
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.781 produits)
- Apoptose(6.260 produits)
- Cycle cellulaire/point de contrôle(4.789 produits)
- Chromatine/Épigénétique(2.437 produits)
- Signalisation du cytosquelette(1.525 produits)
- Altération de l'ADN/réparation de l'ADN(2.967 produits)
- Endocrinologie/Hormones(3.706 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.000 produits)
- Immunologie et Inflammation(3.869 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.249 produits)
- Transporteur membranaire/Canal ionique(3.029 produits)
- Métabolisme(10.207 produits)
- Microbiologie/Virologie(7.583 produits)
- Neuroscience(10.380 produits)
- Autres inhibiteurs(36.059 produits)
- Oxydation-Réduction(43 produits)
- Signalisation PI3K/Akt/mTOR(1.445 produits)
- Protéases/Protéasome(1.725 produits)
- Cellules souche et Dérivés(825 produits)
- Tyrosine Kinase/Adaptateurs(2.037 produits)
- Ubiquitination(1.716 produits)
Affichez 16 plus de sous-catégories
66687 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Paprotrain
CAS :Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.Formule :C16H11N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :245.28Mifepristone
CAS :Mifepristone (C-1073) is a progesterone-receptor (IC50=0.2 nM) and glucocorticoid-receptor antagonist (IC50=2.6 nM). High-Quality, Low-Cost!Formule :C29H35NO2Degré de pureté :98.9% - ≥95%Couleur et forme :Pale Yellow SolidMasse moléculaire :429.59Linaclotide
CAS :Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.Formule :C59H79N15O21S6Degré de pureté :97.93% - 98.71%Couleur et forme :SolidMasse moléculaire :1526.74Gusacitinib
CAS :<p>Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).</p>Formule :C24H28N8O2Degré de pureté :98.06% - 99.94%Couleur et forme :SolidMasse moléculaire :460.53Ethylenediaminetetraacetic acid trisodium salt
CAS :Ethylenediaminetetraacetic acid trisodium salt (EDTA Trisodium) used to bind metal ions in the chelation therapy.Formule :C10H13N2Na3O8Degré de pureté :99.92% - 99.96%Couleur et forme :White CrystalsMasse moléculaire :358.19AX-15836
CAS :AX-15836 is an inhibitor of ERK5 (IC50 : 8 nM).Formule :C32H40N8O5SDegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :648.78Rimonabant
CAS :Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formule :C22H21Cl3N4ODegré de pureté :98% - 99.91%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :463.79Ascorbyl palmitate
CAS :<p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>Formule :C22H38O7Degré de pureté :99.52%Couleur et forme :White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like OdourMasse moléculaire :414.53Desbenzyl Donepezil Hydrochloride
CAS :Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.Formule :C17H24ClNO3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :325.83LY518674
CAS :LY518674 (LY-674) decreases triglycerides and increases HDL-C and is used for the treatment of atherosclerosis.Formule :C23H27N3O4Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :409.48Trospium chloride
CAS :Trospium chloride treats urinary incontinence without causing liver damage.Formule :C25H30ClNO3Degré de pureté :99.84% - >99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :427.964Amcinonide
CAS :Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.Formule :C28H35FO7Degré de pureté :98.33% - 99.62%Couleur et forme :SolidMasse moléculaire :502.57Kira8
CAS :Kira8 (AMG-18) is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity (IC50: 5.9 nM).Formule :C31H29ClN6O3SDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :601.12Lin28-let-7a antagonist 1
CAS :Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formule :C31H29N5O7Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :583.59Promethazine
CAS :Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .Formule :C17H20N2SDegré de pureté :99.76%Couleur et forme :CrystalsMasse moléculaire :284.42Methyl salicylate
CAS :Methyl salicylate (Gaultheria oil) is an organic ester. For acute joint and muscular pain, methyl salicylate is used as a rubefacient and analgesic.Formule :C8H8O3Degré de pureté :99.97%Couleur et forme :Colourless To Slightly Yellow LiquidMasse moléculaire :152.15Procodazole
