Métabolisme

Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.

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8626 produits trouvés pour "Métabolisme"

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ACAT-IN-10 dihydrochloride
CAS :
- 199983-77-2
ACAT-IN-10 dihydrochloride, from EP1236468A1 example 197, inhibits acyl-CoA: cholesterol acyltransferase and reduces NF-κB transcription.
Formule :C₃₅H₅₈Cl₂N₄O₅S
Couleur et forme :Solid
Masse moléculaire :717.83
Ref: TM-T39411
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DSPE-PEG2000-CCK8
DSPE-PEG2000-CCK8 is a PEG compound comprising DSPE and Cholecystokinin-8 (CCK8). Cholecystokinin-8 exhibits peptide activity responsible for regulating gallbladder contractions and digestive system functions. DSPE-PEG2000-CCK8 is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01107
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DSPE-PEG2000-K237
DSPE-PEG2000-K237 is a PEG compound consisting of DSPE and the KDR-targeting peptide (K237). K237 functionally disrupts the interaction between VEGF and KDR receptors, resulting in significant biological effects such as inhibition of angiogenesis and tumor growth. DSPE-PEG2000-K237 is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01136
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N-Demethylerythromycin A
CAS :
- 992-62-1
N-Demethylerythromycin A, a metabolite of erythromycin from S. erythreus, may contaminate its preparations.
Formule :C₃₆H₆₅NO₁₃
Couleur et forme :Solid
Masse moléculaire :719.9
Ref: TM-T35711
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CAY10640
CAS :
- 1208549-68-1
CAY10640 (sEH inhibitor-1) is a potent, orally active, water-soluble epoxide hydrolase (sEH) inhibitor that inhibits sEH in humans and mice with IC50s of 0.4
Formule :C₁₇H₂₀F₃N₃O₃
Degré de pureté :99.63%
Couleur et forme :Solid
Masse moléculaire :371.35
Ref: TM-T38367
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L,L-Dityrosine
CAS :
- 63442-81-9
L,L-Dityrosine, a component found in the acid hydrolysates of various biological materials, such as insect cuticular resilin, plays a significant role in
Formule :C₁₈H₂₀N₂O₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :360.36
Ref: TM-T19396
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α-Glucosidase-IN-22
CAS :
- 2870693-28-8
α-Glucosidase-IN-22 is a selective inhibitor of α-glucosidase (IC50=0.64 μM).
Formule :C₁₄H₁₁N₃O₂S
Degré de pureté :99.66%
Couleur et forme :Soild
Masse moléculaire :285.32
Ref: TM-T67898
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Porfimer Sodium
CAS :
- 87806-31-3
Porfimer sodium, a sodium salt with photodynamic properties, targets tumor cells and induces cytotoxicity with 630 nm laser activation.
Formule :C₆₈H₇₄N₈O₁₁
Couleur et forme :Solid
Masse moléculaire :1179.385
Ref: TM-T34112
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(24R)-MC 976
CAS :
- 112828-09-8
(24R)-MC 976 is a derivative of Vitamin D3.
Formule :C₂₇H₄₂O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :414.62
Ref: TM-T16023L
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Aurantiamide benzoate
Aurantiamide benzoate is a useful organic compound for research related to life sciences and the catalog number is T125778.
Formule :C₃₂H₃₀N₂O₄
Couleur et forme :Solid
Masse moléculaire :506.602
Ref: TM-T125778
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PEG2000-C-DMG
CAS :
- 1019000-64-6
PEG2000-C-DMG is a pegylated lipid for Onpattro, reducing transthyretin production via RNAi.
Formule :C₁₂₆H₂₄₉NO₅₂
Couleur et forme :Solid
Masse moléculaire :2000 (Average)
Ref: TM-T74405
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DSPE-PEG2000-R6H4
DSPE-PEG2000-R6H4 is a PEG compound composed of DSPE and a pH-responsive cell-penetrating peptide (R6H4). The R6H4 component is utilized for pH-responsive anticancer drug delivery. Additionally, DSPE-PEG2000-R6H4 is applicable in drug delivery systems.
Couleur et forme :Odour Solid
Ref: TM-TCL-01155
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Amiquinsin hydrochloride monohydrate
CAS :
- 7125-70-4
Amiquinsin hydrochloride monohydrate is a compound known for its antihypertensive activity. It undergoes metabolism in the body, with its primary metabolite being 4-amino-6,7-dimethoxy-3-quinolineol hydrochloride monohydrate.
Formule :C₁₁H₁₅ClN₂O₃
Couleur et forme :Solid
Masse moléculaire :258.7
Ref: TM-T203204
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CH3OCO-D-CHA-Gly-Arg-pNA acetate
CAS :
- 80895-10-9
CH3OCO-D-CHA-Gly-Arg-pNA acetate serves as a chromogenic substrate for Factor Xa, as documented in sources [1] [2].
Formule :C₂₇H₄₂N₈O₉
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :622.67
Ref: TM-T78424
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Calcineurin Autoinhibitory Peptide
CAS :
- 148067-21-4
Selective inhibitor of Ca2+-calmodulin-dependent protein phosphatase (calcineurin) (IC50 ~ 10 μM). Does not inhibit PP1, PP2A or CaM kinase II (IC50 > 100 mM).
Formule :C₁₂₄H₂₀₅N₃₉O₃₉S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :2930.34
Ref: TM-TP2054
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α-Glycerophosphate Dehydrogenase-Triosephosphate
α-Glycerophosphate Dehydrogenase-Triosephosphate (GDH-TIM) is an enzyme mixture composed of glycerophosphate dehydrogenase (GDH) and triosephosphate isomerase (TIM). This compound is employed to measure transketolase (TK) activity in erythrocyte hemolysates, which helps in assessing vitamin B deficiency.
Ref: TM-TRP-00343
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N1,N12-Diacetylspermine dihydrochloride
CAS :
- 77928-71-3
Diacetylspermine 2HCl, a diacetylated Spermine, is a cancer biomarker linked to the disease's up-regulation.
Formule :C₁₄H₃₂Cl₂N₄O₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :359.34
Ref: TM-T40887
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Bilirubin oxidase
CAS :
- 80619-01-8
Bilirubin oxidase (BOD), a multi-copper enzyme, converts bilirubin to biliverdin, reduces O2 to H2O, and aids porphyrin metabolism.
Couleur et forme :Solid
Ref: TM-T76141
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Sorbitol-6-phosphate 2-dehydrogenase
CAS :
- 37250-69-4
Sorbitol-6-phosphate 2-dehydrogenase, a dehydrogenase enzyme produced by Escherichia coli, catalyzes the interconversion of D-sorbitol 6-phosphate and D-fructose 6-phosphate. The enzyme oxidizes D-sorbitol 6-phosphate at a rate ten times faster than it reduces D-fructose 6-phosphate, playing a role in various cellular processes.
Couleur et forme :Solid
Ref: TM-T200233
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C17 Sphingomyelin (d18:1/17:0)
CAS :
- 121999-64-2
C17 Sphingomyelin is a synthetic derivative of sphingomyelin that has been used as an internal standard for the quantification of sphingomyelin.
Formule :C₄₀H₈₁N₂O₆P
Couleur et forme :Solid
Masse moléculaire :717.05
Ref: TM-T38182
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Coumachlor
CAS :
- 81-82-3
Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.
Formule :C₁₉H₁₅ClO₄
Couleur et forme :Solid
Masse moléculaire :342.77
Ref: TM-T20616
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SHP2-D26
CAS :
- 2458219-65-1
SHP2-D26: potent SHP2 degrader binding VHL-1/SHP2, neddylation & proteasome-dependent.
Formule :C₅₆H₇₉ClN₁₂O₆S₂
Couleur et forme :Solid
Masse moléculaire :1115.9
Ref: TM-T40121
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Endoglycoceramidase I (EGCase I)
CAS :
- 2768502-40-3
EGCase I is a glycosidase used in biochemistry to transfer GSL sugars to 1-alkanols' primary hydroxyl groups.
Couleur et forme :Solid
Ref: TM-T75407
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17β-HSD10-IN-1
CAS :
- 2316765-78-1
17β-HSD10-IN-1 is a 17β-hydroxysteroid dehydrogenase type 10 inhibitor with blood-brain permeability and potency for the study of Alzheimer's disease.
Formule :C₁₆H₁₃ClN₄O₃S
Degré de pureté :98.47%
Couleur et forme :Soild
Masse moléculaire :376.82
Ref: TM-T77576
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(3S,5R)-Fluvastatin D6 sodium
CAS :
- 2249799-35-5
(3S,5R)-Fluvastatin D6 sodium: deuterium-labeled synthetic HMG-CoA reductase inhibitor with 8 nM IC50.
