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Inhibiteurs

Inhibiteurs

Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.

Sous-catégories appartenant à la catégorie "Inhibiteurs"

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  • DREADD agonist 21

    CAS :
    DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
    Formule :C17H18N4
    Degré de pureté :99.94%
    Couleur et forme :Solid
    Masse moléculaire :278.35
  • FSEN1

    CAS :
    FSEN1 is a novel and highly effective non-competitive FSP1 inhibitor with an IC50 value of 313 nM.
    Formule :C22H22BrN5OS
    Degré de pureté :99.54% - 99.97%
    Couleur et forme :Solid
    Masse moléculaire :484.41
  • Hydroxyhexamide

    CAS :
    Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.
    Formule :C15H22N2O4S
    Degré de pureté :98.91%
    Couleur et forme :Solid
    Masse moléculaire :326.41
  • Propafenone

    CAS :
    Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.
    Formule :C21H27NO3
    Degré de pureté :99.02%
    Couleur et forme :Solid
    Masse moléculaire :341.44
  • Imidazole ketone erastin

    CAS :
    View and buy Imidazole ketone erastin from TargetMol.Imidazole ketone erastin (IKE) is an inducer of ferroptosis. It has inhibition of the system Xc- cystine/glutamate transporter.Cited in 22 publications.
    Formule :C35H35ClN6O5
    Degré de pureté :98.48% - 99.87%
    Couleur et forme :Solid
    Masse moléculaire :655.14
  • Vitamin K

    CAS :
    Vitamin K (Kephton) has blood coagulation action and is important for coagulation factors, matrix-Gla protein, and osteocalcin.
    Degré de pureté :97.00% - 99.79%
    Couleur et forme :Solid
  • Rimonabant

    CAS :
    Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.
    Formule :C22H21Cl3N4O
    Degré de pureté :98% - 99.91%
    Couleur et forme :White Or Almost White Crystalline Powder
    Masse moléculaire :463.79
  • Org-26576

    CAS :
    Org-26576 is a positive allosteric modulator of the AMPA receptor.
    Formule :C11H12N2O2
    Degré de pureté :99.67%
    Couleur et forme :Solid
    Masse moléculaire :204.23
  • Penicillamine

    CAS :
    Penicillamine (Artamine), possessing antineoplastic properties, induces apoptosis by a p53-mediated mechanism and inhibits angiogenesis by chelating with copper
    Formule :C5H11NO2S
    Degré de pureté :99.69% - 99.8%
    Couleur et forme :Fine White Or Practically White Crystalline Powder Solid
    Masse moléculaire :149.21
  • Bozitinib

    CAS :
    <p>Bozitinib (PLB-1001) (PLB-1001) is a highly selective inhibitor of the c-MET kinase with blood-brain barrier permeability.</p>
    Formule :C20H15F3N8
    Degré de pureté :99.16%
    Couleur et forme :Solid
    Masse moléculaire :424.38
  • CYM50308

    CAS :
    CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).
    Formule :C20H21F2N3O2S
    Degré de pureté :99.43% - 99.77%
    Couleur et forme :Solid
    Masse moléculaire :405.46
  • Cephalothin sodium

    CAS :
    Cephalothin sodium, a first-gen cephalosporin antibiotic, disrupts bacterial cell walls by inactivating penicillin-binding proteins, leading to cell lysis.
    Formule :C16H15N2NaO6S2
    Degré de pureté :98.19% - 99.17%
    Couleur et forme :Solid Odour
    Masse moléculaire :418.4
  • Boc-Gln-Ala-Arg-AMC hydrochloride

    CAS :
    Boc-Gln-Ala-Arg-AMC HCl: A fluorescent tracer for trypsin and TMPRSS2 protein hydrolysis.
    Formule :C29H43ClN8O8
    Degré de pureté :99.27%
    Couleur et forme :Solid
    Masse moléculaire :667.15
  • Diosgenin

    CAS :
    Diosgenin (Nitogenin) is a spirostan found in DIOSCOREA and other plants.
    Formule :C27H42O3
    Degré de pureté :99.87%
    Couleur et forme :Flaky Or Needle Crystal
    Masse moléculaire :414.62
  • Promethazine

    CAS :
    Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
    Formule :C17H20N2S
    Degré de pureté :99.76%
    Couleur et forme :Crystals
    Masse moléculaire :284.42
  • Ribostamycin sulfate

    CAS :
    Ribostamycin sulfate (Vistamycin sulfate) , an aminoglycoside antibiotic, contains a neutral sugar moiety and is produced by Streptomyces ribosome.
    Formule :C17H34N4O10·H2SO4
    Degré de pureté :99.57%
    Couleur et forme :Coa
    Masse moléculaire :552.55
  • Procodazole

    CAS :
    Procodazole (2-Benzimidazolepropionic acid) is a non-specific active immunoprotective agent against viral and bacterial infections.
    Formule :C10H10N2O2
    Degré de pureté :98% - 99.35%
    Couleur et forme :White To Tan Powder Crystals Or Crystalline Powder And/Or Chunks
    Masse moléculaire :190.2
  • Doxepin hydrochloride

    CAS :
    Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.
    Formule :C19H22ClNO
    Degré de pureté :99.65% - 99.91%
    Couleur et forme :White To Off-White Powder
    Masse moléculaire :315.84
  • Mepiroxol

    CAS :
    <p>Mepiroxol (Lysateril), an antihyperlipidemic, is also called 3-PYRIDINEMETHANOL N-OXIDE.</p>
    Formule :C6H7NO2
    Degré de pureté :98.67%
    Couleur et forme :Solid
    Masse moléculaire :125.13
  • Ciproquazone

    CAS :
    Ciproquazone has analgesic activity and is used to treat spondylitis.
    Formule :C19H18N2O2
    Degré de pureté :99.66%
    Couleur et forme :Solid
    Masse moléculaire :306.36
  • Tiragolumab

    CAS :
    <p>Tiragolumab, a monoclonal antibody, targets TIGIT and is used with Atezolizumab to treat solid tumors like lung cancer.</p>
    Degré de pureté :SDS-PAGE:95.3%;SEC-HPLC:98.8%
    Couleur et forme :Liquid
    Masse moléculaire :148.3 kDa
  • Fezakinumab

    CAS :
    Fezakinumab: a monoclonal antibody targeting IL-22; used in researching psoriasis, arthritis, dermatitis.
    Degré de pureté :> 95%
    Couleur et forme :Liquid
    Masse moléculaire :144.84 kDa
  • Diosmin

    CAS :
    Diosmin (Venosmine) is a bioflavonoid that strengthens vascular walls.
    Formule :C28H32O15
    Degré de pureté :97.90%
    Couleur et forme :Greyish-Yellow Or Light Yellow Hygroscopic Powder
    Masse moléculaire :608.54
  • Bromhexine hydrochloride

    CAS :
    Bromhexine hydrochloride (Bisolvon) is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus.
    Formule :C14H21Br2ClN2
    Degré de pureté :99.98%
    Couleur et forme :White Solid
    Masse moléculaire :412.59
  • Boc-NH-PEG4-CH2COOH

