Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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ω-Conotoxin Bu8
<p>ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges.</p>Formule :C103H174N42O35S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2753.13α-Glucosidase-IN-27
<p>α-Glucosidase-IN-27 (compound 8l), an α-glucosidase inhibitor with an IC50 value of 25.78 μM, demonstrates potential for research into type 2 diabetes (D2M) [1</p>Formule :C22H20N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.482-Pentyl-1H-benzo[d]imidazole
CAS :<p>2-Pentyl-1H-benzo[d]imidazole is a micromolar level inhibitor of Cytochrome P450 1A1 and 2B1 and has antibacterial activity against Fusarium verticillioides.</p>Formule :C12H16N2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :188.27Imatinib Impurity E
CAS :<p>Imatinib Impurity E, a derivative of orally taken Imatinib, inhibits tyrosine kinases BCR/ABL, PDGFR, c-kit, and SARS/MERS-CoV.</p>Formule :C52H48N12O2Couleur et forme :SolidMasse moléculaire :873.02Lacto-N-biose I
CAS :<p>Galβ1-3GlcNAc, a natural metabolite, is a substrate for H. pylori's α1,2-fucosyltransferase.</p>Formule :C14H25NO11Couleur et forme :SolidMasse moléculaire :383.35DSPE-PEG2000-MPG
<p>DSPE-PEG2000-MPG is a PEG compound composed of DSPE and the peptide carrier (MPG). The MPG component is derived from the nuclear localization sequence (NLS) of the SV40 large T antigen and the fusion peptide domain of HIV-1gp41. It effectively delivers short oligonucleotides into cells independently of the endosomal pathway.</p>Couleur et forme :Odour SolidCALP3 TFA(261969-05-5 free base)
<p>CALP3 TFA is a potent Ca2+ channel blocker that activates EF-hand motifs of Ca2+-binding proteins.</p>Formule :C46H69F3N10O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :995.1Coenzyme A
CAS :<p>Coenzyme A is an obligatory cofactor in all living cells synthesized from pantothenate (Vitamin B5), adenosine triphosphate (ATP), and cysteine.</p>Formule :C21H36N7O16P3SDegré de pureté :93.84%Couleur et forme :SolidMasse moléculaire :767.53α-Glucosidase-IN-30
<p>α-Glucosidase-IN-30 (compound 8c) is a potent, orally active competitive inhibitor of α-glucosidase, exhibiting a K i of 40.0 µM and an IC50 of 49.0 µM.</p>Formule :C20H19N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.41Relzomostat
CAS :<p>Relzomostat inhibits MetAP2, with research potential for obesity and type 2 diabetes.</p>Formule :C24H36F2N2O5Couleur et forme :SolidMasse moléculaire :470.558N-Benzoyl-L-Leucine
CAS :<p>N-Benzoyl-L-Leucine is a leucine derivative exhibiting antibacterial activity against Staphylococcus aureus.</p>Formule :C13H17NO3Degré de pureté :99.60%Couleur et forme :SoildMasse moléculaire :235.28Fmoc-Gly-Ser(psi(Me,Me)pro)-OH
CAS :<p>Fmoc-Gly-Ser(psi(Me,Me)pro)-OH is a dipeptide.</p>Formule :C23H24N2O6Couleur et forme :SolidMasse moléculaire :424.45Xanthine oxidase-IN-16
<p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>Couleur et forme :Odour SolidAnirolac
CAS :<p>Anirolac is a nonsteroidal anti-inflammatory agent.</p>Formule :C16H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.29L 645164
CAS :<p>L 645164 is an inhibitor of hydroxymethylglutaryl-CoA reductase.</p>Formule :C22H23FO3Couleur et forme :SolidMasse moléculaire :354.41hCAIX/XII-IN-14
<p>hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.</p>Formule :C16H14F3N3O4SCouleur et forme :SolidMasse moléculaire :401.36α-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Couleur et forme :Odour SolidT3 Acyl glucuronide
CAS :<p>T3 Acyl glucuronide is the acyl glucuronide formation of triiodothyronine (T3). T3 Acyl glucuronide is an endogenous metabolite</p>Formule :C21H20I3NO10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :827.1sEH inhibitor-20
