Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(197 produits)
- Caséine Kinase(139 produits)
- DHFR(30 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(87 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(227 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(56 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(62 produits)
- Lipoxygénase(134 produits)
- MAO(85 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(85 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(17 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(43 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9188 produits trouvés pour "Métabolisme"
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GPX4-IN-16
GPX4-IN-16 ((R)-9i) is a potent inhibitor of GPX4 with a KD value of 20.4 nM, exhibiting cytotoxic properties and anticancer activity.Formule :C29H24N4O3S2Couleur et forme :SolidMasse moléculaire :540.656Decarbamylsaxitoxin
CAS :Decarbamylsaxitoxin is a biochemical.Formule :C9H16N6O3Couleur et forme :SolidMasse moléculaire :256.26Cy3-PEG-DSPE (MW 3400)
Cy3-PEG-DSPE (MW 3400) is a PEG phospholipid that incorporates Cy3 dye, utilized for labeling proteins/nucleic acids and in fluorescence microscopy. It can self-assemble in aqueous solutions to form micelles/lipid bilayers, and is employed in the creation of liposomes or nanoparticles for delivering nutrients such as mRNA or DNA vaccines.Couleur et forme :SolidMasse moléculaire :3400 (Average)Methyl 7(Z)-hexadecenoate
CAS :Methyl 7(Z)-hexadecenoate, a sex pheromone of Trogoderma glabrum, elicits attraction and sexually excitatory responses in male Trogoderma glabrum [1].Formule :C17H32O2Couleur et forme :SolidMasse moléculaire :268.43Trimetazidine-N-oxide
CAS :Trimetazidine-N-oxide, main active metabolite of Trimetazidine, blocks 3-ketoyl CoA thiolase (IC50: 75nM) and has multiple protective properties.Formule :C14H22N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :282.34Suberylglycine
CAS :Suberylglycine is an acyl glycine that is a normally minor metabolite of fatty acid.Formule :C10H17NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.251-Arachidonoyl Lysophosphatidic Acid (ammonium salt)
CAS :1-Arachidonoyl LPA: phospholipid with arachidonic acid, sn-1, LPA2 receptor binder, EC50 ~10 nM, modulates cytokine secretion, affects cell differentiation.Formule :C23H42NO7PCouleur et forme :SolidMasse moléculaire :475.5632MD
CAS :2MD, a vitamin D-like oral drug, enhances bone mass/strength and lowers IOP by gene regulation.Formule :C27H44O3Couleur et forme :SolidMasse moléculaire :416.64Carveol, (-)-
CAS :(-)-Carveol is an unsaturated, cyclic monoterpenoid alcohol; used in cosmetics for fragrance and as a food flavor additive.Formule :C10H16OCouleur et forme :SolidMasse moléculaire :152.23Galactose 1-dehydrogenase
Galactose 1-dehydrogenase, pseudomonas fluorescens, a dehydrogenase found in Pseudomonas fluorescens, facilitates the oxidation of L-arabinose and D-galactose, utilizing NADP+/NAD+ as a cofactor. This enzyme is employed in diagnostic assays to quantify total galactose levels and serves as a biocatalyst in the production of galacturonic acid salts.Couleur et forme :Odour Solid(S)-Salsolidine
CAS :(S)-Salsolidine is a MAO inhibitor with Ki 63μM; its R enantiomer is more effective, Ki 26μM.Formule :C12H17NO2Couleur et forme :SolidMasse moléculaire :207.27α-1,3/4-Fucosyltransferase (α1,3/4FucT)
CAS :alpha-1,3/4-Fucosyltransferase (α1,3/4FucT) (Hp3/4FT) can be found in Helicobacter pylori .Couleur et forme :SolidMPC-IN-1
MPC-IN-1 (compound 4i), a derivative of UK-5099, is a cyanocinnamate-based inhibitor of the mitochondrial pyruvate transporter (MPC). This compound selectively fosters the development of hair follicle stem cells while not impacting normal cells. It enhances cellular lactate production and has shown significant hair growth promotion in mice, suggesting its potential use in combating hair loss.Formule :C18H13N3O2Couleur et forme :SolidMasse moléculaire :303.311-Stearoyl-2-Adrenoyl-sn-glycero-3-PE