    CAS :
    Boc-NH-PEG4-CH2COOH is a cleavable ADC linker used as a linker for antibody-drug conjugates (ADC)[1].
    Formule :C15H29NO8
    Degré de pureté :99.84% - ≥98%
    Couleur et forme :Solid
    Masse moléculaire :351.39
  • Ciclopirox olamine

    CAS :
    Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.
    Formule :C14H24N2O3
    Degré de pureté :99.16% - >99.99%
    Couleur et forme :White To Yellow Solid Solid Particulate/Powder
    Masse moléculaire :268.35
  • Penfluridol

    CAS :
    Penfluridol (TLP-607) is a highly potent antipsychotic.
    Formule :C28H27ClF5NO
    Degré de pureté :98.9% - 99.87%
    Couleur et forme :Off-White To White Crystalline Powder
    Masse moléculaire :523.97
  • Granisetron hydrochloride

    CAS :
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Formule :C18H25ClN4O
    Degré de pureté :99.88% - 99.93%
    Couleur et forme :White To Off-White Crystalline Solid
    Masse moléculaire :348.87
  • Lomefloxacin hydrochloride

    CAS :
    Lomefloxacin hydrochloride (Okacyn) is a fluoroquinolone that inhibits DNA replication in bacteria, causing cell death.
    Formule :C17H20ClF2N3O3
    Degré de pureté :99.43% - 99.75%
    Couleur et forme :White Powder
    Masse moléculaire :387.81
  • 4-Hydroxynonenal

    CAS :
    4-Hydroxynonenal (4-HNE) (4-HNE) is an oxidative/nitrosative stress biomarker. It is a substrate and an inhibitor of acetaldehyde dehydrogenase 2 (ALDH2).
    Formule :C9H16O2
    Degré de pureté :95.12% - 98%
    Couleur et forme :Clear Colorless Liquid
    Masse moléculaire :156.22
  • Gliclazide

    CAS :
    Gliclazide (SE1702), an oral antihyperglycemic agent, belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating beta-cells of the
    Formule :C15H21N3O3S
    Degré de pureté :99.58%
    Couleur et forme :Solid
    Masse moléculaire :323.41
  • 2-Methoxy-5-sulfamoylbenzoic acid

    CAS :
    2-Methoxy-5-sulfamoylbenzoic Acid is a metabolite of the antipsychotic drug, Sulpiride.
    Formule :C8H9NO5S
    Degré de pureté :98.94%
    Couleur et forme :Solid
    Masse moléculaire :231.23
  • Amrinone

    CAS :
    <p>Amrinone (Inocor) is a positive inotropic cardiotonic (cardiotonic agent) with vasodilator properties, phosphodiesterase 3 inhibitory activity.</p>
    Formule :C10H9N3O
    Degré de pureté :98.88% - 99.45%
    Couleur et forme :Solid
    Masse moléculaire :187.2
  • Ethylvanillin

    CAS :
    <p>Ethylvanillin (Rhodiarome) is a flavorant used in the production of chocolate. It is about three times as potent as vanillin.</p>
    Formule :C9H10O3
    Degré de pureté :99.44%
    Couleur et forme :White - Off White Solid Powder
    Masse moléculaire :166.17
  • AZD-8529 mesylate

    CAS :
    AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM).
    Formule :C25H28F3N5O6S
    Degré de pureté :99.19%
    Couleur et forme :Solid
    Masse moléculaire :583.58
  • Toluidine Blue

    CAS :
    <p>Toluidine Blue (Blutene chloride), a phenothiazine, is used as a biological stain, a hemostatic, a dye for silk, and a diagnostic aid for gastric neoplasms.</p>
    Formule :C15H16ClN3S
    Degré de pureté :98%
    Couleur et forme :Dark Green Powder
    Masse moléculaire :305.83
  • NSC781406

    CAS :
    <p>NSC781406 is a highly effective inhibitor of PI3K and mTOR (IC50: 2 nM for PI3Kα).</p>
    Formule :C29H27F2N5O5S2
    Degré de pureté :99.58%
    Couleur et forme :Solid
    Masse moléculaire :627.68
  • Leflunomide

    CAS :
    Leflunomide (HWA486) is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.
    Formule :C12H9F3N2O2
    Degré de pureté :99.52% - 99.96%
    Couleur et forme :Off White Crystalline Solid
    Masse moléculaire :270.21
  • Oxyclozanide

    CAS :
    Oxyclozanide (Oxyclozanid) is a salicylanilide anthelmintic used in grazing animals for fasciola and cestode infestations.
    Formule :C13H6Cl5NO3
    Degré de pureté :99.28%
    Couleur et forme :White To Yellowish Powder
    Masse moléculaire :401.46
  • Desmethyl Celecoxib

    CAS :
    <p>Demethyl celecoxib, a COX-2 inhibitor with 32 nM IC50, is an anti-inflammatory Celecoxib analog with a 75% yield.</p>
    Formule :C16H12F3N3O2S
    Degré de pureté :99.42%
    Couleur et forme :Solid
    Masse moléculaire :367.35
  • Vitamin B6

    CAS :
    Vitamin B6 aids metabolism, especially for amino acids, and helps prevent pregnancy-induced and radiation sickness vomiting.
    Formule :C8H12NO6P
    Degré de pureté :97.81%
    Couleur et forme :Powder
    Masse moléculaire :249.15
  • Seganserin

    CAS :
    <p>Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.</p>
    Formule :C29H27F2N3O
    Degré de pureté :99.22%
    Couleur et forme :Solid
    Masse moléculaire :471.54
  • Mefloquine

    CAS :
    <p>Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor.</p>
    Formule :C17H16F6N2O
    Degré de pureté :99.89%
    Couleur et forme :Solid
    Masse moléculaire :378.31
  • 5,6-Dihydro-5-methyluracil

    CAS :
    <p>5,6-Dihydro-5-methyluracil (Dihydrothymine) is an intermediate breakdown product of thymine.</p>
    Formule :C5H8N2O2
    Degré de pureté :98.53%
    Couleur et forme :Solid
    Masse moléculaire :128.13
  • Agaric acid

    CAS :
    <p>Agaricic acid is an adenine nucleotide translocase antagonist.It is obtained from various plants of the fungous tribe, i.e.</p>
    Formule :C22H40O7
    Degré de pureté :98.99% - ≥98%
    Couleur et forme :Solid
    Masse moléculaire :416.55
  • BMS-905

    CAS :
    BMS-905 is a potent dual inhibitors of TLR7 and TLR8 with good selectivity against TLR9 and other family members.
    Formule :C23H29N3
    Degré de pureté :99.94%
    Couleur et forme :Soild
    Masse moléculaire :347.5
  • Gibberellic acid

    CAS :
    Gibberellic acid (GA3) is a hormone found in plants and fungi.
    Formule :C19H22O6
    Degré de pureté :97.01% - 99.79%
    Couleur et forme :Crystals From Ethyl Acetate Physical Description White Powder (Ntp 1992)
    Masse moléculaire :346.37
  • Etebenecid