<p>sEH inhibitor-20 is a metabolically stable, orally active sEH inhibitor with an IC50 of 0.2 nM. It exhibits significant analgesic and anti-inflammatory properties, making it a promising candidate for researching neuropathic pain.</p>Couleur et forme :Odour Solid(±)-threo-3-Methylglutamic acid
CAS :<p>glutamate transport blocker</p>Formule :C6H11NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :161.16Autophagy inducer 5
<p>Autophagyinducer 5 (compound 21o) serves as a potent inhibitor of MCF-7 (IC50: 2 μM), making it a potential candidate for breast cancer therapy. It induces autophagy by activating the ROS/JNK signaling pathway, which increases ROS production and JNK phosphorylation, ultimately exerting cytotoxic effects.</p>Formule :C41H52N4O3Couleur et forme :SolidMasse moléculaire :648.88Fluazuron
CAS :<p>Fluazuron is an insect growth regulator.</p>Formule :C20H10Cl2F5N3O3Couleur et forme :White PowderMasse moléculaire :506.21CAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Couleur et forme :Odour SolidCrotonyl-CoA tetrasodium
Crotonyl-CoA tetrasodium is the tetrasodium salt form of Crotonyl-CoA. It serves as an intermediate in butyrate fermentation and in the metabolism of lysine and tryptophan. This compound plays a crucial role in the metabolism of fatty acids and amino acids.Formule :C25H36N7Na4O17P3SCouleur et forme :SolidMasse moléculaire :923.54DSPE-PEG2000-CTT2
<p>DSPE-PEG2000-CTT2 is a PEG compound consisting of DSPE and the gelatinase inhibitor CTT2 (CTTHWGFTLC). It possesses the ability to specifically target tumors. DSPE-PEG2000-CTT2 is suitable for drug delivery applications.</p>Couleur et forme :Odour Solid11-epi-Chaetomugilin I
CAS :<p>11-epi-Chaetomugilin I, from Chaetomium globosum, has cytotoxic effects against P388, HL-60, L1210 leukemia, and KB carcinoma cells.</p>Formule :C22H27ClO5Couleur et forme :SolidMasse moléculaire :406.9Ethyl gentisate
CAS :<p>Ethyl gentisate acts as a dual regulator of cell differentiation, promoting osteoblast differentiation while inhibiting osteoclast differentiation.</p>Formule :C9H10O4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :182.17DSPE-PEG5000-CREKA
<p>DSPE-PEG5000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide is utilized for targeting tumor cells and tumor vasculature, exhibiting anti-tumor activity. DSPE-PEG5000-CREKA is applicable in drug delivery systems.</p>Couleur et forme :Odour SolidTpp-CAQK
<p>Tpp-CAQK, a specially engineered mitochondrial compound, has been shown to improve phagocytosis of myelin debris by macrophages, reduce mitochondrial dysfunction and pro-inflammatory features, and enhance tissue repair and functional recovery in mice after spinal cord injury.</p>Formule :C40H54BrN6O7PSCouleur et forme :SolidMasse moléculaire :873.84Phenolic acid
CAS :<p>Phenolic acid is an endogenous metabolite.</p>Formule :C7H8D2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :144.16Tetomilast
CAS :<p>Tetomilast (OPC-6535) is a phosphodiesterase-4 (PDE4) inhibitor, potentially effective in treating inflammatory bowel disease (IBD) and chronic obstructive</p>Formule :C19H18N2O4SCouleur et forme :SolidMasse moléculaire :370.42α-Glucosidase-IN-74
<p>α-Glucosidase-IN-74, a nicotinamide-thiazole derivative, functions as an α-glucosidase (α-glucosidase) inhibitor. It demonstrates antidiabetic activity by reducing blood glucose and triglyceride levels in Streptozotocin-induced diabetic animals.</p>Couleur et forme :Odour Solidβ-Galactose dehydrogenase
CAS :Beta-Galactose dehydrogenase converts galactose to galactonolactone, reducing NAD to fluorescent NADH; useful in galactose measurement.Fexarene
CAS :<p>Fexarene is a non-steroidal FXR agonist.</p>Formule :C32H33NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.62Ercalcidiol
CAS :<p>Ercalcidiol is a metabolite of vitamin D2 and can be used in monitoring vitamin D therapy.</p>Formule :C28H44O2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :412.65α-1,3-N-Acetylgalactosaminyltransferase (Pm1138)