Formule :C₂₄H₂₅FNNaO₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :439.49
Ref: TM-T10128
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DSPE-PEG5000-NYZL1
DSPE-PEG5000-NYZL1 is a PEG compound composed of DSPE and NYZL1, where NYZL1 specifically binds to bladder cancer tissues and cells. DSPE-PEG5000-NYZL1 is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01194
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Gluconapin
CAS :
- 19041-09-9
Gluconapin serves as a precursor to sulforaphane, an effective anticancer isothiocyanate. It has been found to reduce the increase in plasma triglycerides induced by corn oil consumption in mice.
Formule :C₁₁H₁₉NO₉S₂
Couleur et forme :Solid
Masse moléculaire :373.4
Ref: TM-T203029
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KOTX1
CAS :
- 1788963-83-6
KOTX1 is an orally active and selective inhibitor of ALDH1A3. In a diabetic mouse model, KOTX1 improves glucose tolerance, insulin secretion, and blood glucose levels.
Formule :C₁₇H₁₆FN₃O₂
Couleur et forme :Solid
Masse moléculaire :313.33
Ref: TM-T203191
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(±)13(14)-EpDPA
CAS :
- 895127-64-7
Cytochrome P450 metabolism of polyunsaturated fatty acids produces numerous bioactive epoxide regioisomers.
Formule :C₂₂H₃₂O₃
Couleur et forme :Solid
Masse moléculaire :344.495
Ref: TM-T35496
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Oleic Acid-2,6-diisopropylanilide
CAS :
- 140112-65-8
Oleic acid-2,6-diisopropylanilide: ACAT inhibitor, IC50 7 nM; lowers LDL & raises HDL in high-fat fed rabbits/rats at 0.05%.
Formule :C₃₀H₅₁NO
Couleur et forme :Solid
Masse moléculaire :441.744
Ref: TM-T35603
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CTL-12
CTL-12, a fatty acid synthase (FASN) inhibitor (IC50: 2.5 μM), induces apoptosis and disrupts the cell cycle at the Sub-G1/S phase.
Formule :C₂₂H₂₁ClN₄O₄
Couleur et forme :Solid
Masse moléculaire :440.88
Ref: TM-T78873
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Z-Pro-prolinal
CAS :
- 88795-32-8
Z-Pro-prolinal, an orally active PREP inhibitor, IC50: 0.4 nM in porcine.
Formule :C₁₈H₂₂N₂O₄
Couleur et forme :Solid
Masse moléculaire :330.38
Ref: TM-T74044
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ω-Muricholic Acid
CAS :
- 6830-03-1
ω-Muricholic acid (ω-MCA) is a murine-specific secondary bile acid.
Formule :C₂₄H₄₀O₅
Couleur et forme :Solid
Masse moléculaire :408.57
Ref: TM-T40790
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Oglemilast
CAS :
- 778576-62-8
Oglemilast (GRC 3886) suppresses pulmonary cell infiltration, including eosinophilia and neutrophilia in vitro and in vivo.
Formule :C₂₀H₁₃Cl₂F₂N₃O₅S
Degré de pureté :99.82%
Couleur et forme :Solid
Masse moléculaire :516.3
Ref: TM-T16379
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tetranor-12(R)-HETE
CAS :
- 135271-51-1
Corneal metabolism of 12(R)-HETE yields 8(R)-HHxTrE via β-oxidation, losing four carbons from C-1.
Formule :C₁₆H₂₆O₃
Couleur et forme :Solid
Masse moléculaire :266.381
Ref: TM-T37772
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GQ-16
CAS :
- 870554-67-9
GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.
Formule :C₁₉H₁₆BrNO₃S
Degré de pureté :99.84%
Couleur et forme :Solid
Masse moléculaire :418.3
Ref: TM-T21955
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α-1,3-Galactosyltransferase (a1,3GalT)
CAS :
- 128449-51-4
a1,3GalT (GGTA1) synthesizes α-gal glycan by adding galactose from UDP to glycoproteins.
Couleur et forme :Solid
Ref: TM-T75417
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Propiverine N-oxide
CAS :
- 111071-96-6
Propiverine N-oxide is the primary metabolite of propiverine hydrochloride, and it influences bladder contraction and saliva secretion in miniature pigs.
Formule :C₂₃H₂₉NO₄
Couleur et forme :Solid
Masse moléculaire :383.48
Ref: TM-T203473
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PF-07238025
PF-07238025, a potent branched-chain ketoacid dehydrogenase kinase (BDK) inhibitor with an EC50 of 19 nM, enhances the stability of the BDK-BCKDH core E2
Formule :C₁₉H₁₈N₂O₃S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :354.42
Ref: TM-T79357
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Calciseptin
CAS :
- 178805-91-9
Calciseptine, a neurotoxin isolated from the Black Mamba (Dendroaspis p.
Formule :C₂₉₉H₄₆₈N₉₀O₈₇S₁₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :7036.12
Ref: TM-T80078
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Betulin ditosylate
CAS :
- 77265-02-2
Betulinditosylate is a derivative of Betulin, which functions as an SREBP inhibitor.
Formule :C₄₄H₆₂O₆S₂
Couleur et forme :Solid
Masse moléculaire :751.09
Ref: TM-T203693
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α-Glucosidase-IN-26
α-Glucosidase-IN-26 (Compound 7i), with an IC50 value of 4.63 µM, functions as an α-glucosidase inhibitor and is utilized in research related to type 2 diabetes
Formule :C₂₃H₂₂ClN₃O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :455.89
Ref: TM-T78731
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24, 25-Dihydroxy VD2
CAS :
- 58050-55-8
24, 25-Dihydroxy VD2 (24,25-Dihydroxy vitamin D2) is a metabolite of vitamin D2 and is an isomer of 25-hydroxyvitamin D.
Formule :C₂₈H₄₄O₃
Degré de pureté :99.63%
Couleur et forme :Solid
Masse moléculaire :428.65
Ref: TM-T19107
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7-Hydroxydichloromethotrexate
CAS :
- 751-75-7
7-Hydroxydichloromethotrexate is a methotrexate metabolite.
Formule :C₂₀H₂₀Cl₂N₈O₆
Couleur et forme :Solid
Masse moléculaire :539.33
Ref: TM-T29484
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L-Arginyl-L-alanine
CAS :
- 40968-45-4
L-Arginyl-L-alanine is a dipeptide and acts as a vasodilator derived from vascular smooth muscle. It can elevate the levels of cyclic guanosine monophosphate (cGMP) and nitrite in endothelium-denuded artery rings.
Formule :C₉H₁₉N₅O₃
Couleur et forme :Solid
Masse moléculaire :245.28
Ref: TM-TP2963
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PTP1B-IN-22
CAS :
- 86109-60-6
PTP1B-IN-22 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that inhibits glucose uptake in skeletal muscle L6 myotubes.
Formule :C₁₆H₁₂N₂O₃S₂
Degré de pureté :98.35%
Couleur et forme :Soild
Masse moléculaire :344.41
Ref: TM-T67893
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10'-Desmethoxystreptonigrin
CAS :
- 136803-89-9
'10'-Desmethoxystreptonigrin antibiotic derived from streptonigrin combats various bacteria and cancer cells, and inhibits p21ras farnesylation (IC50 = 21 nM).
Formule :C₂₄H₂₀N₄O₇
Couleur et forme :Solid
Masse moléculaire :476.445
Ref: TM-T35607
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Ozolinone
CAS :
- 56784-39-5
Ozolinone, an etozoline metabolite, is a loop diuretic treating hypertension and edema.
Formule :C₁₁H₁₆N₂O₃S
Couleur et forme :Solid
Masse moléculaire :256.32
Ref: TM-T33851
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Deschloro Cetirizine dihydrochloride
CAS :
- 83881-54-3
Deschloro Cetirizine Dihydrochloride: a Cetirizine impurity, second-gen antihistamine, and metabolite of hydroxyzine.
Formule :C₂₁H₂₈Cl₂N₂O₃
Couleur et forme :Solid
Masse moléculaire :427.365
Ref: TM-T73981
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LysoFos Glycerol 14
CAS :
- 326495-21-0
LysoFos Glycerol 14 is a useful organic compound for research related to life sciences. The catalog number is TF0117 and the CAS number is 326495-21-0.
Formule :C₂₀H₄₀NaO₉P
Couleur et forme :Solid
Masse moléculaire :478.495
Ref: TM-TF0117
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Carboxylesterase-IN-1
CAS :
- 2609018-59-7
Carboxylesterase-IN-1, a pesticide inhibits carboxylesterase at 50 μg/mL, akin to triphenyl phosphate.