    CAS :
    Etebenecid (Urelim) reduces uric acid by enhancing kidney excretion and blocks penicillin secretion.
    Formule :C11H15NO4S
    Degré de pureté :99.99%
    Couleur et forme :Solid
    Masse moléculaire :257.31
  • BMS-986158

    CAS :
    BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.
    Formule :C30H33N5O2
    Degré de pureté :98.78%
    Couleur et forme :Solid
    Masse moléculaire :495.62
  • Oxolamine citrate

    CAS :
    Oxolamine citrate (AF-438 citrate) is a cough suppressant that is able to be used as a generic drug in many jurisdictions.
    Formule :C14H19N3O·C6H8O7
    Degré de pureté :99.76%
    Couleur et forme :White Or Off-White Crystalline Powder
    Masse moléculaire :437.44
  • Maritoclax

    CAS :
    Maritoclax (Marinopyrrole A) (Marinopyrrole A) is a novel and specific Mcl-1 inhibitor, shows >8 fold selectivity than BCL-xl (IC50 > 80 μM),with an IC50 value
    Formule :C22H12Cl4N2O4
    Degré de pureté :99.87%
    Couleur et forme :Solid
    Masse moléculaire :510.15
  • Hydroxyurea

    CAS :
    Hydroxyurea (Hydroxycarbamide), an antineoplastic agent, inhibits DNA synthesis through the inhibition of ribonucleoside diphosphate reductase.
    Formule :CH4N2O2
    Degré de pureté :99.85% - 99.92%
    Couleur et forme :Solid
    Masse moléculaire :76.05
  • HaloPROTAC3

    CAS :
    HaloPROTAC3 (HaloPROTAC-3) is a conjugate of ligands for E3 and 16-atom-length linker and a degrader of HaloTag fusion proteins.
    Formule :C41H55ClN4O8S
    Degré de pureté :95.44% - 99.76%
    Couleur et forme :Solid
    Masse moléculaire :799.42
  • Riparin III

    CAS :
    Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.
    Formule :C16H17NO4
    Degré de pureté :95.13%
    Couleur et forme :Solid
    Masse moléculaire :287.31
  • Diaveridine

    CAS :
    Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.
    Formule :C13H16N4O2
    Degré de pureté :99.10%
    Couleur et forme :White Solid
    Masse moléculaire :260.29
  • Dooku1

    CAS :
    Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.
    Formule :C13H9Cl2N3OS
    Degré de pureté :98.87% - 99.74%
    Couleur et forme :Solid
    Masse moléculaire :326.2
  • Etofibrate

    CAS :
    Etofibrate is a combination of clofibrate and niacin, used to treat hyperlipemia.
    Formule :C18H18ClNO5
    Degré de pureté :98.74%
    Couleur et forme :White To Off-White Solid
    Masse moléculaire :363.79
  • 2,5-Dihydroxybenzoic acid

    CAS :
    2,5-Dihydroxybenzoic acid (Gentisic acid) is an active metabolite of salicylic acid degradation with a broad spectrum of biological activity.
    Formule :C7H6O4
    Degré de pureté :99.63%
    Couleur et forme :Solid
    Masse moléculaire :154.12
  • Nitrendipine

    CAS :
    <p>Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.</p>
    Formule :C18H20N2O6
    Degré de pureté :99% - 99.55%
    Couleur et forme :Solid
    Masse moléculaire :360.36
  • AZD5423

    CAS :
    AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.
    Formule :C25H21F4N3O3
    Degré de pureté :98.76%
    Couleur et forme :Solid
    Masse moléculaire :487.45
  • L-Ornithine

    CAS :
    L-Ornithine ((S)-2, 5-diaminopentanoic acid) is a non-protein amino acid. in the urea cycle to remove excess nitrogen from the body. High-Quality, Low-Cost!
    Formule :C5H12N2O2
    Degré de pureté :99.73% - 99.91%
    Couleur et forme :Solid
    Masse moléculaire :132.16
  • Hydralazine hydrochloride

    CAS :
    Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.
    Formule :C8H9ClN4
    Degré de pureté :99.85% - 99.86%
    Couleur et forme :Yellow Crystals White Crystalline Solid
    Masse moléculaire :196.64
  • Deoxycholic acid

    CAS :
    Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.
    Formule :C24H40O4
    Degré de pureté :99.91% - 99.91%
    Couleur et forme :Crystals From Alc Solid
    Masse moléculaire :392.57
  • STAT3-IN-1

    CAS :
    STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumor
    Formule :C28H29NO6
    Degré de pureté :95.89% - 95.89%
    Couleur et forme :Solid
    Masse moléculaire :475.53
  • Ethyleneurea

    CAS :
    Ethyleneurea (Imidazolidinone) is used as a formaldehyde scavenger and intermediate.
    Formule :C3H6N2O
    Degré de pureté :98.47%
    Couleur et forme :White To Pale-Yellow White To Pale-Yellow Powder Or Crystals
    Masse moléculaire :86.09
  • Zolmitriptan

    CAS :
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formule :C16H21N3O2
    Degré de pureté :99.69% - 99.91%
    Couleur et forme :White Or Kind Of White Powder
    Masse moléculaire :287.36
  • MK-8719

    CAS :
    MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .
    Formule :C9H14F2N2O3S
    Degré de pureté :99.67%
    Couleur et forme :Solid
    Masse moléculaire :268.28
  • CXCR7 antagonist-1

    CAS :
    CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.
    Formule :C21H19FN6O
    Degré de pureté :99.93%
    Couleur et forme :Solid
    Masse moléculaire :390.41
  • Oxeladin citrate

    CAS :
    Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.
    Formule :C26H41NO10
    Degré de pureté :97.23%
    Couleur et forme :Solid
    Masse moléculaire :527.6
  • Maltose monohydrate

    CAS :
    D-(+)-Maltose monohydrate (D-(+)-Maltose monohydrate), a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent in
    Formule :C12H2201·H2O
    Degré de pureté :98.41%
    Couleur et forme :Powder
    Masse moléculaire :360.31
  • Pepstatin

    CAS :
    Pepstatin (Pepsin Inhibitor S 735A) is a specific and orally aspartate protease inhibitor that also inhibits HIV protease activity. Cost effective and quality assured.
    Formule :C34H63N5O9
    Degré de pureté :96.74% - 99.94%
    Couleur et forme :Solid
    Masse moléculaire :685.89
  • BRD4 Inhibitor-10

    CAS :
    <p>BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).</p>
    Formule :C25H27N5O2
    Degré de pureté :99.53%
    Couleur et forme :Solid
    Masse moléculaire :429.51
  • Murepavadin acetate(944252-63-5 free base)


    <p>Murepavadin acetate, a strong antibiotic, targets Pseudomonas aeruginosa by hitting its lipopolysaccharide transport.</p>
    Formule :C75H116N22O18
    Degré de pureté :98.057% - 99.72%
    Couleur et forme :Solid
    Masse moléculaire :1613.86
  • Acetohexamide

    CAS :
    Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.
    Formule :C15H20N2O4S
    Degré de pureté :99.19% - 99.85%
    Couleur et forme :Crystals From 90% Aq Ethanol
    Masse moléculaire :324.40
  • Nampt activator-1

