Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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Pi-Methylimidazoleacetic acid
CAS :<p>Pi-Methylimidazoleacetic acid is a potential neurotoxin.</p>Formule :C6H8N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :140.14PNGase F
CAS :<p>PNGase F is an endoglycosidase and amide hydrolase that catalyses the cleavage of internal glycosidic bonds in oligosaccharides.</p>Couleur et forme :SolidGenz-123346
CAS :<p>Genz-123346 is an oral inhibitor of glucosylceramide synthase, blocking ceramide to GL1 conversion, with a 14 nM IC50.</p>Formule :C52H82N4O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :987.23Lasiocarpine
CAS :<p>Lasiocarpine is a pyrrolizidine alkaloid, it has acute cytotoxicity in human and hepatic cell lines.</p>Formule :C21H33NO7Degré de pureté :98%Couleur et forme :Colourless To Beige Crystalline SolidMasse moléculaire :411.49(-)-Dihydroguaiaretic acid
<p>(-)-Dihydroguaiaretic acid is a useful organic compound for research related to life sciences and the catalog number is T126154.</p>Formule :C20H26O4Couleur et forme :SolidMasse moléculaire :330.424α-Glucosidase-IN-65
<p>α-Glucosidase-IN-65 (compound 5) is a Schiff base derivative of 3,4-dihydroxyphenylacetic acid. It acts as a potent α-glucosidase inhibitor with an IC50 of 12.84 μM.</p>Formule :C15H14N2O6Masse moléculaire :318.08519α-Glucosidase-IN-50
<p>α-Glucosidase-IN-50 (compound 8) acts as an inhibitor of α-Glucosidase.</p>Formule :C33H28Cl4N6O6SMasse moléculaire :776.05451Ercalcitriol
CAS :<p>Ercalcitriol, active Vitamin D2 metabolite, boosts immunity by regulating CAMP and DEFB4 genes against infections.</p>Formule :C28H44O3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :428.654,7,10,13,16-Docosapentaenoic acid
CAS :<p>4,7,10,13,16-Docosapentaenoic acid is an endogenous metabolite.</p>Formule :C22H34O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.51Hexokinase II VDAC binding domain peptide, cell-permeable
<p>HexokinaseIIVDACbinding domain peptide (Hxk2VBD peptide) is a cell-permeable peptide derived from the hexokinase II VDAC binding domain. This peptide inhibits the mitochondrial localization of hexokinase 2 (HXK2) and also suppresses neurotrophic factor-induced axon growth.</p>Formule :C188H291N53O40S2Masse moléculaire :3995.18073GZ22-4
<p>GZ22-4 is a near-infrared (NIR) fluorescent probe with a high affinity for carbonic anhydrase IX (CAIX), exhibiting a dissociation constant (Kd) of 0.2 nM. It is applicable in studies for visualizing CAIX-positive tumors.</p>Formule :C88H126F3N6NaO24S4Masse moléculaire :1858.75561PROTAC NAMPT Degrader-1
<p>PROTACNAMPT Degrader-1 is an effective NAMPT-targeting PROTAC with a DC50 value of 217 nM. It exhibits antiproliferative activity, with an IC50 value of 0.12 μM against A2780 cells.</p>Formule :C57H69N13O8S2Masse moléculaire :1127.48335L-Mevalonic acid
CAS :<p>L-Mevalonic acid, a cholesterol precursor, is studied in autoimmune, atherosclerosis, and Alzheimer's research.</p>Formule :C6H12O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :148.16Carbonic anhydrase/AChE-IN-2
<p>Carbonic anhydrase/AChE-IN-2 (compound 19) is a selective inhibitor of acetylcholinesterase (AChE) and carbonic anhydrase (CA), with inhibition efficiencies (Ei) of 8.54 nM, 13.54 nM, and 5.21 nM, respectively.</p>Formule :C17H12BrF3O2Masse moléculaire :383.99728α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid
CAS :<p>α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid was identified as possible dual inhibitors for hLTA4H and hLTC4S enzymes by the computer-aided</p>Formule :C23H23NO3Degré de pureté :97.19% - 99.36%Couleur et forme :SoildMasse moléculaire :361.43Sirtuin modulator 2
CAS :<p>Sirtuin modulator 2 (N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide) exhibits antidiabetic, anti-inflammatory and antitumor activities.</p>Formule :C19H15N3O2SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :349.41α-Amylase/α-Glucosidase-IN-12
<p>α-Amylase/α-Glucosidase-IN-12 (compound 10k) is a dual inhibitor targeting α-glucosidase and α-amylase, with IC50 values of 34.52 nM and 24.62 nM, respectively. This inhibitor is designed based on [triazolo[4,3-b][1,2,4]triazine and holds potential for diabetes research.</p>Formule :C19H13F3N6OSMasse moléculaire :430.08236Yokonoside
CAS :<p>Yokonoside is a biochemical.</p>Formule :C20H21NO11Couleur et forme :SolidMasse moléculaire :451.384α-Glycerophosphate Dehydrogenase-Triosephosphate
<p>α-Glycerophosphate Dehydrogenase-Triosephosphate (GDH-TIM) is an enzyme mixture composed of glycerophosphate dehydrogenase (GDH) and triosephosphate isomerase (TIM). This compound is employed to measure transketolase (TK) activity in erythrocyte hemolysates, which helps in assessing vitamin B deficiency.</p>MPO-IN-7
<p>MPO-IN-7 (compound MDC) is a myeloperoxidase inhibitor with IC50 values of 41 μM for α-glucosidase, 25 μM for dipeptidyl peptidase-4, and 4.5 μM for myeloperoxidase. MPO-IN-7 exhibits antioxidant and anti-inflammatory activities in vitro.</p>Formule :C16H14N2O6Masse moléculaire :330.085191,1,3-Tribromoacetone
CAS :<p>1,1,3-Tribromoacetone (1,1,3-tribromo-2-propanone) is an impurity of methotrexate.</p>Formule :C3H3Br3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.77α-Glucosidase-IN-48
<p>α-Glucosidase-IN-48 (compound 9) is a potent inhibitor of α-Glucosidase, with an IC50 of 1.30 μM.</p>Formule :C15H9Cl2N5O3SMasse moléculaire :408.98032α-Glucosidase-IN-44
<p>α-Glucosidase-IN-44 (compound IT4) is an α-glucosidase inhibitor with an IC50 value of 2.35 μM. This compound is orally active and has the ability to reduce fasting blood glucose levels in diabetic mice.</p>Formule :C23H21N3O3SMasse moléculaire :419.13036JTV-519 Formate
<p>JTV-519 Formate is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA).</p>Formule :C26H34N2O4SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :470.62Amlodipine aspartic acid impurity
