
Ciclo cellulare/Checkpoint
Gli inibitori del ciclo cellulare/dei checkpoint sono composti che interrompono la normale progressione del ciclo cellulare, in particolare nei principali punti di controllo regolatori. Questi inibitori sono fondamentali per studiare la divisione cellulare, comprendere la proliferazione delle cellule cancerose e sviluppare terapie antitumorali. Mirando a fasi specifiche del ciclo cellulare, questi inibitori possono indurre l'arresto del ciclo cellulare, portando all'apoptosi o alla senescenza nelle cellule che si dividono rapidamente. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità del ciclo cellulare/dei checkpoint per supportare le tue ricerche in biologia del cancro, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Ciclo cellulare/Checkpoint"
- Chinasi aurora(111 prodotti)
- CDK(522 prodotti)
- Arresto del ciclo cellulare(4 prodotti)
- Chk(46 prodotti)
- DYRK(49 prodotti)
- Dynamin(26 prodotti)
- Ferroptosi(225 prodotti)
- HSP(180 prodotti)
- Integrina(256 prodotti)
- Chinesina(85 prodotti)
- LIM chinasi(19 prodotti)
- Microtubulo associato(285 prodotti)
- PKC(111 prodotti)
- PLK(25 prodotti)
- ROCK(67 prodotti)
- Rho(2 prodotti)
- Wee1(14 prodotti)
- c-Myc(75 prodotti)
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Trovati 3739 prodotti di "Ciclo cellulare/Checkpoint"
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5'-O-Triphenylmethyl-3'-deoxy-3'-chlorothymidine
CAS:5'-O-Triphenylmethyl-3'-deoxy-3'-chlorothymidine is a Nucleoside Derivative - Halo-nucleoside, 2',3'-Dideoxy nucleoside.Formula:C29H27ClN2O4Colore e forma:SolidPeso molecolare:502.992,8-Dimethyladenosine
CAS:Nucleoside Derivatives - 2-Modified purine nucleosides, 8-Modified purine nucleosides;Naturally modified ribo-nucleosidesFormula:C12H17N5O4Colore e forma:SolidPeso molecolare:295.293'-Deoxy-1,2-O-isopropylidene-5-O-(p-toluoyl)-L-arabinofuranose
CAS:3'-Deoxy-1,2-O-isopropylidene-5-O-(p-toluoyl)-L-arabinofuranose is a purine nucleoside analog that exerts antitumor activity by inhibiting DNA synthesis andFormula:C16H20O5Colore e forma:SolidPeso molecolare:292.335-(Azidomethyl)-2'-O-(2-methoxyethyl)uridine
CAS:Nucleoside Derivatives - Azido-nucleosides, 5-Modified pyrimidine nucleosides, 2’-Modified nucleosidesFormula:C13H19N5O7Colore e forma:SolidPeso molecolare:357.326-Methylpurine-b-D-(3-azido-3-deoxy)riboside
CAS:Nucleoside Derivatives - Azido-nucleoside; 6-Modified purine nucleoside; 3’-Modified nucleosideFormula:C11H13N7O3Colore e forma:SolidPeso molecolare:291.272'-Deoxy-N4-ethyl-5-methylcytidine
CAS:2'-Deoxy-N4-ethyl-5-methylcytidine is a Nucleoside Derivative - N-Methylated alkylated nucleoside.Formula:C12H19N3O4Colore e forma:SolidPeso molecolare:269.32'-Amino-2'-deoxy-b-D-arabinouridine
CAS:Nucleoside Derivatives - Amino-nucleoside; Arabino-nucleoside; 2’-Modified nucleosideFormula:C9H13N3O5Colore e forma:SolidPeso molecolare:243.22N6-Benzoyl-7'-OH-morpholino adenosine
CAS:N6-Benzoyl-7'-OH-morpholino adenosine is a Morpholino-nucleoside.Formula:C17H18N6O3Colore e forma:SolidPeso molecolare:354.367-Allyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl) guanine
CAS:Nucleoside Derivatives - Xylo nucleosides, 8-Modified purine nucleosides; N-Methylated alkylated nucleosidesFormula:C13H17N5O6Colore e forma:SolidPeso molecolare:339.33'-Azido-3'-deoxycytidine
CAS:Nucleoside Derivatives –Azido-nucleosides, 3’-Modified nucleosides; Drugs and Inhibitors; Ribonucleotide reductase inhibitorFormula:C9H12N6O4Colore e forma:SolidPeso molecolare:268.235-(2-Hydroxyethyl)uridine
CAS:5-(2-Hydroxyethyl)uridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside.Formula:C11H16N2O7Colore e forma:SolidPeso molecolare:288.251,3-Dimethyl pseudouridine
CAS:1,3-Dimethyl pseudouridine is a Nucleoside Derivative - C-nucleoside; N-Methylated nucleoside.Formula:C11H16N2O6Colore e forma:SolidPeso molecolare:272.255'-O-TBDPS-2,2'-anhydrouridine
CAS:5'-O-TBDPS-2,2'-anhydrouridine is a Nucleoside Derivative - Protected nucleoside with NH2/OH open.Formula:C25H28N2O5SiColore e forma:SolidPeso molecolare:464.59N1-Ethoxymethyl pseudouridine
CAS:N1-Ethoxymethyl pseudouridine is a Nucleoside Derivative - C-nucleoside;N-Alkylated nucleoside.Formula:C11H16N2O7Colore e forma:SolidPeso molecolare:288.253'-O-(2-Methoxyethyl)guanosine
CAS:3'-O-(2-Methoxyethyl)guanosine is a Nucleoside Derivative - 3'-Modified nucleoside.Formula:C13H19N5O6Colore e forma:SolidPeso molecolare:341.325-Hydroxymethyl-2'-O-(2-methoxyethyl)uridine
CAS:Nucleoside Derivatives - 5-Modified pyrimidine nucleosides, 2’-Modified nucleosidesFormula:C13H20N2O8Colore e forma:SolidPeso molecolare:332.31N6-Dimethylaminomethylidene-2'-deoxyisoguanosine
CAS:N6-Dimethylaminomethylidene-2'-deoxyisoguanosine is a Nucleoside Derivative - Iso-guanosine Derivative.Formula:C13H18N6O4Colore e forma:SolidPeso molecolare:322.323,5-O-Ditoluoyl 6-chloropurine-9-β-D-deoxyriboside
CAS:3,5-O-Ditoluoyl 6-chloropurine-9-β-D-deoxyriboside is a Nucleoside Derivative - Other modified nucleoside.Formula:C26H23ClN4O5Colore e forma:SolidPeso molecolare:506.943',5'-Di-O-benzoyl-2'-deoxy-2'-fluoro-β-D-arabinocytidine