    CAS :
    NAMPT Activator-1, EC50: 3.3-3.7 µM, specific niacinamide phosphotransferase stimulant, shields cells, potential neuroprotectant.
    Formule :C16H17N3O3
    Degré de pureté :99.84% - 99.98%
    Couleur et forme :Soild
    Masse moléculaire :299.32
  • SAR405 R enantiomer

    CAS :
    SAR405 R enantiomer is the less active enantiomer of SAR405. SAR405 is an inhibitor of PIK3C3/Vps34.
    Formule :C19H21ClF3N5O2
    Degré de pureté :98.04%
    Couleur et forme :Solid
    Masse moléculaire :443.85
  • Mucic Acid

    CAS :
    Mucic Acid (Tetrahydroxyadipic acid) is an aldaric acid obtained by nitric acid oxidation of galactose or galactose-containing compounds.
    Formule :C6H10O8
    Degré de pureté :99.31%
    Couleur et forme :Crystalline Powder Solid
    Masse moléculaire :210.14
  • CHK1-IN-4 hydrochloride


    CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).
    Formule :C18H19BrClN7O2
    Degré de pureté :99.29%
    Couleur et forme :Soild
    Masse moléculaire :480.75
  • Adrenosterone

    CAS :
    Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
    Formule :C19H24O3
    Degré de pureté :98.13% - 98.29%
    Couleur et forme :Solid
    Masse moléculaire :300.39
  • Divarasib

    CAS :
    <p>Divarasib (GDC-6036), an investigational KRAS G12C inhibitor for solid tumors, has an IC50 of &lt;0.01 μM.</p>
    Formule :C29H32ClF4N7O2
    Degré de pureté :99.237% - 99.83%
    Couleur et forme :Solid
    Masse moléculaire :622.06
  • AR-C155858

    CAS :
    AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).
    Formule :C21H27N5O5S
    Degré de pureté :98.96% - 99.42%
    Couleur et forme :Solid
    Masse moléculaire :461.53
  • Docusate sodium

    CAS :
    Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation.
    Formule :C20H37NaO7S
    Degré de pureté :99.34%
    Couleur et forme :White Wax-Like Solid With Water (Uscg 1999)
    Masse moléculaire :444.56
  • Moguisteine

    CAS :
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Formule :C16H21NO5S
    Degré de pureté :99.98%
    Couleur et forme :Solid
    Masse moléculaire :339.41
  • IK-930

    CAS :
    IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency.
    Formule :C19H19F3N4O2S
    Degré de pureté :99.89%
    Couleur et forme :Soild
    Masse moléculaire :424.44
  • MK-0533

    CAS :
    <p>MK-0533 is a novel PPARγ partial agonist for the prevention of vascular endothelial dysfunction (VED) and VED-related cardiovascular disease.</p>
    Formule :C28H24F3NO6
    Degré de pureté :99.03%
    Couleur et forme :Soild
    Masse moléculaire :527.49
  • Dexchlorpheniramine Maleate

    CAS :
    Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.
    Formule :C20H23ClN2O4
    Degré de pureté :99.58%
    Couleur et forme :White Or Almost White Crystalline Powder
    Masse moléculaire :390.86
  • Diammonium Glycyrrhizinate

    CAS :
    Diammonium Glycyrrhizinate, a licorice-derived anti-inflammatory, metabolizes to glycyrrhetinic acid, affecting corticosteroid metabolism & blood pressure.
    Formule :C42H62O16·2H3N
    Degré de pureté :90% - 99.93%
    Couleur et forme :Solid
    Masse moléculaire :857
  • Pazopanib

    CAS :
    Pazopanib (GW786034) is an inhibitor of protein tyrosine kinases that inhibits VEGFR1/2/3. Pazopanib has antitumor activity. Cost-effective and quality-assured.
    Formule :C21H23N7O2S
    Degré de pureté :98.78% - 99.85%
    Couleur et forme :White Powder
    Masse moléculaire :437.52
  • Azelaic acid

    CAS :
    Azelaic acid is a naturally occurring compound with antibacterial and anti-inflammatory properties, used to treat acne and rosacea.
    Formule :C9H16O4
    Degré de pureté :98.14%
    Couleur et forme :Monoclinic Prismatic Needles Solid
    Masse moléculaire :188.22
  • ISRIB-A15

    CAS :
    <p>ISRIB-A15 (ISR-IN-2) is an potent inhibitor of the integrated stress response with an EC50 of 0.8 nM.</p>
    Formule :C22H22Cl4N2O4
    Degré de pureté :98.5%
    Couleur et forme :Soild
    Masse moléculaire :520.23
  • Orelabrutinib

    CAS :
    <p>Orelabrutinib (ICP-022) is an orally active and irreversible inhibitor of Bruton's tyrosine kinase (BTK).</p>
    Formule :C26H25N3O3
    Degré de pureté :97.77% - 99.54%
    Couleur et forme :Solid
    Masse moléculaire :427.49
  • Citalopram hydrobromide

    CAS :
    Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby
    Formule :C20H22BrFN2O
    Degré de pureté :99.81%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :405.304
  • Clobetasone butyrate

    CAS :
    Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such as
    Formule :C26H32ClFO5
    Degré de pureté :99.87%
    Couleur et forme :Solid
    Masse moléculaire :478.98
  • AZ084

    CAS :
    AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.
    Formule :C26H34N4O2
    Degré de pureté :97.12%
    Couleur et forme :Solid
    Masse moléculaire :434.57
  • NBD-556

    CAS :
    NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.
    Formule :C17H24ClN3O2
    Degré de pureté :99.79%
    Couleur et forme :Solid
    Masse moléculaire :337.84
  • Topotecan hydrochloride

    CAS :
    Topotecan hydrochloride (NSC609699) is an antineoplastic agent used to treat ovarian cancer.
    Formule :C23H24ClN3O5
    Degré de pureté :97.88% - 99.41%
    Couleur et forme :White Crystalline Solid
    Masse moléculaire :457.92
  • Fmoc-NH-PEG8-NHS ester

    CAS :
    Fmoc-NH-PEG8-NHS ester is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].
    Formule :C38H52N2O14
    Degré de pureté :94.69%
    Couleur et forme :Solid
    Masse moléculaire :760.82
  • Quercetin-3'-o-phosphate TEA


    Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.
    Formule :C21H26NO10P
    Degré de pureté :97.04%
    Couleur et forme :Soild
    Masse moléculaire :483.41
  • Loxeen

    CAS :
    Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.
    Formule :C20H25NO·CH4O3S
    Degré de pureté :99.46%
    Couleur et forme :White To Off-White Crystalline Powder
    Masse moléculaire :391.52
  • Capsaicin

    CAS :
    Capsaicin ((E)-Capsaicin) is a natural product extracted from Capsicum annuum, and is a TRPV1 agonist (EC50=0.29 μM).
    Formule :C18H27NO3
    Degré de pureté :98.24% - 99.88%
    Couleur et forme :Pure Dark Red Solid Solid
    Masse moléculaire :305.41
  • Nevanimibe hydrochloride

