Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(270 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(97 produits)
- Lipides(59 produits)
- Lipoxygénase(125 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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Captopril EP Impurity E
CAS :<p>Captopril EP Impurity E, an ACE inhibitor with antihypertensive properties, has an IC50 of 0.025 μM.</p>Formule :C9H15NO3Couleur et forme :SolidMasse moléculaire :185.22ML266
CAS :<p>ML266: GCase chaperone, non-inhibiting, IC50=2.5 µM, aids mutant protein transport, may help in Gaucher disease study.</p>Formule :C24H22BrN3O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :496.35Fmoc-Cys(Acm)-OH
CAS :<p>Fmoc-Cys(Acm)-OH (Fmoc-S-acetamidomethyl-L-cysteine) is a cysteine derivative.</p>Formule :C21H22N2O5SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :414.47CAY10462
CAS :<p>CAY10462 (CTK8E8405) is an effective and selective inhibitor of the 20-HETE synthase CYP4A11 with an IC50 of 8.8 nM.</p>Formule :C17H27Cl2N3ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :360.32hBChE-IN-3
<p>hBChE-IN-3 (compound 30) serves as both an activator of carbonic anhydrase (CA) and an inhibitor of cholinesterase (ChE), exhibiting IC50 values of 7.4 nM for AchE and 1.9 nM for BchE. This compound is utilized in the research of neurodegenerative and psychiatric disorders.</p>Couleur et forme :Odour Solidβ-Glucosidase
CAS :<p>β-Glucosidase is a glucoside bond hydrolase involved in glucose metabolism and can be used to study diseases caused by abnormal glucose metabolism.</p>Formule :C24H44O12Couleur et forme :SolidMasse moléculaire :524.6Xanthine oxidase-IN-16
<p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>Couleur et forme :Odour SolidHistamine glutarimide
CAS :<p>Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.</p>Formule :C10H13N3O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :207.23γ-glutamyltransferase
CAS :<p>γ-glutamyltransferase (GGT) is an enzyme located on the outer surface of the cell membrane. It maintains physiological concentrations of intracellular glutathione and cellular defense against oxidative stress by cleaving extracellular glutathione and increasing the availability of amino acids. γ-glutamyltransferase can be utilized as a biomaterial or organic compound in life science-related research.</p>Couleur et forme :SolidGlcNAc kinase (EcNagK)
<p>GlcNAc kinase (EcNagK), ATP-dependent, phosphorylates C-6 hydroxyl on GlcNAc, producing GlcNAc-6-P.</p>Couleur et forme :SolidWVSAV
<p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>Formule :C27H40N6O7Couleur et forme :SolidMasse moléculaire :560.64DSPE-PEG5000-NGR
<p>DSPE-PEG5000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide has the capability to target tumor vasculature antigen CD13. DSPE-PEG5000-NGR is applicable in drug delivery.</p>Couleur et forme :Odour SolidPhenacaine
CAS :<p>Phenacaine, also known as Holocaine, is a local anesthetic that blocks certain Ca 2+ enzymes in red blood cells, brain, and heart.</p>Formule :C18H22N2O2Couleur et forme :SolidMasse moléculaire :298.38Leucylproline
CAS :<p>Leucylproline is a peptide that proteolytic breakdown product by larger proteins.</p>Formule :C11H20N2O3Couleur et forme :SolidMasse moléculaire :228.298-Demethyl Ivabradine
CAS :<p>8-Demethyl Ivabradine, a metabolite of Ivabradine, is an oral HCN channel blocker.</p>Formule :C26H34N2O5Couleur et forme :SolidMasse moléculaire :454.567Tacalcitol monohydrate
CAS :<p>Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.</p>Formule :C27H46O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :434.65Lofacimig