CAS:Fluoro-modified nucleoside; arabino-nucleosideFormula:C23H20FN3O6Colore e forma:SolidPeso molecolare:453.425'-O-DMTr-2'-deoxy-5-iodouridine-3'-CED Phosphoramidite
CAS:Nucleoside phosphoramiditeFormula:C39H46IN4O8PColore e forma:SolidPeso molecolare:856.682',3',5'-Tri-O-benzoyl-2'-C-methyl-5-methoxyuridine
CAS:2',3',5'-Tri-O-benzoyl-2'-C-methyl-5-methoxyuridine is a 2'-C-Methyl nucleoside; 5-Modified pyrimidine nucleoside.Formula:C32H28N2O10Colore e forma:SolidPeso molecolare:600.573'-b-Amino-2',3'-dideoxy-5'-O-methoxy trityluridine
CAS:3'-b-Amino-2',3'-dideoxy-5'-O-methoxy trityluridine is a Nucleoside Derivative - Amino-nucleoside, Xylo-nucleoside, 2',3'-Didexoy nucleoside, 3'-ModifiedFormula:C29H29N3O5Colore e forma:SolidPeso molecolare:499.562'-O-(2-Methoxyethyl)-2-aminoadenosine
CAS:Nucleoside Derivatives - 2’-Modified nucleosides, 2-Modified purine nucleosidesFormula:C13H20N6O5Colore e forma:SolidPeso molecolare:340.341-(3'-O-[4,4'-Dimethoxytrityl]-α-L-threofuranosyl)-thymine
CAS:Nucleoside Derivatives - L-Nucleosides; Protected nucleosides w/NH2/OH openFormula:C30H30N2O7Colore e forma:SolidPeso molecolare:530.57N4-Benzoyl-5'-O-DMT-5-methylcytidine
CAS:N4-Benzoyl-5'-O-DMT-5-methylcytidine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open.Formula:C38H37N3O8Colore e forma:SolidPeso molecolare:663.729-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-phenylpurine
CAS:9-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-phenylpurine is a Nucleoside Derivative - Fluoro-modified nucleoside, 6-Modified purine nucleoside, 3'-ModifiedFormula:C16H15FN4O3Colore e forma:SolidPeso molecolare:330.31GDC-0575 dihydrochloride
CAS:GDC-0575 dihydrochloride (ARRY-575 dihydrochloride) is a selective, orally active CHK1 inhibitor (IC50: 1.2 nM) that exhibits antitumour effects.Formula:C16H22BrCl2N5OColore e forma:SolidPeso molecolare:451.194'-α-C-Allyl uridine
CAS:4'-alpha-C-Allyl uridine is a Nucleoside Derivative - 4'-Modified nucleoside.Formula:C12H16N2O6Colore e forma:SolidPeso molecolare:284.27N6-Benzoyl-2'-deoxy-2',2'-diflurocytidine
CAS:N6-Benzoyl-2'-deoxy-2',2'-diflurocytidine is a Nucleoside Derivative - Fluoro-modified nucleoside.Formula:C16H15F2N3O5Colore e forma:SolidPeso molecolare:367.3N1-(1,1,1-Trifluoroethyl)pseudouridine
CAS:Nucleoside Derivatives - C-Nucleosides; N-Alkylated nucleosides; Fluoro-modified nucleosidesFormula:C11H13F3N2O6Colore e forma:SolidPeso molecolare:326.239-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-[5-(propyn-1-yl)pyridin-3-yl]purine
CAS:9-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-[5-(propyn-1-yl)pyridin-3-yl]purine is a Nucleoside Derivative - Fluoro-modified nucleoside, 6-Modified purineFormula:C18H16FN5O3Colore e forma:SolidPeso molecolare:369.355'-O-(4,4'-Dimethoxytrityl)-5-methoxyuridine
CAS:Nucleoside Derivatives - 5-Modified pyrimidine nucleosideFormula:C31H32N2O9Colore e forma:SolidPeso molecolare:576.592,6-Bis(4-morpholinyl)-9-b-D-ribofuranosyl-9H-purine
Nucleoside Derivatives –6-Subtituted nucleosides;2-Substituted nucleosidesColore e forma:Soild2-Chloro-6-methoxypurine -9-β-D-(2'-deoxy-2'-fluoro)-arabinoriboside
CAS:Fluoro-modified nucleoside; Halo-nucleoside; 2/6/8-Modified purine nucleoside; Arabino-nucleoside;Formula:C11H12ClFN4O4Colore e forma:SolidPeso molecolare:318.698-Chloro-2'-β-C-methyl inosine
CAS:Nucleoside Derivatives - 2’-Modified nucleosides; 8-Modified purine nucleosides; Halo-nucleosidesFormula:C11H13ClN4O5Colore e forma:SolidPeso molecolare:316.72'-Deoxy-2'-fluoro-N3-(4-nitrobenzyl)-β-D-arabinouridine
CAS:2'-Deoxy-2'-fluoro-N3-(4-nitrobenzyl)-beta-D-arabinouridine is a Nucleoside Derivative - Fluoro-modified nucleoside,Arabino-nucleoside, 2'-Modified nucleoside.Formula:C16H16FN3O7Colore e forma:SolidPeso molecolare:381.313'-Azido-3'-deoxy-N6,N6-dimethyladenosine
CAS:3'-Azido-3'-deoxy-N6,N6-dimethyladenosine is a Nucleoside Derivative - Azido-nucleoside, 6-Modified purine nucleoside;N-Methylated nucleoside.Formula:C12H16N8O3Colore e forma:SolidPeso molecolare:320.31Ceftriaxone Sodium
CAS:Ceftriaxone Sodium is a sporotaxin antibiotic that inhibits GSK3β and Aurora B. It is used in the study of sepsis and infective endocarditis.Formula:C18H17N8NaO7S3Colore e forma:SolidPeso molecolare:576.5625'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine
CAS:5'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine is a Nucleoside Derivative - 2'-Modified nucleoside; Protected nucleoside with NH2/OH open;Formula:C34H38N2O9Colore e forma:SolidPeso molecolare:618.675'(R)-C-Methyluridine
CAS:5'(R)-C-Methyluridine is a Nucleoside Derivative - 5'-Modified nucleoside.Formula:C10H14N2O6Colore e forma:SolidPeso molecolare:258.233'-O-(2-Methoxyethyl)cytidine
CAS:3'-O-(2-Methoxyethyl)cytidine is a Nucleoside Derivative - 3'-Modified nucleoside.Formula:C12H19N3O6Colore e forma:SolidPeso molecolare:301.35-Azidomethyl-2'-β-methyl-2',3',5'-tri-O-benzoyluridine
CAS:5-Azidomethyl-2'-beta-methyl-2',3',5'-tri-O-benzoyluridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Azido nucleoside; 2'-ModifiedFormula:C32H27N5O9Colore e forma:SolidPeso molecolare:625.596-Amino-4-methoxy-1-(2-deoxy-a-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
