
Ciclo cellulare/Checkpoint
Gli inibitori del ciclo cellulare/dei checkpoint sono composti che interrompono la normale progressione del ciclo cellulare, in particolare nei principali punti di controllo regolatori. Questi inibitori sono fondamentali per studiare la divisione cellulare, comprendere la proliferazione delle cellule cancerose e sviluppare terapie antitumorali. Mirando a fasi specifiche del ciclo cellulare, questi inibitori possono indurre l'arresto del ciclo cellulare, portando all'apoptosi o alla senescenza nelle cellule che si dividono rapidamente. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità del ciclo cellulare/dei checkpoint per supportare le tue ricerche in biologia del cancro, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Ciclo cellulare/Checkpoint"
- Chinasi aurora(111 prodotti)
- CDK(525 prodotti)
- Arresto del ciclo cellulare(4 prodotti)
- Chk(46 prodotti)
- DYRK(49 prodotti)
- Dynamin(26 prodotti)
- Ferroptosi(225 prodotti)
- HSP(180 prodotti)
- Integrina(256 prodotti)
- Chinesina(87 prodotti)
- LIM chinasi(19 prodotti)
- Microtubulo associato(283 prodotti)
- PKC(111 prodotti)
- PLK(25 prodotti)
- ROCK(66 prodotti)
- Rho(2 prodotti)
- Wee1(14 prodotti)
- c-Myc(75 prodotti)
Mostrare 10 più sottocategorie
Trovati 3749 prodotti di "Ciclo cellulare/Checkpoint"
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SNX2-1-108
CAS:SNX2-1-108 is a selective CDK8 and CDK19 inhibitor.Formula:C21H16N4Purezza:98%Colore e forma:SolidPeso molecolare:324.38LIMK-IN-14
CAS:LIMK-IN-14 is an effective and selective inhibitor of LIMK.Formula:C22H27N7O3Purezza:98%Colore e forma:SolidPeso molecolare:437.49N2-Ethylguanosine
CAS:N2-Ethylguanosine is a Nucleoside Derivative - 2-Modified purine nucleoside.Formula:C12H17N5O5Colore e forma:SolidPeso molecolare:311.29S-(N-PhenethylthiocarbaMoyl)-L-cysteine
CAS:PEITC-Cys: anticarcinogenic, antileukemic, inhibits DNA synthesis in HL60, P450 inhibitor.Formula:C12H16N2O2S2Colore e forma:SolidPeso molecolare:284.4Denopterin
CAS:Denopterin is an antineoplastic agent.Formula:C21H23N7O6Purezza:98%Colore e forma:SolidPeso molecolare:469.458-Deazahomofolic acid
CAS:8-Deazahomofolic acid is a potential thymidylate synthase (TS) inhibitor and other folate related enzymes inhibitor.Formula:C21H22N6O6Purezza:98%Colore e forma:SolidPeso molecolare:454.44Direct Black 38 free acid
CAS:Ferristatin II (Direct Black 38 free acid) is a polysulphonated dye and promotes the degradation of transferrin receptor-1 in vitro and in vivo.Formula:C34H27N9O7S2Purezza:98%Colore e forma:SolidPeso molecolare:737.77ProTAME
CAS:ProTAME inhibits APC/CFzr & APC/CCdc20, enhances cell death with doxorubicin/etoposide in primary/MM cells, especially after TOPIIα upregulation.Formula:C34H38N4O12SPurezza:98%Colore e forma:SolidPeso molecolare:726.751-Acetyl-3-o-toluyl-5-fluorouracil
CAS:<p>1-Acetyl-3-o-toluyl-5-fluorouracil is a potent antineoplastic agent.</p>Formula:C14H11FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:290.25RET-IN-19
