Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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Ellagic acid 4-O-β-D-xylopyranoside
CAS :<p>Ellagic acid 4-O-β-D-xylopyranoside, an ellagitannin found naturally, exhibits antimicrobial properties and acts as an inhibitor of xanthine oxidase, displaying</p>Formule :C19H14O12Couleur et forme :SolidMasse moléculaire :434.31Cvs 738
CAS :<p>Cvs 738 is the desmethyl form of CVS 1123, an orally bioavailable inhibitor of thrombin.</p>Formule :C23H40N6O6Couleur et forme :SolidMasse moléculaire :496.6BMT-124110 Formate
<p>BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase</p>Formule :C22H20N2O2Degré de pureté :99.52%Couleur et forme :SoildMasse moléculaire :344.41γ-Acetylenic GABA hydrochloride
CAS :<p>γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.</p>Formule :C6H10ClNO2Degré de pureté :99.28% - 99.64%Couleur et forme :SolidMasse moléculaire :163.6Monoisobutyl phthalic acid
CAS :<p>Monoisobutyl phthalic acid is a metabolite of phthalate that is in human semen and in meconium.</p>Formule :C12H14O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :222.2413,14-dehydro-15-cyclohexyl Carbaprostacyclin
CAS :<p>13,14-dehydro-15-cyclohexyl Carbaprostacyclin, a stable PGI2 analog, impedes ADP-induced platelet aggregation; ED50 ~40 nM in PRP, 77 nM in washed platelets.</p>Formule :C21H30O4Couleur et forme :SolidMasse moléculaire :346.467Cholesteryl Homo-γ-Linolenate
CAS :<p>Cholesteryl homo-γ-linolenate is a cholesterol ester.</p>Formule :C47H78O2Couleur et forme :SolidMasse moléculaire :675.139Diadenosine pentaphosphate pentasodium
CAS :<p>Diadenosine pentaphosphate pentasodium, an endogenous purine from platelets and various cells, has vasoactive properties.</p>Formule :C20H24N10Na5O22P5Couleur et forme :SolidMasse moléculaire :1026.28ERAP1 modulator-1
CAS :<p>ERAP1 modulator-1 (Compound 1) is a regulator of endoplasmic reticulum aminopeptidase 1 (ERAP1) with an IC50 of less than 250 nM.</p>Formule :C23H23F3N2O5SCouleur et forme :SolidMasse moléculaire :496.5MK-8262
CAS :<p>MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.</p>Formule :C35H25F9N2O5Couleur et forme :SolidMasse moléculaire :724.58(±)-threo-3-Methylglutamic acid
CAS :<p>glutamate transport blocker</p>Formule :C6H11NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :161.16DSPE-PEG5000-NYZL1
<p>DSPE-PEG5000-NYZL1 is a PEG compound composed of DSPE and NYZL1, where NYZL1 specifically binds to bladder cancer tissues and cells. DSPE-PEG5000-NYZL1 is applicable for drug delivery.</p>Couleur et forme :Odour SolidBSO-07
<p>BSO-07 is a ROS/JNK activator that exhibits potent anti-cancer properties, demonstrated by an IC50 of 24.81 μM in human breast cancer (BC) cells. The mechanism of action for BSO-07 involves JNK activation and the promotion of increased ROS levels, which lead to the induction of apoptosis (Apoptosis) and tumorigenic apoptosis. This includes enhanced expression of apoptosis-related proteins such as PARP, Bax, phosphorylated p53, ATF4, and CHOP, along with a reduction in the levels of anti-apoptotic proteins (e.g., Bcl-2, Bcl-xL, and Survivin). BSO-07 holds promise for research in the field of breast cancer.</p>Couleur et forme :Odour SolidhBChE-IN-3
<p>hBChE-IN-3 (compound 30) serves as both an activator of carbonic anhydrase (CA) and an inhibitor of cholinesterase (ChE), exhibiting IC50 values of 7.4 nM for AchE and 1.9 nM for BchE. This compound is utilized in the research of neurodegenerative and psychiatric disorders.</p>Couleur et forme :Odour SolidCAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Couleur et forme :Odour Solidβ-Glucosidase