Nucleoside Derivatives - 7-Deaza-8-aza purine nucleosides; alpha-Nucleosides; Scaffolds and TemplatesColore e forma:SoildN6-Benzoyl-2'-O-(2-methoxyethyl)adenosine
CAS:N6-Benzoyl-2'-O-(2-methoxyethyl)adenosine is a Nucleoside Derivative - 2'-Modified nucleoside.Formula:C20H23N5O6Colore e forma:SolidPeso molecolare:429.435-Benzylaminocarbonyl-3'-O-acetyl-2'-O-methyluridine
CAS:5-Benzylaminocarbonyl-3'-O-acetyl-2'-O-methyluridine is a 5-modified pyrimidine nucleoside; 2'-O-Methyl nucleoside.Formula:C20H23N3O8Colore e forma:SolidPeso molecolare:433.417-(N-Acetylaminomethyl)-7-deazaguanosine
Nucleoside Derivatives –7-Deaza-purine nucleosides; Amino nucleosidesColore e forma:Soild3'-O-Propargyladenosine
CAS:3'-O-Propargyladenosine is a Nucleoside Derivative - 3'-Modified nucleoside.Formula:C13H15N5O4Colore e forma:SolidPeso molecolare:305.292'-Deoxy-2'-fluoro-5-trifluoromethyl-arabinouridine
CAS:2'-Deoxy-2'-fluoro-5-trifluoromethyl-arabinouridine is a Nucleoside Derivative - Fluoro-modified nucleoside, Arabino-nucleoside, 5-Modified pyrimidineFormula:C10H10F4N2O5Colore e forma:SolidPeso molecolare:314.192'-Deoxy-2'-fluoroinosine
CAS:2'-Deoxy-2'-fluoroinosine is a Nucleoside Derivative - 2'-Modified nucleoside, Fluoro-modified nucleoside.Formula:C10H11FN4O4Colore e forma:SolidPeso molecolare:270.226-Amino-2,5-dihydro-2-(b-D-ribofuranosyl)-4H-pyrazolo[3,4-d]pyrimidin-4-one
CAS:6-Amino-2,5-dihydro-2-(b-D-ribofuranosyl)-4H-pyrazolo[3,4-d]pyrimidin-4-one is a Nucleoside Derivative - 7-deaza-8-aza purine nucleoside.Formula:C10H13N5O5Colore e forma:SolidPeso molecolare:283.248-Allylthioadenosine
CAS:8-Allylthioadenosine is a Nucleoside Derivative - 8-Modified purine nucleoside; Thio-nucleoside.Formula:C13H17N5O4SColore e forma:SolidPeso molecolare:339.372,3'-Anhydrothymidine
CAS:2,3'-Anhydrothymidine is a Nucleoside Derivative - Anhydro-nucleoside.Formula:C10H12N2O4Colore e forma:SolidPeso molecolare:224.215-Methoxymethyluridine
CAS:5-Methoxymethyluridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside.Formula:C11H16N2O7Colore e forma:SolidPeso molecolare:288.252'-O-Me-C(Bz) Phosphoramidite
CAS:2’-O-Me-C(Bz) Phosphoramidite is a modified phosphoramidite monomer, which can be used for the oligonucleotide synthesis.Formula:C47H54N5O9PColore e forma:SolidPeso molecolare:863.93DTP3
CAS:DTP3 is a selective MKK7/GADD45β inhibitor, which inhibits cancer-selective NF-κB survival pathway.Formula:C26H35N7O5Colore e forma:SolidPeso molecolare:525.63'-Deoxy-3'-fluoro-xylo-5-methoxyuridine
3'-Deoxy-3'-fluoro-xylo-5-methoxyuridine is a Nucleoside Derivative - xylo-nucleoside;Fluoro-modified nucleoside; 5-Modified pyrimidine nucleoside.Colore e forma:Soild5'-DMTr-T-Methyl phosphonamidite
CAS:5'-DMTr-T-Methyl phosphonamidite is a Nucleoside Derivative - phosphonamidite.Formula:C38H48N3O7PColore e forma:SolidPeso molecolare:689.781,2-O-Isopropylidene-3-O-methyl-D-ribofuranose
CAS:1,2-O-Isopropylidene-3-O-methyl-D-ribofuranose is a Carbohydrate.Formula:C9H16O5Colore e forma:SolidPeso molecolare:204.223'-Deoxy-3'-α-C-methylcytidine
CAS:3'-Deoxy-3'-alpha-C-methylcytidine is a Nucleoside; Used for nucleoside and nucleic acid modifications.Formula:C10H15N3O4Colore e forma:SolidPeso molecolare:241.248-Benzyloxyadenosine
CAS:8-Benzyloxyadenosine is a Nucleoside Derivative - 8-Modified purine nucleoside.Formula:C17H19N5O5Colore e forma:SolidPeso molecolare:373.36N6-Benzoylarabinoadenosine
CAS:Nucleoside Derivatives - Arabino-nucleosidesFormula:C17H17N5O5Colore e forma:SolidPeso molecolare:371.354'-C-Methyl-5-methoxyuridine
CAS:Nucleoside Derivatives - 4’-Modified nucleosides; 5-Modified pyrimidine nucleosidesFormula:C11H16N2O7Colore e forma:SolidPeso molecolare:288.252-Amino-6-chloropurine-3',5'-di-O-acetyl-2'-deoxyriboside
CAS:Nucleoside - 2’-deoxy nucleoside; halo nucleosideFormula:C14H16ClN5O5Colore e forma:SolidPeso molecolare:369.765-Bromoarabinouridine
CAS:5-Bromoarabinouridine is a Halo-nucleoside; Arabino-nucleoside.Formula:C9H11BrN2O6Colore e forma:SolidPeso molecolare:323.12',3',5'-Tri-O-acetyl-2-thiouridine
CAS:Nucleosides Derivatives –Thio-nucleosidesFormula:C15H18N2O8SColore e forma:SolidPeso molecolare:386.383'-O-(t-Butyldimethylsilyl)-2'-deoxy-2'-fluorouridine
CAS:Nucleoside Derivatives - Fluoro-Modified nucleosides, 2’-Modified nucleosides; Protected nucleosides with NH2/OH groupFormula:C15H25FN2O5SiColore e forma:SolidPeso molecolare:360.45N2-iso-Butyroyl-2'-O-propargylguanosine
CAS:<p>N2-iso-Butyroyl-2'-O-propargylguanosine is a Nucleoside Derivative - 2'-Modified nucleoside.</p>Formula:C17H21N5O6Colore e forma:SolidPeso molecolare:391.38N1-Methyl-2'-deoxyadenosine
CAS:Nucleoside Derivatives - N-Methylated/ alkylated nucleosides; DNA adductFormula:C11H15N5O3Colore e forma:SolidPeso molecolare:265.27N2-[(N,N-Dimethyl)amino]methylene-N1-methyl-2'-O-Methyl guanosine
CAS:Nucleoside Derivatives - 2’-Modified nucleosides; N-Alkylated nucleosidesFormula:C15H22N6O5Colore e forma:SolidPeso molecolare:366.378-Azido-2'-deoxyadenosine
CAS:Nucleoside Derivatives - 8-Modified purine nucleosides; Azido nucleosidesFormula:C10H12N8O3Colore e forma:SolidPeso molecolare:292.254'-Methyl-5-methyluridine
