Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
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8626 produits trouvés pour "Métabolisme"
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4-Hydroxybenzoic acid-d4
CAS :<p>4-Hydroxybenzoicacid-d4 is a deuterated form of 4-Hydroxybenzoicacid, which is a phenolic derivative of benzoic acid. It is effective in inhibiting most Gram-positive bacteria and some Gram-negative bacteria with an IC50 of 160 μg/mL.</p>Formule :C7H6O3Couleur et forme :SolidMasse moléculaire :142.15WVSAV
<p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>Formule :C27H40N6O7Couleur et forme :SolidMasse moléculaire :560.64hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Formule :C24H17Cl2N3O3S2Couleur et forme :SolidMasse moléculaire :530.446α-Glucosidase-IN-82
<p>α-Glucosidase-IN-82 (compound 8l) is a potent inhibitor of α-glucosidase, with an IC50 value of 13.66 μM. Its inhibitory activity is 52 times greater than that of Acarbose.</p>Formule :C30H24N4O4Couleur et forme :SolidMasse moléculaire :504.536hCAII/IX-IN-1
<p>hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.</p>Formule :C23H22N4O7S2Couleur et forme :SolidMasse moléculaire :530.573MAGL-IN-5
CAS :<p>MAGL-IN-5 is a non-selective lipase inhibitor.</p>Formule :C18H17N3O5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :355.34Fasnall HCl
<p>Fasnall HCl is a selective FASN inhibitor that acts through its co-factor binding sites.</p>Formule :C19H23ClN4SDegré de pureté :99.9%Couleur et forme :SoildMasse moléculaire :374.93DSPE-PEG2000-T7
<p>DSPE-PEG2000-T7 is a PEG compound composed of DSPE and the transferrin receptor peptide (T7). The T7 peptide (HAIYPRH) specifically binds to TfR, making DSPE-PEG2000-T7 useful for drug delivery applications.</p>Couleur et forme :Odour SolidSeco Rapamycin sodium salt
CAS :<p>Seco Rapamycin sodium salt is a ring-opened product of Rapamycin.</p>Formule :C51H79NNaO13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :937.1775-Aminolevulinic acid
CAS :<p>5-Aminolevulinic acid: heme synthesis intermediate, photosensitizer, antineoplastic, prodrug, treats actinic keratosis with blue light.</p>Formule :C5H9NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :131.13CAY10677
CAS :<p>CAY10677 has a wide range of applications in life science related research.</p>Formule :C25H37N5Couleur et forme :SolidMasse moléculaire :407.59Fluticasone dimer impurity
CAS :<p>Fluticasone dimer impurity: a dimer of Fluticasone Propionate, a potent corticosteroid.</p>Formule :C43H51F5O8SCouleur et forme :SolidMasse moléculaire :822.923-Methylcholanthrene
CAS :3-Methylcholanthrene is a carcinogenic polycyclic hydrocarbon formed during combustion, accumulates in prostate tissue, and serves as a prostate cancer model.Formule :C21H16Degré de pureté :99.49%Masse moléculaire :268.35Propionylcarnitine
CAS :<p>Propionylcarnitine (Propionyl carnitine) is a widely used dietary supplement that has been associated with glaucoma and does it ruptu</p>Formule :C10H19NO4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :217.26Desmethylazelastine
CAS :<p>Desmethylazelastine, Azelastine's metabolite; 97% protein bound; 54-hour half-life; treats allergies, asthma, diabetes, SARS-CoV-2.</p>Formule :C21H22ClN3OCouleur et forme :SolidMasse moléculaire :367.87Thalifendine chloride
CAS :Thalifendine chloride is a metabolite of berberine,the methoxy group at the C-10 position undergoes demethylation by CYP51. cytotoxicity against P-388 cells.Formule :C19H16ClNO4Couleur et forme :SolidMasse moléculaire :357.79h-NTPDase-IN-4
CAS :<p>h-NTPDase-IN-4, a pan-inhibitor, targets h-NTPDase1/2/3/8 with IC50s: 3.58, 10.21, 0.13, 13.57 μM.</p>Formule :C22H8F12N2SDegré de pureté :99.92%Couleur et forme :SoildMasse moléculaire :560.36MCI-INI-3
