Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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MTHFD2-IN-4
<p>MTHFD2-IN-4, a tricyclic coumarin derivative, serves as a potent inhibitor of MTHFD2 and has applications in cancer research [1].</p>Formule :C26H21F6N2O5Couleur et forme :SolidMasse moléculaire :555.45Ilexoside O
CAS :<p>Ilexoside O, a root-derived triterpene saponin, modestly blocks XOD with an IC50 of 53.05 μM.</p>Formule :C53H86O22Couleur et forme :SolidMasse moléculaire :1075.249Trihydroxycholestanoic Acid
CAS :<p>Trihydroxycholestanoic acid aids cholic acid creation; high levels indicate Zellweger syndrome due to faulty PEX genes.</p>Formule :C27H46O5Couleur et forme :SolidMasse moléculaire :450.66ONO-8430506
CAS :<p>ONO-8430506 is an orally available, potent autotaxin (ATX)/ENPP2 inhibitor (IC90: 100 nM) that inhibits ATX activity in mouse plasma.</p>Formule :C27H28FN3O3Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :461.53Anti-Cancer Metabolism Compound Library
<p>A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS</p>Couleur et forme :Odour Solid1-Myristoyl-2-hydroxy-sn-glycero-3-PE
CAS :<p>Naturally-occurring lysophospholipid raises intracellular calcium and is higher in breast cancer patients.</p>Formule :C19H40NO7PCouleur et forme :SolidMasse moléculaire :425.50hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Formule :C24H17Cl2N3O3S2Couleur et forme :SolidMasse moléculaire :530.446FASN-IN-4 tosylate
CAS :FASN-IN-4 tosylate: Fatty acid synthase inhibitor, IC50 10 nM; blocks SARS-CoV-2, EC50 18.6 nM.Formule :C33H35N3O7S2Couleur et forme :SolidMasse moléculaire :649.78Paraherquamide E
CAS :<p>Fungal-derived paraherquamide E kills C. elegans and O. fasciatus, reduces T. colubriformis eggs in gerbils.</p>Formule :C28H35N3O4Couleur et forme :SolidMasse moléculaire :477.605Moth Cytochrome C (MCC) (88-103)
CAS :Moth Cytochrome C (88-103) peptide induces positive TCR selection in thymocytes; key for self-tolerant T cell development.Formule :C79H133N23O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1805.04Desoxycarbadox
CAS :<p>Desoxycarbadox, derived from Carbadox, is a quinoxaline-di-N-oxide antibiotic compound.</p>Formule :C11H10N4O2Couleur et forme :SolidMasse moléculaire :230.227(R)-ICMT-IN-3
<p>(R)-ICMT-IN-3 (compound ent 2-27) functions as a potent inhibitor of ICMT, exhibiting an IC50 value of 0.01 μM [1].</p>Couleur et forme :Odour SolidDSPE-PEG2000-VIP
<p>DSPE-PEG2000-VIP is a PEG-based compound composed of DSPE and the vasoactive intestinal peptide (VIP). This compound is useful for drug delivery applications.</p>Couleur et forme :Odour Solidβ-Tetralone
CAS :<p>β-Tetralone (2-Tetralone) is a vital drug synthesis precursor with complex pharmacological properties in combating neurological disorders. Cost-effective and quality-assured.</p>Formule :C10H10ODegré de pureté :97.26% - 99.18%Couleur et forme :Clear To Yellow LiquidMasse moléculaire :146.19Oseltamivir acid methyl ester hydrochloride
CAS :<p>Oseltamivir acid methyl ester hydrochloride, a precursor to oseltamivir, is converted by CES1.</p>Formule :C15H27ClN2O4Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :334.84FCE 28073
CAS :<p>FCE 28073 is a Monoamine oxidase B inibitor with IC50 of 0.45 uM.</p>Formule :C17H19FN2O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :302.34Oleic Acid-2,6-diisopropylanilide
CAS :<p>Oleic acid-2,6-diisopropylanilide: ACAT inhibitor, IC50 7 nM; lowers LDL & raises HDL in high-fat fed rabbits/rats at 0.05%.</p>Formule :C30H51NOCouleur et forme :SolidMasse moléculaire :441.744Camellianin B
CAS :<p>Camellianin B, a flavonoid from Camellianin A, has antioxidant effects and blocks ACE.</p>Formule :C27H30O14Couleur et forme :SolidMasse moléculaire :578.523Chlorothiazide