CAS:Nucleoside Derivatives - 4’-Modified nucleosides, 5-Modified pyrimidine nucleosidesFormula:C11H16N2O6Colore e forma:SolidPeso molecolare:272.252'-Deoxy-2'-fluoro-N3-(4-hydroxybenzyl)uridine
2'-Deoxy-2'-fluoro-N3-(4-hydroxybenzyl)uridine is a Nucleoside Derivative - Fluoro-modified nucleoside, 2'-Modified nucleoside.Colore e forma:Soild4,6-Diamino-1-(b-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
CAS:Nucleoside Derivatives - 8-Aza-7-deaza-purine nucleoside; 2-Modified purine nucleosideFormula:C10H14N6O4Colore e forma:SolidPeso molecolare:282.262'-O-Phthalimidopropyl uridine
CAS:2’-O-Phthalimidopropyl uridine is a useful organic compound for research related to life sciences.Formula:C20H21N3O8Colore e forma:SolidPeso molecolare:431.44'-Cyanouridine
CAS:4'-Cyanouridine is a Nucleoside Derivative - 4'-Modified nucleoside.Formula:C10H11N3O6Colore e forma:SolidPeso molecolare:269.21N6-Ethyl-2'-O-methyladenosine
CAS:N6-Ethyl-2'-O-methyladenosine is a Nucleoside Derivative - 6-Modified purine nucleoside, 2'-Modified nucleoside.Formula:C13H19N5O4Colore e forma:SolidPeso molecolare:309.325-Benzylaminocarbony-3'-O-Ac-2'-O-Me-5'-O-DMT-uridine
CAS:5-Benzylaminocarbony-3'-O-Ac-2'-O-Me-5'-O-DMT-uridine is a 5 modified pyrimidine nucleoside; 2'-O-Methyl nucleoside.Formula:C41H41N3O10Colore e forma:SolidPeso molecolare:735.782',3'-Dideoxy-2',3'-didehydro-uridine
CAS:Nucleoside Derivatives - Didehydro-nucleosideFormula:C9H10N2O4Colore e forma:SolidPeso molecolare:210.193-epi-Azido-3-deoxythymidine
CAS:3’-N-modified nucleoside; Azido-nucleosideFormula:C10H13N5O4Colore e forma:SolidPeso molecolare:267.241-(b-D-Xylofuranosyl)-5-methyluracil
CAS:1-(b-D-Xylofuranosyl)-5-methyluracil is a Nucleoside Derivative - Xylo-nucleoside.Formula:C10H14N2O6Colore e forma:SolidPeso molecolare:258.235-Methoxy-4'-thiouridine
Nucleoside Derivatives - Thio-nucleosides; 5-Modified pyrimidine nucleosidesColore e forma:SoildN2-iso-Butyroyl-5'-O-DMT-3'-O-(methoxyethyl)guanosine
CAS:N2-iso-Butyroyl-5'-O-DMT-3'-O-(methoxyethyl)guanosine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open.Formula:C38H43N5O9Colore e forma:SolidPeso molecolare:713.78N6-Benzoyl-2'-O-methyladdenosine
CAS:N6-Benzoyl-2'-O-methyladdenosine is a 2'-O-Methyl nucleoside.Formula:C18H19N5O5Colore e forma:SolidPeso molecolare:385.373'-Deoxy-3'-fluorouridine
CAS:3'-Deoxy-3'-fluorouridine is a nucleoside, fluoro-modified nucleoside.Formula:C9H11FN2O5Colore e forma:SolidPeso molecolare:246.193'-β-Azido-2',3'-dideoxy-5'-O-(4-methoxytrityl)uridine
CAS:3'-beta-Azido-2',3'-dideoxy-5'-O-(4-methoxytrityl)uridine is a Nucleoside Derivative - 2',3'-Dideoxy nucleoside, 3'-Modified nucleoside, Azido-nucleoside, Xylo-Formula:C29H27N5O5Colore e forma:SolidPeso molecolare:525.562′-Deoxy-6-thioinosine
CAS:2'-Deoxy-6-thioinosine is a Nucleoside Derivative - Thio-nucleoside.Formula:C10H12N4O3SColore e forma:SolidPeso molecolare:268.29N2-(Isopropylphenoxyacetyl)-2'-O-propargylguanosine
CAS:Nucleoside Derivatives - 2’-Modifed NucleosidesFormula:C24H27N5O7Colore e forma:SolidPeso molecolare:497.58-Hydroxy-3'-deoxyguanosine
Nucleoside Derivatives - 3’-Deoxy-nucleosides; 8-Modified purine nucleosidesColore e forma:Soild2',3'-Dideoxy-3'-fluoroadenosine
CAS:Nucleoside Derivatives - Fluoro-modified nucleosides; 2’,3’-Dideoxy nucleosides; Drugs and Inhbitors; Antiviral agentFormula:C10H12FN5O2Colore e forma:SolidPeso molecolare:253.235'-Azido-5'-deoxy-2'-O-methyluridine
CAS:Nucleoside Derivatives - Azido-nucleosides, 5’-Modified nucleosides, 2’-Modified nucleosidesFormula:C10H13N5O5Colore e forma:SolidPeso molecolare:283.242-Chloro-N6-cyclopentyl-2'-deoxy-2'-fluoro-β-D-arabinoadenosine
CAS:Nucleoside Derivatives - 6-Modified purine nucleosides; Halo-nucleosides; Fluoro-modified nucleosidesFormula:C15H19ClFN5O3Colore e forma:SolidPeso molecolare:371.792-Amino-2'-O-(2-methoxy-2-oxoethyl)adenosine
CAS:Nucleosides Derivatives - 2’-Modified nucleosides; 2-Modified purine nucleosidesFormula:C13H18N6O6Colore e forma:SolidPeso molecolare:354.323,5-Bis-O-(4-methylbenzoyl)-2-C-methyl-D-ribonic acid gama-lactone
CAS:3,5-Bis-O-(4-methylbenzoyl)-2-C-methyl-D-ribonic acid gama-lactone is a Carbohydrate Derivative.Formula:C22H22O7Colore e forma:SolidPeso molecolare:398.412-Chloro-2'-C-methyladenosine
CAS:2-Chloro-2'-C-methyladenosine is a 2'-C-Methyl nucleoside; Halo-nucleoside.Formula:C11H14ClN5O4Colore e forma:SolidPeso molecolare:315.712'-Deoxy-2'-fluoro-arabino-tubercidine
CAS:Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, Arabino-nucleosideFormula:C11H13FN4O3Colore e forma:SolidPeso molecolare:268.24N1-Allylpseudouridine
CAS:<p>N1-Allylpseudouridine is a Nucleoside Derivative - C-nucleoside; N-Alkylated nucleoside.</p>Formula:C12H16N2O6Colore e forma:SolidPeso molecolare:284.278-Methyladenosine
CAS:Nucleoside Derivatives - 8-Modified purine nucleosides; Naturally modified ribo-nucleosidesFormula:C11H15N5O4Colore e forma:SolidPeso molecolare:281.27N1-Cyanomethyl pseudouridine
N1-Cyanomethyl pseudouridine is a Nucleoside Derivative - C-nucleoside;N-Alkylated nucleoside.Colore e forma:Soild3'-β-C-Ethynyl inosine