CAS :<p>MCI-INI-3 is a selective competitive inhibitor of human ALDH1A3, with a Ki value of 0.55 μM for ALDH1A3 and 78.2 μM for ALDH1A1. It inhibits retinoic acid biosynthesis and can reduce the viability of glioblastoma cells GSC-83 and GSC-326.</p>Formule :C21H15N3O4Couleur et forme :SolidMasse moléculaire :373.36DSPE-PEG1000-LyP-1
<p>DSPE-PEG1000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). LyP-1 specifically targets tumor-associated lymphatic vessels and macrophages.</p>Couleur et forme :Odour SolidCAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Couleur et forme :Odour SolidHepaxanthin
CAS :<p>Hepaxanthin is a carotenoid.</p>Formule :C20H30O2Couleur et forme :SolidMasse moléculaire :302.4510-Formyldihydrofolate
CAS :<p>10-Formyldihydrofolate is a Methotrexate metabolite. It inhibits thymidylate synthetase and glycinamide ribotide transformylase.</p>Formule :C20H21N7O7Couleur et forme :SolidMasse moléculaire :471.43α-Glucosidase-IN-79
<p>α-Glucosidase-IN-79 (Compound 4d9) is a non-competitive α-glucosidase inhibitor with an IC50 of 2.11 μM, demonstrating greater inhibitory potency than the existing α-glucosidase inhibitors Acarbose (IC50 of 327.0 μM) and HXH8r (IC50 of 15.32 μM). It exhibits no cytotoxicity on normal human liver cells (LO2) and shows good metabolic stability in rat plasma. α-Glucosidase-IN-79 holds promise for research in type 2 diabetes.</p>Formule :C21H22N2O5SCouleur et forme :SolidMasse moléculaire :414.475(Ile8)-Oxytocin acetate
<p>(Ile8)-Oxytocin acetate is a neurohypophysial hormone analog of oxytocin produced in marsupials.</p>Formule :C45H70N12O14S2Couleur et forme :SolidMasse moléculaire :1067.24Anti-ANGPTL4 Antibody
<p>Anti-ANGPTL4 Antibody is a humanized antibody targeting ANGPTL4.</p>Degré de pureté :99.4% (SDS-PAGE); 98.4% (SEC-HPLC) - 99.4% (SDS-PAGE); 98.4% (SEC-HPLC)Couleur et forme :Odour Liquid(R)-SCH 42495
CAS :<p>(R)-SCH 42495, less potent enantiomer of NEP inhibitor SCH 42495, has oral antihypertensive action.</p>Formule :C20H29NO4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.58IDO1/TDO-IN-8
<p>IDO1/TDO-IN-8 (Compound CZ-17) is a dual IDO1 and TDO inhibitor capable of crossing the blood-brain barrier, with EC50 values of 0.33 μM and 1.78 μM, respectively. It modulates the kynurenine pathway of tryptophan metabolism, reducing the kynurenine/tryptophan ratio. IDO1/TDO-IN-8 has neuroprotective effects, alleviating motor dysfunction and improving depressive behavior, making it relevant for research into Parkinson's disease with comorbid depression.</p>Formule :C17H14N2SCouleur et forme :SolidMasse moléculaire :278.371-Naphthyl 3,5-dinitrobenzoate
CAS :<p>1-Naphthyl 3,5-dinitrobenzoate (JMC-4) is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.</p>Formule :C17H10N2O6Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :338.27Transketolase-IN-6
<p>Transketolase-IN-6 (Compound 6bj) serves as a lead compound for herbicides. It achieves approximately 80% root inhibition in redroot pigweed (Amaranthus retroflexus) and green foxtail (Setaria viridis). Moreover, Transketolase-IN-6 is an effective inhibitor of transketolase (TK).</p>Formule :C23H27ClN6OMasse moléculaire :438.19349DSPE-PEG5000-KAA
<p>DSPE-PEG5000-KAA is a PEG compound composed of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically targets the tumor vasculature of RIP-Tag2 transgenic mice. DSPE-PEG5000-KAA can be utilized for drug delivery purposes.</p>Couleur et forme :Odour Solid2-Pentyl-1H-benzo[d]imidazole
CAS :<p>2-Pentyl-1H-benzo[d]imidazole is a micromolar level inhibitor of Cytochrome P450 1A1 and 2B1 and has antibacterial activity against Fusarium verticillioides.</p>Formule :C12H16N2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :188.27TNAP-IN-1