CAS:RET-IN-19, a potent RET inhibitor, anticancer: IC50 6.8 nM (RET-wt), 13.51 nM (RET V804M); for NSCLC research.Formula:C28H28N6O4SColore e forma:SolidPeso molecolare:544.62PF-2771
CAS:PF-2771: potent CENP-E inhibitor, IC50 of 16.1 nM, used in cancer treatment.Formula:C29H36ClN5O4Purezza:98%Colore e forma:SolidPeso molecolare:554.08Cyclapolin 9
CAS:Cyclapolin 9: Selective PLK1 inhibitor, IC50 500 nM, ATP-competitive, inactive against other kinases.Formula:C9H4F3N3O4SPurezza:99.64%Colore e forma:SolidPeso molecolare:307.211-Methylcytosine
CAS:<p>1-Methylcytosine (4-amino-1-methylpyrimidin-2(1H)-one) is a methylated form of the cytosine and can be used as the nucleobase of hachimoji DNA paired with</p>Formula:C5H7N3OPurezza:99.88%Colore e forma:SolidPeso molecolare:125.13CRT5
CAS:CRT5, a selective PKD inhibitor, blocks VEGF effects on histone deacetylase 5, CREB, HSP27, and endothelial functions. IC50s: 1-2 nM for PKD1-3.Formula:C28H30N4O2Colore e forma:SolidPeso molecolare:454.56ANI-7
CAS:ANI-7, an AhR pathway activator, selectively impedes MCF-7 breast cancer cell growth (GI50: 0.56 μM).Formula:C13H8Cl2N2Purezza:99.07%Colore e forma:SolidPeso molecolare:263.12Rabacfosadine succinate
CAS:Rabacfosadine succinate is the acyclic nucleoside phosphonate PMEG double prodrug.Formula:C25H41N8O10PPurezza:98%Colore e forma:SolidPeso molecolare:644.623Thiamiprine
CAS:Thiamiprine is an agent with the activity of antineoplastic.Formula:C9H8N8O2SColore e forma:SolidPeso molecolare:292.28GW8510
CAS:GW8510 is a CDK2 and RRM2 inhibitor that affects DNA synthesis and antiproliferation in tumor cells. In mammalian aging models, GW851 prolongs lifespan.Formula:C21H15N5O3S2Purezza:99.32%Colore e forma:SolidPeso molecolare:449.51Meturedepa
CAS:Meturedepa is an antineoplastic agent.Formula:C11H22N3O3PPurezza:98%Colore e forma:SolidPeso molecolare:275.28Digeranyl bisphosphonate
CAS:Digeranyl bisphosphonate (DGBP) is a potent geranylgeranyl pyrophosphate (GGPP) synthase inhibitor that inhibits geranyl pyrophosphorylation of Rac1.DigeranylFormula:C21H34Na4O6P2Purezza:98.5%Colore e forma:SolidPeso molecolare:536.4(R)-Filanesib
CAS:(R)-Filanesib is the R-enantiomer of ARRY-520. (R)-Filanesib is a synthetic kinesin spindle protein (KSP) inhibitor (IC50: 6 nM).Formula:C20H22F2N4O2SColore e forma:SolidPeso molecolare:420.48Clociguanil
CAS:Clociguanil has antimalarial activity.Formula:C12H15Cl2N5OColore e forma:SolidPeso molecolare:316.19IDD388
CAS:IDD388 is a selective and potent aldose reductase (ALR2) inhibitor with antitumor activity that inhibits the ALR1 receptor.Formula:C16H12BrClFNO4Purezza:99.56%Colore e forma:SolidPeso molecolare:416.63CDK4/6-IN-8
CAS:CDK4/6-IN-8 (Compound 7p) is a selective inhibitor of CDK4 (IC50=5.01 nM) and CDK6 (IC50=3.97 nM).Formula:C18H18N6O5Colore e forma:SolidPeso molecolare:398.37IMB-10
CAS:IMB-10 is an alphaMbeta2 integrin modulator, inhibiting leukocyte migration and recruitment in vitro and in vivo.Formula:C19H15NOS2Colore e forma:SolidPeso molecolare:337.46FRα-IN-1
