2752,3,4,5-Tetrachlorophenol
CAS :<p>2,3,4,5-Tetrachlorophenol, a γ-lindane byproduct, is toxic to minnows, trout (LC50: 0.496, 0.304 mg/L).</p>Formule :C6H2Cl4OCouleur et forme :SolidMasse moléculaire :231.88Mesembrenone
CAS :<p>Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum.</p>Formule :C17H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.35Leukotriene C4 methyl ester
CAS :<p>LTC4, made by neutrophils and others via LTC4 synthase, causes smooth muscle contractions and is involved in asthma/allergic responses.</p>Formule :C31H49N3O9SCouleur et forme :SolidMasse moléculaire :639.81Sandosaponin A
CAS :<p>Sandosaponin A, an olean-12-ene-type triterpene oligoglycoside, is isolated from kidney bean, the seed of Phaseolus vulgaris L.</p>Formule :C48H76O19Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :957.11Leukotriene B3
CAS :<p>LTB3, a LTA3-derived leukotriene, matches LTB4's inflammation effect but is 5x weaker in neutrophil chemotaxis.</p>Formule :C20H34O4Couleur et forme :SolidMasse moléculaire :338.488Nodularin
CAS :<p>Nodularin from N. spumigena is a hepatotoxic pentapeptide that inhibits PP1 and PP2A with IC50s of 1.8 nM and 0.026 nM, respectively.</p>Formule :C41H60N8O10Couleur et forme :SolidMasse moléculaire :824.977Deaminocozymase
CAS :<p>Deaminocozymase also known as Nicotinamide-hypoxanthine dinucleotide, is a biochemical.</p>Formule :C21H26N6O15P2Couleur et forme :SolidMasse moléculaire :664.414Sphingomyelins (buttermilk)
CAS :<p>Sphingomyelins, 2-15% of organ phospholipids, are prevalent in brain and nerve sheaths, regulate cholesterol, and turn into ceramides by hydrolysis.</p>Formule :C46H93N2O6P(fortricosanoyl)Couleur et forme :SolidMasse moléculaire :801.2D-γ-Glutamyl-D-glutamic acid
CAS :D-γ-Glutamyl-D-glutamic acid is a linear polymer with repeating D-glutamic acid units, useful in studies of microbial cell walls and immunological recognition.Formule :C10H16N2O7Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :276.24Casein Kinase Substrates 3
CAS :<p>Casein Kinase Substrates 3 is a substrate of casein kinase.</p>Formule :C85H139N27O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2131.24isomer-CM 352
CAS :<p>isomer-CM 352 is a metalase inhibitor that can be used to slow brain damage.</p>Formule :C24H29N3O6SDegré de pureté :99.65%Couleur et forme :SoildMasse moléculaire :487.57Myxochelin A
CAS :<p>Myxochelin A from A. disciformis fights Gram-positive bacteria, inhibits 5-LO with IC50 of 1.9 μM, and is cytotoxic to colon cancer cells.</p>Formule :C20H24N2O7Couleur et forme :SolidMasse moléculaire :404.419Acremin F
CAS :<p>Acremin F is a useful organic compound for research related to life sciences. The catalog number is T124074 and the CAS number is 863480-61-9.</p>Formule :C12H20O4Couleur et forme :SolidMasse moléculaire :228.288Isariin C
CAS :<p>Isariin C is a flavonoid glucoside derived from the Epimedium plant genus. It stimulates angiogenesis and exhibits antioxidant activity.</p>Formule :C28H49N5O7Couleur et forme :SolidMasse moléculaire :567.72Moth Cytochrome C (MCC) (88-103)
CAS :<p>Moth Cytochrome C (88-103) peptide induces positive TCR selection in thymocytes; key for self-tolerant T cell development.</p>Formule :C79H133N23O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1805.04Mefox
CAS :<p>Mefox is a bioactive chemical.</p>Formule :C20H23N7O7Couleur et forme :SolidMasse moléculaire :473.44AY 9944 dihydrochloride
CAS :<p>AY 9944 dihydrochloride is a intermediate.</p>Formule :C22H30Cl4N2Degré de pureté :99.22% - 99.82%Couleur et forme :SoildMasse moléculaire :464.3C22 Galactosylceramide (d18:1/22:0)
CAS :<p>C22 Galactosylceramide, a CNS sphingolipid, rises in mouse spinal cord on a methionine-restricted diet, found in Alzheimer's hippocampus.</p>Formule :C46H89NO8Couleur et forme :SolidMasse moléculaire :784.20Pancreatic lipase-IN-2
Pancreatic lipase-IN-2 (compound 7r) is a potent inhibitor of pancreatic lipase (PL), with an IC50 value of 2.67 μM, and exhibits anti-obesity effects.Formule :C32H33N3O2SMasse moléculaire :523.22935Mannose 6 phosphate
CAS :Mannose 6-phosphate (M6P) features a type I integral membrane receptor.Formule :C6H13O9PMasse moléculaire :260.14Benzoyl coenzyme A sodium
Benzoyl coenzyme A (sodium) is the sodium salt form of Benzoyl coenzyme A. It is a derivative of coenzyme A (CoA), where the thiol group of CoA is linked to a benzoyl group. This compound serves as a substrate in acyl transfer reactions, playing a role in catalysis. Benzoyl coenzyme A (sodium) is a versatile metabolic intermediate used in studies exploring enzyme substrate specificity, metabolic regulation, and drug metabolism.Formule :C28H39N7NaO17P3SMasse moléculaire :893.12337Arginase
CAS :<p>Arginase (L-Arginine amidinase) is a key hydrolytic enzyme in the urea cycle, which hydrolyzes L-arginine into urea and L-ornithine.</p>Couleur et forme :SolidCreatine Kinase (CPK/CK), Bovine Heart
Creatine Kinase (CPK/CK), Bovine Heart (CK, CPK, Creatine Phosphokinase), is a biological material or organic compound suitable for use in life sciences research.ASP8477