CAS :<p>Alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138) (EC 2.4.1.40(Pm1138)), also known as the ABO system transferase, exhibits glycosyl transferase activity [1</p>Couleur et forme :SolidIPH5201
<p>IPH5201 is a human IgG1 monoclonal antibody (mAb) targeting ENTPD1/CD39. It enhances the accumulation of immunostimulatory ATP released by tumor cells undergoing combination chemotherapy (CT) and reduces the levels of immunosuppressive adenosine (Ado) in the tumor microenvironment (TME). IPH5201 is useful for research on antitumor immunity. Recommended isotype control: Human IgG1 kappa, Isotype Control.</p>Couleur et forme :Odour LiquidSGK1-IN-3 hydrochloride
<p>SGK1-IN-3 hydrochloride (compound 3a) is an efficacious, orally bioavailable SGK1 inhibitor. The serine/threonine kinase SGK1 acts as an activator of the β-catenin pathway and strongly stimulates cartilage degradation, being upregulated under genomic control in diseased osteoarthritic cartilage. SGK1-IN-3 hydrochloride holds potential for osteoarthritis research.</p>Formule :C23H21Cl3N6O3SMasse moléculaire :566.046149AzNue5Ac
CAS :<p>9AzNue5Ac is a Neu5Ac analog that is metabolized in vivo in living cells and in mice.9AzNue5Ac binds to sialoglycans.</p>Formule :C11H18N4O8Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :334.28Ritonavir metabolite
CAS :<p>Ritonavir metabolite is a Ritonavir metabolite, which is a inhibitor of HIV protease.</p>Formule :C32H45N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :579.80D-Sedoheptulose 7-phosphate
CAS :<p>D-Sedoheptulose 7-phosphate, a precursor to group III heptaic acid and group IV hygromycin B, converts to NDP-heptose via similar pathways.</p>Formule :C7H15O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :290.16FABP4-IN-4
<p>FABP4-IN-4 (Compound 30) is an orally effective inhibitor of FABP, with an IC50 value of 1.18 μM against FABP1. In a mouse model of diet-induced obesity, FABP4-IN-4 improves glucose tolerance, reduces levels of blood sugar, lipids, and liver inflammation markers, alleviates hepatic steatosis, and exhibits anti-inflammatory activity.</p>Couleur et forme :Odour Solid(S)-3-Thienylglycine
CAS :<p>(S)-3-Thienylglycine is a thiophene derivative and can be used to investigate the genotoxicity of the similar structures with thiophene derivatives.</p>Formule :C6H7NO2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :157.19PKM2 inhibitor G
CAS :<p>PKM2 inhibitor G is a inhibitor of pyruvate kinase.</p>Formule :C16H15NO3SDegré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :301.36Acesulfame
CAS :<p>Acesulfame inhibits CA9/12 and can be used to study inflammation-related diseases.</p>Formule :C4H5NO4SCouleur et forme :SolidMasse moléculaire :163.15SF2312 ammonium
<p>SF2312 ammonium is the ammonium salt of SF2312, a phosphonate antibiotic and enolase inhibitor derived from the actinomycete Micromonospora and active under</p>Formule :C4H11N2O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :214.11(±)20-HDHA
CAS :<p>(±)20-HDHA is an autoxidation product and is a racemic mixture of Docosahexaenoic acid (DHA).</p>Formule :C22H32O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.49TRH Precursor Peptide
<p>Thyrotropin Releasing Hormone Precursor Peptide</p>Formule :C42H75N19O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1006.17Cholesterol esterase
CAS :<p>Cholesterol esterase breaks down cholesterol ester into cholesterol and free fatty acids, aiding absorption.</p>Couleur et forme :SolidHexasodium phytate
CAS :Hexasodium phytate is used potentially to treat vascular calcification and calciphylaxis.Formule :C6H12Na6O24P6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :791.93
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