CAS:FRα-IN-1 (Compound 4) is a tumour targeting agent. FRα-IN-1 exhibits selective anti-cancer effects on FRα and FRβ expressing cells.Formula:C21H24N6O6Colore e forma:SolidPeso molecolare:456.45Metioprim
CAS:Metioprim is a competitive bacterial dihydrofolate reductases inhibitor.Formula:C14H18N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:306.38L-Cytidine
CAS:L-Cytidine, pyrimidine nucleoside in RNA, regulates glial glutamate, brain lipids, catecholamines, and mitochondria.Formula:C9H13N3O5Colore e forma:SolidPeso molecolare:243.22USP28-IN-2
CAS:USP28-IN-2 selectively inhibits USP28 (IC50=0.3 μM), degrades c-Myc, kills cancer cells, lowers ankyrin-1/2, and enhances Regorafenib effects.Formula:C23H20Cl2N2O3SColore e forma:SolidPeso molecolare:475.39ROCK-IN-4
CAS:ROCK-IN-4: Inhibits ROCK, sustains NO release, disrupts F-actin, hinders HTM cell respiration, aids glaucoma research.Formula:C20H26ClFN4O7SColore e forma:SolidPeso molecolare:520.96TCS 2314
CAS:TCS 2314 is an orally active and selective very late antigen-4 antagonist (IC50: 4.4 nM).Formula:C28H34N4O6Purezza:98%Colore e forma:SolidPeso molecolare:522.59Trimetrexate glucuronate
CAS:Trimetrexate glucuronate, a folic acid foe, blocks DNA/RNA synthesis by inhibiting purine and thymidylic acid production, may fight tumors.Formula:C25H33N5O10Colore e forma:SolidPeso molecolare:563.564Aloisine A
CAS:Aloisine A, a CDK/GSK-3 inhibitor with IC50: Cdk1/B-150nM, Cdk2/A-120nM, Cdk2/E-400nM, Cdk5/25-200nM, Cdk5/35-160nM, GSK-3α-500nM, GSK-3β-650nM, JNK-3-10μM.Formula:C16H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:267.33CDK4/6-IN-14
CAS:CDK4/6-IN-14: potent CDK4/6 inhibitor, IC50s 10/16 nM, >60-fold selectivity over CDKs 1/2/7/9, selective across 205 kinases.Formula:C24H27ClFN7OColore e forma:SolidPeso molecolare:483.97CI-898 HCl
CAS:CI-898 HCl: lipophilic antifolate, DHFR inhibitor, effective on methotrexate-resistant cancers, synergizes with other drugs in advanced P338 leukemia.Formula:C19H26Cl3N5O3Colore e forma:SolidPeso molecolare:478.8XIE18-6
CAS:XIE18-6 is a novel INK4C inhibitor that blocks p18 activity and promotes ex vivo expansion of human and murine hematopoietic stem cells.Formula:C18H15NO6SPurezza:99.712%Colore e forma:SolidPeso molecolare:373.38BA-1049
CAS:BA-1049 is a selective ROCK2 inhibitor.Formula:C16H21N3O2SColore e forma:SolidPeso molecolare:319.42WF-536 Hydrochloride
CAS:WF-536 Hydrochloride, a novel inhibitor of ROCK, inhibits tumour metastasis in some animal models.Formula:C14H16ClN3OColore e forma:SolidPeso molecolare:277.75LY 207702
CAS:LY 207702, a difluorinated purine nucleoside, exhibits antitumor activity in preclinical models.Formula:C10H12F2N6O3Purezza:98%Colore e forma:SolidPeso molecolare:302.24IRE1α kinase-IN-7
CAS:IRE1α kinase-IN-7 is a chemical compound functioning as an inhibitor of IRE1α kinase, primarily utilized in the research of diseases related to endoplasmicFormula:C28H25F3N6OColore e forma:SolidPeso molecolare:518.53DNA Gyrase-IN-4