Formule :C₃₀H₃₇BrN₂O₅
Couleur et forme :Solid
Masse moléculaire :585.539
Ref: TM-T40237
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16,16-dimethyl Prostaglandin A2
CAS :
- 41691-92-3
16,16-dimethyl PGA2, a stable analog of PGA2, greatly reduces Sendai virus growth and helps mice survive influenza and cancer.
Formule :C₂₂H₃₄O₄
Couleur et forme :Solid
Masse moléculaire :362.5
Ref: TM-T36041
+ Info
(R)-Mephenytoin
CAS :
- 71140-51-7
(R)-Mephenytoin ((–)-Mephenytoin) is the the R-enantiomer of Mephenytoin which is an anticonvulsant agent.
Formule :C₁₂H₁₄N₂O₂
Degré de pureté :99.95%
Couleur et forme :Solid
Masse moléculaire :218.25
Ref: TM-T36839
+ Info
Kijanimicin
CAS :
- 78798-08-0
Kijanimicin: antitumor, antibiotic with unique activity against Gram-positive, anaerobic bacteria, and malaria.
Formule :C₆₇H₁₀₀N₂O₂₄
Couleur et forme :Solid
Masse moléculaire :1317.527
Ref: TM-T25579
+ Info
Systemin
CAS :
- 137181-56-7
Systemin is an 18-amino acid polypeptide with the sequence AVQSKPPSKRDPPKMQTD that is found in Solanaceae plants (such as tomato and potato).
Formule :C₈₅H₁₄₄N₂₆O₂₈S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :2010.28
Ref: TM-TP1843
+ Info
13-cis-Retinyl acetate
CAS :
- 34356-31-5
13-cis-Retinyl acetate: active 13-cis isomer of Retinyl acetate, metabolite of vitamin A.
Formule :C₂₂H₃₂O₂
Couleur et forme :Solid
Masse moléculaire :328.49
Ref: TM-T74451
+ Info
Nampt-IN-10 trihydrochloride
Nampt-IN-10 trihydrochloride, a NAMPT inhibitor, is effective on A2780 & CORL23 cells (IC50: 5/19 nM); potential ADC payload.
Formule :C₂₇H₃₁Cl₃FN₅O₂
Couleur et forme :Solid
Masse moléculaire :582.92
Ref: TM-T74562
+ Info
Carboxylesterase
CAS :
- 9016-18-6
CESs are enzymes in mammalian liver hydrolyzing esters and other substrates in biochemical studies.
Couleur et forme :Solid
Ref: TM-T76123
+ Info
Mastoparan
CAS :
- 72093-21-1
Mastoparan is a peptide toxin from wasp venom. It has the chemical structure Ile-Asn-Leu-Lys-Ala-Leu-Ala-Ala-Leu-Ala-Lys-Lys-Ile-Leu-NH2.
Formule :C₇₀H₁₃₁N₁₉O₁₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1478.91
Ref: TM-TP1386
+ Info
α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid
CAS :
- 128253-12-3
α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid was identified as possible dual inhibitors for hLTA4H and hLTC4S enzymes by the computer-aided
Formule :C₂₃H₂₃NO₃
Degré de pureté :97.19% - 99.36%
Couleur et forme :Soild
Masse moléculaire :361.43
Ref: TM-T60040
+ Info
11-cis Retinol
CAS :
- 22737-96-8
11-cisRetinol, a vitamin A isomer, forms from a retinyl ester via RPE65. It's crucial for the visual cycle and cone pigment formation.
Formule :C₂₀H₃₀O
Couleur et forme :Solid
Masse moléculaire :286.459
Ref: TM-T38220
+ Info
Phosmet oxon
CAS :
- 3735-33-9
Phosmet oxon is a toxic byproduct of phosmet, an organophosphate insecticide for apple trees and various crops, targeting moths, aphids, mites, and flies.
Formule :C₁₁H₁₂NO₅PS
Couleur et forme :Solid
Masse moléculaire :301.26
Ref: TM-T34029
+ Info
Cellulose
CAS :
- 9004-34-6
Cellulose, an excipient, aids stability, solubility, and processing of drugs and affects their ADME.
Formule :C₁₂H₂₂O₁₁
Couleur et forme :Solid
Masse moléculaire :342.297
Ref: TM-T75329
+ Info
Diacetinase
Diacetinase, a member of the esterase family, catalyzes the hydrolysis of glyceryl diacetate (Diacetin). It is utilized in the measurement of lipase activity.
Couleur et forme :Odour Solid
Ref: TM-T200253
+ Info
Previtamin D3
CAS :
- 1173-13-3
Previtamin D3 is an intermediate in the production of cholecalciferol (vitamin D3).
Formule :C₂₇H₄₄O
Couleur et forme :Solid
Masse moléculaire :384.648
Ref: TM-T38553
+ Info
Glycerol-3-phosphate dehydrogenase
CAS :
- 9001-49-4
Glycerol-3-phosphate dehydrogenase from Saccharomyces cerevisiae is an enzyme that catalyzes the oxidation of glycerol-3-phosphate (G3P) to dihydroxyacetone phosphate (DHAP), playing a crucial role in glycerol metabolism and energy production. This enzyme acts as the rate-limiting step in glycerol production within Saccharomyces cerevisiae, regulating glycerol formation and accumulation to aid the yeast in adapting to hyperosmotic environments. Additionally, glycerol-3-phosphate dehydrogenase from Saccharomyces cerevisiae is relevant in research within the field of metabolic engineering.
Couleur et forme :Solid
Ref: TM-T89979
+ Info
Endocrocin
CAS :
- 481-70-9
Endocrocin is a useful organic compound for research related to life sciences. The catalog number is T124800 and the CAS number is 481-70-9.
Formule :C₁₆H₁₀O₇
Couleur et forme :Solid
Masse moléculaire :314.249
Ref: TM-T124800
+ Info
Fluticasone dimer impurity
CAS :
- 220589-37-7
Fluticasone dimer impurity: a dimer of Fluticasone Propionate, a potent corticosteroid.
Formule :C₄₃H₅₁F₅O₈S
Couleur et forme :Solid
Masse moléculaire :822.92
Ref: TM-T74169
+ Info
HIF-1 inhibitor-5
HIF-1 inhibitor-5 (Compound 16e) is a potent inhibitor of HIF-1, exhibiting an IC50 value of 2.38 μM and demonstrating significant anti-angiogenic potential [1
Formule :C₂₈H₃₅NO₅
Couleur et forme :Solid
Masse moléculaire :465.58
Ref: TM-T74804
+ Info
Di-O-demethylcurcumin
CAS :
- 60831-46-1
Di-O-demethylcurcumin (Bisdemethylcurcumin) is an intestinal metabolite of curcumin known for its neuroprotective properties.
Formule :C₁₉H₁₆O₆
Couleur et forme :Solid
Masse moléculaire :340.33
Ref: TM-T203667
+ Info
AM6701
CAS :
- 1010096-65-7
AM6701 is a novel highly potent inhibitor of human alpha/beta hydrolase domain 6 (habhd6)
Formule :C₁₇H₁₇N₅O
Degré de pureté :99.25%
Couleur et forme :Solid
Masse moléculaire :307.357
Ref: TM-T72020
+ Info
1-Palmitoyl Lysophosphatidic Acid
CAS :
- 22002-85-3
1-Palmitoyl Lysophosphatidic Acid boosts antibiotics against P. aeruginosa by binding Ca2+ and Mg2+.
Formule :C₁₉H₃₉O₇P
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :410.48
Ref: TM-T37282
+ Info
Imperatoxin A TFA
Imperatoxin A TFA, a peptide toxin derived from the venom of the African scorpion Pandinus imperator, acts as an activator of Ca2+-release channels/ryanodine receptors (RyRs). It facilitates the influx of Ca2+ from the sarcoplasmic reticulum into the cell.
Formule :C₁₄₈H₂₅₄N₅₈O₄₅S₆·xC₂HF₃O₂
Couleur et forme :Solid
Masse moléculaire :3758.35 (free base)
Ref: TM-TP2838
+ Info
IONIS PTP1BRx
CAS :
- 1403406-29-0
IONIS PTP1BRx (ISIS 404173) acts as an antisense inhibitor of protein tyrosine phosphatase 1B (PTP-1B). This compound exhibits anti-diabetic properties, making it suitable for research into insulin resistance related to obesity and type 2 diabetes.
Couleur et forme :Solid
Ref: TM-T200394
+ Info
SGK1-IN-4
CAS :
- 1628048-93-0
SGK1-IN-4 is a selective inhibitor of SGK1 and can be used in studies about osteoarthritis.
