GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.022 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5985 produits trouvés pour "GPCR/G-Protéine"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
H2L 5765834
CAS :H2L 5765834 is a lysophosphatidic acid receptors antagonistFormule :C21H12N2O7Degré de pureté :98.25% - 99.47%Couleur et forme :SolidMasse moléculaire :404.33Ref: TM-T22834
1mg58,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg177,00€25mg334,00€50mg497,00€100mg708,00€Betahistine dihydrochloride
CAS :Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formule :C8H14Cl2N2Degré de pureté :99.22% - 99.88%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :209.12Hydroxyzine dihydrochloride
CAS :Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formule :C21H27ClN2O2·2HClDegré de pureté :99.46% - 99.79%Couleur et forme :Oil PowderMasse moléculaire :447.83Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
2mg35,00€5mg51,00€10mg80,00€25mg131,00€50mg210,00€1mL*10mM (DMSO)215,00€100mg313,00€200mg445,00€Zafirlukast
CAS :Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and anti-inflammatory effects. Cost-effective and quality-assured.Formule :C31H33N3O6SDegré de pureté :99% - 99.83%Couleur et forme :SolidMasse moléculaire :575.68Rizatriptan sulfate
CAS :Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formule :C15H21N5O4SCouleur et forme :SolidMasse moléculaire :367.42Vorapaxar sulfate
CAS :Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.Formule :C29H35FN2O8SDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :590.66Ref: TM-T3098
1mg38,00€2mg49,00€5mg79,00€1mL*10mM (DMSO)99,00€10mg119,00€25mg210,00€50mg354,00€100mg528,00€500mg1.159,00€Tozadenant
CAS :Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5SB 242084
CAS :SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formule :C21H19ClN4O2Degré de pureté :99.75% - ≥98%Couleur et forme :SolidMasse moléculaire :394.85Naftopidil hydrochloride
CAS :Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formule :C24H29ClN2O3Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :428.95Ref: TM-T9220
1mg42,00€5mg82,00€1mL*10mM (DMSO)92,00€10mg111,00€25mg192,00€50mg289,00€100mg414,00€200mg580,00€AnaMorelin hydrochloride
CAS :AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formule :C31H43ClN6O3Degré de pureté :99.18% - ≥98%Couleur et forme :SolidMasse moléculaire :583.16Ref: TM-T7225
1mg34,00€2mg48,00€5mg70,00€10mg90,00€1mL*10mM (DMSO)90,00€25mg138,00€50mg168,00€100mg222,00€Afamelanotide acetate
CAS :Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.
Formule :C80H115N21O21Degré de pureté :98% - 99.494%Couleur et forme :SolidMasse moléculaire :1706.9Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.Formule :C63H104N22O17SDegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :1473.72AVN-492
CAS :AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formule :C17H21N5O2SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :359.45Ref: TM-T5179
1mg37,00€2mg50,00€5mg77,00€1mL*10mM (DMSO)85,00€10mg114,00€25mg225,00€50mg335,00€100mg484,00€Prasugrel Hydrochloride
CAS :Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
Formule :C20H20FNO3S·HClDegré de pureté :99.39% - 99.79%Couleur et forme :SolidMasse moléculaire :409.9RTICBM-189
CAS :RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formule :C15H14Cl2N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :309.19Ref: TM-T9466
2mg34,00€5mg52,00€1mL*10mM (DMSO)67,00€10mg84,00€25mg161,00€50mg250,00€100mg369,00€200mg522,00€FAUC-365
CAS :FAUC-365 is a D3 dopamine receptor agonist.Formule :C23H25Cl2N3OSDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :462.44Ref: TM-T21667
1mg50,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg160,00€25mg305,00€50mg485,00€100mg700,00€500mg1.459,00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormule :C40H67N7O10Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :805.9Melanotan (MT)-II
CAS :Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formule :C50H69N15O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1024.18Diphenhydramine
CAS :Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Formule :C17H21NODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :255.35Dimethocaine
CAS :Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formule :C16H26N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :278.39AC-90179 HCl
CAS :AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formule :C23H31ClN2O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :402.96Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.Formule :C91H143N27O26S4Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :2157RG7713
CAS :RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formule :C25H28ClN3O2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :437.96Bimatoprost