CAS :ASP8477 is a potent and selective FAAH inhibitor. It increases anandamide levels in the brain when administered orally. In rat models of neuropathic and osteoarthritic pain, ASP8477 demonstrates significant efficacy without causing motor coordination issues. A single oral dose of ASP8477 improves thermal hyperalgesia and cold allodynia in rats with chronic constriction nerve injury. Moreover, ASP8477 restores the decreased muscle pressure threshold in a myalgia model induced by reserpine. Research indicates that ASP8477 possesses analgesic effects effective for alleviating neuropathic and functional pain, making its pharmacological properties suitable for chronic pain treatment.Formule :C18H19N3O3Masse moléculaire :325.36(Rac)-BMS-816336
<p>(Rac)-BMS-816336 is a racemic 11β-HSD1 inhibitor; IC50: 10 nM (human), 68 nM (mouse), metabolically stable.</p>Formule :C21H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.44Ferroleuton
<p>Ferroleuton is a selective competitive inhibitor of 5-lipoxygenase with an IC50 of 0.21 μM. It demonstrates antioxidant properties, clearing 86% of DPPH at 50 μM and exhibiting activities in ABTS (EC50 = 19.42 μM) and FRAP (EC50 = 3.32 μM) assays.</p>Formule :C13H16FeN2O2Couleur et forme :SolidMasse moléculaire :288.12GPX4-IN-16
<p>GPX4-IN-16 ((R)-9i) is a potent inhibitor of GPX4 with a KD value of 20.4 nM, exhibiting cytotoxic properties and anticancer activity.</p>Formule :C29H24N4O3S2Couleur et forme :SolidMasse moléculaire :540.656Calcium Channel antagonist 3
CAS :<p>Calcium Channel antagonist 3 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formule :C23H26N2O4SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :426.53Calcium Channel antagonist 2
CAS :<p>Calcium Channel antagonist 2 is a calcium channel antagonist (IC50=5-20 μM) that can be used to study diseases due to Ca2+ channels like pain and diabetes.</p>Formule :C23H25FN2O4SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :444.52MAGL-IN-21
<p>MAGL-IN-21 (Compound (S)-6) is a selective inhibitor of monoacylglycerol lipase (MAGL) with an IC50 of 1.59 nM.</p>Formule :C20H24ClFN2O4Couleur et forme :SolidMasse moléculaire :410.8674-Hydroxy Atorvastatin calcium salt
CAS :<p>4-Hydroxy Atorvastatin calcium salt is metabolised by cytochrome P450 CYP3A4 and has antimicrobial and anti-microbial activity.</p>Formule :C66H68CaF2N4O12Couleur et forme :SolidMasse moléculaire :1187.34α-Glucosidase-IN-82
<p>α-Glucosidase-IN-82 (compound 8l) is a potent inhibitor of α-glucosidase, with an IC50 value of 13.66 μM. Its inhibitory activity is 52 times greater than that of Acarbose.</p>Formule :C30H24N4O4Couleur et forme :SolidMasse moléculaire :504.536CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Formule :C19H16ClN3O5S2Couleur et forme :SolidMasse moléculaire :465.93JTV-519 Formate
<p>JTV-519 Formate is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA).</p>Formule :C26H34N2O4SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :470.62CA Ⅱ-IN-1
<p>CAⅡ-IN-1 (compound 2i) is an inhibitor of the CA Ⅱ isozyme, exhibiting an IC50 of 0.44 µM. This compound is utilized in metabolic research.</p>Formule :C18H19NO6SCouleur et forme :SolidMasse moléculaire :377.41ZG-2305
<p>ZG-2305 is an effective, selective, and orally active inhibitor of FIH (factor inhibiting hypoxia-inducible factor (FIH)), with Ki values of 79.6 nM for FIH and 2786 nM for PHD2. This compound enhances the expression of the EGLN3 gene, reduces cellular triglyceride levels, and decreases lipid accumulation. ZG-2305 holds potential for research into obesity and fatty liver disease.</p>Formule :C17H11Cl2N3O5Couleur et forme :SolidMasse moléculaire :408.19IR-117-17
CAS :<p>IR-117-17 is an ionizable cationic amino lipid that targets the airways. It is degradable via esterase cleavage, making it less likely to accumulate with repeated dosing.</p>Formule :C59H110N2O5Couleur et forme :SolidMasse moléculaire :927.52Pregnenolone Carbonitrile
CAS :<p>Pregnenolone Carbonitrile (5-Pregnen-3β-ol-20-one-16α-carbonitrile) is an activator of rodent-PXR and induces the expression of CYP3A.</p>Formule :C22H31NO2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :341.49Bendroflumethiazide
CAS :<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Formule :C15H14F3N3O4S2Degré de pureté :98% - >99.99%Couleur et forme :Crystals From Dioxane SolidMasse moléculaire :421.41Human Endogenous Metabolite Library
<p>A collection of xnum selected human endogenous metabolites for high throughput and high content screening.</p>Couleur et forme :Odour SolidLactosylsphingosine (d18:1)
CAS :<p>Lactosylsphingosine (d18:1) is a sphingolipid with a lactose moiety that can inhibit fMetLeuPhe-induced cell aggregation at a concentration of 1 μm.</p>Formule :C30H57NO12Couleur et forme :SolidMasse moléculaire :623.77N-Lactoyl-Tyrosine
CAS :<p>N-Lactoyl-Tyrosine is an amino acid derivative and endogenous metabolite, widely used in biochemical experiments and drug synthesis research.</p>Formule :C12H15NO5Degré de pureté :99.59%Couleur et forme :SoildMasse moléculaire :253.25HIF1-IN-3