CAS :Procodazole (2-Benzimidazolepropionic acid) is a non-specific active immunoprotective agent against viral and bacterial infections.Formule :C10H10N2O2Degré de pureté :98% - 99.35%Couleur et forme :White To Tan Powder Crystals Or Crystalline Powder And/Or ChunksMasse moléculaire :190.2EC23
CAS :EC23 (AGN 190205) is a stable synthetic retinoid analogue. It is also induces neuronal differentiation.Formule :C23H24O2Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :332.44Mepiroxol
CAS :<p>Mepiroxol (Lysateril), an antihyperlipidemic, is also called 3-PYRIDINEMETHANOL N-OXIDE.</p>Formule :C6H7NO2Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :125.13Ciproquazone
CAS :Ciproquazone has analgesic activity and is used to treat spondylitis.Formule :C19H18N2O2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :306.36Tiragolumab
CAS :<p>Tiragolumab, a monoclonal antibody, targets TIGIT and is used with Atezolizumab to treat solid tumors like lung cancer.</p>Degré de pureté :SDS-PAGE:95.3%;SEC-HPLC:98.8%Couleur et forme :LiquidMasse moléculaire :148.3 kDaRoxithromycin
CAS :Roxithromycin (RU-28965) is a semi-synthetic derivative of the macrolide antibiotic erythromycin with antibacterial and anti-malarial activities.Formule :C41H76N2O15Degré de pureté :99.29% - 99.98%Couleur et forme :White Crystalline PowderMasse moléculaire :837.05PF-3450074
CAS :PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Formule :C27H27N3O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :425.52Moguisteine
CAS :Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Formule :C16H21NO5SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :339.415-Aminosalicylic Acid
CAS :5-Aminosalicylic Acid (5-ASA) is a specific PPARγ agonist and also inhibits P21-activated kinase 1 (PAK1) and NF-Κb. High-Quality, Low-Cost!Formule :C7H7NO3Degré de pureté :98.88% - 99.49%Couleur et forme :Purplish-Tan Solid PowderMasse moléculaire :153.14Orotic acid
CAS :<p>Orotic acid (Vitamin B13) is an intermediate product in pyrimidine metabolism.</p>Formule :C5H4N2O4Degré de pureté :99.42%Couleur et forme :Crystals Physical Description White Crystals Or Crystalline Powder (Ntp 1992)Masse moléculaire :156.1Arg-Gly-Asp-Ser acetate
Arg-Gly-Asp-Ser acetate targets integrin, binding pro-caspase-8, -9, -3, but not -1; inhibits receptor function.Formule :C17H31N7O10Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :493.47Spectinomycin dihydrochloride
CAS :Spectinomycin dihydrochloride, an antibiotic from Streptomyces spectabilis, treats gonorrhea and targets gram-negative bacteria.Formule :C14H26Cl2N2O7Degré de pureté :99.67% - >99.99%Couleur et forme :PowderMasse moléculaire :405.271AES-135
CAS :AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.Formule :C33H29F6N3O5SDegré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :693.66Flubendazole
CAS :<p>Flubendazole (Flumoxane) is available OTC in Europe that is an anthelmintic using to treat worm infection in humans.</p>Formule :C16H12FN3O3Degré de pureté :98.47% - 99.30%Couleur et forme :White To Pale Yellow PowderMasse moléculaire :313.28Prochlorperazine Maleate
CAS :Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formule :C28H32ClN3O8SDegré de pureté :99.78%Couleur et forme :Off-White PowderMasse moléculaire :606.09Tubulin inhibitor 6
CAS :Tubulin inhibitor 6 (iHAP1) is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines.Formule :C20H14ClNO2SDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :367.85trans-C75
CAS :trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).Formule :C14H22O4Degré de pureté :98.88% - 99.57%Couleur et forme :White To Off-White SolidMasse moléculaire :254.32Endoxifen (E-isomer)
CAS :<p>Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.</p>Formule :C25H27NO2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :373.49Enoxacin
CAS :Enoxacin (NSC-629661) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.Formule :C15H17FN4O3Degré de pureté :98.68% - 99.89%Couleur et forme :Off-White To Yellow CrystalsMasse moléculaire :320.32Nitazoxanide
CAS :Nitazoxanide (NSC-697855) is a synthetic benzamide antiprotozoal; it disrupts pyruvate electron transfer reactions.Formule :C12H9N3O5SDegré de pureté :99% - 99.93%Couleur et forme :SolidMasse moléculaire :307.28Chondroitin sulfate