CAS :Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocularFormule :C25H37NO4Degré de pureté :98% - >99.99%Couleur et forme :Crystalline SolidMasse moléculaire :415.57Ref: TM-T2538
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg127,00€50mg219,00€100mg371,00€200mg547,00€Niaprazine
CAS :Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg90,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formule :C76H117N19O22SDegré de pureté :95.43%Couleur et forme :SolidMasse moléculaire :1680.94Dobutamine tartrate
CAS :Dobutamine tartrate is a cardiotonic.Formule :C22H29NO9Couleur et forme :SolidMasse moléculaire :451.472Enprofylline
CAS :Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Ref: TM-T21389
2mg42,00€1mL*10mM (DMSO)59,00€5mg62,00€10mg88,00€25mg141,00€50mg215,00€100mg318,00€200mg442,00€Fluorogestone acetate
CAS :FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formule :C23H31FO5Degré de pureté :99.47%Couleur et forme :CoaMasse moléculaire :406.49Ref: TM-T21335
2mg39,00€5mg58,00€1mL*10mM (DMSO)74,00€10mg93,00€25mg167,00€50mg245,00€100mg371,00€200mg494,00€Volinanserin
CAS :Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formule :C22H28FNO3Degré de pureté :98.94% - 99.95%Couleur et forme :SolidMasse moléculaire :373.46Ref: TM-T5389
1mg39,00€5mg84,00€1mL*10mM (DMSO)92,00€10mg117,00€25mg220,00€50mg285,00€100mg371,00€200mg530,00€Azaperone
CAS :Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formule :C19H22FN3ODegré de pureté :98.73%Couleur et forme :White Or Off-White CrystallineMasse moléculaire :327.4Elagolix sodium
CAS :Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formule :C32H29F5N3NaO5Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :653.57Ref: TM-T5031
2mg35,00€5mg52,00€1mL*10mM (DMSO)74,00€10mg80,00€25mg144,00€50mg227,00€100mg359,00€200mg532,00€ML 154
CAS :ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.Formule :C29H26BrN2PSDegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :545.47Sigma-LIGAND-1 hydrochloride
CAS :Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formule :C27H34ClNO4Couleur et forme :SolidMasse moléculaire :472.02GLP-1(7-37) acetate(106612-94-6 free base)
CAS :Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Formule :C151H228N40O47Degré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :3355.67Olcegepant
CAS :Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formule :C38H47Br2N9O5Degré de pureté :96.08% - 97.24%Couleur et forme :SolidMasse moléculaire :869.65Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formule :C114H174N34O31Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :2516.81Ref: TM-TP2279L
1mg77,00€2mg97,00€5mg156,00€10mg225,00€25mg375,00€50mg535,00€100mg730,00€200mg938,00€Fluoroclebopride
CAS :Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Formule :C20H23ClFN3O2Degré de pureté :99.68% - 99.91%Couleur et forme :SolidMasse moléculaire :391.87Ref: TM-T3187
1mg34,00€5mg71,00€10mg90,00€1mL*10mM (DMSO)90,00€25mg150,00€50mg222,00€100mg356,00€500mg820,00€Ralinepag
CAS :Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormule :C23H26ClNO5Degré de pureté :99.79% - 99.85%Couleur et forme :SolidMasse moléculaire :431.91Ref: TM-T4635
1mg50,00€2mg71,00€5mg105,00€1mL*10mM (DMSO)117,00€10mg167,00€25mg285,00€50mg401,00€100mg573,00€200mg803,00€ICI 118,551 hydrochloride
CAS :ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3Formule :C17H28ClNO2Degré de pureté :99.296% - 99.76%Couleur et forme :SolidMasse moléculaire :313.86Relugolix
CAS :Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormule :C29H27F2N7O5SDegré de pureté :98.64% - 99.97%Couleur et forme :SolidMasse moléculaire :623.63Ref: TM-T3630
2mg39,00€5mg58,00€1mL*10mM (DMSO)81,00€10mg93,00€25mg167,00€50mg250,00€100mg408,00€200mg585,00€Bupranolol
CAS :Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.Formule :C14H22ClNO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :271.78Ref: TM-T8580
1mg52,00€1mL*10mM (DMSO)96,00€5mg105,00€10mg159,00€25mg309,00€50mg440,00€100mg583,00€200mg785,00€CYM-5541
CAS :CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.Formule :C19H28N2O2Degré de pureté :99.74% - 99.76%Couleur et forme :SolidMasse moléculaire :316.44Ref: TM-T3961
2mg38,00€5mg57,00€1mL*10mM (DMSO)64,00€10mg92,00€25mg160,00€50mg254,00€100mg373,00€500mg873,00€Eprazinone dihydrochloride
CAS :Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.Formule :C24H32N2O2·2HClDegré de pureté :99.25%Couleur et forme :A White Or Almost White CrysMasse moléculaire :453.44Mosapride
CAS :Mosapride (AS-4370) is a selective 5HT4 agonistFormule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89Pridopidine