Formule :C₂₃H₂₁ClFN₅O₄S
Degré de pureté :97.03%
Couleur et forme :Solid
Masse moléculaire :517.96
Ref: TM-T9977
+ Info
Phosphofructokinase
CAS :
- 9001-80-3
Phosphofructokinase, a crucial glycolytic enzyme, catalyzes the conversion of fructose-6-phosphate to fructose-1,6-bisphosphate in the glycolysis pathway. Its activity is inhibited by the binding of Phosphoenolpyruvate (PEP), which regulates the rate of glycolysis. Additionally, Phosphofructokinase is utilized in the measurement of fructose-6-phosphate (fructose-6-phosphate) levels.
Couleur et forme :Solid
Ref: TM-T200040
+ Info
Neo-inositol
CAS :
- 488-54-0
Neo-Inositol, a stable, polar compound, is a rare natural inositol stereoisomer.
Formule :C₆H₁₂O₆
Couleur et forme :Solid
Masse moléculaire :180.16
Ref: TM-T33632
+ Info
Efmoroctocog alfa
CAS :
- 1270012-79-7
Efmoroctocog alfa, a recombinant human coagulation factor VIII-Fc fusion protein (rFVIIIFc), serves as a therapeutic agent for Hemophilia A research [1].
Couleur et forme :Solid
Ref: TM-T82499
+ Info
Bipolamine G
CAS :
- 1357824-71-5
Bipolamine G is an antibacterial polyketide alkaloid [1] .
Formule :C₂₁H₂₈N₂O₄
Couleur et forme :Solid
Masse moléculaire :372.46
Ref: TM-T75482
+ Info
Hexokinase (ScHEX1)
CAS :
- 9001-51-8
ScHEX1, a glycolytic hexokinase, is blocked by n-acetylglucosamine, detaching from the mitochondrial membrane and activating NLRP3 inflammasome.
Couleur et forme :Solid
Ref: TM-T76111
+ Info
Dihydrocarminomycin
CAS :
- 62182-86-9
Dihydrocarminomycin is an anthracycline antibiotics.
Formule :C₂₆H₂₉NO₁₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :515.515
Ref: TM-T24000
+ Info
Penicillinase
CAS :
- 9001-74-5
Penicillinase is a β-lactamase and secretory enzyme capable of degrading and inactivating penicillin and similar compounds.
Couleur et forme :Solid
Ref: TM-T75391
+ Info
2-Chlorophenylboronic acid
CAS :
- 3900-89-8
2-Chlorophenylboronic acid: A monohalogenated phenylboronic acid used in drug synthesis and as a fatty acid amidase inhibitor.
Formule :C₆H₆BClO₂
Degré de pureté :99.42%
Couleur et forme :Solid
Masse moléculaire :156.37
Ref: TM-T77513
+ Info
hCAII/XII-IN-1
hCAII/XII-IN-1 (compound 4l) is a potent inhibitor of hCAXII and hCAII, with Ki values of 8.4 nM and 9.4 nM, respectively. It plays a significant role in cancer research.
Formule :C₂₂H₂₀N₄O₆S₂
Couleur et forme :Solid
Masse moléculaire :500.547
Ref: TM-T204716
+ Info
Fexofenadine Impurity F
CAS :
- 185066-33-5
Fexofenadine Impurity F: byproduct of anti-allergy drug for hay fever and hives.
Formule :C₃₁H₃₇NO₄
Couleur et forme :Solid
Masse moléculaire :487.63
Ref: TM-T73972
+ Info
CAY10581
CAS :
- 1018340-07-2
CAY10581, a derivative of pyranonaphthoquinone, serves as a highly specific and reversible uncompetitive inhibitor of IDO, demonstrating potency with an IC50
Formule :C₂₂H₂₁NO₄
Couleur et forme :Solid
Masse moléculaire :363.41
Ref: TM-T73351
+ Info
C18:1 Ceramide (d18:1/18:1(9Z))
CAS :
- 5966-28-9
C18:1 Ceramide (d18:1/18:1(9Z)) is a ceramide, and C18:1-Ceramide levels are elevated in overweight and insulin-resistant , advanced ovarian cancer.
Formule :C₃₆H₆₉NO₃
Degré de pureté :99.96%
Couleur et forme :Solid
Masse moléculaire :563.94
Ref: TM-T35808
+ Info
Antiproliferative agent-12
Antiproliferative agent-10, a ruthenium(II) complex, inhibits cancer by blocking mitochondrial calcium uptake.
Formule :C₄₆H₄₀Cl₂N₆P₂Ru
Couleur et forme :Solid
Masse moléculaire :910.79
Ref: TM-T74921
+ Info
Folipastatin
CAS :
- 139959-71-0
Folipastatin is a useful organic compound for research related to life sciences. The catalog number is T125927 and the CAS number is 139959-71-0.
Formule :C₂₃H₂₄O₅
Couleur et forme :Solid
Masse moléculaire :380.44
Ref: TM-T125927
+ Info
HMG-CoA Reductase-IN-1
HMG-CoA Reductase-IN-1 is an inhibitor of HMG-CoA reductase, demonstrating strong inhibitory activity on HMGR and affinity for OATP1B1, with pIC50 and pKm
Formule :C₂₇H₂₉N₃O₇
Couleur et forme :Solid
Masse moléculaire :507.54
Ref: TM-T79520
+ Info
Cecropin B
CAS :
- 80451-05-4
Cecropin B is a small antibacterial peptide from the giant silkmoth, Hyalophora cecropia.
Formule :C₁₇₆H₃₀₂N₅₂O₄₁S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :3834.74
Ref: TM-TP1313
+ Info
GLUT1-IN-1
GLUT1-IN-1 inhibits GLUT1; cytotoxic to HeLa, A549, HepG2 (IC50: 5.49, 11.14, 8.73 μM); potential in PDT and cancer research.
Formule :C₂₅H₃₁BF₂I₂N₆O₇
Couleur et forme :Solid
Masse moléculaire :830.17
Ref: TM-T74962
+ Info
MAGL-IN-21
MAGL-IN-21 (Compound (S)-6) is a selective inhibitor of monoacylglycerol lipase (MAGL) with an IC50 of 1.59 nM.
Formule :C₂₀H₂₄ClFN₂O₄
Couleur et forme :Solid
Masse moléculaire :410.867
Ref: TM-T204530
+ Info
Methiocarb
CAS :
- 2032-65-7
Methiocarb is a carbamate insecticide acting as a reversible AChE or ChE inhibitor, inducing oxidative stress in rats.
Formule :C₁₁H₁₅NO₂S
Degré de pureté :98.49%
Couleur et forme :Colorless Crystals Immobilizing Agent For Birds Acaricide And Molluscicide (Epa 1998)
Masse moléculaire :225.31
Ref: TM-T21464
+ Info
DOSPA (hydrochlorid)
CAS :
- 913194-16-8
DOSPA hydrochloride is a cationic lipid utilized in the formation of lipid nanoparticles.
Formule :C₅₄H₁₁₅Cl₅N₆O₃
Couleur et forme :Solid
Masse moléculaire :1073.79
Ref: TM-TYD-02047
+ Info
FASN-IN-6
FASN-IN-6 (compound 44), a potent fatty acid biosynthesis (FAB) inhibitor, serves as an antibacterial agent, exhibiting minimum inhibitory concentrations (MICs
Formule :C₂₄H₁₆BrF₄N₃O₂
Couleur et forme :Solid
Masse moléculaire :534.3
Ref: TM-T79416
+ Info
PROTAC SGK3 degrader-1
CAS :
- 2381320-35-8
PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC coupler that targets SGK3 and binds ligands to VH032 VHL to induce endogenous SGK3 degradation.
Formule :C₅₇H₇₃FN₁₀O₁₁S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1157.38
Ref: TM-T13847
+ Info
Prostaglandin D1
CAS :
- 17968-82-0
Prostaglandin D1 is a prostaglandin that has contraction and relaxation effects on isolated human arteries and can inhibit ADP-induced platelet aggregation (
Formule :C₂₀H₃₄O₅
Couleur et forme :Solid
Masse moléculaire :354.48
Ref: TM-T36544
+ Info
Cholesterol nervonate
CAS :
- 60758-73-8
Cholesterol nervonate is a cholesterol ester found in human meibum, used experimentally in synthetic liposomes for biophysics and drug delivery research.