CAS :Phospholipid with stearic acid at sn-1, adrenic acid at sn-2; less in older human hippocampal mitochondria.Formule :C45H82NO8PCouleur et forme :SolidMasse moléculaire :796.124PtdIns-(3)-P1 (1,2-dioctanoyl) (sodium salt)
CAS :PtdIns phosphates are minor but crucial in cell signaling. PtdIns-(3)-P1 with C8:0 mimics natural lipids and can be phosphorylated to PIP2 or PIP3.Formule :C25H46Na2O16P2Couleur et forme :SolidMasse moléculaire :710.55Fluazifop-P-butyl
CAS :Fluazifop-P-butyl is an arylophenoxypropionate group graminicide that functions as an inhibitor of acetyl-CoA carboxylase (ACCase)[1].Formule :C19H20F3NO4Couleur et forme :Light Yellow LiquidMasse moléculaire :383.36Ot-730
CAS :Ot-730（QLT 091568） is a novel selective beta-blocker prodrug for the study of ocular diseases.Cost-effective and quality-assured.Formule :C25H36N2O8Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :492.56m-PEG8-DSPE
m-PEG8-DSPE is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.Formule :C59H116NO17PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1142.52DSPE-PEG2000-KAA
DSPE-PEG2000-KAA is a PEG compound composed of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically binds to the tumor vasculature of RIP-Tag2 transgenic mice. DSPE-PEG2000-KAA can be used for drug delivery.Couleur et forme :Odour SolidDapagliflozin-3-O-β-D-Glucuronide
CAS :Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin .Formule :C27H33ClO12Couleur et forme :SolidMasse moléculaire :585Citreoindole
CAS :Citreoindole: a diketopiperazine from P. citreovirde, cytotoxic against HeLa cells at 8.4 μM.Formule :C29H28N4O4Couleur et forme :SolidMasse moléculaire :496.567DSPE-PEG3400-PP1
DSPE-PEG3400-PP1 is a PEG compound composed of DSPE and PP1 peptide. The PP1 peptide targets inflammatory atherosclerotic plaques. DSPE-PEG3400-PP1 can be utilized for drug delivery.Couleur et forme :Odour Solidm-Tyramine
CAS :m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator.Formule :C8H11NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :137.18D-Erythrose 4-phosphate sodium
CAS :D-erythrose 4-sodium phosphate: sodium salt of monosaccharide, made from erythritol via 3 isomerases.Formule :C4H8NaO7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :222.07Jasmone, (E)-
CAS :Jasmone, (E)- is a type of perfuming agent.Formule :C11H16OCouleur et forme :Oil SolidMasse moléculaire :164.24ESI1
ESI1 is a small molecule inhibitor of epigenetic silencing. This compound induces the formation of nuclear aggregates of the key lipid metabolism regulator SREBP1/2, thereby concentrating transcription co-activators to drive lipid/cholesterol biosynthesis. Additionally, ESI1 promotes myelin regeneration in demyelination animal models and facilitates de novo myelination on regenerating CNS axons, reversing age-related cognitive decline.Formule :C18H18ClN5OCouleur et forme :SolidMasse moléculaire :355.823-hydroxy Darifenacin
CAS :3-hydroxy Darifenacin, darifenacin metabolite, blocks M1-5 muscarinic receptors with varying potency (Kis: 2.24-79.43 nM) in CHO cells.Formule :C28H30N2O3Couleur et forme :SolidMasse moléculaire :442.559ATP ditromethamine
CAS :ATP ditromethamine is key for energy storage, metabolism, and acts as a coenzyme and signaling molecule in immunity and inflammation.Formule :C18H38N7O19P3Couleur et forme :SolidMasse moléculaire :749.45XW-032
XW-032 is an apo-IDO1 inhibitor with an IC50 of 21 nM. In the CT26 syngeneic mouse model, XW-032 demonstrates significant in vivo antitumor efficacy with a TGI of 63%, showing potential for cancer research applications.Couleur et forme :Odour SolidSaccharopine hydrochloride
Saccharopine hydrochloride, from lysine degradation, disrupts mitochondria and hinders development.Formule :C11H21ClN2O6Couleur et forme :SolidMasse moléculaire :312.75Etonitazene N-oxide
Etonitazene N-oxide (EtN-NOX) is a metabolite of the opioid compound Etonitazene.Couleur et forme :Odour SolidSethoxydim
CAS :Sethoxydim is an effective herbicide.Formule :C17H29NO3SCouleur et forme :Oily Liquid Sethoxydim Is An Oily Odorless Liquid Non Corrosive Used As An HerbicideMasse moléculaire :327.48CE(20:5(5Z,8Z,11Z,14Z,17Z)