CAS:DNA Gyrase-IN-4 inhibits DNA cyclooxygenase (IC50: 0.13 μM) and is effective against Salmonella and E. coli.Formula:C22H15Cl2NO4SColore e forma:SolidPeso molecolare:460.33Codon readthrough inducer 1
CAS:Codon readthrough inducer 1 contains pyrimidine bases and shows good readthrough activity.Formula:C15H11N3O5Purezza:98%Colore e forma:SolidPeso molecolare:313.26Binucleine 2
CAS:Binucleine 2: Drosophila Aurora B kinase inhibitor (Ki=0.36μM), dose-dependent, minimal effect on human/X. laevis kinases, disrupts mitosis in fly cells.Formula:C13H11ClFN5Colore e forma:SolidPeso molecolare:291.71FUBP1-IN-2
CAS:FUBP1-IN-2 hinders FUBP1, affects c-Myc and p21 expression, and depletes polyamines.Formula:C26H26ClN3O4Colore e forma:SolidPeso molecolare:479.96MS0017509
CAS:MS0017509 is a DNA damage repair inhibitor.Formula:C11H10N4Purezza:98%Colore e forma:SolidPeso molecolare:198.22Cylindrospermopsin
CAS:Cylindrospermopsin: a toxic cyanobacterial uracil derivative, disrupts protein/glutathione synthesis in hepatocytes, and is genotoxic.Formula:C15H21N5O7SColore e forma:SolidPeso molecolare:415.42MDK6204
CAS:MDK6204 is a selective inhibitor of CLK1 and CLK2.Formula:C20H20N6OPurezza:98%Colore e forma:SolidPeso molecolare:360.41Zalunfiban
CAS:RUC-4 is an aIIb 3 antagonist. It is also used for prehospital therapy of myocardial infarction.Formula:C16H18N8O2SColore e forma:SolidPeso molecolare:386.43Syntelin
CAS:Syntelin: a selective CENP-E inhibitor with an IC50 of 160 nM; distinct from GSK923295, effective on resistant mutants.Formula:C21H20N6O2S3Colore e forma:SolidPeso molecolare:484.62DNA Gyrase-IN-5
CAS:DNA Gyrase-IN-5 is a potent inhibitor of DNA gyrase (IC50: 0.10 μM) and has an antibacterial effect on both wild-type and drug-resistant strains.Formula:C25H15BrClN5Colore e forma:SolidPeso molecolare:500.78BSJ-01-175
CAS:BSJ-01-175: Selective, potent covalent inhibitor of CDK12/13, targets cancer cells, inhibits phosphorylated RNA polymerase II, downregulates CDK12 genes.Formula:C30H33ClN6O2Colore e forma:SolidPeso molecolare:545.08DENV-IN-7
CAS:DENV-IN-7, a flavone analog, inhibits dengue virus at 70 nM EC50 with low toxicity to normal cells.Formula:C24H22O8Colore e forma:SolidPeso molecolare:438.43P1788
CAS:P1788 is a dihydroorotate dehydrogenase (DHODH) inhibitor that can induce DNA damage [1].Formula:C15H17NO3Colore e forma:SolidPeso molecolare:259.35,10-Dideazaaminopterin
CAS:5,10-Dideazaaminopterin is an antileukemic drug.Formula:C21H22N6O5Purezza:98%Colore e forma:SolidPeso molecolare:438.44Antibacterial agent 89
CAS:Antibacterial agent 89 blocks bacterial transcription and clostridial cytotoxins, inhibiting β'CH-σ interactions.Formula:C21H10Cl2F3NO5SColore e forma:SolidPeso molecolare:516.27HBV-IN-14
CAS:HBV-IN-14: a pyridinopyrimidinone, potent cccDNA inhibitor for HBV study (patent WO2021190502A1, comp 5).Formula:C22H21ClN2O5Colore e forma:SolidPeso molecolare:428.87BMH-23