CAS :<p>Amlodipine aspartic acid: a calcium blocker with antihypertensive effects; contains specific impurities.</p>Formule :C24H29ClN2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.95Carbonic anhydrase inhibitor 18
<p>Carbonic anhydrase inhibitor18 (Compound 9) is an inhibitor of human carbonic anhydrase (hCA) isozymes, with Ki values of 604.8 nM for hCA I, 333.6 nM for hCA II, 1.9 nM for hCA IX, and 6.7 nM for hCA XII. Carbonic anhydrase inhibitor18 is applicable in cancer research.</p>Formule :C26H28N4O6S2Masse moléculaire :556.14503L-Amino acid oxidase
CAS :<p>L-Amino acid oxidase catalyzes the oxidative deamination of L-amino acids, which have local oxidative effects as well as potent antimicrobial effects.</p>Couleur et forme :SolidFellutanine A
CAS :<p>Fellutanine A is a useful organic compound for research related to life sciences. The catalog number is T129801 and the CAS number is 175414-35-4.</p>Couleur et forme :SoildAllotetrahydrocortisol
CAS :<p>Allotetrahydrocortisol (5a-Tetrahydrocortisol) is a metabolite of Cortisol. Cortisol is the main glucocorticoid in human.</p>Formule :C21H34O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :366.49NU223612
CAS :<p>"NU223612 is a potent IDO1-degrading PROTAC with Kd 640 nM, binds CRBN at 290 nM, and crosses the BBB."</p>Formule :C49H55FN6O9Couleur et forme :SolidMasse moléculaire :890.99Nucleocidin
CAS :<p>Nucleocidin, an antitrypanosomal antibiotic, inhibits the transfer of labeled amino acids from S-RNA to protein.</p>Formule :C10H13FN6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.31Melittin Acetate
<p>Melittin Acetate, a PLA2 activator, enhances low-weight PLA2 activity but not high-weight PLA2.</p>Formule :C133H233N39O33Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :2906.51N-Methyl pemetrexed
CAS :<p>N-Methyl pemetrexed, an impurity found in Pemetrexed, serves as an antifolate cytotoxic agent utilized in cancer research [1].</p>Formule :C21H23N5O6Couleur et forme :SolidMasse moléculaire :441.44Milpocitide
CAS :<p>Milpocitide, a (293-333)-peptide fragment of the human low-density lipoprotein receptor (LDLR), specifically corresponds to the EGF-like domain 1 [1].</p>Formule :C255H413N63O86S6Couleur et forme :SolidMasse moléculaire :5929.75LDHA-IN-8
CAS :<p>LDHA-IN-8, an inhibitor, inhibits the proliferation of pancreatic and lung cancer cells, decreasing the intracellular lactate content and increasing ROS levels.</p>Formule :C15H14N4O2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :282.3O-Demethyl Lenvatinib hydrochloride
<p>O-Demethyl Lenvatinib HCl is a Lenvatinib metabolite; an oral inhibitor targeting VEGFR, FGFR, PDGFR, KIT, RET with antitumor properties.</p>Formule :C20H18Cl2N4O4Couleur et forme :SolidMasse moléculaire :449.29Gluconapin
CAS :<p>Gluconapin serves as a precursor to sulforaphane, an effective anticancer isothiocyanate. It has been found to reduce the increase in plasma triglycerides induced by corn oil consumption in mice.</p>Formule :C11H19NO9S2Couleur et forme :SolidMasse moléculaire :373.4Saccharopine
CAS :<p>L-Saccharopine is a product of the breakdown of essential amino acid Lysine.</p>Formule :C11H20N2O6Couleur et forme :SolidMasse moléculaire :276.29Pyridindolol
CAS :<p>Pyrindolol, a S. alboverticillatus metabolite, inhibits bovine β-galactosidase at 2 μg/ml in acid; not effective on other species' enzymes.</p>Formule :C14H14N2O3Couleur et forme :SolidMasse moléculaire :258.2778-Isoprostaglandin F2α
CAS :<p>8-Isoprostaglandin F2α is a natural product for research related to life sciences. The catalog number is T37164 and the CAS number is 27415-26-5.</p>Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.489(S)-HOTrE
CAS :<p>9(S)-HOTrE is a plant metabolite and octadecatrienoic acid produced by the action of 5-lipoxygenase (5-LO) on α-linolenic acid.</p>Formule :C18H30O3Couleur et forme :SolidMasse moléculaire :294.43D-Threonine
CAS :<p>D-Threonine (H-D-Thr-OH) is one of the metabolites of Saccharomyces cerevisiae.</p>Formule :C4H9NO3Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :119.12Porcine Factor Xa
CAS :<p>PorcineFactor Xa is obtained by activating purified Porcine Factor X using Russells' Viper Venom, after which the venom is removed.</p>Couleur et forme :SolidFXIIa-IN-4
<p>FXIIa-IN-4 (compound 22) is a potent and selective human FXIIa inhibitor, exhibiting IC50 values of 0.032 μM for FXIIa, 0.30 μM for thrombin, and >50 μM for FXIa. It is utilized in anticoagulant research.</p>Formule :C11H9FN4O3Masse moléculaire :264.06587DSPE-PEG2000-CSTSMLKAC
<p>DSPE-PEG2000-CSTSMLKAC is a PEG compound composed of DSPE and CSTSMLKAC. CSTSMLKAC can mediate phage selective homing to ischemic heart tissue. DSPE-PEG2000-CSTSMLKAC is suitable for drug delivery.</p>Couleur et forme :Odour SolidFZQ-21
<p>FZQ-21 (Compound 70P) is an inhibitor of the water-soluble epoxide hydrolase (sEH), with an IC50 value of 4 nM. The IC50 for inhibiting human sEH is 1.5 nM, which is comparable to that of EC5026 (1.7 nM). FZQ-21 is utilized in sepsis research.</p>Formule :C28H30N4O3Masse moléculaire :470.23179PTP1B-IN-27
<p>PTP1B-IN-27 (Compound 7i) is an inhibitor of protein tyrosine phosphatase 1-B (PTP-1B) with an IC50 of 8.2 µM. Additionally, it inhibits α-glucosidase with an IC50 of 120 µM and exhibits competitive inhibition characteristics (Ki=118 µM).</p>Formule :C26H24FN7O2SMasse moléculaire :517.16962(R,S)-Carvedilol Glucuronide
CAS :<p>(R,S)-Carvedilol glucuronide is a racemic mix, metabolized by UGT1A1, UGT2B4, and UGT2B7.</p>Formule :C30H34N2O10Couleur et forme :SolidMasse moléculaire :582.606E 6080 HCl
CAS :<p>E 6080 HCl is a 5-lipoxygenase inhibitor and can be used to study bronchial diseases.</p>Formule :C17H20ClN3O3S2Degré de pureté :99.80%Couleur et forme :SoildMasse moléculaire :413.94Carvedilol metabolite 4-Hydroxyphenyl Carvedilol
