Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(197 produits)
- Caséine Kinase(139 produits)
- DHFR(30 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(63 produits)
- Facteur Xa(87 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(233 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(56 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(36 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(62 produits)
- Lipoxygénase(134 produits)
- MAO(84 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(84 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(17 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(43 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9198 produits trouvés pour "Métabolisme"
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CM121
CAS :CM121, a reversible ALDH1A2 inhibitor, targets active site with IC50=0.54μM, Kd=1.1μM, using hydrophobic interactions.Formule :C24H17FN4O3SCouleur et forme :SolidMasse moléculaire :460.4828-Epirapamycin
CAS :28-Epirapamycin, an impurity of Rapamycin, serves as a potent and specific mTOR inhibitor, exhibiting an IC50 value of 0.1 nM in HEK293 cells [1].Formule :C51H79NO13Couleur et forme :SolidMasse moléculaire :914.17(3E,8Z,11Z)-Tetradeca-3,8,11-trienyl acetate
CAS :(3E,8Z,11Z)-Tetradeca-3,8,11-trienyl acetate is an additive to tobacco products and a vegetable pest pheromone.Formule :C16H26O2Degré de pureté :83.13%Couleur et forme :SolidMasse moléculaire :250.38N-Pivaloyl-L-tyrosine
CAS :N-Pivaloyl-L-tyrosine is an N-pivaloyl amino acid ester.Formule :C14H19NO4Couleur et forme :SolidMasse moléculaire :265.30T-705RMP
CAS :T-705RMP, a T-705 byproduct, mildly inhibits IMPDH in host cells; IC50 = 601 μM.Formule :C10H13FN3O9PCouleur et forme :SolidMasse moléculaire :369.20Aspercolorin
CAS :Aspercolorin is a fungal metabolite produced by Aspergillus.Formule :C25H28N4O5Couleur et forme :SolidMasse moléculaire :464.51N-Desalkyludenafil
CAS :N-Desalkyludenafil, a metabolite of Udenafil, functions as a PDE5 inhibitor and is utilized in the study of erectile dysfunction [1].Formule :C18H23N5O4SCouleur et forme :SolidMasse moléculaire :405.47Coproporphyrin I
CAS :Coproporphyrin I, an endogenous metabolite found in urine and blood, is utilized in researching liver disease and porphyria [1] [2] [3] [4].Formule :C36H38N4O8Couleur et forme :SolidMasse moléculaire :654.71Zifcasiran
CAS :Zifcasiran reduces HIF synthesis, has antitumor properties, useful in renal carcinoma studies.Formule :C737H972F20N211O349P43S8Couleur et forme :SolidMasse moléculaire :20339.13Dibutyl-3-Hydroxybutyl Phosphate
CAS :Dibutyl 3-hydroxybutyl phosphate forms from tributyl phosphate metabolism, goldfish liver microsomes, and TBP radiolysis.Formule :C12H27O5PCouleur et forme :SolidMasse moléculaire :282.31Febuxostat dicarboxylic acid impurity
CAS :Febuxostat dicarboxylic acid impurity is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1] .Formule :C16H17NO5SCouleur et forme :SolidMasse moléculaire :335.38KF-52
KF-52 is an inhibitor of phosphofructokinase-1 (PFK1), possessing an IC50 value of 2.1 μM. It significantly enhances the ratio of oxygen consumption rate (OCR) to extracellular acidification rate (ECAR).Formule :C21H19F3N2O3Couleur et forme :SolidMasse moléculaire :404.382URB754
CAS :"URB754 inhibits rat MAGL with an IC50 of 200 nM, possibly due to impurity. Weak FAAH and CB1 binding, no COX inhibition. Potential pain management target."Formule :C16H14N2O2Couleur et forme :SolidMasse moléculaire :266.29Deoxycholic acid 3-sulfate
CAS :Deoxycholic acid 3-sulfate is a sulphonated bile acid and endogenous metabolite, suitable for biochemical experiments and drug synthesis research.Formule :C24H40O7SCouleur et forme :SoildMasse moléculaire :472.64LysoFos Glycerol 14
CAS :LysoFos Glycerol 14 is a useful organic compound for research related to life sciences. The catalog number is TF0117 and the CAS number is 326495-21-0.Formule :C20H40NaO9PCouleur et forme :SolidMasse moléculaire :478.4951,2,3-Trioctanoyl-rac-glycerol-13C3