CAS :<p>HIF1-IN-3 (Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-) is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in</p>Formule :C26H24N2O3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :412.4816α-hydroxy Dehydroepiandrosterone
CAS :<p>16α-hydroxy Dehydroepiandrosterone (16α-OH-DHEA) is a neurosteroid found in the brain and a precursor in the biosynthesis of placental estriol.</p>Formule :C19H28O3Couleur et forme :SolidMasse moléculaire :304.42Orotidine
CAS :<p>Orotidine (Uridin-6-carboxylic acid) is a nucleoside found in bacteria, fungi, and plants. In humans, orotidine occurs as its 5'-phosphate (orotidylic acid).</p>Formule :C10H12N2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.21SW209049
CAS :<p>SW209049 is a stearoyl-CoA 9-desaturase inhibitor. SW209049 exhivits potent activity against H2122 cell with IC50 of 0.13uM.</p>Formule :C25H18N2O4SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :442.49Catestatin acetate
<p>Catestatin acetate is a non-competitive antagonist of nAChR and inhibits catecholamine release.</p>Formule :C109H177N37O28SDegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :2485.87IPI-9119
CAS :<p>IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).</p>Formule :C24H19F2N5O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :495.43BC 11-38
CAS :<p>BC 11-38 is a potent, selective PDE biodepressant which is mainly effective against PDE11 (IC50 : 0.28 μM).</p>Formule :C15H16N2OS2Degré de pureté :98.95% - 99.28%Couleur et forme :SolidMasse moléculaire :304.43Lalistat 2
CAS :<p>Lalistat 2: selective lysosomal acid lipase inhibitor, IC50 152 nM, no effect on pancreatic/milk lipase <10 μM.</p>Formule :C13H20N4O2SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :296.39(Ile8)-Oxytocin acetate
<p>(Ile8)-Oxytocin acetate is a neurohypophysial hormone analog of oxytocin produced in marsupials.</p>Formule :C45H70N12O14S2Couleur et forme :SolidMasse moléculaire :1067.24SR-4995
CAS :<p>SR-4995 (CID 16016685) is an ABHD5 ligand, directly binding to ABHD5 and stimulating lipolysis by releasing it from PLIN.</p>Formule :C19H21N3O2SCouleur et forme :SoildMasse moléculaire :355.45α-glucosidase/PTP1B-IN-1
<p>α-glucosidase/PTP1B-IN-1 (compound 8a) is an effective inhibitor of both α-glucosidase and PTP1B, with IC50 values of 66.3 μM and 47.0 μM, respectively. It also exhibits strong inhibitory activity against α-amylase, having an IC50 of 30.62 μM. This compound is capable of binding to the active sites of α-glucosidase and PTP1B. α-glucosidase/PTP1B-IN-1 holds potential for reducing postprandial blood glucose levels and may be useful in managing type 2 diabetes.</p>Formule :C23H20Cl2O5Couleur et forme :SolidMasse moléculaire :447.31Lofacimig
<p>Lofacimig is a bispecific antibody of VH-VH-G1(h-CH2-CH3) dimer type that targets FXI/PTA.</p>Couleur et forme :Odour LiquidWVSAV
<p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>Formule :C27H40N6O7Couleur et forme :SolidMasse moléculaire :560.64CYP1B1-IN-7
CAS :<p>CYP1B1-IN-7 is a CYP1B1 inhibitor that can be used in synergy with anticancer compounds for the treatment of cancers.</p>Formule :C19H13ClODegré de pureté :99.49%Couleur et forme :SoildMasse moléculaire :292.76TC HSD 21
CAS :<p>TC HSD 21 is a potent and highly selective inhibitor of 17β-hydroxysteroid dehydrogenase type 3 (IC50 = 14 nM).</p>Formule :C17H12BrNO3S2Degré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :422.32Fmoc-L-Proline
CAS :<p>Fmoc-L-Proline (Fmoc-Pro-OH) is a proline derivative.</p>Formule :C20H19NO4Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :337.37GQ-16
CAS :<p>GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.</p>Formule :C19H16BrNO3SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :418.3BI 1015550
CAS :<p>Nerandomilast (BI 1015550) is an orally active PDE4B inhibitor with IC50 of 7.2 nM.Cost-effective and quality-assured.</p>Formule :C20H25ClN6O2SDegré de pureté :98.06% - 99.71%Couleur et forme :SoildMasse moléculaire :448.97α-Hydroxyglutaric Acid Lithium
<p>α-Hydroxyglutaric Acid Lithium is an α-ketoglutarate-dependent dioxygenase and 5-methylcytosine hydroxylase inhibitor of ATP synthase.</p>Formule :C5H6Li2O5Degré de pureté :≥98%Couleur et forme :SoildMasse moléculaire :159.98N-Lactoyl-Phenylalanine
CAS :<p>N-Lactoyl-Phenylalanine (Lac-Phe) is a peptide coupling of lactic acid and phenylalanine that can be used in the study of obesity and metabolic off diseases.</p>Formule :C12H15NO4Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :237.25L-739750 2HCl
<p>L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.</p>Formule :C23H41Cl2N3O6S2Degré de pureté :98.69% - 99.16%Couleur et forme :SoildMasse moléculaire :590.62MSNBA
CAS :MSNBA inhibits GLUT5 fructose uptake (KI: 3.2±0.4 μM) in MCF7 cells, serving as a potent GLUT5 probe.Formule :C14H12N2O6SDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :336.32Atagabalin HCl
CAS :<p>Atagabalin HCl is a novel voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) ligand that affects slow-wave sleep and can be used to treat insomnia.</p>Formule :C10H20ClNO2Degré de pureté :99.96% - ≥98%Couleur et forme :SoildMasse moléculaire :221.72BNTA