    CAS :
    Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50
    Formule :C27H40ClN3O
    Degré de pureté :99.75%
    Couleur et forme :Solid
    Masse moléculaire :458.08
  • Simvastatin

    CAS :
    Simvastatin (MK 733) is an HMG-CoA reductase inhibitor (Ki=0.2 nM) with oral activity.
    Formule :C25H38O5
    Degré de pureté :98.54% - 99.13%
    Couleur et forme :Solid
    Masse moléculaire :418.57
  • Ciprofloxacin

    CAS :
    Ciprofloxacin (Bay-09867) mainly targets bacterial DNA Gyrase (IC50=0.22-0.31 µM) and topoisomerase IV (IC50=0.3-1.9 µM). antibiotic. High-Quality, Low-Cost!
    Formule :C17H18FN3O3
    Degré de pureté :98.77% - 99.91%
    Couleur et forme :White Powder
    Masse moléculaire :331.34
  • (S)-AK-242

    CAS :
    (S)-AK-242 ((S)-Resatorvid) is a cytokine inhibitor used in the treatment of heart disease, autoimmune disease, and inflammatory disease.
    Formule :C15H17ClFNO4S
    Degré de pureté :99.86%
    Couleur et forme :Soild
    Masse moléculaire :361.82
  • Lysipressin acetate(50-57-7(fb_acetate))

    CAS :
    <p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction &amp; activates adenylate cyclase, is an antidiuretic in pigs &amp; marsupials.</p>
    Formule :C48H69N13O14S2
    Degré de pureté :98.08%
    Couleur et forme :Solid
    Masse moléculaire :1116.28
  • Heptaminol hydrochloride

    CAS :
    Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.
    Formule :C8H20ClNO
    Degré de pureté :98.61%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :181.71
  • Thermolysin

    CAS :
    Thermolysin is an extracellular metalloendopeptidase from Bacillus thermolysinophilus that selectively catalyzes short peptides.
    Couleur et forme :Solid
  • 5-hydroxytryptophan

    CAS :
    5-hydroxytryptophan (NSC-92523) is the immediate precursor in the biosynthesis of SEROTONIN from tryptophan. It is used as an antiepileptic and antidepressant.
    Formule :C11H12N2O3
    Degré de pureté :99.52%
    Couleur et forme :Minute Rods Or Needles From Ethanol White Solid
    Masse moléculaire :220.22
  • 2-(Acetyloxy)-3-Methylbenzoic Acid

    CAS :
    2-(Acetyloxy)-3-Methylbenzoic Acid is used in qHTS Assay for Inhibitors of hydroxysteroid (17-beta) dehydrogenase 4, HSD17B4 with activity value of 19.95 μM
    Formule :C10H10O4
    Degré de pureté :97.15%
    Couleur et forme :Solid
    Masse moléculaire :194.18
  • Mianserin hydrochloride

    CAS :
    Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.
    Formule :C18H21ClN2
    Degré de pureté :99.63% - 99.82%
    Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
    Masse moléculaire :300.83
  • L-Ascorbic acid

    CAS :
    L-Ascorbic acid (Vitamin C) is a natural product that is a potent reducing agent and antioxidant.
    Formule :C6H8O6
    Degré de pureté :99.85% - 99.89%
    Couleur et forme :Crystals (Usually Plates Sometimes Needles Mon°Clinic System) Taste Almost Odorless (Ntp 1992)
    Masse moléculaire :176.12
  • Brivudine

    CAS :
    <p>Brivudine (BVDU), an antiviral medicine, is used in the therapy of herpes zoster.</p>
    Formule :C11H13BrN2O5
    Degré de pureté :99.51% - 99.85%
    Couleur et forme :Solid
    Masse moléculaire :333.14
  • Ac-FLTD-CMK

    CAS :
    <p>Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.</p>
    Formule :C26H37ClN4O8
    Degré de pureté :95.17%
    Couleur et forme :Solid
    Masse moléculaire :569.05
  • Mizoribine

    CAS :
    Mizoribine (NSC-289637) belongs to the family of 1-Ribosyl-imidazolecarboxamides. Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.
    Formule :C9H13N3O6
    Degré de pureté :98.38% - 99.95%
    Couleur et forme :White To Off-White Crystalline Powder
    Masse moléculaire :259.22
  • Unesbulin

    CAS :
    <p>Unesbulin (PTC596) is an orally active and selective inhibitor of B-cell-specific Moloney murine leukemia virus integration site 1 (BMI-1).</p>
    Formule :C19H13F5N6
    Degré de pureté :98.71%
    Couleur et forme :Solid
    Masse moléculaire :420.34
  • Alarelin Acetate

    CAS :
    Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
    Formule :C56H78N16O12
    Degré de pureté :99.81% - >99.99%
    Couleur et forme :White Powder
    Masse moléculaire :1167.34
  • Desbenzyl Donepezil Hydrochloride

    CAS :
    Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.
    Formule :C17H24ClNO3
    Degré de pureté :99.39%
    Couleur et forme :Solid
    Masse moléculaire :325.83
  • RMC-7977

    CAS :
    RMC-7977 is a inhibitor of the active (GTP-bound) forms of KRAS, HRAS, and NRAS with anticancer activity for the study of solid tumors with KRAS G12C mutations.
    Formule :C47H60N8O6S
    Degré de pureté :97.11% - 99.86%
    Couleur et forme :Solid
    Masse moléculaire :865.09
  • Zileuton

    CAS :
    Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.
    Formule :C11H12N2O2S
    Degré de pureté :98.72% - 99.43%
    Couleur et forme :Crystalline Solid
    Masse moléculaire :236.29
  • 4'-Demethylepipodophyllotoxin

    CAS :
    4'-Demethylepipodophyllotoxin (DMEP) is a potent inhibitor of microtubule assembly.
    Formule :C21H20O8
    Degré de pureté :98.49% - 99.72%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :400.38
  • Pulrodemstat benzenesulfonate

    CAS :
    Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.
    Formule :C30H29F2N5O5S
    Degré de pureté :97.67%
    Couleur et forme :Solid
    Masse moléculaire :609.64
  • Elacestrant

    CAS :
    Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
    Formule :C30H38N2O2
    Degré de pureté :98.31%
    Couleur et forme :Solid
    Masse moléculaire :458.63
  • Eletriptan hydrobromide

    CAS :
    Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.
    Formule :C22H27BrN2O2S
    Degré de pureté :99.69% - 99.85%
    Couleur et forme :Tan Solid
    Masse moléculaire :463.43
  • Deferoxamine Mesylate

    CAS :
    Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.
    Formule :C26H52N6O11S
    Degré de pureté :94.68% - 99.8%
    Couleur et forme :Solid
    Masse moléculaire :656.79
  • Procurcumadiol

    CAS :
    Procurcumadiol (5-Hydroxyprocurcumenol) is a natural product found in Curcuma longa and Curcuma phaeocaulis.
    Formule :C15H22O3
    Degré de pureté :99.88%
    Couleur et forme :Solid
    Masse moléculaire :250.33
  • Ceftazidime