3'-beta-C-Ethynyl inosine is a Nucleoside Derivative - 3'-Modified nucleoside.Colore e forma:SoildDMTr-LNA-U-3-CED-phosphoramidite
CAS:Nucleoside Phosphoramidites; Nucleoside Derivatives - LNA-related nucleosidesFormula:C40H47N4O9PColore e forma:SolidPeso molecolare:758.83'-Deoxy-3'-fluoro-xyloadenosine
CAS:3'-Deoxy-3'-fluoro-xyloadenosine is a Nucleoside Derivative - Xylo-nucleoside, Fluoro-modified nucleoside, 3'-Modified nucleoside.Formula:C10H12FN5O3Colore e forma:SolidPeso molecolare:269.232',3'-Dideoxy-5-fluorocytidine
CAS:Nucleoside Derivatives - 2’,3’-Dideoxy-nucleoside; Fluoro-modified nucleoside; Drugs and Inhibitors; HIV-1 inhibitorsFormula:C9H12FN3O3Colore e forma:SolidPeso molecolare:229.215'-Amino-5'-deoxythymidine
CAS:5'-Amino-5'-deoxythymidine is a thymidine derivative widely used in biochemical experiments and drug synthesis research.Formula:C10H15N3O4Purezza:99.89%Colore e forma:SolidPeso molecolare:241.242-Amino-6-chloropurine-9-β-D-(2'-deoxy)riboside
CAS:2-Amino-6-chloropurine-9-beta-D-(2'-deoxy)riboside is a 2'-Deoxy nucleoside; Halo-nucleoside.Formula:C10H12ClN5O3Colore e forma:SolidPeso molecolare:285.693',5'-Di-O-acetyl-2'-deoxy-N3-methyl uridine
CAS:3',5'-Di-O-acetyl-2'-deoxy-N3-methyl uridine is a Nucleoside Derivative - N-Alkylated nucleoside.Formula:C14H18N2O7Colore e forma:SolidPeso molecolare:326.33'-β-C-Methyl-5-methylcytidine
3'-beta-C-Methyl-5-methylcytidine is a Nucleoside Derivative - 3'-Modified nucleoside.Colore e forma:Soild2'-O-Phthalimidopropyl cytidine
CAS:2’-O-Phthalimidopropyl cytidine is a useful organic compound for research related to life sciences.Formula:C20H22N4O7Colore e forma:SolidPeso molecolare:430.413'-Deoxy-5-methoxyuridine
CAS:Nucleoside Derivatives - 3’-Deoxy nucleosides, 5-Modified pyrimidine nucleosidesFormula:C10H14N2O6Colore e forma:SolidPeso molecolare:258.23N1-Methyl-N3-[(2S)-2-(t-butoxycarbonyl)amino-3-(t-butoxycarbonyl)] propylpseudouridine
CAS:N1-Methyl-N3-[(2S)-2-(t-butoxycarbonyl)amino-3-(t-butoxycarbonyl)] propylpseudouridine is a Nucleoside Derivative - C-nucleoside; N-Alkylated nucleoside.Formula:C23H37N3O10Colore e forma:SolidPeso molecolare:515.55α-inosine
CAS:Alpha-inosine is a useful organic compound for research related to life sciences. The catalog number is TNU1638 and the CAS number is 38183-47-0.Formula:C10H12N4O5Colore e forma:SolidPeso molecolare:268.237,8-Dihydro-8-oxo-7-propargyl-3'-deoxy-3'-fluoro-xylo-guanosine
CAS:7,8-Dihydro-8-oxo-7-propargyl-3’-deoxy-3’-fluoro-xylo-guanosine is a useful organic compound for research related to life sciences.Formula:C13H14FN5O5Colore e forma:SolidPeso molecolare:339.282'-Deoxy-2'-fluoro-ara-uridine
2'-Deoxy-2'-fluoro-ara-uridine is a Nucleoside Derivative - 2'-Modified nucleoside, Fluoro-modified nucleoside, N-Methylated/ alkylated nucleoside.Colore e forma:Soild4,6-Diamino-2-(b-D-ribofuranosyl)-2H-pyrazolo[3,4-d]pyrimidine
CAS:4,6-Diamino-2-(b-D-ribofuranosyl)-2H-pyrazolo[3,4-d]pyrimidine is a Nucleoside Derivative - 7-deaza-8-aza purine nucleoside.Formula:C10H14N6O4Colore e forma:SolidPeso molecolare:282.265'-Azido-5'-deoxy-2'-O-methyl-5-methyluridine
CAS:Nucleoside Derivatives - 5’-Modified nucleosides, Azido-nucleosides, 2’-Modified nucleosidesFormula:C11H15N5O5Colore e forma:SolidPeso molecolare:297.272'-O-MOE-A(Bz)-3'-phosphoramidite
CAS:2'-O-MOE-A(Bz)-3'-phosphoramidite is a Nucleoside Phosphoramidite;Nucleoside Derivative - 2'-Modified nucleoside;.Formula:C50H58N7O9PColore e forma:SolidPeso molecolare:932.013'-β-C-Ethynyl-N6,N6-dimethyladenosine
CAS:Nucleoside Derivatives - 3’-Modified purine nucleosides; 6-Modified purine nucleosidesFormula:C14H17N5O4Colore e forma:SolidPeso molecolare:319.325'-O-DMT-2'-TBDMS-Uridine
CAS:5’-O-DMT-2’-TBDMS-Uridine is a deoxyribonucleoside used for the oligonucleotide synthesis.Formula:C36H44N2O8SiColore e forma:SolidPeso molecolare:660.83N1-(N,N-Dimethylaminocarbonyl)-pseudouridine
N1-(N,N-Dimethylaminocarbonyl)-pseudouridine is a Nucleoside Derivative - C-nucleoside.Colore e forma:Soild2'-Deoxy-2'-fluoro-N3-(n-dodecyl)-β-D-arabinouridine
CAS:2'-Deoxy-2'-fluoro-N3-(n-dodecyl)-beta-D-arabinouridine is a Nucleoside Derivative - Fluoro-modified nucleoside,Arabino-nucleoside, 2'-Modified nucleoside.Formula:C21H35FN2O5Colore e forma:SolidPeso molecolare:414.513'-O-(2-Methoxyethyl)uridine
CAS:3'-O-(2-Methoxyethyl)uridine is a Nucleoside Derivative - 3'-Modified nucleoside.Formula:C12H18N2O7Colore e forma:SolidPeso molecolare:302.281,2-Di-O-acetyl-5-O-benzoyl-3-deoxy-3-fluoro-D-xylofuranose
CAS:1,2-Di-O-acetyl-5-O-benzoyl-3-deoxy-3-fluoro-D-xylofuranose is a Carbohydrate Derivative.Formula:C16H17FO7Colore e forma:SolidPeso molecolare:340.3360A
CAS:<p>360A is a stabilizing G-Quadruplex ligand, and also inhibits telomerase activity for telomerase in TRAP-G4 assay(IC50 : 300 nM).</p>Formula:C27H23N5O2Purezza:98.68%Colore e forma:SolidPeso molecolare:449.5Dasabuvir
CAS:<p>Dasabuvir (ABT-333) blocks HCV replication by inhibiting the essential NS5B RNA polymerase.</p>Formula:C26H27N3O5SPurezza:99.54% - 99.62%Colore e forma:SolidPeso molecolare:493.57Apcin