CAS :<p>4-Hydroxyphenyl Carvedilol is a metabolite of Carvedilol. Carvedilol is a beta-blocker/alpha-1 blocker.</p>Formule :C24H26N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :422.47IDO1-IN-12
CAS :<p>IDO1-IN-12 is a potent and orally available IDO1 inhibitor.</p>Formule :C21H19F3N2O2Couleur et forme :SolidMasse moléculaire :388.39LYP-IN-1
CAS :<p>LYP-IN-1 is a potent, selective inhibitor of lymphoid-specific tyrosine phosphatase useful for studying autoimmune disorders and immune signaling.</p>Formule :C28H20ClNO6Degré de pureté :92.43%Couleur et forme :SolidMasse moléculaire :501.92GS-493
CAS :<p>GS-493: Specific SHP2 inhibitor, very potent (IC50=71 nM), 29x affinity vs. SHP1, 45x vs. PTP1B; hinders cancer cell growth/movement.</p>Formule :C21H14N6O8SCouleur et forme :SolidMasse moléculaire :510.44α-2,6-Sialyltransferase (Pd26ST)
CAS :<p>Alpha-2,6-Sialyltransferase (Pd26ST) efficiently catalyzes the sialylation of both terminal and internal galactose and N-acetylgalactosamine residues, resulting</p>Couleur et forme :SolidCurcumin monoglucuronide
CAS :<p>Curcumin monoglucuronide, curcumin's in vivo metabolite, useful for metabolic research and cancer study.</p>Formule :C27H28O12Couleur et forme :SolidMasse moléculaire :544.50β-Cryptoxanthin
CAS :<p>β-Cryptoxanthin is isolated from Satsuma mandarin orange with an anti-stress effect. It is an oxygenated carotenoid and an antioxidant.</p>Formule :C40H56ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.87ARL67156 triethylamine
<p>ARL67156, a selective ecto-ATPase inhibitor, blocks NTPDase1, 3, and NPP1; used in calcific valve, asthma research. Ki: 11-18 μM.</p>Formule :C15H24Br2N5O12P3·3C6H15N)Couleur et forme :SolidMasse moléculaire :1154.231-β-D-Glucosylsphingadienine (d18:2 (4E,8E))
CAS :<p>1-β-D-Glucosylsphingadienine is a glucosylsphingosine, which are deacetylated lysolipid derivatives of glucosylcerebrosides .</p>Formule :C24H45NO7Couleur et forme :SolidMasse moléculaire :459.624DSPE-PEG2000-EB1
<p>DSPE-PEG2000-EB1 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (EB1). It is utilized for drug delivery.</p>Couleur et forme :Odour SolidXanthine oxidase-IN-13
<p>Xanthine oxidase-IN-13 (Compound 10) is a selective inhibitor of xanthine oxidase, with an IC50 of 149.56 μM for bovine xanthine oxidase. It is utilized in the study of inflammatory arthritis.</p>Formule :C14H13NOMasse moléculaire :211.09971Maltodextrin, dextrose equivalent 16.5-19.5
CAS :<p>Maltodextrin (DE 16.5-19.5) is an inactive pharma excipient that enhances drug stability, solubility, and processing.</p>Formule :(C6H10O5)n·xH2OCouleur et forme :SolidDSPE-PEG5000-CCK8
<p>DSPE-PEG5000-CCK8 is a PEGylated compound comprised of DSPE and Cholecystokinin-8 (CCK8). Cholecystokinin-8 exhibits peptide activity that regulates gallbladder contraction and the functioning of the digestive system. DSPE-PEG5000-CCK8 can be applied in drug delivery systems.</p>Couleur et forme :Odour SolidARL67156 trisodium hydrate
<p>ARL67156 trisodium hydrate inhibits ecto-ATPase, NTPDase1, NTPDase3, NPP1 (Kis 11-18µM), for calcific valve disease, asthma research.</p>Formule :C15H23Br2N5Na3O13P3Couleur et forme :SolidMasse moléculaire :834.61Cellobiosan
CAS :<p>Cellobiosan is an anhydro sugar formed during biofuel production from the fast pyrolysis of wood.</p>Formule :C12H20O10Couleur et forme :SolidMasse moléculaire :324.282SCD1 inhibitor-3
CAS :<p>SCD1 inhibitor-3 (ML-270) is a highly effective and orally available compound that inhibits SCD1 with remarkable safety.</p>Formule :C19H16FN7O2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :393.37PTP Inhibitor IV
CAS :<p>PTP Inhibitor IV selectively inhibits DUSP14 (IC50=5.21µM) and other PTPs, affecting cellular signaling.</p>Formule :C26H26F6N2O4S2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :608.62DSPE-PEG2000-R9
<p>DSPE-PEG2000-R9 is a PEG compound composed of DSPE and polyarginine-9 peptide (R9) peptide. It can be used for drug delivery.</p>Couleur et forme :Odour Solid5-hydroxy Thiabendazole
CAS :<p>5-OH TBZ, a thiabendazole metabolite, lacks anthelmintic effect on A. caninum larvae growth.</p>Formule :C10H7N3OSCouleur et forme :SolidMasse moléculaire :217.247α-1,3-Galactosyltransferase (GTB)
CAS :<p>alpha-1,3-Galactosyltransferase (GTB) synthesizes α-Gal epitopes by transferring galactose to specific acceptors.</p>Couleur et forme :SolidSDUY817
<p>SDUY817 is a dual APN/NEP inhibitor with IC50 values of 0.29 μM for APN and 7.4 μM for NEP. It exhibits analgesic effects in a concentration- and time-dependent manner, making it a potential candidate for research in the field of neuropathic pain disorders.</p>Formule :C18H16IN3O3Couleur et forme :SolidMasse moléculaire :449.24Spirolaxine
CAS :<p>Spirolaxine from Sporotrichum laxum shows anti-Helicobacter pylori activity.</p>Formule :C23H32O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :404.5Stephacidin B
CAS :<p>Stephacidin B, from A. ochraceus, forms avrainvillamide in vitro. Cytotoxic to various cancer cells; induces apoptosis in hepatocarcinoma at 4 μM.</p>Formule :C52H54N6O8Couleur et forme :SolidMasse moléculaire :891.038PTP1B-IN-22
CAS :<p>PTP1B-IN-22 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that inhibits glucose uptake in skeletal muscle L6 myotubes.</p>Formule :C16H12N2O3S2Degré de pureté :98.35%Couleur et forme :SoildMasse moléculaire :344.41Larsucosterol sodium
CAS :<p>Larsucosterol sodium: a liver-derived cholesterol byproduct; modulates lipid synthesis, inflammation, and cell death regulation.</p>Formule :C27H46NaO5SCouleur et forme :SolidMasse moléculaire :505.7110'-Desmethoxystreptonigrin
CAS :<p>'10'-Desmethoxystreptonigrin antibiotic derived from streptonigrin combats various bacteria and cancer cells, and inhibits p21ras farnesylation (IC50 = 21 nM).</p>Formule :C24H20N4O7Couleur et forme :SolidMasse moléculaire :476.445Febuxostat sec-butoxy acid