CAS :<p>TNAP-IN-1 is a specific inhibitor of tissue-nonspecific alkaline phosphatase (TNAP) and is utilized in studying diseases related to soft tissue calcification.</p>Formule :C17H16N2O4SDegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :344.39Roridin L2
CAS :<p>Roridin L2 is a natural product for research related to life sciences. The catalog number is T41264 and the CAS number is 85124-22-7.</p>Formule :C29H38O9Couleur et forme :SolidMasse moléculaire :530.614Daclatasvir Impurity C
CAS :<p>Daclatasvir Impurity C is an impurity found in Daclatasvir, a robust inhibitor of the HCV NS5A protein [1].</p>Formule :C29H32N6O3Couleur et forme :SolidMasse moléculaire :512.611R-CaN-AID
CAS :<p>11R-CaN-AID is a potent, cell-permeant inhibitor of calcineurin [1] [2].</p>Formule :C135H248N70O34S2Couleur et forme :SolidMasse moléculaire :3459.99Ionizable Lipid 4
CAS :<p>Ionizable Lipid 4 is an ionizable cationic lipid that forms as a product of the rearrangement of cationic lipid CA-lipid 5 under hydrogen peroxide induction.</p>Formule :C48H85NO7Couleur et forme :SolidMasse moléculaire :788.19(S)-Higenamine hydrobromide
CAS :<p>(S)-Higenamine hydrobromide, S-enantiomer for benzylisoquinoline synthesis, results from dopamine and 4-HPAA condensation by NCS.</p>Formule :C16H18BrNO3Couleur et forme :SolidMasse moléculaire :352.222-Hydroxyquinoline
CAS :<p>Compound PDK0291, with CAS No. 59-31-4, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0291 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C9H7NOCouleur et forme :White SolidMasse moléculaire :145.15MTHFD2-IN-2
<p>MTHFD2-IN-2 (compound 13) serves as a potent inhibitor of methylenetetrahydrofolate dehydrogenase (MTHFD2) [1].</p>Formule :C22H18N4O5Couleur et forme :SolidMasse moléculaire :418.4Phenylsulfamide
CAS :<p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>Formule :C6H8N2O2SCouleur et forme :SolidMasse moléculaire :172.2Pectin
CAS :<p>Pectin, a plant cell wall derived heteropolysaccharide, forms nanoparticles for delivery and acts as an antimicrobial adsorbent.</p>Couleur et forme :SolidIlaprazole sulfone
CAS :<p>Ilaprazole sulfone, main Ilaprazole metabolite, formed mostly by CYP3A4/5, is an oral proton pump inhibitor.</p>Formule :C19H18N4O3SCouleur et forme :SolidMasse moléculaire :382.44Carbazeran citrate
CAS :<p>aldehyde oxidase (AO) substrate</p>Formule :C24H32N4O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.53DSPE-PEG5000-RVG29
<p>DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.</p>Couleur et forme :Odour SolidPDE5-IN-9
CAS :<p>WAY-639921 treats cardiovascular and respiratory conditions by inhibiting PDE1c.</p>Formule :C18H14N4SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :318.4N-Desethyl Bimatoprost
CAS :<p>N-Desethyl Bimatoprost (17-phenyl trinor PGF2α amide) is an F-series PG analog in which the C-1 carboxyl group has been modified to an unsubstituted amide.</p>Formule :C23H33NO4Couleur et forme :SolidMasse moléculaire :387.51Herbicidal agent 6
<p>Herbicidal agent 6 (D15) functions as a Transketolase (TKL) inhibitor and exhibits herbicidal activity.</p>Couleur et forme :Odour SolidCUDA
CAS :<p>CUDA is an effective soluble cyclohydrolase inhibitor with IC50 of 11.1 nM and 112 nM for mouse sEH and human sEH, respectively.</p>Formule :C19H36N2O3Degré de pureté :97.585%Couleur et forme :SolidMasse moléculaire :340.5Cortisol sulfate
CAS :<p>Cortisol sulfate (Cortisol 21-sulfate) is a metabolite of Cortisol . Cortisol sulfate is a specific ligand for intracellular transcortin [1] [2] [3] .</p>Formule :C21H30O8SCouleur et forme :SolidMasse moléculaire :442.5211β-HSD1 inibitor 19
CAS :<p>3-chloro-4-sulfonyl-Benzonitrile inhibits hHSD1/mHSD1, IC50: 16nM/10nM.</p>Formule :C19H16ClF4N3O2SDegré de pureté :99.58%Couleur et forme :SoildMasse moléculaire :461.86
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