CAS:Apcin: potent APC/C(Cdc20) E3 ligase inhibitor, blocks substrate recognition & mitosis, synergizes with Ts-Arg-OMe.Formula:C13H14Cl3N7O4Purezza:96.74%Colore e forma:SolidPeso molecolare:438.65Preq1-Dihydrochloride
CAS:Preq1-Dihydrochloride, a queuosine pathway intermediate, binds strongly to PreQ1 riboswitch aptamer, suppressing protein expression.Formula:C7H11Cl2N5OPurezza:99.46%Colore e forma:SolidPeso molecolare:252.1TH588
CAS:TH588 is nudix hydrolase family inhibitor that effectively and selectively engages and inhibits the MTH1(IC50: 5 nM) in cells.Formula:C13H12Cl2N4Purezza:96.05% - 99.82%Colore e forma:SolidPeso molecolare:295.17Besifloxacin Hydrochloride
CAS:Besifloxacin Hydrochloride (BOL-303224-A) is a fourth-generation fluoroquinolone antibiotic.Formula:C19H21ClFN3O3·HClPurezza:99.20%Colore e forma:Pale Yellow SolidPeso molecolare:430.3TH287 hydrochloride
CAS:<p>TH287 inhibits MTH1 (IC50: 0.8 nM), causing DNA damage in cancer cells through oxidized dNTP incorporation, leading to cytotoxicity in mouse xenografts.</p>Formula:C11H11Cl3N4Purezza:>99.99%Colore e forma:SolidPeso molecolare:305.59FUBP1-IN-1
CAS:FUBP1-in-1: Potent FUBP1 inhibitor with 11.0 M IC50, disrupts FUBP1-DNA binding.Formula:C19H14F3N3O2SPurezza:99.7%Colore e forma:SolidPeso molecolare:405.39(1E)-CFI-400437 dihydrochloride
CAS:(1E)-CFI-400437 dihydrochloride (CFI-400437 dihydrochloride) is a selective and potent polo-like kinase 4 (PLK4) inhibitor.Formula:C29H30Cl2N6O2Purezza:97.08%Colore e forma:SolidPeso molecolare:565.5APY29
CAS:APY29 is an allosteric modulator of IRE1α; inhibits IRE1α autophosphorylation (IC50 = 280 nM) and activates IRE1α RNase activity.Formula:C17H16N8Purezza:96.51% - 98.46%Colore e forma:SolidPeso molecolare:332.36TH-257
CAS:TH-257 is a Potent and selective allosteric LIMK 1/2 inhibitor(LIMK1 and LIMK2, IC50 of 84 nM and 39 nM).Formula:C24H26N2O3SPurezza:98.23%Colore e forma:SolidPeso molecolare:422.54CRT0044876
CAS:CRT0044876 (7-NO2-ICA) is a potent and selective APE1 inhibitor with IC50 of ~3 μM.Formula:C9H6N2O4Purezza:98.27% - 98.98%Colore e forma:Brown PowderPeso molecolare:206.15URMC-099
CAS:URMC-099: oral, brain-accessible MLK/LRRK2 inhibitor; IC50 – MLK1/2/3/DLK: 19/42/14/150 nM, LRRK2: 11 nM.Formula:C27H27N5Purezza:99.32% - 99.98%Colore e forma:SolidPeso molecolare:421.54Adavosertib
CAS:Adavosertib (MK-1775) is a small molecule inhibitor of the checkpoint kinase WEE1 (IC50: 5.2 nM). It hinders the G2 DNA damage checkpoint.Formula:C27H32N8O2Purezza:98.65% - 99.86%Colore e forma:SolidPeso molecolare:500.6SNS-314 Mesylate
CAS:SNS-314 Mesylate (SNS-314) is an effective and specific Aurora A/B/C inhibitor. SNS-314 is less inhibition of Trk A/B, Fms, Flt4, c-Raf, Axl, and DDR2.Formula:C18H15ClN6OS2·CH4O3SPurezza:99.44% - 99.92%Colore e forma:SolidPeso molecolare:527.04ILK-IN-3
CAS:ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.Formula:C10H12N6OPurezza:99.69%Colore e forma:SolidPeso molecolare:232.24XMD8-92
CAS:XMD8-92 is an effective and specific BMK1/ERK5 inhibitor (Kd: 80 nM).Formula:C26H30N6O3Purezza:98.21%Colore e forma:SolidPeso molecolare:474.55Dalpiciclib hydrochloride
Dalpiciclib (SHR-6390) HCl is an oral CDK4/6 inhibitor with IC50s of 12.4/9.9 nM, an antitumor for breast and esophageal cancers.Formula:C25H31ClN6O2Colore e forma:SolidPeso molecolare:483.015-Fluoroorotic acid
CAS:5-Fluoroorotic acid is an inhibitor of thymidylate synthase.Formula:C5H3FN2O4Purezza:99.7% - >99.99%Colore e forma:White To Pale Yellow PowderPeso molecolare:174.09Favipiravir
CAS:<p>Favipiravir is a potent and selective RNA-dependent RNA polymerase inhibitor for the treatment of influenza virus infections.Cost-effective and quality-assured.</p>Formula:C5H4FN3O2Purezza:97.32% - 99.90%Colore e forma:SolidPeso molecolare:157.1Simeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purezza:99.45% - 99.92%Colore e forma:SolidPeso molecolare:749.94MNS
CAS:MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.Formula:C9H7NO4Purezza:98.53%Colore e forma:Yellow PowderPeso molecolare:193.16CID-797718
CAS:CID-797718 is a protein kinase D1 (PKD1) inhibitor.Formula:C12H11NO3Purezza:98.91% - 99.21%Colore e forma:SolidPeso molecolare:217.22NSAH
CAS:NSAH (2-hydroxy-N'-[(E)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide) is a nonnucleoside inhibitor of human ribonucleotide reductase (hRR).with cell-Formula:C18H14N2O3Purezza:99.27%Colore e forma:SolidPeso molecolare:306.32RI-2
CAS:RI-2, a potent RAD51 inhibitor, has a 44.17 μM IC50 and selectively blocks human HR repair.Formula:C21H18Cl2N2O4Purezza:99.63% - 99.86%Colore e forma:SolidPeso molecolare:433.28SBC-115337
CAS:SBC-115337 is a PCSK9 inhibitor.Formula:C29H19N3O4Purezza:99.41%Colore e forma:SolidPeso molecolare:473.48CID755673
CAS:CID755673 inhibits PKD (IC50: 182 nM), with selectivity over PLK1, AKT, CAMKIIα, CAK, PKC.Formula:C12H11NO3Purezza:97.68% - 99.84%Colore e forma:SolidPeso molecolare:217.226-Thio-2'-Deoxyguanosine
CAS:6-Thio-2'-Deoxyguanosine (β-TGdR) is a nucleoside analog and telomerase substrate.Formula:C10H13N5O3SPurezza:97.52%Colore e forma:SolidPeso molecolare:283.31Carotegrast methyl HCl