CAS :<p>BNTA is a potent extracellular matrix (ECM) modulator.</p>Formule :C17H11BrClNO3S2Degré de pureté :98.87% - 99.79%Couleur et forme :SolidMasse moléculaire :456.76α-Glucosidase-IN-22
CAS :<p>α-Glucosidase-IN-22 is a selective inhibitor of α-glucosidase (IC50=0.64 μM).</p>Formule :C14H11N3O2SDegré de pureté :99.66%Couleur et forme :SoildMasse moléculaire :285.32TMP-778
CAS :<p>TMP-778 is a selective inverse agonist of RORγt.</p>Formule :C31H30N2O4Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :494.58BAY 2666605
CAS :<p>BAY 2666605 is an orally active inhibitor of PDE3A and PDE3B with IC50s of 87 nM and 50 nM, respectively. BAY 2666605 has anticancer effects.</p>Formule :C17H12F4N2O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :352.28CAY10640
CAS :<p>CAY10640 (sEH inhibitor-1) is a potent, orally active, water-soluble epoxide hydrolase (sEH) inhibitor that inhibits sEH in humans and mice with IC50s of 0.4</p>Formule :C17H20F3N3O3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :371.35Isobutyryl-L-carnitine chloride
CAS :<p>Isobutyryl-L-carnitine chloride is a potential clinical OCT1 biomarker for DDI evaluation and can be used to study heart failure.</p>Formule :C11H22ClNO4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :267.75Nordoxepin hydrochloride
CAS :<p>Nordoxepin hydrochloride (Desmethyldoxepin hydrochloride) has antidepressant activity and is useful for studying depression and peptic ulcer disease.</p>Formule :C18H20ClNODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :301.81TDI-11055
<p>TDI-11055 is a chromatin reader 11-19 leukemia inhibitor and can be used to study acute myeloid leukemia (AML).</p>Formule :C22H24N6ODegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :388.47POPG sodium salt
CAS :<p>POPG sodium salt is a phospholipid and a component of biological membranes and can be used to study the function of biological membranes.</p>Formule :C40H76NaO10PDegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :770.99FXR agonist 5
CAS :<p>FXR agonist 5 is an FXR agonist used in the study of liver diseases or diseases mediated by metabolic inflammation.</p>Formule :C40H53N5O5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :683.88OPC 8490 free base
CAS :<p>OPC 8490 free base is a positive inotropic vasodilator and a cardiotonic agent that can be used to study cardiovascular diseases.</p>Formule :C24H27N3O3Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :405.491-Salicylate Glucuronide
CAS :<p>1-Salicylate Glucuronide (Salicylic Acid b-D-O-Glucuronide) is a metabolite of salicylic acid after glucuronidation, promoting excretion.</p>Formule :C13H14O9Couleur et forme :SolidMasse moléculaire :314.25DPPD-Q
CAS :<p>DPPD-Q, an antioxidant and an oxidative derivative of substituted p-phenylenediamine (DPPD), is identified in tire wear particles, rubber debris, particulate matter 2.5 (PM2.5), and wastewater influents and effluents. At a concentration of 5 µM, DPPD-Q inhibits soybean urease by 91.4%.</p>Formule :C18H14N2O2Couleur et forme :SolidMasse moléculaire :290.32N-Desmethyl Bendamustine
CAS :<p>N-DesmethylBendamustine is a metabolite of Bendamustine. It exerts cytotoxic effects on various lymphoma cell lines and peripheral blood lymphocytes.</p>Formule :C15H19Cl2N3O2Couleur et forme :SolidMasse moléculaire :344.24APP-018
CAS :<p>APP-018 (D-4F) is an 18 D-amino acid peptide that mimics apolipoprotein A-I (apoA-I). It enhances the anti-inflammatory properties of high-density lipoprotein (HDL) and is applicable in cardiovascular disease research.</p>Formule :C114H156N24O28Couleur et forme :SolidMasse moléculaire :2310.611-Hydroxy cannabinol
CAS :<p>11-Hydroxy cannabinol (Compound 5b) is an active metabolite of cannabinol.</p>Formule :C21H26O3Couleur et forme :SolidMasse moléculaire :326.43b-Cortolone
CAS :<p>b-Cortolone, a metabolite of Cortisol, exhibits relatively lower biological activity.</p>Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.49Cyano-myracrylamide
CAS :<p>Cyano-myracrylamide is an inhibitor of zinc finger DHHC domain-containing palmitoyltransferase 20 (zDHHC20) with an IC50 value of 1.35 µM. It also inhibits the S-palmitoylation of EGFR and CD36. In HEK293T cells expressing recombinant E. coli GobX, recombinant human MyD88, or endogenous Ras, Cyano-myracrylamide inhibits the S-palmitoylation of E. coli E3 ligase GobX, MyD88, and Ras, which are substrates of zDHHC20, zDHHC9, and zDHHC6.</p>Formule :C19H34N2OCouleur et forme :SolidMasse moléculaire :306.49ZG-2033
CAS :<p>ZG-2033 (Compound 26) is an orally active HIF-2α agonist that exhibits nanomolar activity (EC50 = 490 nM) in a luciferase reporter assay. It demonstrates an anti-anemic effect and shows synergistic effects with AKB-6548 in anemia, making it useful for the study of renal anemia.</p>Formule :C15H14N2O2SCouleur et forme :SolidMasse moléculaire :286.35YYLLVR
CAS :<p>YYLLVR is an inhibitory peptide of angiotensin-converting enzyme (ACE) with an inhibition rate of 89.10%. It demonstrates a low binding energy to ACE at -35.98 kcal/mol. YYLLVR can be utilized in hypertension research.</p>Formule :C41H63N9O9Couleur et forme :SolidMasse moléculaire :825.99Resinacein L