CAS :<p>Febuxostat sec-butoxy acid is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1] .</p>Formule :C16H16N2O3SCouleur et forme :SolidMasse moléculaire :316.37Tanshinone IIA anhydride
CAS :<p>Tanshinone IIA anhydride: irreversible inhibitor for human CE1 (Ki=1.9 nM) and hiCE (Ki=1.4 nM).</p>Formule :C19H18O4Couleur et forme :SolidMasse moléculaire :310.34LYP-8
<p>LYP-8 is a potent NAMPT degrader that achieves a maximum degradation rate of 97% in NAMPT within SKOV-3 cells at a concentration of 0.5 μM. LYP-8 also demonstrates anticancer activity both in vitro and in vivo.</p>Formule :C56H74N8O10SMasse moléculaire :1050.52486CD13-IN-1
<p>CD13-IN-1 (Compound 5f) is a CD13 inhibitor with an IC50 value of 1.71 μM. It effectively suppresses the proliferation of various tumor cells, demonstrating antitumor activity.</p>Couleur et forme :Odour SolidCTL26
<p>CTL26 is an effective, orally active α-glucosidase inhibitor, with an IC50 value of 2.81 µM, demonstrating antidiabetic properties.</p>Formule :C25H18N6O3SMasse moléculaire :482.1161111,12-DiHETrE
CAS :<p>11,12-DiHETrE: Endogenous P450 eicosanoid, used in preterm labor study and NAFL/NASH differentiation.</p>Formule :C20H34O4Couleur et forme :SolidMasse moléculaire :338.48Calcitetrol
CAS :<p>Calcitetrol is the hormonally active form of vitamin D with three hydroxyl groups.</p>Formule :C27H44O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.64Doxorubicinol
CAS :<p>Doxorubicinol is the major circulating metabolite of doxorubicin with antineoplastic acitivity.</p>Formule :C27H31NO11Couleur et forme :SolidMasse moléculaire :545.54trans-5-Hydroxyferulic acid
CAS :<p>trans-5-Hydroxyferulic acid is a useful organic compound for research related to life sciences. The catalog number is T126397 and the CAS number is 110642-42-7.</p>Formule :C10H10O5Couleur et forme :SolidMasse moléculaire :210.185DSPE-PEG5000-ANG
<p>DSPE-PEG5000-ANG is a PEGylated compound formed by DSPE and the dual-targeting ligand (Angiopep-2, ANG). ANG exhibits high binding efficacy to LRP1 and has been utilized for targeting glioma delivery. DSPE-PEG5000-ANG is applicable in drug delivery.</p>Couleur et forme :Odour SolidBBOX-IN-1
<p>BBOX-IN-1 (compound 58) is a potent BBOX inhibitor with an IC50 of 0.02 μM, and it is applicable in research related to triple-negative breast cancer (TNBC).</p>Formule :C18H17N3O6SCouleur et forme :SolidMasse moléculaire :403.41ER 50891 quarterhydrate
<p>ER 50891 quarterhydrate is a potent RARα (retinoic acid receptor α) antagonist that markedly diminishes the inhibitory effects of ATRA (all-trans retinoic acid</p>Formule :C29H24N2O2H2OCouleur et forme :SolidMasse moléculaire :437.02Adenosine deaminase
CAS :<p>Adenosine deaminase is an enzyme that catalyzes the irreversible deamination of 2'-deoxyadenosine and adenosine to 2'-deoxyinosine and inosine, respectively.</p>Degré de pureté :98%Couleur et forme :Solid16,16-dimethyl Prostaglandin A2
CAS :<p>16,16-dimethyl PGA2, a stable analog of PGA2, greatly reduces Sendai virus growth and helps mice survive influenza and cancer.</p>Formule :C22H34O4Couleur et forme :SolidMasse moléculaire :362.5IOX2-NH2-1
CAS :<p>IOX2-NH2-1 inhibits E. coli EGLN-3 (prolyl hydroxylase) with an IC50 of 0.02–1 μM.</p>Formule :C19H17N3O5Degré de pureté :98.77% - 99.91%Couleur et forme :SoildMasse moléculaire :367.3624R-Calcipotriol
CAS :<p>24R-Calcipotriol(PRI 2202) is an impurity of Calcipotriol which is a ligand of VDR-like receptors.</p>Formule :C27H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.60DSPE-PEG2000-LTLRWVGLMS
<p>DSPE-PEG2000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 is the receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG2000-LTLRWVGLMS can be utilized for drug delivery.</p>Couleur et forme :Odour SolidCP-LC-1422
<p>CP-LC-1422 is a homocysteine-derived ionizable amino lipid known for its efficient RNA delivery capabilities, enabling high-level protein expression in vivo. When formulated in lipid nanoparticles (LNP) and administered intravenously, it demonstrates significant spleen-targeting properties without observed notable toxicity.</p>Formule :C51H97N3O8S3Couleur et forme :SolidMasse moléculaire :975.64378Cholesterol glucuronide
CAS :<p>Cholesterol glucuronide is an endogenous metabolite of lipid generated by UDP glucuonyltransferase in the liver.</p>Formule :C33H54O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.78PTP1B-IN-25
<p>PTP1B-IN-25 (Compound 19) is an inhibitor of PTP1B with notable antiviral, antibacterial, and antidiabetic activities. It exhibits IC50 values of 0.37 μM for PTP1B, 8.6 μM for HIV, 3.7 μM for α-Glucosidase, and 29 μM for methicillin-resistant Staphylococcus aureus (MRSA).</p>Formule :C44H66O17Masse moléculaire :866.432-Nitrophenyl a-D-glucopyranoside
CAS :<p>2-Nitrophenyl a-D-glucopyranoside is a substrate of β-glucosidase [1] .</p>Formule :C12H15NO8Couleur et forme :SolidMasse moléculaire :301.25Creatine-d3
CAS :<p>Creatine-d3 is an isotopically labeled version of creatine. Creatine is an endogenous amino acid metabolite that plays a crucial role in cellular energy, particularly within muscles and the brain.</p>Formule :C4H9N3O2Couleur et forme :SolidMasse moléculaire :134.15DSPE-PEG1000-TH
<p>DSPE-PEG1000-TH is a PEG compound composed of DSPE and a pH-responsive cell-penetrating peptide (TH). In acidic environments, such as the tumor microenvironment, TH is activated, enabling the selective delivery of small molecules, oligonucleotides, proteins, and other agents into tumor cells.</p>Couleur et forme :Odour Solid11(R)-HETE
CAS :<p>11(R)-HETE aids in oocyte maturation in sea urchins and tentacle regeneration in hydras; it is also made by aspirin-influenced COX-2 and arachidonic acid.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473Sp-cAMPS triethylamine
CAS :<p>Sp-cAMPS triethylamine activates PKA I/II and inhibits PDE3A (Ki 47.6µM), binds PDE10 GAF (EC50 40µM).</p>Formule :C16H27N6O5PSCouleur et forme :SolidMasse moléculaire :446.46Hydroxy ritonavir