CAS:BMH-23 is an RNA polymerase I inhibitor that acts by causing nucleolar stress and showing potent anticancer activity across many tumor types.Formula:C15H15N3Purezza:98%Colore e forma:SolidPeso molecolare:237.3Indirubin-3'-monoxime-5-sulphonic acid
CAS:Indirubin-3'-monoxime-5-sulphonic acid is a potent and selective inhibitor of GSK-3β, CDK5, and CDK1 with IC50s of 80nM,5 nM, and 7 nM, respectively.Formula:C16H11N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:357.34MMV688845
CAS:MMV688845: NTM RNA polymerase inhibitor, kills Mycobacterium abscessus, and fights TB.Formula:C24H25N3O3SColore e forma:SolidPeso molecolare:435.54CDK7-IN-13
CAS:CDK7-IN-13 (compound 1) is an effective CDK7 inhibitor for investigating cancers associated with transcriptional dysregulation.Formula:C20H23F3N6OSPurezza:99.22%Colore e forma:SolidPeso molecolare:452.5TP1287
CAS:TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.Formula:C21H21ClNO8PColore e forma:SolidPeso molecolare:481.825,10-Dideazafolic acid
CAS:5,10-Dideazafolic acid is an antileukemic drug.Formula:C21H21N5O6Colore e forma:SolidPeso molecolare:439.422'-Fluorothymidine
CAS:<p>2'-Fluorothymidine is a selective substrate for TK2, related to thymidine and methyluridine.</p>Formula:C10H13FN2O5Purezza:99.67%Colore e forma:SolidPeso molecolare:260.228RK64
CAS:8RK64 is a covalent UCHL1 inhibitor ( IC 50 : 0.32 μM) .Formula:C14H16N8O2SColore e forma:SolidPeso molecolare:360.4Chrysotobibenzyl
CAS:Chrysotobibenzyl from Dendrobium pulchellum stems may trigger cell death in detached cells and hinder lung cancer growth.Formula:C19H24O5Colore e forma:SolidPeso molecolare:332.39Antibacterial agent 124
CAS:Antibacterial agent 124 inhibits Sa ProRS with an IC50 of 0.18 μM.Formula:C16H17ClFN3O2Colore e forma:SolidPeso molecolare:337.78JA2131
CAS:JA2131: Small PARG inhibitor, IC50 0.4μM, induces DNA damage, stalls replication, kills cancer cells.Formula:C13H19N5O2S2Colore e forma:SolidPeso molecolare:341.45Poloxipan
CAS:Poloxipan inhibits PLK1 (IC50: 3.2µM), PLK2 (1.7µM), PLK3 (3µM); minimal effect on Chk2, STAT1, STAT5b, Lck.Formula:C14H10BrN3O3SColore e forma:SolidPeso molecolare:380.22Integrin modulator 1
CAS:Integrin modulator 1 is a selective α4β1 integrin agonist (IC50 9.8 nM) that enhances adhesion with EC50 12.9 nM, aiding integrin-dependent studies.Formula:C13H14N2O4Purezza:99.61%Colore e forma:SolidPeso molecolare:262.26CDK7-IN-20
CDK7-IN-20: potent, irreversible CDK7 inhibitor, IC50 of 4nM, 206x selectivity vs. other CDKs, potential for ADPKD study.Formula:C30H26N6O3Colore e forma:SolidPeso molecolare:518.57Zelpolib
CAS:Zelpolib is a specific inhibitor of DNA polymerase δ (Pol δ), inhibiting DNA replication. antiproliferative.Formula:C22H21N3O5S2Purezza:98.79%Colore e forma:SolidPeso molecolare:471.55c-Myc inhibitor 9
CAS:c-Myc inhibitor 9 (compound 332) with logEC50 ≥6, suppresses tumors in mice, useful for cancer research.Formula:C27H31N5OSColore e forma:SolidPeso molecolare:473.63BMS-587101