CAS :<p>Resinacein L is an inhibitor of α-glucosidase with an IC50 of 0.635 mM. This compound can slow the digestion and absorption of carbohydrates, thereby reducing postprandial blood glucose levels.</p>Formule :C30H40O8Couleur et forme :SolidMasse moléculaire :528.63DPTIP hydrochloride
CAS :<p>DPTIP hydrochloride is a potent inhibitor of neutral sphingomyelinase (N-SMase 2) that can cross the blood-brain barrier. It acts as an exosome inhibitor with an IC50 value of 30 nM.</p>Formule :C21H19ClN2O3SCouleur et forme :SolidMasse moléculaire :414.91SH7s
<p>SH7s is an effective carbonic anhydrase inhibitor, exhibiting Ki values of 15.9 nM for hCA IX and 55.2 nM for hCA XII. Additionally, SH7s acts as a hypoxia-mediated chemosensitizer in colorectal cancer cells.</p>Formule :C24H19ClF3N5O4SCouleur et forme :SolidMasse moléculaire :565.95α-Glucosidase-IN-77
<p>α-Glucosidase-IN-77 (Compound H7) is a non-competitive α-glucosidase inhibitor with an IC50 of 1.25 μM. It reduces blood glucose levels, improves glucose tolerance, regulates gut microbiota, and exhibits hepatoprotective effects in a mouse model of type 2 diabetes.</p>Formule :C25H16F3NO5SCouleur et forme :SolidMasse moléculaire :499.46N-Desmethyl clotiazepam
CAS :<p>N-Desmethyl clotiazepam (Desmethylclotiazepam) is an active metabolite of Clotiazepam.</p>Formule :C15H13ClN2OSCouleur et forme :SolidMasse moléculaire :304.8O-Desmethylcarvedilol
CAS :<p>O-Desmethylcarvedilol (Desmethylcarvedilol) is an active metabolite of Carvedilol, a non-selective β-adrenergic receptor (β-AR) antagonist. This compound inhibits store overload-induced calcium release in HEK293 cells expressing the RyR2 R4496C mutation (IC50= 7.62 µM). Additionally, O-Desmethylcarvedilol slows the increase in heart rate and prevents diastolic pressure reduction induced by Isoproterenol in conscious rabbits (ED50s = 32 and 5 µg/kg).</p>Formule :C23H24N2O4Couleur et forme :SolidMasse moléculaire :392.45Inostamycin A
CAS :<p>Inostamycin A, a anticancer bacterial metabolite isolated from Streptomyces, is a selective inhibitor of CDP-diacylglycerol:inositol 3-phosphatidyltransferase.</p>Formule :C38H68O11Couleur et forme :SolidMasse moléculaire :700.94LYP-IN-3
<p>LYP-IN-3 (compound D34) is a selective Lymphoid-tyrosine phosphatase (LYP) inhibitor (Ki=0.93 μM) that modulates the T-cell receptor (TCR) signaling pathway</p>Formule :C35H27NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.66ω-Conotoxin CVIF
<p>ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value of 34.3 nM in isolated rat DRG neurons.</p>Formule :C101H170N40O33S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2665.07L-Isoleucyl-L-arginine
CAS :<p>L-Isoleucyl-L-arginine, a dipeptide composed of L-isoleucine and L-arginine, acts as a potent angiotensin-converting enzyme (ACE) inhibitor and is utilized in</p>Formule :C12H25N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.36PTPσ Inhibitor, ISP
<p>PTPσ Inhibitor ISP is a compound that binds to recombinant human PTPs, thereby inhibiting PTPσ signaling.</p>Formule :C177H306N66O54S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4318.93Erythronic acid potassium
<p>Potassium erythronate is an intrinsic carbohydrate metabolite utilized in researching metabolic diseases.</p>Formule :C4H7KO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :173.99305Imperatoxin A
CAS :<p>Imperatoxin A, a peptide toxin sourced from the African scorpion Pandinus imperator, functions as an activator of Ca2+-release channels/ryanodine receptors (</p>Formule :C148H254N58O45S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3758.35nSMase2-IN-1
<p>nSMase2-IN-1 is an orally active inhibitor of Neutral sphingomyelinase 2 (nSMase2) with a potent IC50 value of 0.13 ± 0.06 μM.</p>Formule :C12H17N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.3hCAXII-IN-7
<p>hCAXII-IN-7 (compound 6e) functions as an inhibitor of human carbonic anhydrase XII (hCA XII) and possesses blood-brain barrier (BBB) permeability.</p>Formule :C26H25N5O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.645-LOX-IN-5
<p>Compound 29, also known as 5-LOX-IN-5, is a 5-lipoxygenase (5-LOX) inhibitor with an inhibitory concentration 50 (IC50) of 56 nM, utilized in research</p>Formule :C19H18BrN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.33RPR132595A hydrochloride
<p>RPR132595A (NPC) hydrochloride, an active metabolite of CPT-11, is produced via cytochrome P-450 3A4 (CYP3A4) metabolism and is ultimately eliminated via</p>Formule :C28H31ClN4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :555.02NAMPT degrader-3
<p>NAMPT Degrader-3 (compound C5) is a NAMPT degrader that functions through a VHL- and proteasome-dependent mechanism.</p>Formule :C56H74N8O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1003.3A3373
CAS :<p>A3373 is a novel inhibitor targeting both Phospholipase D1 (PLD1) and Phospholipase D2 (PLD2), demonstrating half maximal inhibitory concentrations (IC50) of</p>Formule :C17H9F7N2ODegré de pureté :98%Couleur et forme :SoildMasse moléculaire :390.26α-Glucosidase-IN-31