CAS :<p>Hydroxy ritonavir, a metabolite of ritonavir, functions as an inhibitor of the HIV protease, thereby serving as a treatment for HIV infection and AIDS [1].</p>Formule :C37H48N6O6S2Couleur et forme :SolidMasse moléculaire :736.94Equilenin
CAS :<p>Equilenin (E 400) is a natural estrogen that is an endocrine disruptor and has been used in breast cancer research.</p>Formule :C18H18O2Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :266.33Hepaxanthin
CAS :<p>Hepaxanthin is a carotenoid.</p>Formule :C20H30O2Couleur et forme :SolidMasse moléculaire :302.45RXP-407
CAS :<p>RXP 407 selectively inhibits ACE N-domain, preserving acetyl-Ser-Asp-Lys-Pro and not affecting angiotensin I in vivo.</p>Formule :C21H31N4O8PCouleur et forme :SolidMasse moléculaire :498.47DSPE-PEG1000-APRPG
<p>DSPE-PEG1000-APRPG is a PEG compound composed of DSPE and the APRPG peptide. It is applicable for drug delivery.</p>Couleur et forme :Odour Solid(+)-Menthofuran
<p>(+)-Menthofuran is a useful organic compound for research related to life sciences and the catalog number is T125544.</p>Formule :C10H14OCouleur et forme :SolidMasse moléculaire :150.221Deoxyadenosine diphosphate sodium
CAS :<p>Deoxyadenosine diphosphate sodium is a diphosphate nucleoside featuring deoxyadenosine as its nucleoside component. It plays a role in the synthesis and repair of DNA. Deoxyadenosine diphosphate sodium acts as an inhibitor of polynucleotide phosphorylase, thereby interfering with the polymerization of ADP and CDP.</p>Formule :C10H12N5Na3O9P2Couleur et forme :SolidMasse moléculaire :477.15DSPE-PEG5000-VIP
<p>DSPE-PEG5000-PP1 is a PEG compound composed of DSPE and the cell-penetrating peptide (TAT) peptide. DSPE-PEG2000-TAT is applicable for drug delivery.</p>Couleur et forme :Odour SolidDSPE-PEG5000-APRPG
<p>DSPE-PEG5000-APRPG is a PEG compound composed of DSPE and the APRPG peptide, utilized for drug delivery.</p>Couleur et forme :Odour SolidCefetamet Hydrochloride
CAS :<p>Cefetamet is a potent antibiotic to treat respiratory and urinary tract infections.</p>Formule :C14H16ClN5O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.89Leucomyosuppressin
CAS :<p>Leucomyosuppressin, isolated from head extracts of the cockroach Leucophaea maderae, inhibits evoked transmitter release at the mealworm neuromuscular junction.</p>Formule :C59H84N16O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1257.4182,3,4,6,7,8-Hexachlorodibenzofuran
CAS :<p>2,3,4,6,7,8-Hexachlorodibenzofuran (2,3,4,6,7,8-HxCDF) is a type of polychlorinated dibenzofuran (PCDF). It induces the expression of aryl hydrocarbon hydroxylase (AHH) and ethoxyresorufin-o-deethylase (EROD) genes in H-4-II-E rat hepatoma cells, with EC50 values of 0.687 and 0.575 nM, respectively.</p>Formule :C12H2Cl6OCouleur et forme :SolidMasse moléculaire :374.86Carbonic anhydrase inhibitor 29
<p>Carbonic anhydrase inhibitor29 (Compound 5d) is an inhibitor targeting carbonic anhydrase IX and XII, with an inhibition constant (Ki) of 26.6 nM for carbonic anhydrase IX and a Ki of 10.9 nM for carbonic anhydrase XII. Carbonic anhydrase inhibitor29 can be used in cancer research.</p>Couleur et forme :Odour SolidL-Proline-15N
CAS :<p>L-Proline-15N is an isotopically labeled amino acid suitable for metabolic research, aiding in the exploration of amino acid metabolism pathways and mechanisms.</p>Formule :C5H9NO2Couleur et forme :SolidMasse moléculaire :116.12ERAP1-IN-3
<p>ERAP1-IN-3 (compound 13) is a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1), with a pIC50 value of 8.6. ERAP1-IN-3 shows potential for research in cancer immunotherapy and autoimmune disease studies.</p>Formule :C22H22N2O4SCouleur et forme :SolidMasse moléculaire :410.49Probestin
CAS :<p>Probestin is an aminopeptidase M inhibitor, isolated from Streptomyces azureus MH663-2F6.</p>Formule :C26H38N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :502.60hCAII/IX-IN-1
<p>hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.</p>Formule :C23H22N4O7S2Couleur et forme :SolidMasse moléculaire :530.573SLC7A11-IN-3
<p>SLC7A11-IN-3 (Compound 42711_11) acts as an inhibitor of SLC7A11.</p>Couleur et forme :Odour Solid2,3-Dehydrosilybin B
CAS :<p>2,3-Dehydrosilybin B is a useful organic compound for research related to life sciences and the catalog number is T125883.</p>Formule :C25H20O10Couleur et forme :SolidMasse moléculaire :480.4218-Hydroxycorticosterone
CAS :<p>18-Hydroxycorticosterone is a corticosteroid and corticosterone derivative, which can lead to serious electrolyte imbalances.</p>Formule :C21H30O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :362.46Plipastatin A1
CAS :<p>Plipastatin A1, a lipopeptide isolated from B.</p>Formule :C72H110N12O20Couleur et forme :SolidMasse moléculaire :1463.71hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Formule :C24H17Cl2N3O3S2Couleur et forme :SolidMasse moléculaire :530.446O-Methyl Atorvastatin hemicalcium
CAS :<p>O-Methyl Atorvastatin, an Atorvastatin impurity, orally inhibits HMG-CoA reductase to lower blood lipids.</p>Formule :C68H76CaF2N4O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1187.449Acetildenafil
CAS :<p>Acetildenafil is an analog of the phosphodiesterase inhibitor sildenafil.</p>Formule :C25H34N6O3Couleur et forme :Off-White To Pale Yelow SolidMasse moléculaire :466.58α-Glucosidase-IN-73
<p>α-Glucosidase-IN-73 (compound 16b), an α-Glucosidase inhibitor, exhibits an IC 50 value of 0.158 μM and possesses the ability to activate PPAR γ. This compound is applicable in studies focusing on anti-diabetic and anti-inflammatory treatments.</p>Formule :C24H21N3O2SCouleur et forme :SolidMasse moléculaire :415.51Calcitroic acid