CAS :1,2,3-Trioctanoyl-rac-glycerol-13C3 is intended for use as an internal standard for the quantification of 1,2,3-trioctanoyl-rac-glycerol by GC- or LC-MS.Formule :C27H50O6Couleur et forme :SolidMasse moléculaire :473.668N-β-alanyldopamine hydrochloride
CAS :N-β-Alanyldopamine hydrochloride (NBAD hydrochloride) represents the primary dopamine derivative found in haemolymph [1].Formule :C11H17ClN2O3Couleur et forme :SolidMasse moléculaire :260.72Z-Pro-Ala
CAS :Z-Pro-Ala, an acid carboxypeptidase, can be isolated from the grains and leaves of Triticum aestivum L. (wheat) [1].Formule :C16H20N2O5Couleur et forme :SolidMasse moléculaire :320.34trans-4,5-epoxy-2(E)-Decenal
CAS :Essential fatty acids like arachidonate can oxidize, forming trans-4,5-epoxy-2(E)-decanal, which imparts a metallic taste and harms cell proteins.Formule :C10H16O2Couleur et forme :SolidMasse moléculaire :168.236Neuron-specific enolase, Human
Neuron-specific enolase, Human (EC 4.2.1.11), is an enolase enzyme that serves as a biomarker for traumatic brain injury (TBI), stroke following cardiac arrest, hypoxic encephalopathy, and acute spinal cord injury (SCI).Couleur et forme :Odour SolidRawsonol
CAS :Rawsonol is a HMG-CoA reductase inhibitor from the tropical green alga Avrainvillea rawsoni.Formule :C29H24Br4O7Couleur et forme :SolidMasse moléculaire :804.11Posaconazole D-glucuronide
Posaconazole D-glucuronide (SCH 56592 D-glucuronide) is the glucuronide metabolite of the antifungal agent Posaconazole. It is formed in human liver microsomes through catalysis by UGT1A4.Couleur et forme :Odour Solidα-Glucosidase-IN-24
CAS :α-Glucosidase-IN-24 (Compound 13), an α-Glucosidase inhibitor, exhibits an IC50 value of 451 μM and can be derived from Swertia kouitchensis [1].Formule :C26H30O15Couleur et forme :SolidMasse moléculaire :582.515,6-Dihydroabiraterone
CAS :5,6-Dihydroabiraterone, a metabolite of Abiraterone, is a strong, irreversible CYP17A1 inhibitor, effective in CRPC.Formule :C24H33NOCouleur et forme :SolidMasse moléculaire :351.52Adipokinetic hormone I (Locusta migratoria)
CAS :Lom-AKH-I is an AKH from Locusta migratoria that boosts fat body cAMP and mobilizes energy for insect flight.Formule :C54H74N14O15Couleur et forme :SolidMasse moléculaire :1159.25DMPG sodium
CAS :DMPG sodium is a phospholipid analog commonly used in the preparation of artificial lipid bilayers to mimic the structure and function of biological membranes.Formule :C34H66NaO10PDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :688.85LL P880 β
CAS :LL P880 beta is a fungal metabolite.Formule :C11H18O5Couleur et forme :SolidMasse moléculaire :230.26Sarcophine
CAS :Sarcophine is a natural cembranoid from the Red Sea soft coral Sarcophyton glaucum.Formule :C20H28O3Couleur et forme :SolidMasse moléculaire :316.441NMTCA
CAS :NMTCA (NMTPRO) is a sulfur-containing N-nitrosamino acid utilized as an endogenous nitrosation indicator in gas chromatography-thermal energy analysis.Formule :C5H8N2O3SCouleur et forme :SolidMasse moléculaire :176.19Remisporine B
CAS :Remisporine B, a polyketide found in Penicillium, inhibits mouse lymphocyte proliferation (IC50 = 30-32.4 μg/ml).Formule :C30H24O12Couleur et forme :SolidMasse moléculaire :576.5β-1,4-Galactosyltransferase 1 (Y285L)
Beta-1,4-Galactosyltransferase 1 (Y285L) is capable of enzymatically synthesizing the LacdiNAc motif. Additionally, Beta-1,4-Galactosyltransferase 1 (Y285L) can transfer GalNAc from UDP-GalNAc.Febuxostat amide impurity
CAS :Febuxostat amide impurity is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1]Formule :C16H18N2O4SCouleur et forme :SolidMasse moléculaire :334.392-oxo Clopidogrel
CAS :2-oxo Clopidogrel SR-121683 is a metabolite of Clopidogrel,catalyzed by P450 enzyme via CYP3A oxidation, ydrolysis to the active metabolite CAM.antithrombotic.Formule :C16H16ClNO3SCouleur et forme :SolidMasse moléculaire :337.82Phospholipase D
CAS :PLD is an enzyme in the phospholipase family, found across many life forms, and linked to diseases like diabetes and cancer.Couleur et forme :Solidα-1,3-N-Acetylgalactosaminyltransferase (Pm1138)