CAS :CE(20:5(5Z,8Z,11Z,14Z,17Z) is an endogenous metabolite.Formule :C47H74O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :671.09Nucleocidin
CAS :Nucleocidin, an antitrypanosomal antibiotic, inhibits the transfer of labeled amino acids from S-RNA to protein.Formule :C10H13FN6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.31ARC19499
CAS :ARC19499, an aptamer, inhibits TFPI to aid clotting through the extrinsic pathway, enhancing thrombin in hemophilia.Couleur et forme :SolidPhenylpyropene A
CAS :Phenylpyropene A, a P. griseofulvum fungus product, blocks ACAT (IC50=0.8μM) and DGAT, kills M. persicae at 5ppm.Formule :C32H38O10Couleur et forme :SolidMasse moléculaire :582.64BRD8518
CAS :BRD8518, a PCSK9 inhibitor (EC50=0.23 μM), effectively lowers lipid levels by upregulating LDLR expression and enhancing the uptake of LDL. This compound is utilized in cardiovascular disease research.Formule :C33H32F3N3O5Couleur et forme :SolidMasse moléculaire :607.62cis-Ferulic acid 4-O-β-D-glucopyranoside
CAS :Cis-Ferulic acid 4-O-β-D-glucopyranoside (compound 7), a phenolic glycoside derived from Nitraria sibirica, demonstrates antioxidant properties and a potentFormule :C16H20O9Couleur et forme :SolidMasse moléculaire :356.32IONIS PTP1BRx sodium
IONIS PTP1BRx (ISIS 404173) sodium, an antisense inhibitor of protein tyrene phosphatase 1B (PTP-1B), exhibits antidiabetic properties. This compound is utilzed in researching insulin resistance and type 2 diabetes mellitus associated with obesity.Couleur et forme :Odour SolidAcetate kinase (ACK)
CAS :ACK, found in bacteria/archaea, phosphorylates acetate with ATP and cations, yielding acetyl-CoA; used in biochemistry.Couleur et forme :Solid(+)-Menthofuran
(+)-Menthofuran is a useful organic compound for research related to life sciences and the catalog number is T125544.Formule :C10H14OCouleur et forme :SolidMasse moléculaire :150.221Phosphoglycerate kinase
CAS :PGK is an enzyme that catalyzes phosphate transfer between 1,3-BPG and ADP, vital in glycolysis and gluconeogenesis.Couleur et forme :SolidLagunamycin
CAS :Lagunamycin is used as a novel 5-lipoxygenase inhibitor.Formule :C19H21N3O4Couleur et forme :SolidMasse moléculaire :355.39Desmethylazelastine
CAS :Desmethylazelastine, Azelastine's metabolite; 97% protein bound; 54-hour half-life; treats allergies, asthma, diabetes, SARS-CoV-2.Formule :C21H22ClN3OCouleur et forme :SolidMasse moléculaire :367.87Doxorubicinone
CAS :Adriamycin Aglycone, also known as Doxorubicinone, is an oncolytic agent. It is a metabolite of Doxorubicin which binds to the DNA minor-groove.Formule :C21H18O9Couleur et forme :SolidMasse moléculaire :414.36Trichodecenin I
CAS :Trichodecenin I is a peptaibol isolated from Trichoderma viride.Formule :C38H69N7O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :752.011Arylsulfatase
CAS :Arylsulfatase is an enzyme that catalyzes the hydrolysis of aryl sulfates, specifically recognizes and cleaves sulfated bonds.Couleur et forme :SolidNeoechinulin C
CAS :Neoechinulin C, a neuroprotective indolediketopiperazine, guards neurons against paraquat in Parkinson's.Formule :C24H27N3O2Couleur et forme :SolidMasse moléculaire :389.49Epoxide hydrolase
CAS :Epoxide hydrolase, an enzyme responsible for catalyzing the reaction of epoxides with water to convert epoxy groups into diols, plays a crucial role in the metabolism of environmental pollutants and lipids. It is instrumental in detoxification, inflammatory responses, and regulating the health of the cardiovascular system. Additionally, Epoxide hydrolase is used in asymmetric catalytic reactions, such as the asymmetric ring-opening of epoxides, which are important for the synthesis of chiral pharmaceutical molecules.Couleur et forme :Solid3-Nitro-L-tyrosine ethyl ester hydrochloride
3-Nitro-L-tyrosine ethyl ester hydrochloride is a useful organic compound for research related to life sciences and the catalog number is T124433.Formule :C11H15ClN2O5Couleur et forme :SolidMasse moléculaire :290.7