CAS :Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formule :C15H23NO2SDegré de pureté :95.2% - 99.89%Couleur et forme :SolidMasse moléculaire :281.41Org 27569
CAS :Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormule :C24H28ClN3ODegré de pureté :>99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :409.95Isocorynoxeine
CAS :Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formule :C22H26N2O4Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T6S0654
1mg62,00€2mg89,00€5mg132,00€1mL*10mM (DMSO)146,00€10mg226,00€25mg384,00€50mg557,00€100mg785,00€200mg1.054,00€Cilansetron Hydrochloride
CAS :Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formule :C20H24ClN3O2Couleur et forme :SolidMasse moléculaire :373.88Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.Formule :C169H276N52O55S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :3980.45Quipazine maleate
CAS :Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formule :C17H19N3O4Couleur et forme :SolidMasse moléculaire :329.356Piperoxan hydrochloride
CAS :Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formule :C14H20ClNO2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :269.77Ref: TM-T4526
2mg39,00€1mL*10mM (DMSO)55,00€5mg62,00€10mg92,00€25mg128,00€50mg166,00€100mg200,00€200mg299,00€TRAP-6
CAS :TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).Formule :C34H56N10O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :748.87Ref: TM-T7625
1mg40,00€2mg52,00€5mg88,00€10mg126,00€1mL*10mM (DMSO)126,00€25mg274,00€50mg411,00€100mg550,00€200mg785,00€Carbazochrome
CAS :Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.Formule :C10H12N4O3Degré de pureté :98.36%Couleur et forme :Nacarat Crystalline PowderMasse moléculaire :236.23AM-2232
CAS :AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formule :C24H20N2ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :352.43TCS-OX2-29
CAS :TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formule :C23H31N3O3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :397.51Ref: TM-T4965
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg147,00€50mg203,00€100mg286,00€200mg425,00€CCG-50014
CAS :CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.Formule :C16H13FN2O2SDegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :316.35Xanthotoxol
CAS :Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formule :C11H6O4Degré de pureté :98.44% - 99.97%Couleur et forme :SolidMasse moléculaire :202.16Piperacetazine
CAS :Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Dazoxiben
CAS :Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase
Formule :C12H13ClN2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :268.7Anisotropine Methylbromide
CAS :Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formule :C17H32BrNO2Degré de pureté :99.73%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :362.35NPS ALX Compound 4a
CAS :NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formule :C25H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.55ML221
CAS :ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormule :C17H11N3O6SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :385.35Ref: TM-T4390
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg80,00€25mg137,00€50mg215,00€100mg349,00€200mg512,00€WIN 55,212-2 Mesylate
CAS :WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formule :C28H30N2O6SDegré de pureté :98% - 99.71%Couleur et forme :White To Off-White SolidMasse moléculaire :522.61Dobutamine hydrochloride
CAS :Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.Formule :C18H24ClNO3Degré de pureté :97.15% - 99.94%Couleur et forme :SolidMasse moléculaire :337.84MEN 10207 acetate
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.Formule :C59H72N14O12Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :1169.29Phenylephrine
CAS :Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).Formule :C9H13NO2Degré de pureté :99.5% - 99.89%Couleur et forme :SolidMasse moléculaire :167.21[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS :[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.Formule :C190H286N54O56Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :4223Benorilate
CAS :Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formule :C17H15NO5Degré de pureté :98.39% - 99.85%Couleur et forme :SolidMasse moléculaire :313.35-HT1A modulator 2 hydrochloride
CAS :5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formule :C11H16ClNODegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :213.7E7046
CAS :E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.Formule :C22H18F5N3O4Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :483.4Netupitant
CAS :Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).Formule :C30H32F6N4ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :578.59Lodoxamide