CAS :<p>Chondroitin sulfate (Chonsurid) is extracted from shark bone;Store the product in sealed, cool and dry condition</p>Formule :(C14H21NO14S)nDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :30,000-50,0005-Feruloylquinic acid
CAS :5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.Formule :C17H20O9Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :368.34Oxyclozanide
CAS :Oxyclozanide (Oxyclozanid) is a salicylanilide anthelmintic used in grazing animals for fasciola and cestode infestations.Formule :C13H6Cl5NO3Degré de pureté :99.28%Couleur et forme :White To Yellowish PowderMasse moléculaire :401.46Bromhexine hydrochloride
CAS :Bromhexine hydrochloride (Bisolvon) is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus.Formule :C14H21Br2ClN2Degré de pureté :99.98%Couleur et forme :White SolidMasse moléculaire :412.59Vitamin B6
CAS :Vitamin B6 aids metabolism, especially for amino acids, and helps prevent pregnancy-induced and radiation sickness vomiting.Formule :C8H12NO6PDegré de pureté :97.81%Couleur et forme :PowderMasse moléculaire :249.15SLU-PP-332
CAS :SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,Formule :C18H14N2O2Degré de pureté :97.53% - 98.60%Couleur et forme :SoildMasse moléculaire :290.32Ozagrel
CAS :<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formule :C13H12N2O2Degré de pureté :97.90% - 99.38%Couleur et forme :White PowderMasse moléculaire :228.25Capreomycin sulfate
CAS :Capreomycin sulfate (Capastat sulfate) , a cyclic peptide antibiotic, binds to the 70S ribosomal unit leading to inhibition of protein synthesis.Formule :C25H46N14O11SDegré de pureté :98% - 99.54%Couleur et forme :White PowderMasse moléculaire :752.76Dabuzalgron
CAS :Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence.Formule :C12H16ClN3O3SDegré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :317.79Terpin hydrate
CAS :<p>Terpin hydrate is derived from sources such as oil of turpentine, oregano, thyme, and eucalyptus. Terpin is used as an insect repellent and expectorant.</p>Formule :C10H22O3Degré de pureté :99.73%Couleur et forme :Colorless Lustrous Crystal Or White PowderMasse moléculaire :190.29Febantel
CAS :Febantel is an anthelmintic. It is used for veterinary use on dogs, cats, cattle, sheep, goats, pig, and poultry against roundworms and tapeworms.Formule :C20H22N4O6SDegré de pureté :99.85%Couleur et forme :White To Off-White PowderMasse moléculaire :446.48Quinine
CAS :Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria.Formule :C20H24N2O2Degré de pureté :99.93% - 99.97%Couleur et forme :White Solid PowderMasse moléculaire :324.42Telomerase-IN-2
CAS :Telomerase-IN-2 (Telomerase inhibitor 2) shows potent inhibitory activity against telomerase by decreasing the expression of dyskerin (IC50: 0.89 µM).Formule :C34H39N3O9Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :633.69Hydroxyhexamide
CAS :Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.Formule :C15H22N2O4SDegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :326.412'-Deoxyinosine
CAS :2'-Deoxyinosine (Guanine deoxyriboside) inhibits the growth of human colon-carcinoma cell lines and is associated with PNP deficiency.Formule :C10H12N4O4Degré de pureté :99.87% - 99.89%Couleur et forme :SolidMasse moléculaire :252.23AZ7550 hydrochloride
CAS :AZ7550 hydrochloride (AZ7550 hydrochloride ), an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).Formule :C27H32ClN7O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :522.04LY2940094
CAS :LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.Formule :C22H23ClF2N4O2SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :480.96β-Elemene
CAS :β-Elemene (Levo-β-elemene) is a natural product isolated from Curcuma wenyujin, with an antitumor activity and induce cell apoptosis.Formule :C15H24Degré de pureté :99.165% - 99.35%Couleur et forme :SolidMasse moléculaire :204.35NH2-PEG6-Boc
CAS :NH2-PEG6-Boc is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Formule :C19H39NO8Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :409.51MK-8719
CAS :MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .Formule :C9H14F2N2O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.28Citalopram hydrobromide