    CAS :
    Ceftazidime (GR20263) is a beta-lactam, cephalosporin antibiotic with bactericidal activity.
    Formule :C22H22N6O7S2
    Degré de pureté :99.1% - 99.85%
    Couleur et forme :Solid
    Masse moléculaire :546.58
  • NS-2028

    CAS :
    NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.
    Formule :C9H5BrN2O3
    Degré de pureté :99.44%
    Couleur et forme :A Crystalline Solid
    Masse moléculaire :269.05
  • Labetalol hydrochloride

    CAS :
    Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
    Formule :C19H25ClN2O3
    Degré de pureté :99.54% - 99.85%
    Couleur et forme :Solid
    Masse moléculaire :364.87
  • Ticagrelor

    CAS :
    Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.
    Formule :C23H28F2N6O4S
    Degré de pureté :98.08% - 99.77%
    Couleur et forme :Solid
    Masse moléculaire :522.57
  • Sulfamethoxazole

    CAS :
    Sulfamethoxazole (STX 608), a sulfonamide antimicrobial, inhibits Cytochrome P450 2C9.
    Formule :C10H11N3O3S
    Degré de pureté :99.71% - 99.92%
    Couleur et forme :Crystals Or White Powder
    Masse moléculaire :253.28
  • Zonisamide

    CAS :
    <p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>
    Formule :C8H8N2O3S
    Degré de pureté :99.05% - 99.9%
    Couleur et forme :Off-White Powder
    Masse moléculaire :212.23
  • Lotilaner

    CAS :
    Lotilaner is a parasiticide.
    Formule :C20H14Cl3F6N3O3S
    Degré de pureté :99.56%
    Couleur et forme :Solid
    Masse moléculaire :596.76
  • Florfenicol

    CAS :
    <p>Florfenicol treats BRD in cattle, effective against Mannheimia, Pasteurella, Haemophilus, Fusobacterium, and Bacteroides.</p>
    Formule :C12H14Cl2FNO4S
    Degré de pureté :98.93%
    Couleur et forme :Solid
    Masse moléculaire :358.21
  • Xylitol

    CAS :
    Xylitol (Ribitol) is a five-carbon sugar alcohol derived from XYLOSE by reduction of the carbonyl group.
    Formule :C5H12O5
    Degré de pureté :99.89% - 99.96%
    Couleur et forme :White Solid Powder
    Masse moléculaire :152.15
  • GPX-100

    CAS :
    GPX-100 (13-deoxydoxorubicin) is an anthracycline antitumour antibiotic that inhibits DNA replication by interacting with topoisomerase II.
    Formule :C27H31NO10
    Degré de pureté :95.91%
    Couleur et forme :Solid
    Masse moléculaire :529.54
  • Diphenylacetonitrile

    CAS :
    Diphenylacetonitrile (Dipan) is used as herbicide and industrial intermediate.
    Formule :C14H11N
    Degré de pureté :98.56%
    Couleur et forme :White Crystal
    Masse moléculaire :193.24
  • DUPA(OtBu)-OH

    CAS :
    DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.
    Formule :C23H40N2O9
    Degré de pureté :97.29%
    Couleur et forme :Solid
    Masse moléculaire :488.57
  • Uracil

    CAS :
    Uracil, a pyrimidine in RNA, pairs with adenine, becomes thymine when methylated, and aids enzyme synthesis.
    Formule :C4H4N2O2
    Degré de pureté :99.51% - 99.97%
    Couleur et forme :Fine Off-White Crystalline Powder
    Masse moléculaire :112.09
  • Dibenzosuberone

    CAS :
    Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline.
    Formule :C15H12O
    Degré de pureté :99.83%
    Couleur et forme :Clear To Yellow Liquid
    Masse moléculaire :208.26
  • Mifepristone

    CAS :
    Mifepristone (C-1073) is a progesterone-receptor (IC50=0.2 nM) and glucocorticoid-receptor antagonist (IC50=2.6 nM). High-Quality, Low-Cost!
    Formule :C29H35NO2
    Degré de pureté :98.9% - ≥95%
    Couleur et forme :Pale Yellow Solid
    Masse moléculaire :429.59
  • GNF351

    CAS :
    GNF351: Full AHR antagonist, inhibits DRE-dependent/independent activity, low toxicity, binds AHR (IC50: 62 nM).
    Formule :C24H25N7
    Degré de pureté :98.43%
    Couleur et forme :Solid
    Masse moléculaire :411.5
  • Frovatriptan succinate hydrate

    CAS :
    Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.
    Formule :C18H25N3O6
    Degré de pureté :99.66%
    Couleur et forme :Solid
    Masse moléculaire :379.41
  • Aliskiren hemifumarate

    CAS :
    <p>Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.</p>
    Formule :C30H53N3O6C4H4O4
    Degré de pureté :96.18% - 99.21%
    Couleur et forme :Solid
    Masse moléculaire :1219.6
  • hGPR91 antagonist 1

    CAS :
    hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
    Formule :C31H23F4N3O
    Degré de pureté :98.89%
    Couleur et forme :Solid
    Masse moléculaire :529.53
  • HPPH

    CAS :
    HPPH (Photochlor) (Photochlor) is a second-generation photosensitizer. It is used as photodynamic therapy (PDT) agent.
    Formule :C39H48N4O4
    Degré de pureté :99.72%
    Couleur et forme :Black Solid Powder
    Masse moléculaire :636.82
  • Carbazochrome sodium sulfonate

    CAS :
    Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
    Formule :C10H11N4NaO5S
    Degré de pureté :99.63%
    Couleur et forme :Orange Yellow Crystalline Powder
    Masse moléculaire :322.03
  • Mycophenolic acid

    CAS :
    Mycophenolic acid (Mycophenolate) is an inosine monophosphate dehydrogenase(IMPDH) inhibitor with anti-proliferative activity.
    Formule :C17H20O6
    Degré de pureté :98.79% - 99.77%
    Couleur et forme :Solid
    Masse moléculaire :320.34
  • ZT 52656A hydrochloride

    CAS :
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Formule :C19H26ClF3N2O
    Degré de pureté :98.78%
    Couleur et forme :Solid
    Masse moléculaire :390.87
  • Arjungenin

    CAS :
    Arjungenin, a triterpene derived from Terminalia arjuna, exhibits insect feeding-deterrent and growth inhibitory properties.
    Formule :C30H48O6
    Degré de pureté :99.76%
    Couleur et forme :Solid
    Masse moléculaire :504.70
  • Pomisartan 2HCl


    <p>Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.</p>
    Formule :C31H32Cl2N4O2
    Degré de pureté :99.88%
    Couleur et forme :Soild
    Masse moléculaire :563.52
  • Fostemsavir Tris

    CAS :
    Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.
    Formule :C29H37N8O11P
    Degré de pureté :99.45%
    Couleur et forme :Solid
    Masse moléculaire :704.62
  • MRT-83

    CAS :
    MRT-83 is a potent Smo antagonist.
    Formule :C31H30N4O5
    Degré de pureté :99.81%
    Couleur et forme :Solid
    Masse moléculaire :538.59
  • Bifonazole