CAS:Carotegrast methyl (AJM300/PTC-100) is an oral α4 integrin blocker reducing inflammation and experimental colitis.Formula:C25H20Cl3N3O5Colore e forma:SolidPeso molecolare:548.801Tegafur-Uracil
CAS:Tegafur-Uracil, an oral anticancer agent for solid tumor research, inhibits thymidylate synthase.Formula:C12H13FN4O5Colore e forma:SolidPeso molecolare:312.257Seliciclib
CAS:Seliciclib (Roscovitine) is a potent inhibitor of Cdk2/cyclin E, also inhibits Cdk7, Cdk5 and Cdc2. Seliciclib has antitumor effect. Cost-effective, quality assurance.Formula:C19H26N6OPurezza:97.15% - 99.89%Colore e forma:White To Off-White SolidPeso molecolare:354.45CK7
CAS:CK7, a Cdk2/9 inhibitor, is instrumental in the synthesis of Nek1 inhibitors BSc5231 and BSc5367.Formula:C14H12N6O2SPurezza:99.54%Colore e forma:SolidPeso molecolare:328.35Quarfloxin
CAS:<p>Quarfloxin (CX-3543), a fluoroquinolone, inhibits neuroblastoma with nanomolar IC50, disrupting nucleolin and G-quadruplex DNA.</p>Formula:C35H33FN6O3Purezza:99.77%Colore e forma:SolidPeso molecolare:604.67Ganciclovir hydrate
CAS:Ganciclovir hydrate: oral anti-cytomegalovirus; inhibits HSV 1/2, CMV, adenoviruses, FHV-1; brain-penetrating.Formula:C9H15N5O5Colore e forma:SolidPeso molecolare:273.249Alovudine
CAS:<p>3'-Fluoro-3'-deoxythymidine (3'-Deoxy-3'-fluorothymidine) is a marker of DNA synthesis,which is less susceptible to inflammatory changes than FDG.</p>Formula:C10H13FN2O4Purezza:99.41%Colore e forma:Less Solid Colourless SolidPeso molecolare:244.22FDI-6
CAS:FDI-6 is an effective and selective inhibitor of FOXM1 that blocks DNA binding. FDI-6 binds to the FOXM1 protein and downregulates FOXM1-activated genes.Formula:C19H11F4N3OS2Purezza:98.92% - >99.99%Colore e forma:SolidPeso molecolare:437.43BSJ-03-123
CAS:BSJ-03-123 is a potent, CDK6-selective small-molecule degrader.Formula:C47H56N10O11Purezza:97.78% - 99.38%Colore e forma:SolidPeso molecolare:937.01LIMK-IN-22j
CAS:LIMK-IN-22j (LIMK inhibitor 22j) is an effective and selective inhibitor of LIMK.Formula:C20H21BrN8Purezza:99.165%Colore e forma:SolidPeso molecolare:453.34Ro5-3335
CAS:Ro5-3335 (CBFβ-Runx1 inhibitor II) is core binding factor (CBF) inhibitor; preferentially kills human leukemia cell lines with CBF fusion proteins.Formula:C13H10ClN3OPurezza:99.42% - 99.87%Colore e forma:SolidPeso molecolare:259.69AT9283
CAS:<p>AT9283 (J-504568) is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora B and Abl(T315I).</p>Formula:C19H23N7O2Purezza:99.83% - 99.98%Colore e forma:SolidPeso molecolare:381.43XL228
CAS:XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).Formula:C22H31N9OPurezza:99.07%Colore e forma:SolidPeso molecolare:437.54Simeprevir sodium
CAS:Simeprevir is a drug for the treatment and cure of hepatitis C.Formula:C38H46N5NaO7S2Purezza:98%Colore e forma:SolidPeso molecolare:771.92Tozasertib
CAS:Tozasertib (MK-0457) is a pan-Aurora kinase inhibitor (Kis: 0.6/18/4.6 nM for Aurora A/Aurora B/Aurora C).Formula:C23H28N8OSPurezza:99.99%Colore e forma:SolidPeso molecolare:464.59Pritelivir
CAS:Pritelivir (BAY 57-1293) (BAY 57-1293) is a potent helicase-primase inhibitor with active against HSV-1 and HSV-2 (IC50: 20 nM).Formula:C18H18N4O3S2Purezza:97.96% - 99.42%Colore e forma:SolidPeso molecolare:402.49Voruciclib
CAS:Voruciclib: oral, selective CDK inhibitor (Ki: 0.626-9.1 nM), reduces MCL-1, targets CDK9 in diffuse large B-cell lymphoma.Formula:C22H19ClF3NO5Purezza:99.89% - 99.99%Colore e forma:SolidPeso molecolare:469.84SAR-020106
CAS:SAR-020106 is a potent, ATP-competitive, and selective CHK1 inhibitor with an IC50 of 13.3 nmol/L on the isolated human enzyme.Formula:C19H19ClN6OPurezza:97.78%Colore e forma:SolidPeso molecolare:382.85Pyridostatin TFA
CAS:Pyridostatin Trifluoroacetate Salt is a G-quadruplexe stabilizer with Kd of 490 nM in a cell-free assay, which targets a series of proto-oncogenes including c-Formula:C37H35F9N8O11Purezza:97.09% - 99.84%Colore e forma:SolidPeso molecolare:938.71AZ3146
CAS:<p>AZ3146 is a selective Mps1 inhibitor with IC50 of ~35 nM.</p>Formula:C24H32N6O3Purezza:97.84% - >99.99%Colore e forma:SolidPeso molecolare:452.55GSK-923295
CAS:GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).Formula:C32H38ClN5O4Purezza:96.22% - 98.02%Colore e forma:SolidPeso molecolare:592.13WNK463
CAS:WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Formula:C21H24F3N7O2Purezza:>99.99% - ≥95%Colore e forma:SolidPeso molecolare:463.46Tipiracil hydrochloride
CAS:Tipiracil hydrochloride (MA-1 hydrochloride) is a thymidine phosphorylase inhibitor (TPI).Formula:C9H12Cl2N4O2Purezza:98.13% - ≥95%Colore e forma:SolidPeso molecolare:279.12InhA-IN-2
CAS:N-[3-(Aminomethyl)phenyl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide inhibits InhA without KatG activation.Formula:C16H15ClN2O2S2Purezza:98.4%Colore e forma:SolidPeso molecolare:366.89THZ2
CAS:THZ2 (CDK7-IN-1), an analog of THZ1, is a potent and selective CDK7 inhibitor(IC50:13.9 nM),with the potential to treat Triple-negative breast cancer (TNBC).Formula:C31H28ClN7O2Purezza:98.28%Colore e forma:SolidPeso molecolare:566.05GSK461364