<p>Lofacimig is a bispecific antibody of VH-VH-G1(h-CH2-CH3) dimer type that targets FXI/PTA.</p>Couleur et forme :Odour LiquidD-(+)-Trehalose-13C12
CAS :<p>D-(+)-Trehalose-13C12 is an isotopic label of D-(+)-Trehalose, enriched with 13C. This compound is pervasively found and often employed as a food ingredient and a shape-forming agent for active molecules.</p>Formule :C12H22O11Couleur et forme :SolidMasse moléculaire :354.21Lysylglutamic acid
CAS :<p>Lysylglutamic acid is a dipeptide composed of the amino acids lysine (Lysine, Lys) and glutamic acid (Glutamic acid, Glu), with an inhibitory constant (Ki) of 1.3 mM for the membrane transport protein PEPT1.</p>Formule :C11H21N3O5Couleur et forme :SolidMasse moléculaire :275.3NAADP sodium
<p>NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.</p>Formule :C21H27N6O18P3Couleur et forme :SolidMasse moléculaire :744.39Inulobiose
CAS :<p>Inulobiose, a difructan disaccharide isolated from Pistacia vera L., demonstrates inhibitory effects on α-glycosidase (α-glycosidase) and α-amylase (α-amylase) activities, with IC50 values of 1.87 and 40.72 mg/mL respectively. It is utilized in research related to diabetes and glomerular filtration rate testing.</p>Formule :C12H22O11Couleur et forme :SolidMasse moléculaire :342.3Sphingolipid ceramide N-deacylase (SCDase)
CAS :<p>SCDase splits fatty acids from sphingosine in glycosphingolipids, forming lysoglycosphingolipids.</p>Couleur et forme :SolidLysylcysteine TFA
<p>Lysylcysteine (L-Lysyl-L-cysteine)TFA is a dipeptide composed of lysine and cysteine.</p>Formule :C13H21F6N3O7SCouleur et forme :SolidMasse moléculaire :477.10044GLUT1-IN-1
<p>GLUT1-IN-1 inhibits GLUT1; cytotoxic to HeLa, A549, HepG2 (IC50: 5.49, 11.14, 8.73 μM); potential in PDT and cancer research.</p>Formule :C25H31BF2I2N6O7Couleur et forme :SolidMasse moléculaire :830.171-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine
CAS :<p>Endogenous metabolite: 1-myristoyl-2-stearoyl-sn-glycero-3-phosphocholine, a phosphatidylcholine example.</p>Formule :C40H80NO8PDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :734.04Vardenafil dihydrochloride
CAS :<p>Vardenafil dihydrochloride (Levitra) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>Formule :C23H34Cl2N6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :561.52Enterostatin(human,mouse,rat)
CAS :<p>Enterostatin, human, mouse, rat is a pentapeptide that reduces fat intake.</p>Formule :C21H36N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :496.569ML171
CAS :<p>Compound PDK0326, with CAS No. 6631-94-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0326 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C14H11NOSCouleur et forme :Mustard-Colored PowderMasse moléculaire :241.3Senecionine acetate
CAS :<p>Senecionine acetate, a pyrrolizidine alkaloid, blocks Ca2+ storage in cells by inactivating sulfhydryl groups.</p>Formule :C20H27NO6Couleur et forme :SolidMasse moléculaire :377.432-Methoxy-4-propylphenol
CAS :<p>2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.</p>Formule :C10H14O2Couleur et forme :SolidMasse moléculaire :166.22Rennin
CAS :<p>Rennin or Chymosin, a stomach enzyme in some animals, curdles milk by cleaving K-casein; key in cheese making.</p>Couleur et forme :SolidRibulose, L-
CAS :<p>Ribulose: key in pentose metabolism, aids L-ribose isomerase study, yeast engineering, and chiral compound research.</p>Formule :C5H10O5Couleur et forme :SolidMasse moléculaire :150.13A32390A
CAS :<p>A32390A, an antibiotic inhibitor, shows antimicrobial activity against gram-positive bacteria and fungi.</p>Formule :C18H24N2O8Couleur et forme :SolidMasse moléculaire :396.39γ-Glu-Gly TFA