Formule :C₅₁H₉₀O₂
Couleur et forme :Solid
Masse moléculaire :735.26
Ref: TM-T77231
+ Info
DSPE-PEG3000-R6H4
DSPE-PEG3000-R6H4 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (R6H4). R6H4 is applicable for pH-responsive anticancer drug delivery. DSPE-PEG3000-R6H4 can be utilized for drug delivery purposes.
Couleur et forme :Odour Solid
Ref: TM-TCL-01092
+ Info
Desbutyl Lumefantrine D9
CAS :
- 1346606-35-6
Desbutyl Lumefantrine D9, a deuterium-labeled metabolite of Lumefantrine, exhibits the incorporation of deuterium atoms.
Formule :C₂₆H₂₄Cl₃NO
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :481.89
Ref: TM-T19275
+ Info
Cystocholic acid
CAS :
- 73386-01-3
Cystocholic acid is a metabolite of bile acids, possessing antimicrobial potential.
Formule :C₂₇H₄₅NO₇
Couleur et forme :Solid
Masse moléculaire :495.65
Ref: TM-T203240
+ Info
Citrulline malate
CAS :
- 70796-17-7
Citrulline malate is a cpd of anti-fatigue.
Formule :C₁₀H₁₉N₃O₈
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :309.27
Ref: TM-T20200
+ Info
(±)16-HDHA
CAS :
- 90780-51-1
(±)16-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.
Formule :C₂₂H₃₂O₃
Couleur et forme :Solid
Masse moléculaire :344.495
Ref: TM-T35512
+ Info
ACAT-IN-4 hydrochloride
CAS :
- 199984-46-8
ACAT-IN-4 hydrochloride is a potent ACAT inhibitor and blocks NF-κB transcription.
Formule :C₃₂H₅₁ClN₂O₅S
Couleur et forme :Solid
Masse moléculaire :611.28
Ref: TM-T39416
+ Info
Desoxycarbadox
CAS :
- 55456-55-8
Desoxycarbadox, derived from Carbadox, is a quinoxaline-di-N-oxide antibiotic compound.
Formule :C₁₁H₁₀N₄O₂
Couleur et forme :Solid
Masse moléculaire :230.227
Ref: TM-T40635
+ Info
β-Tetralone
CAS :
- 530-93-8
β-Tetralone (2-Tetralone) is a vital drug synthesis precursor with complex pharmacological properties in combating neurological disorders. Cost-effective and quality-assured.
Formule :C₁₀H₁₀O
Degré de pureté :97.26% - 99.18%
Couleur et forme :Clear To Yellow Liquid
Masse moléculaire :146.19
Ref: TM-T0660
+ Info
(+)-Menthofuran
(+)-Menthofuran is a useful organic compound for research related to life sciences and the catalog number is T125544.
Formule :C₁₀H₁₄O
Couleur et forme :Solid
Masse moléculaire :150.221
Ref: TM-T125544
+ Info
N-acetyl Dapsone
CAS :
- 565-20-8
N-acetyl Dapsone is an anti-inflammatory and antimicrobial compound widely used in the treatment of leprosy, malaria, acne and various immune disorders.
Formule :C₁₄H₁₄N₂O₃S
Degré de pureté :99.86%
Couleur et forme :White
Masse moléculaire :290.34
Ref: TM-T35903
+ Info
TRH Precursor Peptide
Thyrotropin Releasing Hormone Precursor Peptide
Formule :C₄₂H₇₅N₁₉O₁₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1006.17
Ref: TM-TP2201
+ Info
1α, 24, 25-Trihydroxy VD2
CAS :
- 457048-34-9
1alpha, 24, 25-Trihydroxy VD2 is a vitamin D analog.
Formule :C₂₈H₄₄O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :444.65
Ref: TM-T19090
+ Info
5-Formylcytosine
CAS :
- 4425-59-6
5-Formylcytosine (5FC) is a rare mammalian DNA base aiding in demethylation, altering helix structure, and affecting RNA polymerase II activity.
Formule :C₅H₅N₃O₂
Couleur et forme :Solid
Masse moléculaire :139.11
Ref: TM-T29453
+ Info
Galactosylhydroxylysine hydrochloride
Galactosylhydroxylysine hydrochloride, found in bone collagen, is higher in metabolic bone loss due to resorption.
Formule :C₁₂H₂₅ClN₂O₈
Couleur et forme :Solid
Masse moléculaire :360.79
Ref: TM-T73770
+ Info
AP-III-a4 hydrochloride
CAS :
- 2070014-95-6
AP-III-a4 hydrochloride (ENOblock hydrochloride) is a direct enolase (enolase) inhibitor that inhibit metastasis and affect glucose homeostasis.
Formule :C₃₁H₄₄ClFN₈O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :631.18
Ref: TM-T6759L
+ Info
trans-2-Hexadecenoyl-L-carnitine
CAS :
- 26145-55-1
trans-2-Hexadecenoyl-L-carnitine is an endogenous metabolite in urine[1].
Formule :C₂₃H₄₃NO₄
Couleur et forme :Solid
Masse moléculaire :397.59
Ref: TM-T37640
+ Info
4''-C18 EGCG
4''-C18 EGCG is an effective inhibitor of α-amylase and α-glucosidase, with IC50 values of 3.74 and 0.81 μM, respectively. This compound suppresses carbohydrate-hydrolyzing enzymes, reduces oxidative stress and inflammation, and exhibits anti-diabetic activity. Moreover, 4''-C18 EGCG downregulates pro-inflammatory cytokines and demonstrates cytotoxicity at 50 μM against primary human peripheral blood mononuclear cells (PBMC), as well as non-cancerous cell lines 3T3-L1 and HEK 293.
Formule :C₄₀H₅₄O₁₁
Couleur et forme :Solid
Masse moléculaire :710.85
Ref: TM-T200812
+ Info
hCAII/IX-IN-1
hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.
Formule :C₂₃H₂₂N₄O₇S₂
Couleur et forme :Solid
Masse moléculaire :530.573
Ref: TM-T204640
+ Info
GGACK hydrochloride
GGACK (H-Glu-Gly-Arg-CMK) hydrochloride is an irreversible substrate-like inhibitor of the serine protease urokinase-type plasminogen activator (uPA).
Formule :C₁₄H₂₆Cl₂N₆O₅
Couleur et forme :Solid
Masse moléculaire :428.13417
Ref: TM-T207613
+ Info
MK-8262
CAS :
- 1432054-03-9
MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.
Formule :C₃₅H₂₅F₉N₂O₅
Couleur et forme :Solid
Masse moléculaire :724.58
Ref: TM-T38908
+ Info
hCAIX/XII-IN-7
Compound 3e (hCAIX/XII-IN-7) is a potent inhibitor of human carbonic anhydrase (hCA) isozymes IX and XII, displaying inhibitory constants (Kis) of 503.7 nM for
Formule :C₁₇H₁₄N₆O₃S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :382.4
Ref: TM-T79748
+ Info
γ-Globulins from human blood
CAS :
- 9007-83-4
γ-Globulins, a protein fraction found in human blood, comprise a class of proteins with potent antibody activity that safeguards against bacterial and viral
Couleur et forme :Solid
Ref: TM-T41030
+ Info
(±)7(8)-EpDPA
CAS :
- 895127-66-9
Docosahexaenoic acid is the most abundant ω-3 fatty acid in neural tissues, especially in the brain and retina.
Formule :C₂₂H₃₂O₃
Couleur et forme :Solid
Masse moléculaire :344.495
Ref: TM-T35497
+ Info
SHP2-IN-36
SHP2-IN-36 (Compound B8) is an allosteric inhibitor of SHP2 with an IC50 of 9.0 nM, and it exhibits an IC50 of 40 nM against p-ERK. Moreover, SHP2-IN-36 demonstrates significant antitumor activity in the KYSE520 xenograft mouse model and is applicable for research in the field of antitumor studies.
Couleur et forme :Odour Solid
Ref: TM-T206615
+ Info
Epicoccamide
CAS :
- 606139-26-8
Epicoccamide is a marine fungal metabolite originally isolated from E. purpurascens.
Formule :C₂₉H₅₁NO₉
Couleur et forme :Solid
Masse moléculaire :557.72
Ref: TM-T31651
+ Info
IPH5201
IPH5201 is a human IgG1 monoclonal antibody (mAb) targeting ENTPD1/CD39. It enhances the accumulation of immunostimulatory ATP released by tumor cells undergoing combination chemotherapy (CT) and reduces the levels of immunosuppressive adenosine (Ado) in the tumor microenvironment (TME). IPH5201 is useful for research on antitumor immunity. Recommended isotype control: Human IgG1 kappa, Isotype Control.
Couleur et forme :Odour Liquid
Ref: TM-T9901A-1061
+ Info
NAADP sodium
NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.