CAS :Alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138) (EC 2.4.1.40(Pm1138)), also known as the ABO system transferase, exhibits glycosyl transferase activity [1Couleur et forme :Solid3-Indoleacetic acid-d4
CAS :3-Indoleacetic acid-d4 (Indole-3-acetic acid-d4; 3-IAA-d4) is a deuterium-labeled form of 3-Indoleacetic acid. It is the most prevalent natural plant growth hormone within the auxin class. When added to cell culture media, it can stimulate the elongation and division of plant cells.Formule :C10H9NO2Couleur et forme :SolidMasse moléculaire :179.21Formate dehydrogenase
CAS :Formate dehydrogenase, found in all life forms, converts formate to CO2 and is categorized by metal content for research.Couleur et forme :SolidDMPS-Na
CAS :DMPS-Na is an arsenicolytic agent with toxicity that can be used to study cell membranes.Formule :C34H65NNaO10PDegré de pureté :≥98%Couleur et forme :SoildMasse moléculaire :701.84NY-ESO-1 (157-165) peptide
CAS :NY-ESO-1 (157–165) peptide is a peptide derived from the NY-ESO-1 protein and has the ability to activate the immune system. It is particularly effective in individuals positive for HLA-A2, as it can be recognized by CD8+ T cells, thus triggering an immune response. The presence of NY-ESO-1 (157–165) peptide in various tumors makes it a potential target for cancer immunotherapy. This peptide is also utilized in research focusing on cancer immunotherapy.Formule :C49H79N11O13S2Masse moléculaire :1094.35DSPE-PEG5000-YIGSR
DSPE-PEG5000-YIGSR is a PEG compound comprised of DSPE and the biomimetic peptide YIGSR. YIGSR interacts with the 67 kDa laminin-binding protein (LBP), enhancing the adhesion and proliferation of various cell types, such as endothelial cells, fibroblasts, and smooth muscle cells. DSPE-PEG5000-YIGSR is applicable for drug delivery.Couleur et forme :Odour SolidAP219
CAS :AP39 boosts mitochondrial H2S with triphenylphosphonium and dithiolethione; AP219 lacks H2S-donating part.Formule :C28H34O2PCouleur et forme :SolidMasse moléculaire :433.551Penicillide
CAS :Penicillide: fungal metabolite, inhibits calpain 2/ACAT (IC50 = 7.1/22.9 μM), blocks oxytocin receptors (IC50 = 67 μM), stops RNA synthesis in P388 cells.Formule :C21H24O6Couleur et forme :SolidMasse moléculaire :372.417DPP IV/hCA II-IN-1
CAS :DPP IV/hCA II-IN-1: strong DPP IV & CA inhibitor, IC50=0.049μM (DPP IV), Ki=0.0361-3.034μM (CA II-IV).Formule :C17H20N2O5SCouleur et forme :SolidMasse moléculaire :364.42Ganglioside sialidase (AuSialidase S)
CAS :AuSialidase S is an endogenous metabolite involved in neuronal differentiation and neurite outgrowth.Couleur et forme :SolidPKM2 activator 7
PKM2 activator 7 (Compd B4) is a PKM2 activator with an AC50 value of 0.144 μM. It functions by inhibiting the growth of T cells, thereby alleviating DSS-induced colitis in mice.Formule :C16H19F3O4Masse moléculaire :332.12354α-D-Glucose-1-phosphate disodium hydrate
CAS :α-D-Glucose-1-phosphate disodium hydrate serves multiple roles in medical and biochemical applications, including as a precursor in the synthesis of glucuronicFormule :C6H15Na2O11PCouleur et forme :SolidMasse moléculaire :340.13Mycestericin G
CAS :Mycestericin G, a sphingosine-like fungal metabolite, demonstrates immunosuppressive activity [1].Formule :C21H41NO5Couleur et forme :SolidMasse moléculaire :387.55SB-435495
CAS :SB-435495 is a compound characterized by its potent, selective, reversible, and non-covalent inhibition of Lp-PLA2, demonstrating an IC50 value of 0.06 nM.Formule :C38H40F4N6O2SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :720.82PDE5-IN-9
CAS :WAY-639921 treats cardiovascular and respiratory conditions by inhibiting PDE1c.Formule :C18H14N4SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :318.4Cy3-PEG-DSPE (MW 3400)
Cy3-PEG-DSPE (MW 3400) is a PEG phospholipid that incorporates Cy3 dye, utilized for labeling proteins/nucleic acids and in fluorescence microscopy. It can self-assemble in aqueous solutions to form micelles/lipid bilayers, and is employed in the creation of liposomes or nanoparticles for delivering nutrients such as mRNA or DNA vaccines.Couleur et forme :SolidMasse moléculaire :3400 (Average)