CAS :<p>Calcitroic acid is a vitamin D receptor (VDR) agonist that activates VDR-mediated transcription. It is the primary metabolite of 1,25-dihydroxyvitamin D3, showing the highest concentrations in the liver and mucosa of mice. The compound exhibits metabolic stability and extremely low toxicity.</p>Formule :C23H34O4Couleur et forme :SolidMasse moléculaire :374.514Terpendole I
CAS :<p>Terpendole I, from A. yamanashiensis, inhibits ACAT (IC50=145 μM), fights B. cereus/subtilis (MIC=100 μg/ml), and kills HeLa cells (IC50=52.6 μM).</p>Formule :C27H35NO5Couleur et forme :SolidMasse moléculaire :453.579UDP-glucosamine disodium
CAS :<p>UDP-GlcNAc disodium is a substrate for O-GlcNAc transferase and removed by O-GlcNAcase, produced in the hexosamine pathway regulated by GFAT.</p>Formule :C15H23N3Na2O16P2Couleur et forme :SolidMasse moléculaire :609.28tetranor-PGAM
CAS :<p>PGE2 is a biomarker for inflammation and disease; its unstable urinary metabolite, tetranor-PGEM, and its byproduct, tetranor-PGAM, indicate biosynthesis.</p>Formule :C16H22O6Couleur et forme :SolidMasse moléculaire :310.346(±)13(14)-DiHDPA
CAS :<p>(±)13(14)-DiHDPA is a metabolite of docosahexaenoic acid that is produced via oxidation by cytochrome P450 epoxygenases.</p>Formule :C22H34O4Couleur et forme :SolidMasse moléculaire :362.51FASN-IN-4 tosylate
CAS :<p>FASN-IN-4 tosylate: Fatty acid synthase inhibitor, IC50 10 nM; blocks SARS-CoV-2, EC50 18.6 nM.</p>Formule :C33H35N3O7S2Couleur et forme :SolidMasse moléculaire :649.782-Pentyl-1H-benzo[d]imidazole
CAS :<p>2-Pentyl-1H-benzo[d]imidazole is a micromolar level inhibitor of Cytochrome P450 1A1 and 2B1 and has antibacterial activity against Fusarium verticillioides.</p>Formule :C12H16N2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :188.27Tpp-CAQK
<p>Tpp-CAQK, a specially engineered mitochondrial compound, has been shown to improve phagocytosis of myelin debris by macrophages, reduce mitochondrial dysfunction and pro-inflammatory features, and enhance tissue repair and functional recovery in mice after spinal cord injury.</p>Formule :C40H54BrN6O7PSCouleur et forme :SolidMasse moléculaire :873.84Angiotensin I-13C6,15N (human, mouse, rat) TFA
<p>Angiotensin I-13C6,15N (human, mouse, rat) TFA is a labeled version of Angiotensin I, using isotopes 13C and 15N, specifically targeted for human, mouse, and rat studies. This compound serves as a precursor to angiotensin II, which is formed through the cleavage by angiotensin-converting enzyme (ACE).</p>Formule :C5713C6H89N1615NO14·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1303.42 (free base)Ninerafaxstat trihydrochloride
CAS :<p>Ninerafaxstat trihydrochloride shifts cellular metabolism to glucose oxidation from fatty acid oxidation.</p>Formule :C22H32Cl3N3O5Degré de pureté :99.71%Couleur et forme :SoildMasse moléculaire :524.878-iso Prostaglandin A1
CAS :<p>8-iso PGA1: an isoprostane, non-COX prostanoid, minor PGE1 impurity, biological effects unstudied.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472CAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formule :C23H21N5O3SCouleur et forme :SolidMasse moléculaire :447.51DJ-53
<p>DJ-53 (compound 68) is an orally active, phenyl-quinoline-based soluble epoxide hydrolase inhibitor.</p>Couleur et forme :Odour Solidα-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Couleur et forme :Odour SolidsEH inhibitor-20
<p>sEH inhibitor-20 is a metabolically stable, orally active sEH inhibitor with an IC50 of 0.2 nM. It exhibits significant analgesic and anti-inflammatory properties, making it a promising candidate for researching neuropathic pain.</p>Couleur et forme :Odour SolidKKII5
CAS :<p>KKII5 is a potent inhibitor of the lipoxygenase LOX-1 with an IC50 of 19 μM.KKII5 inhibits lipid peroxidation and enhances the ability of the active centers of</p>Formule :C16H14N2SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :266.36DSPE-PEG1000-THRPPMWSPVWP
<p>DSPE-PEG1000-THRPPMWSPVWP is a PEG compound composed of DSPE and the transferrin receptor (TfR) peptide. The THRPPMWSPVWP peptide binds to TfR and is subsequently internalized into cells expressing TfR.</p>Couleur et forme :Odour SolidDSPE-PEG2000-CTT2
<p>DSPE-PEG2000-CTT2 is a PEG compound consisting of DSPE and the gelatinase inhibitor CTT2 (CTTHWGFTLC). It possesses the ability to specifically target tumors. DSPE-PEG2000-CTT2 is suitable for drug delivery applications.</p>Couleur et forme :Odour SolidPantothenoylcysteine
CAS :<p>Pantothenoylcysteine is a bioactive chemical.</p>Formule :C12H22N2O6SCouleur et forme :SolidMasse moléculaire :322.3818:0,18:1 PS sodium
CAS :<p>18:0,18:1 PS sodium, a lipid found in synaptic vesicles and cholesterol, serves a role in metabolic research [1].</p>Formule :C42H79NNaO10PCouleur et forme :SolidMasse moléculaire :812.04DSPE-PEG5000-CREKA
<p>DSPE-PEG5000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide is utilized for targeting tumor cells and tumor vasculature, exhibiting anti-tumor activity. DSPE-PEG5000-CREKA is applicable in drug delivery systems.</p>Couleur et forme :Odour SolidHistamine glutarimide
CAS :<p>Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.</p>Formule :C10H13N3O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :207.23UK 227786
CAS :<p>UK 227786 is an inhibitor of phosphodiesterase 5 (PDE5), used for treatment of prostatic diseases.</p>Formule :C22H22Cl2N4O4Degré de pureté :99.9%Couleur et forme :SoildMasse moléculaire :477.34CBS-1114 HCl
CAS :<p>CBS-1114 HCl: 5-lipoxygenase inhibitor, anti-inflammatory, improves heart function, reduces heart's fat.</p>Formule :C13H14ClN3Degré de pureté :99.36%Couleur et forme :SoildMasse moléculaire :247.72Penicitide A
CAS :<p>Penicitide A: marine metabolite, moderately cytotoxic to A. brassicae, HepG2 cells.</p>Formule :C18H34O4Couleur et forme :SolidMasse moléculaire :314.46Diphenamid
CAS :<p>Diphenamid is a chemical compound from the group of acetamides and a herbicide. The effect is based on the inhibition of acetyl-CoA carboxylase.</p>Formule :C16H17NODegré de pureté :98%Couleur et forme :White Diphenamid Is A Colorless To Off-White Crystals Used As An HerbicideMasse moléculaire :239.31Fructosyl-lysine dihydrochloride