Formule :C₂₁H₂₇N₆O₁₈P₃
Couleur et forme :Solid
Masse moléculaire :744.39
Ref: TM-T35922
+ Info
CP-LC-1422
CP-LC-1422 is a homocysteine-derived ionizable amino lipid known for its efficient RNA delivery capabilities, enabling high-level protein expression in vivo. When formulated in lipid nanoparticles (LNP) and administered intravenously, it demonstrates significant spleen-targeting properties without observed notable toxicity.
Formule :C₅₁H₉₇N₃O₈S₃
Couleur et forme :Solid
Masse moléculaire :975.64378
Ref: TM-TCL-01213
+ Info
DSPE-PEG2000-T7
DSPE-PEG2000-T7 is a PEG compound composed of DSPE and the transferrin receptor peptide (T7). The T7 peptide (HAIYPRH) specifically binds to TfR, making DSPE-PEG2000-T7 useful for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01139
+ Info
Myristelaidic Acid
CAS :
- 50286-30-1
Myristelaidic Acid is a natural product for research related to life sciences. The catalog number is T37358 and the CAS number is 50286-30-1.
Formule :C₁₄H₂₆O₂
Couleur et forme :Solid
Masse moléculaire :226.35
Ref: TM-T37358
+ Info
LL P880 β
CAS :
- 41164-59-4
LL P880 beta is a fungal metabolite.
Formule :C₁₁H₁₈O₅
Couleur et forme :Solid
Masse moléculaire :230.26
Ref: TM-T32808
+ Info
VDR agonist 2
VDR agonist 2 (compound 16i), a vitamin D receptor (VDR) agonist, effectively inhibits TGF-β1-induced hepatic stellate cell (HSC) activation, demonstrating
Formule :C₂₀H₂₁F₃O₃
Couleur et forme :Solid
Masse moléculaire :366.37
Ref: TM-T78944
+ Info
Butyryl-Coenzyme A trisodium
Butyryl-Coenzyme A (trisodium) is a microbial metabolite that can be synthesized into butyric acid or butyrate.
Formule :C₂₅H₃₉N₇Na₃O₁₇P₃S
Masse moléculaire :903.10291
Ref: TM-TYD-02789
+ Info
DL-TBOA ammonium
CAS :
- 2093503-71-8
DL-TBOA ammonium is a potent EAAT inhibitor with IC50 (6-70 μM) and Ki (3.2-42 μM) against EAAT1-5, blocking [14C]glutamate uptake.
Formule :C₁₁H₁₆N₂O₅
Couleur et forme :Solid
Masse moléculaire :256.258
Ref: TM-T39510
+ Info
DSPE-PEG1000-EB1
DSPE-PEG1000-EB1 is a PEG compound composed of DSPE and a pH-responsive cell-penetrating peptide (EB1). It is utilized for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01134
+ Info
MS1262-C3-amide-C10-amine
MS1262-C3-amide-C10-amine is an E3 Ligase Ligand-Linker conjugate. It includes a GLP ligand targeting the E3 ligase SPOP and a PROTAC linker. This compound can be utilized in designing PROTACs such as example [MS479].
Couleur et forme :Odour Solid
Ref: TM-T206748
+ Info
Trimipramine N-oxide
CAS :
- 14171-70-1
Trimipramine N-oxide, a trimipramine metabolite, inhibits hNAT, hSERT, hDAT, and hOCT1/2 with IC50s 11.7-27.4 nM; for depression/anxiety research.
Formule :C₂₀H₂₆N₂O
Couleur et forme :Solid
Masse moléculaire :310.43
Ref: TM-T74582
+ Info
11-epi-Chaetomugilin I
CAS :
- 1319729-88-8
11-epi-Chaetomugilin I, from Chaetomium globosum, has cytotoxic effects against P388, HL-60, L1210 leukemia, and KB carcinoma cells.
Formule :C₂₂H₂₇ClO₅
Couleur et forme :Solid
Masse moléculaire :406.9
Ref: TM-T75453
+ Info
Cellohexaose
CAS :
- 2478-35-5
Cellohexaose, a cellulose-derived polymer, comprises at least two β(1-4) linked D-glucose units.
Formule :C₃₆H₆₂O₃₁
Couleur et forme :Solid
Masse moléculaire :990.86
Ref: TM-T75639
+ Info
Sirtuin modulator 2
CAS :
- 667910-69-2
Sirtuin modulator 2 (N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide) exhibits antidiabetic, anti-inflammatory and antitumor activities.
Formule :C₁₉H₁₅N₃O₂S
Degré de pureté :99.67%
Couleur et forme :Solid
Masse moléculaire :349.41
Ref: TM-T9999
+ Info
MPO-IN-6
MPO-IN-6 (compound ADC) is an electrophilic agent with excellent antioxidant and anti-inflammatory properties. It acts as an inhibitor of myeloperoxidase (MPO), dipeptidyl peptidase-4 (DPP-4), and α-glucosidase (α-GD), with IC50 values of 10 μM, 31.02 μM, and 46.05 μM, respectively. MPO-IN-6 may serve as a potential cardiovascular protective agent.
Formule :C₁₆H₁₂N₂O₆
Masse moléculaire :328.06954
Ref: TM-T209254
+ Info
α-Amylase-IN-11
α-Amylase-IN-11 (compound C5f) is an α-amylase inhibitor with an IC50 of 0.56 μM, effective in reducing glucose levels in vivo. Additionally, it exhibits moderate inhibitory activity against α-glucosidase with an IC50 of 11.03 μM. In mouse models, α-Amylase-IN-11 significantly decreases glucose concentrations, indicating its potential for diabetes research.
Formule :C₂₂H₁₈N₄OS
Couleur et forme :Solid
Masse moléculaire :386.47
Ref: TM-T205363
+ Info
Mitochondrial respiration-IN-1 hydrobromide
Mitochondrial inhibitor 49 (respiration-IN-1 hydrobromide, IC50=8.8 mg/mL) from US20110301180A1 reduces platelet respiration.
Couleur et forme :Solid
Ref: TM-T37657
+ Info
Coproporphyrin III
CAS :
- 14643-66-4
Coproporphyrin III is a derivative of porphyrin.
Formule :C₃₆H₃₈N₄O₈
Degré de pureté :98%
Couleur et forme :Purple Xtl
Masse moléculaire :654.72
Ref: TM-T19247
+ Info
Laprafylline
CAS :
- 90749-32-9
Laprafylline: Xanthine derivative, blocks bronchoconstriction & tumor growth, competes with serotonin, resists histamine at high levels.
Formule :C₂₉H₃₆N₆O₂
Degré de pureté :>99.99%
Couleur et forme :Solid
Masse moléculaire :500.64
Ref: TM-T68090
+ Info
2-Methoxy-4-propylphenol
CAS :
- 2785-87-7
2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.
Formule :C₁₀H₁₄O₂
Couleur et forme :Solid
Masse moléculaire :166.22
Ref: TM-TN9775
+ Info
DSPE-PEG1000-YIGSR
DSPE-PEG1000-YIGSR is a PEG compound consisting of DSPE and the biomimetic peptide YIGSR. YIGSR interacts with the 67 kDa laminin-binding protein (LBP) to enhance adhesion and spreading of various cell types, including endothelial cells, fibroblasts, and smooth muscle cells. DSPE-PEG1000-YIGSR is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01157
+ Info
(R,S)-Carvedilol Glucuronide
CAS :
- 114869-83-9
(R,S)-Carvedilol glucuronide is a racemic mix, metabolized by UGT1A1, UGT2B4, and UGT2B7.
Formule :C₃₀H₃₄N₂O₁₀
Couleur et forme :Solid
Masse moléculaire :582.606
Ref: TM-T35845
+ Info
CNBCA
CNBCA, a selective and potent competitive inhibitor of the SHP2 enzyme, exhibits an IC50 value of 0.87 μM.
Formule :C₂₆H₃₄O₅
Couleur et forme :Solid
Masse moléculaire :426.55
Ref: TM-T79311
+ Info
PDE5-IN-10
PDE5-IN-10 (compound 4b), a potent phosphodiesterase type 5 (PDE5) inhibitor, exhibits an effective half-maximal inhibitory concentration (IC50) of 20 nM,
Formule :C₂₁H₂₀N₄O₂
Couleur et forme :Solid
Masse moléculaire :360.41
Ref: TM-T79533
+ Info
1-Palmitoyl-2-linoleoyl PE
CAS :
- 26662-95-3
Phosphatidylethanolamine PLPE: a cell membrane component, studied for anandamide biosynthesis, sPLA2-IIA activity substrate.