<p>α-Glucosidase-IN-31 (compound R1) is a potent oral α-Glucosidase inhibitor with an IC50 of 10.1 μM, demonstrating significant blood glucose reduction and</p>Formule :C18H18N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :290.36RORγt inverse agonist 31
<p>RORγt inverse agonist 31 (14g) is a potent antagonist of the retinoic acid receptor-related orphan receptor γt (RORγt), exhibiting an inhibitory concentration (</p>Formule :C23H15Cl2F3N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :555.36Eurestobart
CAS :<p>Eurestobart is a humanized IgG1κ (IgG1 kappa) monoclonal antibody that specifically targets the enzyme ectonucleoside triphosphate diphosphohydrolase (ENTPDase</p>Degré de pureté :98%Couleur et forme :Liquidα-Glucosidase-IN-38
<p>α-Glucosidase-IN-38 (Compound 11j) is a potent α-glucosidase inhibitor, demonstrating an IC50 of 12.44±0.38 μM, and is significant in the context of Diabetes</p>Degré de pureté :98%Couleur et forme :Odour SolidAlternaphenol B2
<p>Alternaphenol B2, a selective inhibitor of mutant isocitrate dehydrogenase 1 (IDH1m), is sourced from the coral-derived fungus Parengyodontium album SCSIO</p>Degré de pureté :98%Couleur et forme :Odour SolidVHL-IN-1
<p>VHL-IN-1 (compound 30), a ubiquitin E3 ligase von Hippel-Lindau (VHL) inhibitor with a dissociation constant (Kd) of 37 nM, potently stabilizes HIF-1α and</p>Formule :C28H37FN4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :544.68Myoregulin TFA
<p>Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics.</p>Formule :C239H391N53O67S3·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5175.17 (free base)α-Glucosidase-IN-36
<p>α-Glucosidase-IN-36 (compound 5g) is a potent inhibitor of α-glucosidase, exhibiting an IC50 value of 6.69 ± 0.18 μM and inhibition constants Ki and Kis of 1.65</p>Formule :C26H24BrN5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :566.47Ovotransferrin (328-332)
CAS :<p>Ovotransferrin (328-332), with an IC50 of 20 μM, exhibits protective activity against hypertension by inhibiting the Angiotensin-Converting Enzyme (ACE) and</p>Formule :C25H46N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :570.68Hepcidin-25 (human) (acetate)
CAS :<p>Hepcidin-25 (human) acetate is a modulator of iron metabolism that demonstrates anti-inflammatory and antibacterial effects through the modulation of iron-</p>Formule :C113H170N34O31S9·xC2H4O2Degré de pureté :98%Couleur et forme :Solidω-Conotoxin MVIID
<p>ω-Conotoxin MVIID (SNX-238) is a peptide from the Conus genus that inhibits the ω-Conotoxin-GVIA-sensitive, high-threshold calcium (Ca 2+) current in fish</p>Formule :C99H164N42O33S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2695.08ω-Conotoxin CVIA
CAS :<p>ω-Conotoxin CVIA, a 27-amino acid neuropeptide, functions as a blocker of voltage-sensitive calcium channels (VSCCs) [1].</p>Formule :C97H161N39O36S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2641.95Casuarictin
CAS :<p>Casuarictin, a potent competitive inhibitor of α-glucosidase, exhibits an IC50 of 0.21 μg/mL and functions as a presenilin stabilization factor-like (PSFL)</p>Formule :C41H28O26Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :936.65Flaccidoside III
CAS :<p>Flaccidoside III, a flavonoid and triterpenoid compound extracted from the aerial parts of N.</p>Formule :C59H96O26Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1221.38Stevisaliosides D
<p>Stevisaliosides D (Compound 5), extracted from the roots of Stevia serrata, exhibits inhibition of PTP1B with an IC50 of 31.8 μM and has applications in</p>Formule :C35H54O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :730.79Glucocerebrosidase
CAS :<p>Glucocerebrosidase (Glucosylceramidase; GBA), a lysosomal enzyme, catalyzes the hydrolysis of the β-glucosidic linkage in glucocerebroside (GC) to yield glucose</p>Degré de pureté :98%Couleur et forme :SolidPF-07238025
<p>PF-07238025, a potent branched-chain ketoacid dehydrogenase kinase (BDK) inhibitor with an EC50 of 19 nM, enhances the stability of the BDK-BCKDH core E2</p>Formule :C19H18N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :354.42Alanine aminotransferase
CAS :<p>Alanine aminotransferase (ALT), a pyridoxal-dependent enzyme, catalyzes the reversible interconversion of L-alanine and 2-oxoglutarate into pyruvate and L-</p>Degré de pureté :98%Couleur et forme :SolidCalciseptin
CAS :<p>Calciseptine, a neurotoxin isolated from the Black Mamba (Dendroaspis p.</p>Formule :C299H468N90O87S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7036.12HIF-1α-IN-6
<p>HIF-1α-IN-6 (compound 3s) is a potent inhibitor of HIF-1α, demonstrating IC50 values of 0.6 nM and 53.3 nM in MiaPaCa-2 and MDA-MB-231 cells, respectively.</p>Degré de pureté :98%Couleur et forme :Odour SolidIDO1-IN-23
<p>IDO1-IN-23 (compound 41) is a potent inhibitor of human indoleamine 2,3-dioxygenase 1 (IDO1), exhibiting an IC50 of 13 μM [1].</p>Degré de pureté :98%Couleur et forme :Odour SolidAmidase
CAS :<p>Amidases, belonging to the nitrilase superfamily, catalyze amide hydrolysis to yield carboxylic acid and ammonia.</p>Degré de pureté :98%Couleur et forme :SolidD-Pro-Phe-Arg-Chloromethylketone