CAS :<p>Fructoselysine dihydrochloride, a Maillard reaction product and precursor to diabetes marker glucosepane.</p>Formule :C12H26Cl2N2O7Couleur et forme :SolidMasse moléculaire :381.25Glycerol-3-phosphate oxidase
CAS :<p>Glycerol-3-phosphate oxidase, from E. coli, is crucial in glycerol metabolism and phospholipid formation, producing electrons via oxidation.</p>Couleur et forme :SolidMP 518
CAS :<p>MP 518 is a PDE inhibitor with antihypertensive properties. It prevents the degradation of cAMP, leading to increased ICa levels, and counteracts the effects of β-adrenergic stimulation, resulting in vasodilation.</p>Formule :C10H11ClN2O2Couleur et forme :SolidMasse moléculaire :226.661α-Hydroxy VD4
CAS :<p>1alpha-Hydroxy VD4 can effectively induce the differentiation of monoblastic leukaemia U937, P39/TSU, and P31/FUJ cells.</p>Formule :C28H46O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.66PKM2-IN-3
CAS :<p>PKM2-IN-3 inhibits PKM2 kinase with 4.1 μM IC50, curbing glycolysis and NLRP3, reducing neuroinflammation.</p>Formule :C21H22O4Couleur et forme :SolidMasse moléculaire :338.403(+)-Geodin
CAS :<p>(+)-Geodin, a fungal metabolite, boosts fibrinolysis in BAECs (50-150 μM) and glucose uptake in rat adipocytes (1-100 μg/ml).</p>Formule :C17H12Cl2O7Couleur et forme :SolidMasse moléculaire :399.18Bromacil
CAS :<p>Bromacil, a substituted uracil herbicide used worldwide, is not readily biodegradable and therefore has consequences to the environment.</p>Formule :C9H13BrN2O2Couleur et forme :SolidMasse moléculaire :261.12Ono EI-601
CAS :<p>Ono EI-601 is the main metabolite of ONO-5046, the human neutrophil elastase inhibitor .</p>Formule :C15H14N2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.35TPH1-IN-1
<p>TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.</p>Formule :C21H18N6O4SCouleur et forme :SolidMasse moléculaire :450.47GLX481369
<p>GLX481369 is a redox-active substance that functions as an NOX4 inhibitor, exhibiting antioxidant effects [1].</p>Formule :C21H24ClN7OCouleur et forme :SolidMasse moléculaire :425.91Muvalaplin tetrahydrochloride
CAS :<p>Muvalaplin tetrahydrochloride (LY3473329) is an orally active lipoprotein (a)Lp(a) agent currently under investigation. Research on the oral formulation of Muvalaplin tetrahydrochloride is ongoing.</p>Formule :C42H58Cl4N4O6Couleur et forme :SolidMasse moléculaire :856.75Biotin sodium
CAS :<p>Biotin (Vitamin B7) sodium aids in metabolism, cell growth, fatty acid synthesis, and gluconeogenesis.</p>Formule :C10H15N2NaO3SCouleur et forme :SolidMasse moléculaire :266.29Quinaprilat hydrate
CAS :<p>Quinaprilat: active form of quinapril; treats heart failure, hypertension.</p>Formule :C23H28N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.481,2-Dihexadecyl-sn-glycero-3-PC
CAS :<p>1,2-Dihexadecyl-sn-glycero-3-PC can be used in related research in the field of life sciences. Its product number is T37043 and CAS number is 36314-47-3.</p>Formule :C40H84NO6PCouleur et forme :SolidMasse moléculaire :706.07Epicoccamide
CAS :<p>Epicoccamide is a marine fungal metabolite originally isolated from E. purpurascens.</p>Formule :C29H51NO9Couleur et forme :SolidMasse moléculaire :557.72DSPE-PEG1000-octreotide
<p>DSPE-PEG1000-Octreotide, a PEG compound formed from DSPE and Octreotide, acts as a somatostatin receptor agonist. Octreotide exhibits antitumor properties and induces apoptosis, making it useful in researching acromegaly. Additionally, DSPE-PEG1000-Octreotide is applicable in drug delivery.</p>Couleur et forme :Odour Solid4-Ethylbenzonitrile
CAS :<p>4-Ethylbenzonitrile is a micromolar level inhibitor of Cytochrome P450 2A6 with an IC50 value of 7.4 渭M.</p>Formule :C9H9NCouleur et forme :SolidMasse moléculaire :131.17Phospholipase D
CAS :<p>PLD is an enzyme in the phospholipase family, found across many life forms, and linked to diseases like diabetes and cancer.</p>Couleur et forme :SolidCoenzyme Q6
CAS :<p>Coenzyme Q6, also Ubiquinone 30, is a benzoquinone lipid aiding respiration and acting as an antioxidant.</p>Formule :C39H58O4Couleur et forme :SolidMasse moléculaire :590.882,3-Dihydroxybenzaldehyde
CAS :<p>2,3-Dihydroxybenzaldehyde exhibits activity against NADH dehydrogenase (Km = 35 µM) and can be used in biochemical experiments and drug synthesis.</p>Formule :C7H6O3Couleur et forme :SolidMasse moléculaire :138.12Estrone 3-glucuronide
CAS :<p>Deuterium-labeled Estrone 3-glucuronide is a key urinary marker for predicting fertility.</p>Formule :C24H30O8Couleur et forme :SolidMasse moléculaire :446.49Hydroorotic acid
CAS :<p>Hydroorotic acid（Dihydroorotic acid） is an endogenous metabolite，a potential biomarker for diabetic nephropathy and adrenal pheochromocytoma.</p>Formule :C5H6N2O4Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :158.11Benzo[b]furan-2-carboxaldehyde
CAS :<p>Benzo[b]furan-2-carboxaldehyde is a CYP2A6 inhibitor and can be used in biochemical experiments and drug synthesis.</p>Formule :C9H6O2Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :146.14Fumiquinazoline D
CAS :<p>Fumiquinazoline D, from A. fumigatus, inhibits Gram-positive/negative bacteria (MIC 8-16 μg/ml) and F. solani, C. albicans (MIC 32, 64 μg/ml).</p>Formule :C24H21N5O4Couleur et forme :SolidMasse moléculaire :443.4631,2,3,6,7,8-Hexachlorodibenzofuran
CAS :<p>1,2,3,6,7,8-Hexachlorodibenzofuran (1,2,3,6,7,8-HxCDF) is a type of polychlorinated dibenzofuran (PCDF). It promotes the expression of aryl hydrocarbon hydroxylase (AHH) and ethoxyresorufin-O-deethylase (EROD) genes in H-4-II-E rat hepatoma cells with EC50 values of 1.47 and 1.24 nM, respectively. 1,2,3,6,7,8-HxCDF also reduces rat body weight, causes thymic atrophy, and induces the expression of cytochrome P450 (CYP) subtype CYP1A1 and 4-chlorobiphenyl hydroxylase genes with EC50 values of 3.2, 0.9, 0.35, and 0.21 µmol/kg.</p>Formule :C12H2Cl6OCouleur et forme :SolidMasse moléculaire :374.86DSPE-PEG5000-LTLRWVGLMS