CAS :Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formule :C11H6ClN3O6Degré de pureté :99.13% - 99.96%Couleur et forme :SolidMasse moléculaire :311.63Cerlapirdine hydrochloride
CAS :Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formule :C22H24ClN3O3SCouleur et forme :SolidMasse moléculaire :445.96ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.42% - 98.98%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg58,00€2mg82,00€5mg113,00€1mL*10mM (DMSO)133,00€10mg177,00€25mg333,00€50mg502,00€100mg710,00€500mg1.494,00€Betazole dihydrochloride
CAS :Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.Formule :C5H11Cl2N3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :184.067Ref: TM-T8599
1mg34,00€5mg57,00€1mL*10mM (DMSO)57,00€10mg90,00€25mg167,00€50mg290,00€100mg378,00€200mg538,00€Bevantolol
CAS :Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formule :C20H27NO4Couleur et forme :SolidMasse moléculaire :345.43Dolasetron
CAS :Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formule :C19H20N2O3Degré de pureté :99.84% - 99.86%Couleur et forme :White PowderMasse moléculaire :324.37Decloxizine dihydrochloride
CAS :Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Formule :C21H28N2O2·2ClHDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :413.39Picotamide
CAS :Picotamide has anticoagulant and fibrinolytic properties.Formule :C21H20N4O3Degré de pureté :98.90%Couleur et forme :SolidMasse moléculaire :376.41Ref: TM-T9153
1mg38,00€5mg92,00€1mL*10mM (DMSO)94,00€10mg147,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€5-Hydroxy-1-methylhydantoin
CAS :5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formule :C4H6N2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :130.1SKF 38393 hydrochloride
CAS :SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formule :C16H17NO2·HClDegré de pureté :99.1% - 99.51%Couleur et forme :SolidMasse moléculaire :291.77Betazole
CAS :Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formule :C5H9N3Couleur et forme :SolidMasse moléculaire :111.15SB-200646
CAS :SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormule :C15H14N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :266.3A-582941 dihydrochloride
CAS :A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFormule :C17H22Cl2N4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :353.29Ref: TM-T22016
1mg42,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg533,00€200mg743,00€MK-571 sodium
CAS :MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formule :C26H27ClN2O3S2·NaDegré de pureté :97.86% - 99.58%Couleur et forme :SolidMasse moléculaire :537.07Fenspiride
CAS :Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.Formule :C15H20N2O2Couleur et forme :SolidMasse moléculaire :260.33ESI-09
CAS :ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Formule :C16H15ClN4O2Degré de pureté :97.24% - 99.57%Couleur et forme :SolidMasse moléculaire :330.77CRT0273750
CAS :CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formule :C25H22ClF3N4O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :502.92idalopirdine
CAS :Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formule :C20H19F5N2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :398.37Ref: TM-T7103
1mg88,00€2mg118,00€1mL*10mM (DMSO)187,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€Olanzapine HCl
CAS :Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formule :C17H21ClN4SCouleur et forme :SolidMasse moléculaire :348.89Azepexole
CAS :Azepexole is a selective α2-adrenoceptor agonist that exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor.Formule :C9H15N3OCouleur et forme :SolidMasse moléculaire :181.23Pirenperone
CAS :Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formule :C23H24FN3O2Degré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :393.45ICI 89406
CAS :ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.Formule :C19H22N4O3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :354.4Alprenolol hydrochloride
CAS :Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formule :C15H24ClNO2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :285.81Prazosin
CAS :Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Formule :C19H21N5O4Degré de pureté :99.86%Couleur et forme :White To Tan Powder SolidMasse moléculaire :383.4Neurotensin
CAS :Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formule :C78H121N21O20Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1672.927-Amino-4-(trifluoromethyl)coumarin
CAS :7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formule :C10H6F3NO2Degré de pureté :97.31% - 97.84%Couleur et forme :Yellow PowderMasse moléculaire :229.16
![[Leu31,Pro34]-Neuropeptide Y (porcine)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2206.webp&w=3840&q=75)