Formule :C₃₉H₇₄NO₈P
Couleur et forme :Solid
Masse moléculaire :715.994
Ref: TM-T37785
+ Info
GS-704277
CAS :
- 1911579-04-8
GS-704277, a Remdesivir metabolite, shows potent in vitro effects against COVID-19.
Formule :C₁₅H₁₉N₆O₈P
Couleur et forme :Solid
Masse moléculaire :442.325
Ref: TM-T37959
+ Info
Trifluoperazine N-Glucuronide
CAS :
- 165602-90-4
Trifluoperazine N-Glucuronide is a metabolite of Trifluoperazine with antidepressant and antipsychotic activity.
Formule :C₂₇H₃₂F₃N₃O₆S
Couleur et forme :Solid
Masse moléculaire :583.62
Ref: TM-T29009
+ Info
Forrestiacids K
CAS :
- 2920898-65-1
Forrestiacid K, a terpenoid derived from Pseudotsuga forrestii, functions as an inhibitor of ATP-citrate lyase (ACL) [1].
Formule :C₅₀H₇₄O₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :771.12
Ref: TM-T79936
+ Info
UCM-13207
CAS :
- 1621536-10-4
UCM-13207 is a specific ICMT inhibitor that improves progeria.
Formule :C₂₄H₃₂N₂O₂
Degré de pureté :99.83%
Couleur et forme :Soild
Masse moléculaire :380.52
Ref: TM-T80677
+ Info
3-Oxo-7-hydroxychol-4-enoic acid
CAS :
- 14772-95-3
3-Oxo-7-hydroxychol-4-enoic acid, a body metabolite, may signal bad liver disease prognosis.
Formule :C₂₄H₃₆O₄
Couleur et forme :Solid
Masse moléculaire :388.54
Ref: TM-T75703
+ Info
HBPC-GSH
CAS :
- 1055039-06-9
HBPC-GSH, a derivative of glutathione, functions as an inhibitor for the glyoxalase system, specifically inhibiting cGloI and cGloII with IC50 values of 0.6μM
Formule :C₁₇H₂₃BrN₄O₈S
Couleur et forme :Solid
Masse moléculaire :523.36
Ref: TM-T74658
+ Info
CHEMBL1276927
CAS :
- 305357-89-5
CHEMBL1276927 (N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide) shows antibacterial and antiparasitic activities against Chlamydia pneumoniae and
Formule :C₂₁H₁₇N₃O
Degré de pureté :99.86%
Couleur et forme :Solid
Masse moléculaire :327.38
Ref: TM-T60092
+ Info
PROTAC IDO1 Degrader-1
CAS :
- 2488851-89-2
First potent PROTAC IDO1 degrader; links IDO1 to CRBN E3 ligase for UPS-induced degradation (DC50=2.84 μM), boosts H ER2 CAR-T cell efficacy.
Formule :C₄₀H₅₃BrFN₉O₁₃
Couleur et forme :Solid
Masse moléculaire :966.816
Ref: TM-T37329
+ Info
DSPE-PEG5000-LTLRWVGLMS
DSPE-PEG5000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 serves as a receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG5000-LTLRWVGLMS can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01178
+ Info
S32826
CAS :
- 1096770-84-1
S32826, a potent autotaxin inhibitor with an IC50 of 8.8 nM, blocks LPA release and targets α, β, γ isoforms.
Formule :C₂₁H₃₆NO₄P
Couleur et forme :Solid
Masse moléculaire :397.496
Ref: TM-T38488
+ Info
DSPE-PEG5000-MPG
DSPE-PEG5000-MPG is a PEG compound composed of DSPE and a peptide carrier (MPG). MPG is derived from the nuclear localization sequence (NLS) of the SV40 large T antigen and the fusion peptide domain of HIV-1 gp41. This compound effectively delivers short oligonucleotides into cells independently of the endosomal pathway.
Couleur et forme :Odour Solid
Ref: TM-TCL-01146
+ Info
H-Pro-Phe-OH
CAS :
- 13589-02-1
H-Pro-Phe-OH is a dipeptide formed from proline and phenylalanine, serving as a substrate for prolylase and in peptide synthesis.
Formule :C₁₄H₁₈N₂O₃
Couleur et forme :Solid
Masse moléculaire :262.30
Ref: TM-T76613
+ Info
Vitamin K1 2,3-epoxide
CAS :
- 25486-55-9
Vitamin K1 2,3-epoxide (Phylloquinone oxide) is reduced to vitamin k and is involved in the vitamin k cycle.
Formule :C₃₁H₄₆O₃
Degré de pureté :98% - 98.05%
Couleur et forme :Solid
Masse moléculaire :466.7
Ref: TM-T36730
+ Info
SHP2-IN-16
SHP2-IN-16 (compound 222) is a potent SHP2 inhibitor exhibiting an IC50 of 1 nM, and is applicable in glioblastoma research [1].
Formule :C₂₅H₂₄F₂N₆O
Couleur et forme :Solid
Masse moléculaire :462.49
Ref: TM-T79412
+ Info
15-LOX-1 inhibitor 1
CAS :
- 2349374-37-2
9c(i472) blocks 15-LO-1 (IC50=0.19μM), lowers NF-κB in RAW-Blue cells, & cuts Nos2/lipid peroxidation in RAW 264.7 at 0.2-5μM.
Formule :C₂₂H₂₁ClN₂O₄
Couleur et forme :Solid
Masse moléculaire :412.87
Ref: TM-T36169
+ Info
Ascorbate oxidase
CAS :
- 9029-44-1
Ascorbate oxidase, a REDOX enzyme, catalyzes ascorbic acid and oxygen to dehydroascorbic acid, regulating the extracellular matrix.
Couleur et forme :Solid
Ref: TM-T76101
+ Info
α-Hydroxytamoxifen
CAS :
- 97151-02-5
α-Hydroxytamoxifen is a metabolite of tamoxifen. It reacts with DNA and causes the formation of DNA adducts.
Formule :C₂₆H₂₉NO₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :387.51
Ref: TM-T19192
+ Info
ACAT-IN-8
CAS :
- 199984-35-5
ACAT-IN-8 is an ACAT inhibitor which regulates cholesterol and blocks NF-κB mediated transcription.
Formule :C₃₂H₄₉N₃O₅S
Couleur et forme :Solid
Masse moléculaire :587.82
Ref: TM-T39413
+ Info
Previridicatumtoxin
CAS :
- 1379585-81-5
Previridicatumtoxin, found in P. aethiopicum, fights MRSA, VRE, C. albicans, S. cerevisiae, and kills NCI H460, KB-3-1, SW620 cancer cells.
Formule :C₃₀H₃₃NO₁₀
Couleur et forme :Solid
Masse moléculaire :567.58
Ref: TM-T37006
+ Info
Pectin
CAS :
- 9000-69-5
Pectin, a plant cell wall derived heteropolysaccharide, forms nanoparticles for delivery and acts as an antimicrobial adsorbent.
Couleur et forme :Solid
Ref: TM-T77242
+ Info
CAIX Inhibitor S4
CAS :
- 1330061-67-0
CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.
Formule :C₁₅H₁₇N₃O₄S
Degré de pureté :99.07%
Couleur et forme :Solid
Masse moléculaire :335.38
Ref: TM-T36758
+ Info
DSPE-PEG2000-M2pep
DSPE-PEG2000-M2pep is a PEG compound formed from DSPE and the M2-polarized macrophage-targeting peptide (M2pep). M2pep acts as a monovalent or multivalent ligand conjugated with pro-apoptotic peptides to specifically target M2 macrophages with toxic effects. DSPE-PEG2000-M2pep is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01085
+ Info
DSPE-PEG5000-pPB
DSPE-PEG5000-pPB is a PEG compound composed of DSPE and the cyclic oligopeptide (pPB). The pPB component has high binding affinity to PDGFRβ, which is overexpressed on activated hepatic stellate cells (HSC). DSPE-PEG5000-pPB is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01144
+ Info
2'-Rhamnoechinacoside
CAS :
- 1422390-59-7
2'-Rhamnoechinacoside is a naturally occurring compound sourced from Cistanche tubulosa.
Formule :C₄₁H₅₆O₂₄
Couleur et forme :Solid
Masse moléculaire :932.9
Ref: TM-TN7431
+ Info
α-Glucosidase-IN-74
α-Glucosidase-IN-74, a nicotinamide-thiazole derivative, functions as an α-glucosidase (α-glucosidase) inhibitor. It demonstrates antidiabetic activity by reducing blood glucose and triglyceride levels in Streptozotocin-induced diabetic animals.