CAS :Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFormule :C20H22BrFN2ODegré de pureté :99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :405.304L-Cycloserine
CAS :L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formule :C3H6N2O2Degré de pureté :99.75% - 99.99%Couleur et forme :Crystals White PowderMasse moléculaire :102.09Nitrendipine
CAS :<p>Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.</p>Formule :C18H20N2O6Degré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :360.36Lysipressin acetate(50-57-7(fb_acetate))
CAS :<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formule :C48H69N13O14S2Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1116.28L-Ornithine
CAS :L-Ornithine ((S)-2, 5-diaminopentanoic acid) is a non-protein amino acid. in the urea cycle to remove excess nitrogen from the body. High-Quality, Low-Cost!Formule :C5H12N2O2Degré de pureté :99.73% - 99.91%Couleur et forme :SolidMasse moléculaire :132.166-Methoxy-2-naphthoic acid
CAS :6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.Formule :C12H10O3Degré de pureté :99.25%Couleur et forme :White To Off-White Powder Crystals Crystalline Powder And/Or ChunksMasse moléculaire :202.21Procurcumadiol
CAS :Procurcumadiol (5-Hydroxyprocurcumenol) is a natural product found in Curcuma longa and Curcuma phaeocaulis.Formule :C15H22O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :250.33NE 10790
CAS :NE 10790, similar to risedronate, is a mild bone resorption inhibitor but poorly blocks FPP synthase.Formule :C8H10NO6PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :247.14Ethyleneurea
CAS :Ethyleneurea (Imidazolidinone) is used as a formaldehyde scavenger and intermediate.Formule :C3H6N2ODegré de pureté :98.47%Couleur et forme :White To Pale-Yellow White To Pale-Yellow Powder Or CrystalsMasse moléculaire :86.09Imazamox
CAS :Imazamox: a selective, safe, broad-spectrum systemic herbicide inhibiting ALS, stops plant growth, causing death.Formule :C15H19N3O4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :305.33FSEN1
CAS :FSEN1 is a novel and highly effective non-competitive FSP1 inhibitor with an IC50 value of 313 nM.Formule :C22H22BrN5OSDegré de pureté :99.54% - 99.97%Couleur et forme :SolidMasse moléculaire :484.41CXCR7 antagonist-1
CAS :CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.Formule :C21H19FN6ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :390.41Articaine hydrochloride
CAS :Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.Formule :C13H21ClN2O3SDegré de pureté :99.76%Couleur et forme :White Crystalline PowderMasse moléculaire :320.84CYM50308
CAS :CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).Formule :C20H21F2N3O2SDegré de pureté :99.43% - 99.77%Couleur et forme :SolidMasse moléculaire :405.46Zolmitriptan
CAS :<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36BRD4 Inhibitor-10
CAS :<p>BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).</p>Formule :C25H27N5O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :429.51Boc-NH-PEG4-CH2COOH
CAS :Boc-NH-PEG4-CH2COOH is a cleavable ADC linker used as a linker for antibody-drug conjugates (ADC)[1].Formule :C15H29NO8Degré de pureté :99.84% - ≥98%Couleur et forme :SolidMasse moléculaire :351.39p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Captopril
CAS :Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.Formule :C9H15NO3SDegré de pureté :98.34% - 99.85%Couleur et forme :White To Off-White Crystalline Powder SolidMasse moléculaire :217.29DNA2 inhibitor C5
CAS :DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.Formule :C10H6N2O5Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :234.16Adenosine 5'-monophosphate monohydrate
CAS :<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24CHK1-IN-4 hydrochloride
CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).Formule :C18H19BrClN7O2Degré de pureté :99.29%Couleur et forme :SoildMasse moléculaire :480.75Niclosamide olamine
CAS :<p>Niclosamide olamine (Niclosamide Ethanolamine salt) is an Repellent, Insect Attractant and Chemosterilant.</p>Formule :C15H15Cl2N3O5Degré de pureté :99.89%Couleur et forme :Bright Yellow Crystalline Physical Description Yellow Solid Insoluble In Water (Ntp 1992)Masse moléculaire :388.20D-Mannitol