CAS :D-Pro-Phe-Arg-Chloromethylketone, an inhibitor of coagulation factor XII and plasma kallikrein, is significant in the regulation of thrombosis and inflammationFormule :C21H31ClN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.96α-Glucosidase-IN-26
<p>α-Glucosidase-IN-26 (Compound 7i), with an IC50 value of 4.63 µM, functions as an α-glucosidase inhibitor and is utilized in research related to type 2 diabetes</p>Formule :C23H22ClN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.89hCA XII-IN-6
<p>Compound 4d, known as hCA XII-IN-6, is a potent inhibitor of human carbonic anhydrase XII (hCA XII) with a Ki value of 84.2 nM and exhibits anti-proliferative</p>Formule :C11H9N5O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.35wt hMLN
<p>Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump (SERCA), playing a crucial role in the regulation of</p>Formule :C245H404N54O66SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :5194.22PROTAC SGK3 degrader-1
CAS :<p>PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC coupler that targets SGK3 and binds ligands to VH032 VHL to induce endogenous SGK3 degradation.</p>Formule :C57H73FN10O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1157.38Glutamate dehydrogenase (NAD(P))
CAS :<p>GLDH, found in liver/kidney/brain/muscle/intestine, catalyzes glutamate to α-KG in urea cycle.</p>Couleur et forme :SolidN-Desethyl Sunitinib hydrochloride
<p>N-Desethyl Sunitinib hydrochloride (SU-12662 hydrochloride) has potential anticancer activity and can be used to study cancer.</p>Formule :C20H24ClFN4O2Couleur et forme :SolidMasse moléculaire :406.89IFB-088 acetate
CAS :<p>IFB-088 acetate targets PPP1R15A-related diseases, including cancers and protein misfolding disorders.</p>Formule :C10H13ClN4O2Degré de pureté :90%Couleur et forme :SolidMasse moléculaire :256.69SB-435495
CAS :<p>SB-435495 is a compound characterized by its potent, selective, reversible, and non-covalent inhibition of Lp-PLA2, demonstrating an IC50 value of 0.06 nM.</p>Formule :C38H40F4N6O2SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :720.82Carbonic anhydrase
CAS :<p>Carbonic anhydrase, a zinc enzyme in all life forms, converts CO2 to bicarbonate; studied for cancer, glaucoma, obesity, epilepsy.</p>Couleur et forme :SolidN-Acetyl lysyltyrosylcysteine amide acetate
<p>N-Acetyl lysyltyrosylcysteine amide acetate is an effective and selective tripeptide inhibitor of myeloperoxidase (MPO).</p>Formule :C22H35N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.61PKR activator 4
CAS :<p>PKR activator 4 (example 7A), a potent activator of pyruvate kinase R (PKR), holds promise for blood disorder research [1].</p>Formule :C18H24N6O2SSiCouleur et forme :SolidMasse moléculaire :416.57Cavosonstat
CAS :<p>Cavosonstat (N91115) is an oral GSNOR inhibitor aiding CFTR in cystic fibrosis.</p>Formule :C16H10ClNO3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :299.71O-Desmethyl apixaban sulfate sodium
<p>O-Desmethyl apixaban sulfate sodium inhibits factor X (FXa) with a Ki of 58 μM,and is a major circulating metabolite of Apixaban in humans.</p>Formule :C24H22N5NaO7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :547.52(S,S)-GSK321
CAS :<p>(S,S)-GSK321 is a (S,S)-enantiomer of GSK321 [1] .</p>Formule :C28H28FN5O3Couleur et forme :SolidMasse moléculaire :501.55MAGL-IN-5
CAS :<p>MAGL-IN-5 is a non-selective lipase inhibitor.</p>Formule :C18H17N3O5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :355.34Angstrom6
CAS :<p>Angstrom6 (A-6 peptide) is an 8 amino acid peptide derived from single chain urokinase fibrinogen activator (scuPA) that interferes with the uPA/uPAR cascade</p>Formule :C39H62N10O15Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :910.97Alphitonin
CAS :<p>Alphitonin: a flavonoid in L. leptolepis wood, metabolized from quercetin by E. ramulus in the gut.</p>Formule :C15H12O7Couleur et forme :SolidMasse moléculaire :304.25Aldose 1-epimerase
CAS :<p>Aldose 1-epimerase facilitates the conversion of α- to β-sugars like glucose, crucial for carbohydrate processing.</p>Couleur et forme :Solid5-Lipoxygenase-IN-3
CAS :<p>Compound 14, a <1 μM 5-lipoxygenase inhibitor, researches inflammation, cancer, stroke, Alzheimer's.</p>Formule :C19H16ClN5OCouleur et forme :SolidMasse moléculaire :365.82hMAO-B-IN-5
CAS :<p>hMAO-B-IN-5: potent, selective hMAO-B inhibitor (IC50: 0.12μM), crosses blood-brain barrier, for Parkinson's research.</p>Formule :C24H22O3Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :358.43HPA-IN-1
<p>HPA-IN-1: potent human pancreatic α-amylase inhibitor; IC50: 12.0 μM for HPA, 410.4 μM for α-glucosidase.</p>Formule :C33H32N4O11Couleur et forme :SolidMasse moléculaire :660.63N-Stearoylsphingomyelin
CAS :<p>N-Stearoylsphingomyelin (N-Stearoyl-D-sphingomyelin), a sphingolipid, inhibits Phospholipase Cδ1 (PLCδ1) [1].</p>Formule :C41H83N2O6PCouleur et forme :SolidMasse moléculaire :731.08(±)10(11)-DiHDPA
CAS :<p>(±)10(11)-DiHDPA is produced from cytochrome P450 epoxygenase action on docosahexaenoic acid .</p>Formule :C22H34O4Couleur et forme :SolidMasse moléculaire :362.51Oseltamivir acid methyl ester hydrochloride