    CAS :
    Bifonazole (Bay H-4502) inhibits fungal enzyme cytochrome p450 51, halting ergosterol synthesis, causing cell membrane damage and fungal cell lysis.
    Formule :C22H18N2
    Degré de pureté :99.29% - 99.87%
    Couleur et forme :Solid
    Masse moléculaire :310.39
  • Amcinonide

    CAS :
    Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
    Formule :C28H35FO7
    Degré de pureté :98.33% - 99.62%
    Couleur et forme :Solid
    Masse moléculaire :502.57
  • Deferiprone

    CAS :
    Deferiprone (Deferidone) is an Iron Chelator. The mechanism of action of deferiprone is as an Iron Chelating Activity.
    Formule :C7H9NO2
    Degré de pureté :99.58% - ≥95%
    Couleur et forme :White Needles
    Masse moléculaire :139.15
  • ATG7-IN-1

    CAS :
    <p>ATG7-IN-1 is a selective ATG7 inhibitor with an IC50 of 62 nM.</p>
    Formule :C17H19FN6O5S2
    Degré de pureté :99.85% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :470.5
  • Sonepcizumab

    CAS :
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.90%
    Couleur et forme :Liquid
    Masse moléculaire :146.43 kDa
  • AB-680

    CAS :
    AB-680 is a highly potent, reversible, and selective inhibitor of CD73 (an ectonucleotidase, Ki: 4.9 pM for hCD73) with anti-tumor activity, displays >10,000-
    Formule :C20H24ClFN4O9P2
    Degré de pureté :97.51% - 97.98%
    Couleur et forme :Solid
    Masse moléculaire :580.82
  • EC23

    CAS :
    <p>EC23 (AGN 190205) is a stable synthetic retinoid analogue. It is also induces neuronal differentiation.</p>
    Formule :C23H24O2
    Degré de pureté :99.64%
    Couleur et forme :Solid
    Masse moléculaire :332.44
  • Spesolimab

    CAS :
    Spesolimab (BI 655130) is an antibody targeting IL-36 receptor, key in immunity, for systemic pustular psoriasis and dermatitis studies.
    Degré de pureté :> 95%
    Couleur et forme :Liquid
    Masse moléculaire :150 kDa
  • Tirbanibulin Mesylate

    CAS :
    Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).
    Formule :C27H33N3O6S
    Degré de pureté :99%
    Couleur et forme :Solid
    Masse moléculaire :527.63
  • Tea polyphenol

    CAS :
    <p>Tea polyphenol, also called green tea extract, are a mixture of chemical compounds, such as flavanoids and tannins, found naturally in tea.</p>
    Formule :C17H19N3O
    Degré de pureté :98%
    Couleur et forme :Yelloish Green Free Flowing Powder
    Masse moléculaire :281.36
  • Larazotide acetate

    CAS :
    Larazotide acetate is a synthetic peptide. It functions as a tight junction regulator and reverses leaky junctions to their normally closed state.
    Formule :C34H59N9O12
    Degré de pureté :95.53% - 99.425%
    Couleur et forme :Solid
    Masse moléculaire :785.89
  • Reserpine

    CAS :
    Reserpine, an alkaloid from Rauwolfia roots, depletes neurotransmitters, used in treating hypertension and psychosis, but side effects restrict use.
    Formule :C33H40N2O9
    Degré de pureté :98.85% - 99.99%
    Couleur et forme :White Or Pale Buff To Slightly Yellowish Powder With A Bitter Taste (Ntp 1992)
    Masse moléculaire :608.68
  • Glucagon (1-29), bovine, human, porcine hydrochloride

    CAS :
    Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.
    Formule :C153H225N43O49S·ClH
    Degré de pureté :95.65% - 98.03%
    Couleur et forme :Solid
    Masse moléculaire :3519.21
  • Roxithromycin

    CAS :
    Roxithromycin (RU-28965) is a semi-synthetic derivative of the macrolide antibiotic erythromycin with antibacterial and anti-malarial activities.
    Formule :C41H76N2O15
    Degré de pureté :99.29% - 99.98%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :837.05
  • Trospium chloride

    CAS :
    Trospium chloride treats urinary incontinence without causing liver damage.
    Formule :C25H30ClNO3
    Degré de pureté :99.84% - >99.99%
    Couleur et forme :White To Off-White Powder
    Masse moléculaire :427.964
  • Aldose reductase-IN-1

    CAS :
    Aldose reductase-IN-1 (AT-001, Caficrestat) is a highly potent inhibitor of aldose reductase.Cost-effective and quality-assured.
    Formule :C17H10F3N5O3S
    Degré de pureté :99.82%
    Couleur et forme :Solid
    Masse moléculaire :421.35
  • KukoaMine B

    CAS :
    Kukoamine B, as a constituent of Lycii Cortex, exhibits anti-acute inflammatory, anti-oxidant, and anti-diabetic characteristics.
    Formule :C28H42N4O6
    Degré de pureté :95% - 99.59%
    Couleur et forme :Solid
    Masse moléculaire :530.66
  • Desvenlafaxine

    CAS :
    Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.
    Formule :C16H25NO2
    Degré de pureté :99.46% - 99.81%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :263.38
  • Kira8

    CAS :
    Kira8 (AMG-18) is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity (IC50: 5.9 nM).
    Formule :C31H29ClN6O3S
    Degré de pureté :98.07%
    Couleur et forme :Solid
    Masse moléculaire :601.12
  • Pidotimod

    CAS :
    <p>Pidotimod is a synthetic dipeptide with immunomodulatory properties.</p>
    Formule :C9H12N2O4S
    Degré de pureté :97.56% - 99.74%
    Couleur et forme :Almost White To White Crystalline Powder
    Masse moléculaire :244.27
  • NIC3

    CAS :
    NIC3 is a selective nucleus accumbens-associated protein-1 (NAC1) inhibitor, with anti-cancer activity.
    Formule :C26H36N2O4
    Degré de pureté :98.06%
    Couleur et forme :Solid
    Masse moléculaire :440.58
  • NE 10790

    CAS :
    NE 10790, similar to risedronate, is a mild bone resorption inhibitor but poorly blocks FPP synthase.
    Formule :C8H10NO6P
    Degré de pureté :>99.99%
    Couleur et forme :Solid
    Masse moléculaire :247.14
  • Silodosin

    CAS :
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Formule :C25H32F3N3O4
    Degré de pureté :99.282% - 99.76%
    Couleur et forme :Colorless To Pink Solid
    Masse moléculaire :495.53
  • GSK3145095

    CAS :
    GSK3145095 is an orally active inhibitor of RIPK1 with IC50 of 5 nM, with potential immunomodulatory activities and antineoplastic.
    Formule :C20H17F2N5O2
    Degré de pureté :99.50%
    Couleur et forme :Solid
    Masse moléculaire :397.38
  • Lin28-let-7a antagonist 1

    CAS :
    Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.
    Formule :C31H29N5O7
    Degré de pureté :99.44%
    Couleur et forme :Solid
    Masse moléculaire :583.59
  • Col003