CAS :D-Mannitol (Mannitol) is a diuretic and renal diagnostic aid related to sorbitol.Formule :C6H14O6Degré de pureté :99.66% - 99.68%Couleur et forme :Orthorhombic Needles From Alc (Ntp 1992)Masse moléculaire :182.17LTURM34
CAS :LTURM34 is an inhibitor of DNA-PK with IC50 of 34 nM.Formule :C24H18N2O3SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :414.48Aldose reductase-IN-1
CAS :Aldose reductase-IN-1 (AT-001, Caficrestat) is a highly potent inhibitor of aldose reductase.Cost-effective and quality-assured.Formule :C17H10F3N5O3SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :421.35Desmethyl Celecoxib
CAS :<p>Demethyl celecoxib, a COX-2 inhibitor with 32 nM IC50, is an anti-inflammatory Celecoxib analog with a 75% yield.</p>Formule :C16H12F3N3O2SDegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :367.35Capsaicin
CAS :Capsaicin ((E)-Capsaicin) is a natural product extracted from Capsicum annuum, and is a TRPV1 agonist (EC50=0.29 μM).Formule :C18H27NO3Degré de pureté :98.24% - 99.88%Couleur et forme :Pure Dark Red Solid SolidMasse moléculaire :305.41Tramiprosate
CAS :<p>Tramiprosate (Alzhemed) is an orally active, BBB-crossing, naturally occurring amino acid that binds soluble Aβ and maintains it in a non-protofibrillar form.</p>Formule :C3H9NO3SDegré de pureté :99%Couleur et forme :White Crystals Or Crystalline PowerMasse moléculaire :139.17Clioquinol
CAS :<p>Clioquinol: oral, lipophilic copper-binder; halogenated quinoline with antifungal, antiparasitic, and possible antitumor uses.</p>Formule :C9H5ClINODegré de pureté :97.02%Couleur et forme :Brownish-Yellow Bulky Powder Decomposes At 178-179°C Used As A Topical Anti-InfectiveMasse moléculaire :305.5BAY-2402234
CAS :BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.Formule :C21H18ClF5N4O4Degré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :520.84MRT-83
CAS :MRT-83 is a potent Smo antagonist.Formule :C31H30N4O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :538.59AZD5423
CAS :AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.Formule :C25H21F4N3O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :487.45ISRIB-A15
CAS :<p>ISRIB-A15 (ISR-IN-2) is an potent inhibitor of the integrated stress response with an EC50 of 0.8 nM.</p>Formule :C22H22Cl4N2O4Degré de pureté :98.5%Couleur et forme :SoildMasse moléculaire :520.23Canrenone
CAS :Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.Formule :C22H28O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :340.46Samidorphan HCl
CAS :<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formule :C21H27ClN2O4Degré de pureté :96.79% - 97.85%Couleur et forme :SoildMasse moléculaire :406.9(R)-Terazosin
CAS :R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).Formule :C19H25N5O4Degré de pureté :98.96% - 99.79%Couleur et forme :SolidMasse moléculaire :387.43HLY78
CAS :HLY78, a Wnt/β-catenin activator, enhances Axin-LRP6 binding by targeting Axin's DIX domain.Formule :C17H17NO2Degré de pureté :99.548%Couleur et forme :SolidMasse moléculaire :267.32NBD-556
CAS :NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Formule :C17H24ClN3O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :337.84Maltose monohydrate
CAS :D-(+)-Maltose monohydrate (D-(+)-Maltose monohydrate), a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent inFormule :C12H2201·H2ODegré de pureté :98.41%Couleur et forme :PowderMasse moléculaire :360.31K-604 dihydrochloride
CAS :K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.Formule :C23H32Cl2N6OS3Degré de pureté :99.10% - 99.74%Couleur et forme :SolidMasse moléculaire :575.64Amoxapine
CAS :<p>Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a lesser degree, of serotonin, at adrenergic nerve</p>Formule :C17H16ClN3ODegré de pureté :98.25% - 98.80%Couleur et forme :SolidMasse moléculaire :313.78Loxeen
CAS :Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.Formule :C20H25NO·CH4O3SDegré de pureté :99.46%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.52Mirtazapine
CAS :Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formule :C17H19N3Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :265.35