CAS:BMS-587101 is a small molecule antagonist of LFA-1, which can reduce inflammation and joint destruction in the mouse model of arthritis.Formula:C26H20Cl2N4O4SColore e forma:SolidPeso molecolare:555.43ML372
CAS:ML372 is a potent and selective SMN Modulator (EC50 = 12 nM, 325% increase inSMN2) with good potency, pharmacokinetics, tolerance, and CNS penetration.Formula:C18H20N2O4SColore e forma:SolidPeso molecolare:360.43RSK-IN-1
CAS:RSK-IN-1 (compound 7d) shows anti-tumor activity. RSK-IN-1 is an inhibitor of RSK that inhibits the phosphorylation of YB-1 [1].Formula:C22H17NO2Colore e forma:SolidPeso molecolare:327.38ERCC1-XPF-IN-1
CAS:ERCC1-XPF-IN-1: potent ERCC1-XPF inhibitor (IC50: 0.49 μM), hampers CPD removal, boosts UV toxicity, hinders DNA repair.Formula:C28H32ClN5O2Colore e forma:SolidPeso molecolare:506.04MtTMPK-IN-6
CAS:MtTMPK-IN-6 inhibits M. tuberculosis thymidylate kinase with IC50 of 29 μM, promising for TB research.Formula:C23H25N3O3Colore e forma:SolidPeso molecolare:391.46DIF-3
CAS:DIF-3 activates GSK-3β, degrades cyclin D1/c-Myc, and inhibits Wnt/β-catenin in DLD-1 cells, curbing HeLa cell proliferation.Formula:C13H17ClO4Purezza:99.57%Colore e forma:SolidPeso molecolare:272.72Eprociclovir
CAS:Eprociclovir (A-5021) is a novel acyclovir analog that is a potent inhibitor of EHV1 replication and may be used for the treatment and/or prevention ofFormula:C11H15N5O3Purezza:98.50% - 99.86%Colore e forma:SolidPeso molecolare:265.27SEL120-34A
CAS:SEL120-34A inhibits CDK8 (IC50: 4.4 nM) & CDK19 (10.4 nM), less on CDK9 (1070 nM), has antitumor properties.Formula:C15H18Br2N4Purezza:99.764% - 99.84%Colore e forma:SolidPeso molecolare:414.14Cytembena
CAS:Cytembena is a cytostatic and a carcinogenic compound that may increase the incidence of fibroadenomas.Cytembena broadly inhibits DNA biosynthesis.Formula:C11H8BrNaO4Purezza:99.7%Colore e forma:White PowderPeso molecolare:307.07CD532
CAS:CD532: Potent Aurora A inhibitor, IC50=45 nM, blocks kinase activity, degrades MYCN, interacts with AURKA, studies cancer.Formula:C26H25F3N8OPurezza:99.99%Colore e forma:SolidPeso molecolare:522.52CDK4/6/1 Inhibitor
CAS:CDK4/6/1 Inhibitor (Crozbaciclib) is a type of CDK4/6 inhibitor (IC50s: 3 and 1 nM).Formula:C28H30F2N6Purezza:97.25% - 99.72%Colore e forma:SolidPeso molecolare:488.57D-I03
CAS:D-I03 is a selective RAD52 inhibitor with a Kd of 25.8 µM.Formula:C23H36N6SPurezza:99.65%Colore e forma:SolidPeso molecolare:428.649-Isopropylolomoucine
CAS:9-Isopropylolomoucine (N9-Isopropylolomoucine), a cell cycle protein-dependent kinase inhibitor, is a thiopurine.Formula:C17H22N6OPurezza:99.82%Colore e forma:SolidPeso molecolare:326.4PCSK9-IN-10
CAS:<p>PCSK9-IN-10: potent oral PCSK9 inhibitor (IC50 = 6.4 µM), upregulates LDLR, curbs atherosclerosis, for hyperlipidemia research.</p>Formula:C18H23N5O4Purezza:99.06%Colore e forma:SoildPeso molecolare:373.41DS18561882
CAS:DS18561882: Potent MTHFD2 inhibitor (IC50=0.0063), inhibits MTHFD1 (IC50=0.57), good oral kinetics.Formula:C28H31F3N4O6SPurezza:98.19% - >99.99%Colore e forma:SolidPeso molecolare:608.63116-9e