CAS :<p>Oseltamivir acid methyl ester hydrochloride, a precursor to oseltamivir, is converted by CES1.</p>Formule :C15H27ClN2O4Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :334.84Fmoc-Cys(Acm)-OH
CAS :<p>Fmoc-Cys(Acm)-OH (Fmoc-S-acetamidomethyl-L-cysteine) is a cysteine derivative.</p>Formule :C21H22N2O5SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :414.478′-Hydroxy ABA
CAS :<p>8′-Hydroxy ABA (8'-OH-ABA), a key metabolite of abscisic acid (ABA), exhibits hormonal activity by promoting enhanced oil synthesis.</p>Formule :C15H20O5Couleur et forme :SolidMasse moléculaire :280.32ML266
CAS :<p>ML266: GCase chaperone, non-inhibiting, IC50=2.5 µM, aids mutant protein transport, may help in Gaucher disease study.</p>Formule :C24H22BrN3O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :496.35Coumachlor
CAS :<p>Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.</p>Formule :C19H15ClO4Couleur et forme :SolidMasse moléculaire :342.77sEH inhibitor-20
<p>sEH inhibitor-20 is a metabolically stable, orally active sEH inhibitor with an IC50 of 0.2 nM. It exhibits significant analgesic and anti-inflammatory properties, making it a promising candidate for researching neuropathic pain.</p>Couleur et forme :Odour SolidL,L-Dityrosine
CAS :<p>L,L-Dityrosine, a component found in the acid hydrolysates of various biological materials, such as insect cuticular resilin, plays a significant role in</p>Formule :C18H20N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.36Octachlorodibenzo-p-dioxin
CAS :<p>Octachlorodibenzo-p-dioxin (OCDD) is an environmental contaminant with no acute toxicity when administered. In rats, the systemic elimination half-life of Octachlorodibenzo-p-dioxin (50 μg/kg intravenously or 50-5000 μg/kg orally) is 3-5 months. It can accumulate and concentrate in the liver and adipose tissue after low-dose, repeated exposure. Repeated dosing of Octachlorodibenzo-p-dioxin leads to increased activity of 7-ethoxyresorufin-O-deethylase (7-EROD) and elevated total cytochrome P-450 levels.</p>Formule :C12Cl8O2Couleur et forme :SolidMasse moléculaire :459.75Lacto-N-biose I
CAS :<p>Galβ1-3GlcNAc, a natural metabolite, is a substrate for H. pylori's α1,2-fucosyltransferase.</p>Formule :C14H25NO11Couleur et forme :SolidMasse moléculaire :383.35Monononadecanoin
CAS :<p>Monononadecanoin is a lipid compound known for its anti-inflammatory and antioxidant properties. It is frequently used in skincare products as a moisturizer and skin-repairing agent. Additionally, Monononadecanoin serves as a flavor enhancer and preservative in food additives.</p>Formule :C22H46O5Couleur et forme :SolidMasse moléculaire :390.6N-Trifluoroacetyladriamycin
CAS :<p>N-Trifluoroacetyladriamycin, Valrubicin's metabolite, treats bladder cancer; it's an analog of doxorubicin, infused into the bladder.</p>Formule :C29H28F3NO12Couleur et forme :SolidMasse moléculaire :639.533DSPE-PEG1000-CREKA
<p>DSPE-PEG1000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide has the capability to target tumor cells and tumor vasculature, exhibiting anti-tumor activity. Additionally, DSPE-PEG1000-CREKA can be utilized for drug delivery.</p>Couleur et forme :Odour Solidα-1,4-Galactosyltransferase (LgtC)
CAS :<p>A4GALT (LgtC) adds galactose to lactosylceramide, forming globotriaosylceramide; used in P1 antigen synthesis.</p>Couleur et forme :SolidSucunamostat hydrochloride
<p>Sucunamostat (SCO-792) hydrochloride is an orally active, reversible inhibitor of enteropeptidase, displaying inhibition constants (IC50) of 4.6 nM for rat</p>Formule :C22H23ClN4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.89Nepetalactone
CAS :<p>Nepetalactone is found in the plant Nepeta parnassica and has high mosquito repellency properties.</p>Formule :C10H14O2Couleur et forme :SolidMasse moléculaire :166.22trans-hydroxy Glimepiride
CAS :<p>trans-Hydroxy Glimepiride, an active sulfonylurea glimepiride metabolite, is primarily synthesized in the liver by CYP2C9.</p>Formule :C24H34N4O6SCouleur et forme :SolidMasse moléculaire :506.62(S)-Higenamine hydrobromide
CAS :<p>(S)-Higenamine hydrobromide, S-enantiomer for benzylisoquinoline synthesis, results from dopamine and 4-HPAA condensation by NCS.</p>Formule :C16H18BrNO3Couleur et forme :SolidMasse moléculaire :352.2213-cis-Retinyl acetate
CAS :<p>13-cis-Retinyl acetate: active 13-cis isomer of Retinyl acetate, metabolite of vitamin A.</p>Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.49Perflubutane
CAS :<p>Perfluorobutane is a gas that is colorless.</p>Formule :C4F10Degré de pureté :98%Couleur et forme :Colorless Gas Colorless GasMasse moléculaire :238.03Hydroxydehydro Nifedipine Carboxylate
CAS :<p>Hydroxydehydro nifedipine carboxylate is a metabolite of nifedipine .1</p>Formule :C16H14N2O7Couleur et forme :SolidMasse moléculaire :346.2955β-Androstan-3β-ol-17-one
CAS :<p>5β-Androstan-3β-ol-17-one (3β-Etiocholanolone; 5β-Epiandrosterone), a 5β-reduced steroid and a significant metabolic derivative of dehydroepiandrosterone (DHEA</p>Formule :C19H30O2Couleur et forme :SolidMasse moléculaire :290.44
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