CAS :<p>β-Glucosidase is a glucoside bond hydrolase involved in glucose metabolism and can be used to study diseases caused by abnormal glucose metabolism.</p>Formule :C24H44O12Couleur et forme :SolidMasse moléculaire :524.6Caffeoylcalleryanin
CAS :<p>Caffeoylcalleryanin demonstrated potent inhibitory activity against 15-lipoxygenase (15-LOX), with an IC50 value of 1.59 μM. Furthermore, ethanol extract from A. pulchra leaves (EEAPL) was found to contain compounds exhibiting antiviral properties, particularly effective against Dengue virus type 2 (DENV-2). Among these compounds, Caffeoylcalleryanin emerged as the most potent anti-DENV-2 agent, achieving a selectivity index (SI) of 20.0.</p>Formule :C22H24O11Couleur et forme :SolidMasse moléculaire :464.4TRH Precursor Peptide
<p>Thyrotropin Releasing Hormone Precursor Peptide</p>Formule :C42H75N19O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1006.17CTL-12
<p>CTL-12, a fatty acid synthase (FASN) inhibitor (IC50: 2.5 μM), induces apoptosis and disrupts the cell cycle at the Sub-G1/S phase.</p>Formule :C22H21ClN4O4Couleur et forme :SolidMasse moléculaire :440.88ω-Conotoxin CVIF
<p>ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value of 34.3 nM in isolated rat DRG neurons.</p>Formule :C101H170N40O33S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2665.07O-desmethyl Mebeverine acid
CAS :<p>O-desmethyl Mebeverine acid is a metabolite of Mebeverine.</p>Formule :C15H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.35Xanthine oxidase-IN-16
<p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>Couleur et forme :Odour SolidProstaglandin F2β
CAS :<p>Prostaglandin F2β (PGF2β) is the 9β-hydroxy stereoisomer of PGF2α.</p>Formule :C20H34O5Couleur et forme :White SolidMasse moléculaire :354.48WXC-25
<p>WXC-25 is an α-glucosidase inhibitor with an IC50 value of 2.02 μM.</p>Couleur et forme :Odour SolidPyruvate carboxylase
CAS :<p>Pyruvate carboxylase, a biotin-containing enzyme, catalyzes the carboxylation of pyruvate to oxaloacetate, a reaction dependent on HCO3− and MgATP.</p>Degré de pureté :98%Couleur et forme :Solidα-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Couleur et forme :Odour Solid3α-Hydroxy pravastatin sodium
CAS :<p>3α-Hydroxy pravastatin sodium, the primary metabolite of Pravastatin, is a potent competitive inhibitor of HMG-CoA reductase.</p>Formule :C23H36NaO7Couleur et forme :SolidMasse moléculaire :447.524Paeoniflorgenin
CAS :<p>Paeoniflorgenin is a deglucosylated metabolite of Paeoniflorin[1].</p>Formule :C17H18O6Couleur et forme :SolidMasse moléculaire :318.3251-Naphthyl 3,5-dinitrobenzoate
CAS :<p>1-Naphthyl 3,5-dinitrobenzoate (JMC-4) is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.</p>Formule :C17H10N2O6Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :338.27PKM2 activator 6
<p>Compound Z10 (PKM2 activator 6) serves as both a PKM2 activator and a PDK1 inhibitor, exhibiting dissociation constants (K D ) of 121 μM and 19.6 μM,</p>Couleur et forme :Odour SolidDefensin HNP-2 human
CAS :<p>Defensin HNP-2 is a naturally occurring antibiotic and monocyte chemotactic peptide synthesized by human neutrophils.</p>Formule :C147H223N43O37S6Couleur et forme :SolidMasse moléculaire :3377.03SX29
<p>SX29 is a non-competitive α-glucosidase inhibitor with oral activity, exhibiting an IC50 of 2.12 μM. It possesses hypoglycemic properties; oral administration of SX29 reduces blood glucose levels and enhances glucose tolerance in diabetic mice.</p>Couleur et forme :Odour Solidα-Glucosidase-IN-74