CAS:116-9e (MAL2-11B) is an Hsp70 chaperone DNAJA1 inhibitor with antiviral properties, inhibits SV40 replication, and can be used to study cancer drug resistance.Formula:C31H32N2O5Purezza:99.55%Colore e forma:SolidPeso molecolare:512.6Talviraline
CAS:Talviraline (Bay 10-8979) is an RNA-induced DNA polymerase inhibitor.Talviraline is a potent inhibitor of HIV-1-induced cell killing and HIV-1 replication in aFormula:C15H20N2O3S2Purezza:99.88%Colore e forma:SolidPeso molecolare:340.46UMK57
CAS:UMK57 is a CENP-Ei and MCAK enhancer, selectively promoting k-MT attachment error correction to inhibit chromosome missegregation of small molecule compounds,Formula:C17H17N3SPurezza:99.86%Colore e forma:SolidPeso molecolare:295.4Galocitabine
CAS:Galocitabine (Neofrutulon), a thymidylate synthase inhibitor, is used potentially for the treatment of cancer.Formula:C19H22FN3O8Purezza:99.89%Colore e forma:SolidPeso molecolare:439.39hDHODH-IN-7
CAS:hDHODH-IN-7 (DHODH-IN-9) is a nitrogen-containing analog and is a human dihydrorotatory dehydrogenase inhibitor.Formula:C21H23FN4OPurezza:99.87%Colore e forma:SolidPeso molecolare:366.43hSMG-1 inhibitor 11e
CAS:hSMG-1 inhibitor 11e is an effective and selective inhibitor of hSMG-1 (IC50 <0.05 nM) and can be used in studies about cancer treatment.Formula:C26H27N7O3SPurezza:99.89%Colore e forma:SolidPeso molecolare:517.6DENV-IN-5
CAS:Denv-in-5 is an effective and selective dengue virus (DENV) inhibitor with EC50 values of 1.47, 9.23, 7.08, 8.91 μM for denV-I-IV and 0.1512 μM for HIV-1IIIB.Formula:C23H25ClF2N4OSPurezza:99.42%Colore e forma:SolidPeso molecolare:478.99ITX3
CAS:ITX3 is a specific, non-toxic, active and selective TrioN RhoGEF inhibitor with IC50 of 76 μM.Formula:C22H17N3OSPurezza:97.28%Colore e forma:SolidPeso molecolare:371.45AzddMeC
CAS:<p>AzddMeC (Az-Dcme) is an HIV-1 reverse transcriptase and HIV-1 replication inhibitor with antiretroviral activity.AzddMeC is used in the study of HIV-1 infection</p>Formula:C10H14N6O3Purezza:97.14% - 99.62%Colore e forma:SolidPeso molecolare:266.2610-Formylfolic acid
CAS:10-Formylfolic acid is a novel and potent inhibitor of dihydrofolate reductase, which can be used in leukemia research.Formula:C20H19N7O7Purezza:99.97%Colore e forma:SolidPeso molecolare:469.41Poloxin-2
CAS:Poloxin-2 is a potent and selective Plk1 PBD inhibitor with anti-tumour activity that reduces the protein level of Plk1 in HeLa cells.Formula:C16H15NO3Purezza:99.67%Colore e forma:SolidPeso molecolare:269.3GRK6-IN-1
CAS:GRK6-IN-1 (compound 18) is a potent GRK6 blocker, with an IC50 of 120 nM, showing promise for multiple myeloma research.Formula:C22H23ClN6O2Purezza:99.37%Colore e forma:SolidPeso molecolare:438.91Haspin-IN-3
CAS:<p>Haspin-IN-3 is a potent haspin inhibitor with an IC50 of 14 nM.Haspin-IN-3 has anticancer activity.</p>Formula:C16H10N2O3Purezza:98.78%Colore e forma:SolidPeso molecolare:278.26