CAS :<p>Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.</p>Formule :C7H6ClN3O4S2Degré de pureté :98.46% - 98.91%Couleur et forme :Crystals Physical Description Crystals; White Powder (Ntp 1992)Masse moléculaire :295.7220,26-Dihydroxyecdysone
CAS :<p>20,26-Dihydroxyecdysone is a predominant ecdysteroid metabolite [1] .</p>Formule :C27H44O8Couleur et forme :SolidMasse moléculaire :496.63Acetoacetic acid
CAS :<p>Acetoacetic acid(3-oxobutanoic acid) is a oxidative stress inducer, gluconeogenesis, and can be used as an indicator of in ketoacidosis.</p>Formule :C4H6O3Degré de pureté :99.59% - 99.85%Couleur et forme :SolidMasse moléculaire :102.09LDHA-IN-3
CAS :<p>LDHA-IN-3 is a potent selenobenzene-based LDHA inhibitor with a 145.2 nM IC50, useful in cancer research.</p>Formule :C13H9F3SeDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :301.173-keto Fusidic Acid
CAS :<p>3-keto Fusidic acid (3-keto FA) is an active metabolite of the antibiotic fusidic acid .13-keto FA is active againstM. tuberculosis(MIC99= 1.25 μM).</p>Formule :C31H46O6Couleur et forme :SolidMasse moléculaire :514.703N-Stearoylsphingomyelin
CAS :<p>N-Stearoylsphingomyelin (N-Stearoyl-D-sphingomyelin), a sphingolipid, inhibits Phospholipase Cδ1 (PLCδ1) [1].</p>Formule :C41H83N2O6PCouleur et forme :SolidMasse moléculaire :731.08Acremin F
CAS :<p>Acremin F is a useful organic compound for research related to life sciences. The catalog number is T124074 and the CAS number is 863480-61-9.</p>Formule :C12H20O4Couleur et forme :SolidMasse moléculaire :228.288(Rac)-5-Keto Fluvastatin
CAS :<p>(Rac)-5-Keto Fluvastatin (rac 5-Keto Fluvastatin) is an impurity of Fluvastatin which is an inhibitor of HMG-CoA reductase.</p>Formule :C24H24FNO4Degré de pureté :95.04%Couleur et forme :SolidMasse moléculaire :409.45D-Fructose 1-phosphate disodium
CAS :<p>D-Fructose 1-phosphate disodium salt, a derivative of fructose, serves as a crucial intermediate in glucose metabolism.</p>Formule :C6H11Na2O9PCouleur et forme :SolidMasse moléculaire :304.10SGK1-IN-4
CAS :<p>SGK1-IN-4 is a selective inhibitor of SGK1 and can be used in studies about osteoarthritis.</p>Formule :C23H21ClFN5O4SDegré de pureté :97.03%Couleur et forme :SolidMasse moléculaire :517.96α-Glucosidase-IN-54
CAS :<p>α-Glucosidase-IN-54 (compound 2) functions as an α-glucosidase inhibitor, exhibiting an IC 50 value of 0.011 mM, and is derived from Syzygium jambos (L.). This compound is employed in diabetes research [1].</p>Formule :C24H36O3Couleur et forme :SolidMasse moléculaire :372.54Ellagic acid 4-O-β-D-xylopyranoside
CAS :<p>Ellagic acid 4-O-β-D-xylopyranoside, an ellagitannin found naturally, exhibits antimicrobial properties and acts as an inhibitor of xanthine oxidase, displaying</p>Formule :C19H14O12Couleur et forme :SolidMasse moléculaire :434.31DSPE-PEG5000-pPB
<p>DSPE-PEG5000-pPB is a PEG compound composed of DSPE and the cyclic oligopeptide (pPB). The pPB component has high binding affinity to PDGFRβ, which is overexpressed on activated hepatic stellate cells (HSC). DSPE-PEG5000-pPB is applicable for drug delivery.</p>Couleur et forme :Odour SolidHIV-IN-9
<p>HIV-IN-9 (Compound 2b) is an HIV inhibitor with an IC50 value of 6.65 μg/mL, demonstrating high binding affinity for HIV-RT.</p>Couleur et forme :Odour SolidCTL-12
<p>CTL-12, a fatty acid synthase (FASN) inhibitor (IC50: 2.5 μM), induces apoptosis and disrupts the cell cycle at the Sub-G1/S phase.</p>Formule :C22H21ClN4O4Couleur et forme :SolidMasse moléculaire :440.88(±)-Hexanoylcarnitine chloride