<p>α-Glucosidase-IN-74, a nicotinamide-thiazole derivative, functions as an α-glucosidase (α-glucosidase) inhibitor. It demonstrates antidiabetic activity by reducing blood glucose and triglyceride levels in Streptozotocin-induced diabetic animals.</p>Couleur et forme :Odour SolidIsomer-Turosteride
<p>Isomer-Turosteride, a novel 5α-reductase inhibitor, reduces prostate DHT and has anticancer properties without raising T levels.</p>Formule :C27H45N3O3Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :459.67D-Lactate dehydrogenase
CAS :<p>D-LDH is an oxidoreductase turning D-lactate into pyruvate, using NAD+/NADP+; prevalent in bacteria and fungi, key for biochemical research.</p>Couleur et forme :SolidDSPE-PEG5000-R8
<p>DSPE-PEG5000-R8 is a PEG compound composed of DSPE and the cell-penetrating peptide (R8). It is utilized for drug delivery applications.</p>Couleur et forme :Odour SolidNIM811
CAS :<p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>Formule :C62H111N11O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1202.635DSPE-PEG5000-NGR
<p>DSPE-PEG5000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide has the capability to target tumor vasculature antigen CD13. DSPE-PEG5000-NGR is applicable in drug delivery.</p>Couleur et forme :Odour SolidPhenacaine
CAS :<p>Phenacaine, also known as Holocaine, is a local anesthetic that blocks certain Ca 2+ enzymes in red blood cells, brain, and heart.</p>Formule :C18H22N2O2Couleur et forme :SolidMasse moléculaire :298.38PEG2000-C-DMG
CAS :<p>PEG2000-C-DMG is a pegylated lipid for Onpattro, reducing transthyretin production via RNAi.</p>Formule :C126H249NO52Couleur et forme :SolidMasse moléculaire :2000 (Average)POPG sodium salt
CAS :<p>POPG sodium salt is a phospholipid and a component of biological membranes and can be used to study the function of biological membranes.</p>Formule :C40H76NaO10PDegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :770.99PK-10
<p>PK-10, when combined with Fluconazole, exhibits potent synergistic antifungal activity against multiple Fluconazole-resistant Candida albicans strains.</p>Formule :C35H36F3N5OCouleur et forme :SolidMasse moléculaire :599.69Leucylproline
CAS :<p>Leucylproline is a peptide that proteolytic breakdown product by larger proteins.</p>Formule :C11H20N2O3Couleur et forme :SolidMasse moléculaire :228.298-Demethyl Ivabradine
CAS :<p>8-Demethyl Ivabradine, a metabolite of Ivabradine, is an oral HCN channel blocker.</p>Formule :C26H34N2O5Couleur et forme :SolidMasse moléculaire :454.5676α-hydroxy Paclitaxel
CAS :<p>6α-hydroxy Paclitaxel (6α-OH-PTX) is a major metabolite of the anticancer compound paclitaxel and is partially cytotoxic.</p>Formule :C47H51NO15Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :869.91Pectin
CAS :<p>Pectin, a plant cell wall derived heteropolysaccharide, forms nanoparticles for delivery and acts as an antimicrobial adsorbent.</p>Couleur et forme :SolidTacalcitol monohydrate
CAS :<p>Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.</p>Formule :C27H46O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :434.65Camellianin B
CAS :<p>Camellianin B, a flavonoid from Camellianin A, has antioxidant effects and blocks ACE.</p>Formule :C27H30O14Couleur et forme :SolidMasse moléculaire :578.523BAY-277
<p>BAY-277 is a degrader of METAP2, with IC50 values of 5.8 nM for human METAP2 (hMETAP2) and 5.9 nM for mouse METAP2 (mMETAP2).</p>Formule :C44H52N8O5Couleur et forme :SolidMasse moléculaire :772.93Secalciferol
CAS :<p>Secalciferol is a Vitamin D metabolite,Secalciferol is a possibly anti-inflammatory steroid which is involved in bone ossification.</p>Formule :C27H44O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.64