<p>DSPE-PEG5000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 serves as a receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG5000-LTLRWVGLMS can be utilized for drug delivery.</p>Couleur et forme :Odour Solid4-Hydroxybenzoic acid-d4
CAS :<p>4-Hydroxybenzoicacid-d4 is a deuterated form of 4-Hydroxybenzoicacid, which is a phenolic derivative of benzoic acid. It is effective in inhibiting most Gram-positive bacteria and some Gram-negative bacteria with an IC50 of 160 μg/mL.</p>Formule :C7H6O3Couleur et forme :SolidMasse moléculaire :142.15Cysteinylglycine acetate
<p>Cysteinylglycine acetate (Cys-Gly Acetate) is an acetate salt of Cysteinylglycine.</p>Formule :C7H14N2O5SDegré de pureté :99.49%Couleur et forme :SoildMasse moléculaire :238.26Doxorubicinol hydrochloride
CAS :<p>Doxorubicinol hydrochloride, also known as 13-Dihydroadriamycin hydrochloride, is a secondary alcohol metabolite derived from Doxorubicin.</p>Formule :C27H32ClNO11Couleur et forme :SolidMasse moléculaire :582.0Histone acetyltransferase p300 Inhibitor 4c
CAS :<p>2-Amino-4-(4-chlorophenyl)thiazole blocks hCA I/II, AChE, BChE with Ki: ~0.008, 0.124, 0.129, 0.083 µM.</p>Formule :C9H7ClN2SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :210.68DSPE-PEG5000-ESBP
<p>DSPE-PEG5000-ESBP is a PEG compound composed of DSPE and E-selectin binding peptide (ESBP). Acting as a tumor-targeting peptide, ESBP has the ability to specifically recognize and bind to receptors or markers on the surface of tumor cells.</p>Couleur et forme :Odour SolidDSPE-PEG2000-octreotide
<p>DSPE-PEG2000-Octreotide is a PEG compound composed of DSPE and Octreotide. Octreotide serves as a somatostatin receptor agonist with antitumor properties, mediating apoptosis and applicable in acromegaly research. DSPE-PEG2000-Octreotide is employed in drug delivery systems.</p>Couleur et forme :Odour SolidAcrihellin
CAS :<p>Acrihellin is a cardioactive steroid, a cardiotonic drug.</p>Formule :C29H38O7Couleur et forme :SolidMasse moléculaire :498.61PTP1B-IN-14
CAS :<p>PTP1B-IN-14 is a selective inhibitor of Protein Tyrosine Phosphatase 1B (PTP1B) that targets the allosteric site, exhibiting an inhibitory concentration (IC50)</p>Formule :C27H19N5O3S4Couleur et forme :SolidMasse moléculaire :589.73Reduced Haloperidol
CAS :<p>Reduced haloperidol, an active metabolite of haloperidol, binds dopamine D2/sigma-1 receptors and inhibits neurotransmitter reuptake.</p>Formule :C21H25ClFNO2Couleur et forme :SolidMasse moléculaire :377.88Cy3 IRGD-PEG-DSPE
<p>Cy3 IRGD-PEG-DSPE is a PEG phospholipid containing Cy3 dye, applicable for protein/nucleic acid labeling and fluorescence microscopy. It self-assembles in aqueous solutions to form micelles or lipid bilayers, which are useful for creating liposomes or nanoparticles for the delivery of nutrients, such as mRNA or DNA vaccines.</p>Couleur et forme :Odour Solid2′,3′-Di-O-acetyl-5′-deoxy-5-fluorocytidine
CAS :<p>2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine is a derivative of capecitabine.</p>Formule :C13H16FN3O6Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :329.28PDE5-IN-11
<p>PDE5-IN-11 is a potent PDE5 inhibitor, exhibiting an IC50 of 40 nM, and also displays inhibitory activity against PDE4 and PDE6 with IC50 values of 1.78 μM and</p>Couleur et forme :Odour SolidFASN-IN-6
<p>FASN-IN-6 (compound 44), a potent fatty acid biosynthesis (FAB) inhibitor, serves as an antibacterial agent, exhibiting minimum inhibitory concentrations (MICs</p>Formule :C24H16BrF4N3O2Couleur et forme :SolidMasse moléculaire :534.3Liarozole fumarate
CAS :<p>Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.</p>Formule :C17H13ClN4C4H4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.88Dilaurylglycerosulfate
CAS :<p>Dilauryl glycerol sulfate is an auxiliary emulsifier for lipase determination.</p>Formule :C27H56O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.8(Iso)-Dehydroemetine
CAS :<p>(Iso)-Dehydroemetine (Dehydroisoemetine, (+/-)-) is a compound with antispasmolytic effect on smooth muscle.</p>Formule :C29H38N2O4Degré de pureté :98.26% - 98.31%Couleur et forme :SoildMasse moléculaire :478.62SPL-334
CAS :<p>SPL-334 is an inhibitor of S-nitrosoglutathione reductase.</p>Formule :C22H15N3O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.50Crotonyl-CoA
CAS :<p>Crotonyl-CoA: key in butyric acid fermentation, lysine and tryptophan metabolism, crucial for fatty and amino acid processing.</p>Formule :C25H40N7O17P3SCouleur et forme :SolidMasse moléculaire :835.61PDK-IN-2
<p>PDK-IN-2 (Compound 1F), with an IC50 of 68 nM, is a potent PDK inhibitor that downregulates the expression of PDK1 and PDK4 in cells.</p>Formule :C17H23AsCl2N2O2S2Couleur et forme :SolidMasse moléculaire :497.33CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Formule :C19H16ClN3O5S2Couleur et forme :SolidMasse moléculaire :465.93BE2647
<p>BE2647 is a selective inhibitor of the mitochondrial pyruvate carrier (MPC), with an EC50 of 70 nM. It exhibits good metabolic stability in mouse liver microsomes. BE2647 can be utilized in research related to metabolic diseases, metabolic-associated steatotic liver disease (MASLD), or metabolic-associated steatohepatitis (MASH).</p>Formule :C13H7Br2N3O2Couleur et forme :SolidMasse moléculaire :397.022WAY-311610
CAS :<p>WAY-311610 is an HSD11B1 inhibitor targeting 11β-HSD1 enzyme with 0.34 μM IC; used for neuropathic and inflammatory pain research.</p>Formule :C16H13F3N4O2Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :350.3Reticulol
CAS :<p>Reticulol is an isocoumarin derivative produced by certain species of Streptomyces.</p>Formule :C11H10O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :222.19
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