CAS:GSK461364 (GSK461364A)(Ki=2.2 nM) inhibits purified Plk1 .The specificity of GSK461364 for Plk1 is more than 1000-fold over Plk2/3.Formula:C27H28F3N5O2SPurezza:99% - 99.73%Colore e forma:SolidPeso molecolare:543.6BMS-1001
CAS:BMS-1001 is a potent inhibitor of PD-1/PD-L1 interaction(IC50 : 2.25 nM, in a homogenous time-resolved fluorescence binding assay).Formula:C35H34N2O7Purezza:98.43%Colore e forma:SolidPeso molecolare:594.7Madrasin
CAS:<p>Madrasin (DDD00107587) is a potent and cell penetrant splicing inhibitor that interferes with the early stages of spliceosome assembly.</p>Formula:C16H17N5O2Purezza:99.06% - 99.61%Colore e forma:SolidPeso molecolare:311.34Dimethylenastron
CAS:Dimethylenastron, an Eg5 inhibitor, arrests cells with monopolar spindles to which all chromosomes attach in a syntelic manner.Formula:C16H18N2O2SPurezza:98.07%Colore e forma:SolidPeso molecolare:302.39Senexin A
CAS:Senexin A is an effective and selective CDK8 inhibitor that also inhibits CDK19 with Kd values of 0.83 microns and 0.31 microns, respectively.Formula:C17H14N4Purezza:99.74%Colore e forma:SolidPeso molecolare:274.32Nemorubicin HCL
CAS:Nemorubicin HCL, a PNU152243A salt, acts on resistant tumors via topoisomerase I inhibition and targets NER pathway upregulated cells.Formula:C32H38ClNO13Colore e forma:SolidPeso molecolare:680.1SCH900776 (S-isomer)
CAS:SCH900776 S-isomer (MK-8776 S-isomer) is an effective, specific and orally bioavailable inhibitor of checkpoint kinase Chk1 (IC50: 3 nM).Formula:C15H18BrN7Purezza:99.88%Colore e forma:SolidPeso molecolare:376.25Indisulam
CAS:Indisulam (E 7070) is a dual-action anticancer drug, blocking G1/S cell cycle transition by degrading cyclin E and activating p53/p21.Formula:C14H12ClN3O4S2Purezza:98.68% - 99.77%Colore e forma:SolidPeso molecolare:385.85GDC-0575
CAS:<p>GDC-0575 (ARRY-575) is a highly-selective oral small-molecule Chk1 inhibitor(IC50 of 1.2 nM).</p>Formula:C16H20BrN5OPurezza:≥95%Colore e forma:SolidPeso molecolare:378.27Trilaciclib
CAS:Trilaciclib is a short-acting, orally effective CDK4/6 inhibitor with IC₅₀ values of 1 nM and 4 nM respectively. enhances antitumour immunity.Formula:C24H30N8OPurezza:99.624%Colore e forma:SolidPeso molecolare:446.55THZ531
CAS:THZ531 is a covalent inhibitor of both CDK12(IC50=158 nM) and CDK13(IC50=69 nM).Formula:C30H32ClN7O2Purezza:97.17% - 99.86%Colore e forma:SolidPeso molecolare:558.07VX-11e
CAS:VX-11e (TCS ERK 11e) is a potent, selective, and orally bioavailable ERK(Extracellular Signal-Regulated Kinase) inhibitor; antitumor agent.Formula:C24H20Cl2FN5O2Purezza:98.92% - ≥98%Colore e forma:SolidPeso molecolare:500.35Cetraxate hydrochloride
CAS:Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.Formula:C17H24ClNO4Purezza:99.75%Colore e forma:SolidPeso molecolare:341.83BTB-1
CAS:BTB-1 (NSC156750) is a novel small molecule inhibitor of the mitotic motor protein Kif18A.Formula:C12H8ClNO4SPurezza:99.71%Colore e forma:SolidPeso molecolare:297.71BUR1
CAS:BUR1 is a Saccharomyces cerevisiae cyclin-dependent kinase (CDK) and is homologous to mammalian Cdk9, which functions in transcriptional elongation.Formula:C16H17N5Purezza:90%Colore e forma:SolidPeso molecolare:279.34Adefovir dipivoxil
CAS:Adefovir dipivoxil (GS 0840) is a dipivoxil formulation of adefovir, a nucleoside reverse transcriptase inhibitor analog of adenosine with activity againstFormula:C20H32N5O8PPurezza:98% - 99.80%Colore e forma:It Has Broad-Spectrum Antiviral ActivityPeso molecolare:501.4710074-G5
CAS:<p>10074-G5 is an inhibitor of c-Myc-Max dimerization.</p>Formula:C18H12N4O3Purezza:99.51% - 99.67%Colore e forma:SolidPeso molecolare:332.31MTOB
CAS:MTOB, a CtBP substrate, inhibits CtBP-linked cancer activity in cells/mice and regulates TCF-4, affecting CSC proliferation.Formula:C5H7NaO3SPurezza:98.23%Colore e forma:SolidPeso molecolare:170.16ILK-IN-2
CAS:<p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>Formula:C30H30F3N5OPurezza:99.30%Colore e forma:SolidPeso molecolare:533.59LY2334737
CAS:LY2334737 is an orally available prodrug of gemcitabine with antineoplastic activity.Formula:C17H25F2N3O5Purezza:98.82%Colore e forma:SolidPeso molecolare:389.39BTYNB
CAS:BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1. MDK6620 downregulates β-TrCP1 mRNA and reduces activation of NF-κB.Formula:C12H9BrN2OSPurezza:≥95%Colore e forma:SolidPeso molecolare:309.18BS-181 dihydrochloride
CAS:BS-181 dihydrochloride: Potent CDK7 inhibitor (IC50: 21 nM), less effective on CDK2/5/9, no impact on CDK1/4/6, halts cancer cell growth, triggers apoptosis.Formula:C22H34Cl2N6Colore e forma:SolidPeso molecolare:453.46IMP-1088
CAS:IMP-1088 is a potent inhibitor of human N-myristoyltransferases NMT1 and NMT2 dual.Formula:C25H29F2N5OPurezza:98.48% - 99.52%Colore e forma:SolidPeso molecolare:453.533-AP
CAS:3-AP (Triapine) is a novel inhibitor of the M2 subunit of ribonucleotide reductase (RR).Formula:C7H9N5SPurezza:97.33% - 99.87%Colore e forma:SolidPeso molecolare:195.24GPRP acetate (67869-62-9 free base)
CAS:<p>GPRP acetate (Pefabloc FG) is fibrinogen-related peptides, which inhibit the interaction of fibrinogen with the platelet membrane glycoprotein IIbIIIa complex.</p>Formula:C20H35N7O7Purezza:>99.99%Colore e forma:SolidPeso molecolare:485.53