Couleur et forme :Odour Solid
Ref: TM-T200727
+ Info
DSPE-PEG5000-octreotide
DSPE-PEG5000-Octreotide is a PEG compound composed of DSPE and Octreotide. Octreotide serves as a somatostatin receptor agonist and exhibits anti-tumor properties, induces apoptosis, and is applicable for acromegaly research. DSPE-PEG5000-Octreotide can be utilized in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01159
+ Info
Mycophenolic acid-β-D-glucuronide
CAS :
- 31528-44-6
Mycophenolic acid glucuronide is the glucuronide metabolite of mycophenolic acid in human plasma.
Formule :C₂₃H₂₈O₁₂
Degré de pureté :98.29%
Couleur et forme :Solid
Masse moléculaire :496.46
Ref: TM-T60104
+ Info
Angiotensin I-13C6,15N (human, mouse, rat) TFA
Angiotensin I-13C6,15N (human, mouse, rat) TFA is a labeled version of Angiotensin I, using isotopes 13C and 15N, specifically targeted for human, mouse, and rat studies. This compound serves as a precursor to angiotensin II, which is formed through the cleavage by angiotensin-converting enzyme (ACE).
Formule :C₅₇₁₃C₆H₈₉N₁₆₁₅NO₁₄·xC₂HF₃O₂
Couleur et forme :Solid
Masse moléculaire :1303.42 (free base)
Ref: TM-T201458
+ Info
Histone acetyltransferase p300 Inhibitor 4c
CAS :
- 2103-99-3
2-Amino-4-(4-chlorophenyl)thiazole blocks hCA I/II, AChE, BChE with Ki: ~0.008, 0.124, 0.129, 0.083 µM.
Formule :C₉H₇ClN₂S
Degré de pureté :99.76%
Couleur et forme :Solid
Masse moléculaire :210.68
Ref: TM-T77560
+ Info
Galactonic acid
CAS :
- 13382-27-9
Galactonic acid, derived from galactose metabolism, is converted from galactonolactone.
Formule :C₆H₁₂O₇
Couleur et forme :Solid
Masse moléculaire :196.16
Ref: TM-T73756
+ Info
Palitantin
CAS :
- 15265-28-8
Palitantin is a useful organic compound for research related to life sciences. The catalog number is T125757 and the CAS number is 15265-28-8.
Formule :C₁₄H₂₂O₄
Couleur et forme :Solid
Masse moléculaire :254.326
Ref: TM-T125757
+ Info
PDE11A4-IN-1
PDE11A4-IN-1 (compound 23b) is a potent, selective inhibitor of PDE11A4, demonstrating an IC50 of 12 nM and exhibiting high selectivity against PDE1, PDE2,
Couleur et forme :Odour Solid
Ref: TM-T81534
+ Info
2-(2',3',4'-Trihydroxybutyl)quinoxaline
CAS :
- 42015-38-3
2-(2',3',4'-Trihydroxybutyl)quinoxaline is a food metabolite.
Formule :C₁₂H₁₄N₂O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :234.25
Ref: TM-T19091
+ Info
1,2-Dihexadecyl-sn-glycero-3-PC
CAS :
- 36314-47-3
1,2-Dihexadecyl-sn-glycero-3-PC can be used in related research in the field of life sciences. Its product number is T37043 and CAS number is 36314-47-3.
Formule :C₄₀H₈₄NO₆P
Couleur et forme :Solid
Masse moléculaire :706.07
Ref: TM-T37043
+ Info
5(S)-HPETE
CAS :
- 71774-08-8
5(S)-HpETE is a PUFA made by 5-LO from arachidonic acid, metabolized into LTA4, a key leukotriene precursor.
Formule :C₂₀H₃₂O₄
Couleur et forme :Solid
Masse moléculaire :336.472
Ref: TM-T40826
+ Info
Arginase
CAS :
- 9000-96-8
Arginase (L-Arginine amidinase) is a key hydrolytic enzyme in the urea cycle, which hydrolyzes L-arginine into urea and L-ornithine.
Couleur et forme :Solid
Ref: TM-T76208
+ Info
Beauverolide Ka
CAS :
- 76265-42-4
Beauverolide Ka, from Beauveria bassiana, enhances glucose uptake and protects HEI-OC1 cells; active in L6 cells/myotubes.
Formule :C₃₇H₅₀N₄O₅
Couleur et forme :Solid
Masse moléculaire :630.82
Ref: TM-T74199
+ Info
Fmoc-Gly-Ser(psi(Me,Me)pro)-OH
CAS :
- 1095952-22-9
Fmoc-Gly-Ser(psi(Me,Me)pro)-OH is a dipeptide.
Formule :C₂₃H₂₄N₂O₆
Couleur et forme :Solid
Masse moléculaire :424.45
Ref: TM-T38485
+ Info
NU223612
CAS :
- 2759420-43-2
"NU223612 is a potent IDO1-degrading PROTAC with Kd 640 nM, binds CRBN at 290 nM, and crosses the BBB."
Formule :C₄₉H₅₅FN₆O₉
Couleur et forme :Solid
Masse moléculaire :890.99
Ref: TM-T74992
+ Info
DSPE-PEG2000-R9
DSPE-PEG2000-R9 is a PEG compound composed of DSPE and polyarginine-9 peptide (R9) peptide. It can be used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01119
+ Info
Trichodecenin I
CAS :
- 141024-74-0
Trichodecenin I is a peptaibol isolated from Trichoderma viride.
Formule :C₃₈H₆₉N₇O₈
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :752.011
Ref: TM-TP2474
+ Info
HLF1-11
CAS :
- 183623-03-2
HLF1-11: human lactoferrin peptide, antimicrobial, inhibits MPO, steers monocytes to macrophages, boosts immunity.
Formule :C₅₆H₉₅N₂₅O₁₄S
Couleur et forme :Solid
Masse moléculaire :1374.58
Ref: TM-T73659
+ Info
Carvedilol metabolite 4-Hydroxyphenyl Carvedilol
CAS :
- 142227-49-4
4-Hydroxyphenyl Carvedilol is a metabolite of Carvedilol. Carvedilol is a beta-blocker/alpha-1 blocker.
Formule :C₂₄H₂₆N₂O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :422.47
Ref: TM-T10686
+ Info
h15-LOX-2 inhibitor 2
Compound 10 (h15-LOX-2 inhibitor 2) suppresses h15-LOX activity, exhibiting IC 50 and K i values of 26.9 μM and 16.4 μM, respectively.
Formule :C₂₂H₃₀Cl₂N₆O₃
Couleur et forme :Solid
Masse moléculaire :497.42
Ref: TM-T200017
+ Info
α-2,3-Sialyltransferase (PmST3)
CAS :
- 71124-51-1
PmST3 is a beta-galactoside enzyme adding sialic acid to glycoproteins and glycolipids.
Couleur et forme :Solid
Ref: TM-T75421
+ Info
3'-sulfo Galactosylsphingosine (ammonium salt)
CAS :
- 1246681-32-2
Sulfatide derivative inhibits cell migration, adhesion, PKC, cytochrome c; accumulates in metachromatic leukodystrophy; used for LC-MS quantification.
Formule :C₂₄H₅₀N₂O₁₀S
Couleur et forme :Solid
Masse moléculaire :558.73
Ref: TM-T38090
+ Info
α-Glucosidase-IN-85
α-Glucosidase-IN-85 (Compound 8D1) functions as an inhibitor of α-Glucosidase, with an IC50 of 5.43 μM. This compound is useful for research related to type 2 diabetes.
Couleur et forme :Odour Solid
Ref: TM-T206275
+ Info
LYP-IN-1
CAS :
- 1404436-51-6
LYP-IN-1 is a potent, selective inhibitor of lymphoid-specific tyrosine phosphatase useful for studying autoimmune disorders and immune signaling.
Formule :C₂₈H₂₀ClNO₆
Degré de pureté :92.43%
Couleur et forme :Solid
Masse moléculaire :501.92
Ref: TM-T38834
+ Info
Abieslactone
CAS :
- 33869-93-1
Abieslacton possesses anti-tumor promoting activity isolated from several Abies genus.
Formule :C₃₁H₄₈O₃
Couleur et forme :Solid
Masse moléculaire :468.722
Ref: TM-T24996
+ Info
FZQ-21
FZQ-21 (Compound 70P) is an inhibitor of the water-soluble epoxide hydrolase (sEH), with an IC50 value of 4 nM. The IC50 for inhibiting human sEH is 1.5 nM, which is comparable to that of EC5026 (1.7 nM). FZQ-21 is utilized in sepsis research.
Formule :C₂₈H₃₀N₄O₃
Masse moléculaire :470.23179
Ref: TM-T209090