<p>γ-Glu-Gly TFA, a γ-glutamyl dipeptide, is a human lipid metabolite with a structure resembling GABA (γ-aminobutyric acid).</p>Couleur et forme :LiquidTrimipramine N-oxide
CAS :<p>Trimipramine N-oxide, a trimipramine metabolite, inhibits hNAT, hSERT, hDAT, and hOCT1/2 with IC50s 11.7-27.4 nM; for depression/anxiety research.</p>Formule :C20H26N2OCouleur et forme :SolidMasse moléculaire :310.431-(2-Quinoxalinyl)-1,2,3,4-butanetetrol
CAS :<p>1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is a quinoxaline derivative and endogenous metabolite applicable to biochemical experiments and drug synthesis research.</p>Formule :C12H14N2O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :250.25DSPE-PEG3000-R6H4
<p>DSPE-PEG3000-R6H4 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (R6H4). R6H4 is applicable for pH-responsive anticancer drug delivery. DSPE-PEG3000-R6H4 can be utilized for drug delivery purposes.</p>Couleur et forme :Odour SolidAnti-osteoporosis agent-10
<p>Anti-osteoporosis agent-10 is an inhibitor of osteoporosis that suppresses the formation of osteoclasts with an IC50 of 0.042 μM. It also exhibits antagonistic activity towards PPARγ, with an EC50 value of 0.75 μM.</p>Couleur et forme :Odour SolidIPI-9119
CAS :<p>IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).</p>Formule :C24H19F2N5O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :495.43MCC-555
CAS :<p>MCC-555 (Isaglitazone) is a PPARα and PPARγ agonist exerting antihyperglycemic effects.</p>Formule :C21H16FNO3SDegré de pureté :99.07% - 99.82%Couleur et forme :SolidMasse moléculaire :381.42Viridicatin
CAS :<p>Viridicatin is a natural product for research related to life sciences. The catalog number is T38335 and the CAS number is 129-24-8.</p>Formule :C15H11NO2Couleur et forme :SolidMasse moléculaire :237.255-Lipoxygenase-IN-3
CAS :<p>Compound 14, a <1 μM 5-lipoxygenase inhibitor, researches inflammation, cancer, stroke, Alzheimer's.</p>Formule :C19H16ClN5OCouleur et forme :SolidMasse moléculaire :365.82Canine Factor Xa
<p>CanineFactor Xa is derived from purified Canine Factor X through activation by Russell's Viper Venom, after which the venom is removed.</p>Couleur et forme :Odour SolidPepticinnamin E
CAS :<p>Pepticinnamin E is a naturally occurring bisubstrate farnesyltransferase inhibitor.</p>Formule :C49H54ClN5O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :908.43Carbonic anhydrase inhibitor 30
<p>Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].</p>Formule :C23H22FN3O5SCouleur et forme :SolidMasse moléculaire :471.12642(±)16-HDHA
CAS :<p>(±)16-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.</p>Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.495Creatine kinase (OcCK)
CAS :<p>Creatine kinase (OcCK) converts creatine and ATP into phosphocreatine and ADP, crucial for ATP/ADP balance during high energy demand.</p>Couleur et forme :Solid15-keto Latanoprost (free acid)
CAS :<p>15-keto Latanoprost, a less potent metabolite and impurity of latanoprost, lowers intraocular pressure in monkeys and constricts pupils in cats.</p>Formule :C23H32O5Couleur et forme :SolidMasse moléculaire :388.55-Formylcytosine
CAS :<p>5-Formylcytosine (5FC) is a rare mammalian DNA base aiding in demethylation, altering helix structure, and affecting RNA polymerase II activity.</p>Formule :C5H5N3O2Couleur et forme :SolidMasse moléculaire :139.11Fasnall HCl
<p>Fasnall HCl is a selective FASN inhibitor that acts through its co-factor binding sites.</p>Formule :C19H23ClN4SDegré de pureté :99.9%Couleur et forme :SoildMasse moléculaire :374.93