CAS :<p>(±)-Hexanoylcarnitine chloride is a fatty acid metabolite that breaks down fatty acids into small compounds that can be utilized by the body.</p>Formule :C13H26ClNO4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :295.8Carbonic anhydrase inhibitor 29
<p>Carbonic anhydrase inhibitor29 (Compound 5d) is an inhibitor targeting carbonic anhydrase IX and XII, with an inhibition constant (Ki) of 26.6 nM for carbonic anhydrase IX and a Ki of 10.9 nM for carbonic anhydrase XII. Carbonic anhydrase inhibitor29 can be used in cancer research.</p>Couleur et forme :Odour SolidCAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Couleur et forme :Odour SolidSHP2-IN-36
<p>SHP2-IN-36 (Compound B8) is an allosteric inhibitor of SHP2 with an IC50 of 9.0 nM, and it exhibits an IC50 of 40 nM against p-ERK. Moreover, SHP2-IN-36 demonstrates significant antitumor activity in the KYSE520 xenograft mouse model and is applicable for research in the field of antitumor studies.</p>Couleur et forme :Odour Solid1,3-Dipalmitoleoyl-rac-glycerol
CAS :<p>1,3-Dipalmitoleoyl-rac-glycerol: a diacylglycerol inhibiting yeast α-glucosidase over rat's (IC50s: 4.45 vs 9326.5 μM). Used to study membrane potentials.</p>Formule :C35H64O5Couleur et forme :SolidMasse moléculaire :564.892Hydroxydehydro Nifedipine Carboxylate
CAS :<p>Hydroxydehydro nifedipine carboxylate is a metabolite of nifedipine .1</p>Formule :C16H14N2O7Couleur et forme :SolidMasse moléculaire :346.295Xanthine oxidase-IN-16
<p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>Couleur et forme :Odour SolidMefox
CAS :<p>Mefox is a bioactive chemical.</p>Formule :C20H23N7O7Couleur et forme :SolidMasse moléculaire :473.44WXC-25
<p>WXC-25 is an α-glucosidase inhibitor with an IC50 value of 2.02 μM.</p>Couleur et forme :Odour Solid1-Naphthyl 3,5-dinitrobenzoate
CAS :<p>1-Naphthyl 3,5-dinitrobenzoate (JMC-4) is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.</p>Formule :C17H10N2O6Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :338.27D-Lactate dehydrogenase
CAS :<p>D-LDH is an oxidoreductase turning D-lactate into pyruvate, using NAD+/NADP+; prevalent in bacteria and fungi, key for biochemical research.</p>Couleur et forme :SolidSX29
<p>SX29 is a non-competitive α-glucosidase inhibitor with oral activity, exhibiting an IC50 of 2.12 μM. It possesses hypoglycemic properties; oral administration of SX29 reduces blood glucose levels and enhances glucose tolerance in diabetic mice.</p>Couleur et forme :Odour SolidATX inhibitor 7
CAS :<p>ATX inhibitor 7 is a autotaxin inhibitor and shows good oral exposure.</p>Formule :C21H22F3N7O2Couleur et forme :SolidMasse moléculaire :461.449(±)-Geosmin
CAS :(±)-Geosmin, a natural compound, is biologically active in producing an earthy aroma. It plays a crucial role in microbial metabolism and is frequently used as a flavoring agent in food and fragrance in air. Additionally, (±)-Geosmin is under investigation for its potential to detect contamination in soil and water bodies.Formule :C12H22OCouleur et forme :SolidMasse moléculaire :182.3DSPE-PEG5000-NGR
<p>DSPE-PEG5000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide has the capability to target tumor vasculature antigen CD13. DSPE-PEG5000-NGR is applicable in drug delivery.</p>Couleur et forme :Odour SolidPhenacaine
CAS :<p>Phenacaine, also known as Holocaine, is a local anesthetic that blocks certain Ca 2+ enzymes in red blood cells, brain, and heart.</p>Formule :C18H22N2O2Couleur et forme :SolidMasse moléculaire :298.38PK-10
<p>PK-10, when combined with Fluconazole, exhibits potent synergistic antifungal activity against multiple Fluconazole-resistant Candida albicans strains.</p>Formule :C35H36F3N5OCouleur et forme :SolidMasse moléculaire :599.69