    CAS :
    Col003 is a selective and potent inhibitor of Hsp47 and competitively binds to the collagen-binding site on Hsp47 (IC50: 1.8 μM).
    Formule :C14H11NO4
    Degré de pureté :99.03% - 99.96%
    Couleur et forme :Solid
    Masse moléculaire :257.24
  • Epalrestat

    CAS :
    Epalrestat (ONO2235), an aldose reductase inhibitor, helps manage diabetic neuropathy symptoms and slows disease progression.
    Formule :C15H13NO3S2
    Degré de pureté :99.2% - 99.54%
    Couleur et forme :Deep Red Acicular Crystal
    Masse moléculaire :319.4
  • Isomaltose

    CAS :
    Isomaltose (D-Isomaltose) is a reducing disaccharide, similar to maltose, but with an α-(1-6)-linkage instead of the α-(1-4)-linkage.
    Formule :C12H22O11
    Degré de pureté :99.98% - ≥95%
    Couleur et forme :Coloured Solution
    Masse moléculaire :342.30
  • Pefloxacin Mesylate Dihydrate

    CAS :
    Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).
    Formule :C17H20FN3O3·CH4O3S·2H2O
    Degré de pureté :99.79%
    Couleur et forme :Solid
    Masse moléculaire :465.49
  • Folic acid

    CAS :
    <p>Folic acid (Vitamin B9) is a vitamin B9 that is essential for the synthesis of DNA/RNA and for the production new cells. Cost-effective and quality-assured.</p>
    Formule :C19H19N7O6
    Degré de pureté :99.19% - 99.27%
    Couleur et forme :Yellowish-Orange Crystals; Extremely Thin Platelets (Elongated @ 2 Ends) From Hot Water 482°F
    Masse moléculaire :441.40
  • Hydrocortisone

    CAS :
    Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.
    Formule :C21H30O5
    Degré de pureté :98.4% - 99.95%
    Couleur et forme :Plates From Alc Or Iso-Propyl Alc Solid
    Masse moléculaire :362.46
  • Tramiprosate

    CAS :
    <p>Tramiprosate (Alzhemed) is an orally active, BBB-crossing, naturally occurring amino acid that binds soluble Aβ and maintains it in a non-protofibrillar form.</p>
    Formule :C3H9NO3S
    Degré de pureté :99%
    Couleur et forme :White Crystals Or Crystalline Power
    Masse moléculaire :139.17
  • Ascorbyl palmitate

    CAS :
    <p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>
    Formule :C22H38O7
    Degré de pureté :99.52%
    Couleur et forme :White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like Odour
    Masse moléculaire :414.53
  • Orphenadrine hydrochloride

    CAS :
    Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
    Formule :C18H23NO·HCl
    Degré de pureté :99.88%
    Couleur et forme :Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)
    Masse moléculaire :305.85
  • PEG300

    CAS :
    PEG300 (Polyethylene glycol 300) is a polymer formed from repeating units of ethylene glycol that is water soluble, low immunogenicity, and biocompatible.
    Formule :C5H15NO2
    Degré de pureté :FW~300 - mw~300
    Couleur et forme :Transparent Liquid Viscous
    Masse moléculaire :10000
  • VUF11207 fumarate

    CAS :
    VUF11207 fumarate is an agonist of CXCR7 and a high-potency ligand of CXCR7 (pKi: 8.1).
    Formule :C31H39FN2O8
    Degré de pureté :97.98%
    Couleur et forme :Solid
    Masse moléculaire :586.65
  • p-Coumaric acid

    CAS :
    p-Coumaric acid (para-Coumaric Acid) is the abundant isomer of cinnamic acid, with antitumor and anti-mutagenic activities.
    Formule :C9H8O3
    Degré de pureté :99.51% - 99.64%
    Couleur et forme :White Crystal
    Masse moléculaire :164.16
  • SLU-PP-332

    CAS :
    SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,
    Formule :C18H14N2O2
    Degré de pureté :97.53% - 98.60%
    Couleur et forme :Soild
    Masse moléculaire :290.32
  • Cyclamic acid

    CAS :
    <p>Cyclamic acid, a synthetic sweetener (NSC-220327), often used as Na/Ca cyclamate. Banned in USA over disputed cancer risk.</p>
    Formule :C6H13NO3S
    Degré de pureté :98.42%
    Couleur et forme :White Crystals
    Masse moléculaire :179.24
  • Ozagrel

    CAS :
    <p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>
    Formule :C13H12N2O2
    Degré de pureté :97.90% - 99.38%
    Couleur et forme :White Powder
    Masse moléculaire :228.25
  • 6-Methoxy-2-naphthoic acid

    CAS :
    6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.
    Formule :C12H10O3
    Degré de pureté :99.25%
    Couleur et forme :White To Off-White Powder Crystals Crystalline Powder And/Or Chunks
    Masse moléculaire :202.21
  • Irbesartan

    CAS :
    Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.
    Formule :C25H28N6O
    Degré de pureté :99.79% - 99.81%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :428.53
  • Homosalate

    CAS :
    Homosalate is an organic UV filter, an ester of salicylic acid and 3,3,5-trimethylcyclohexanol.
    Formule :C16H22O3
    Degré de pureté :99.48%
    Couleur et forme :Physical Description Viscous Or Light Yellow To Slightly Tan Liquid Or Oil (Ntp 1992)
    Masse moléculaire :262.34
  • Terpin hydrate

    CAS :
    <p>Terpin hydrate is derived from sources such as oil of turpentine, oregano, thyme, and eucalyptus. Terpin is used as an insect repellent and expectorant.</p>
    Formule :C10H22O3
    Degré de pureté :99.73%
    Couleur et forme :Colorless Lustrous Crystal Or White Powder
    Masse moléculaire :190.29
  • Broxyquinoline

    CAS :
    Broxyquinoline (5,7-Dibromo-8-hydroxyquinoline) is an antiprotozoal agent, and it can release oxygen free radicals from the water in mucous membranes.
    Formule :C9H5Br2NO
    Degré de pureté :99.71%
    Couleur et forme :Almost White Powder
    Masse moléculaire :302.95
  • Metyrapone

    CAS :
    Metyrapone (NSC-25265) blocks steroid 11β-monooxygenase, used to diagnose Cushing's syndrome.
    Formule :C14H14N2O
    Degré de pureté :99.03% - ≥95%
    Couleur et forme :Crystals From Ether & Pentane Solid
    Masse moléculaire :226.27
  • Amphotericin B

    CAS :
    Amphotericin B (NSC-527017) is a polyene antifungal agent with broad-spectrum activity against many fungal species.
    Formule :C47H73NO17
    Degré de pureté :99.75% - ≥98%
    Couleur et forme :Deep Yellow Prisms Or Needles From N N-Dimethylformamide Physical Description Bright Yellow Powder (Ntp 1992)
    Masse moléculaire :924.08
  • HG106

    CAS :
    <p>HG106 is an anti-inflammatory that may treat RAS gene-related malignant tumor growth.</p>
    Formule :C15H13ClN4O2
    Degré de pureté :99.51% - 99.62%
    Couleur et forme :Soild
    Masse moléculaire :316.74