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Ciclo cellulare/Checkpoint

Ciclo cellulare/Checkpoint

Gli inibitori del ciclo cellulare/dei checkpoint sono composti che interrompono la normale progressione del ciclo cellulare, in particolare nei principali punti di controllo regolatori. Questi inibitori sono fondamentali per studiare la divisione cellulare, comprendere la proliferazione delle cellule cancerose e sviluppare terapie antitumorali. Mirando a fasi specifiche del ciclo cellulare, questi inibitori possono indurre l'arresto del ciclo cellulare, portando all'apoptosi o alla senescenza nelle cellule che si dividono rapidamente. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità del ciclo cellulare/dei checkpoint per supportare le tue ricerche in biologia del cancro, biologia cellulare e sviluppo di farmaci.

Sottocategorie di "Ciclo cellulare/Checkpoint"

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Trovati 3739 prodotti di "Ciclo cellulare/Checkpoint"

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  • 5'-O-DMT-2'-O-TBDMS-Ac-rC

    CAS:
    5’-O-DMT-2’-O-TBDMS-Ac-rC is a modified nucleoside and can be used to synthesize DNA or RNA.
    Formula:C38H47N3O8Si
    Colore e forma:Solid
    Peso molecolare:701.892
  • DNA Gyrase-IN-6


    Agent 138: soluble benzothiazole, inhibits DNA gyrase/topoisomerase IV, targets Gram+ & Gram- bacteria, binds plasma proteins.
    Formula:C18H16Cl2N4O4S
    Colore e forma:Solid
    Peso molecolare:455.32
  • 5'-O-TBDMS-N2-ibu-dG

    CAS:
    <p>5'-O-TBDMS-N2-ibu-dG: a nucleoside derivative with strong anti-BVDV activity, useful in lead compound synthesis.</p>
    Formula:C20H33N5O5Si
    Colore e forma:Solid
    Peso molecolare:451.59
  • XT17


    XT17 is an anthrone compound with broad-spectrum antibacterial activity, exerting its effects by disrupting the cell wall and inhibiting DNA synthesis. It demonstrates weak hemolytic activity, low cytotoxicity to mammalian cell lines, and a low rate of resistance development. Additionally, XT17 shows in vivo efficacy in a mouse corneal infection model induced by Staphylococcus aureus or Pseudomonas aeruginosa. Further docking studies confirm that XT17 forms a stable complex with bacterial gyrase. XT17 is suitable for research in the field of anti-infective agents.
    Colore e forma:Odour Solid
  • Nogalamycin

    CAS:
    Nogalamycin is an anthracycline antibiotic with antitumor properties produced by soil bacteria Streptomyces nogalater.
    Formula:C39H49NO16
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:787.812
  • 4-Amino-1-(β-D-ribofuranosyl)-7H-pyrrolo[2.3-d]pyrimidine-5-carboxamide


    4-Amino-1-(β-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide is a purine nucleoside analog with broad antitumor activity against indolent lymphoid
    Formula:C12H15N5O5
    Colore e forma:Solid
    Peso molecolare:309.28
  • Bz-rC Phosphoramidite

    CAS:
    <p>Bz-rC Phosphoramidite is a phosphinamide monomer utilized for oligonucleotide synthesis.</p>
    Formula:C52H66N5O9PSi
    Colore e forma:Solid
    Peso molecolare:964.185
  • Pseudorabies virus-IN-1


    <p>Pseudorabies virus-IN-1 is a potent inhibitor of pseudorabies virus (PRV) with an EC50 of 0.29 nM, acting by targeting PRV deoxyribonucleic acid polymerase (DNA pol) to suppress PRV replication. It effectively inhibits PRV replication even at low concentrations (MIC80: 1.6-8 nM) and is useful for research on PRV infections.</p>
    Formula:C27H23ClF2N4O2
    Colore e forma:Solid
    Peso molecolare:508.947
  • ONX 0801 trisodium

    CAS:
    <p>ONX 0801 (BGC 945) trisodium is a targeted thymidylate synthase (TS) inhibitor specifically designed to act against tumors overexpressing the α-folate receptor.</p>
    Formula:C32H30N5Na3O10
    Colore e forma:Solid
    Peso molecolare:713.58
  • c-Myc inhibitor 7

    CAS:
    c-Myc inhibitor 7 degrades c-MYC, CK1α, GSPT1, IKZF1/2/3 proteins in tumors, for research on related diseases.
    Formula:C35H30N6O5
    Colore e forma:Soild
    Peso molecolare:614.65
  • JB-11 isethionate

    CAS:
    JB-11 isethionate is a bioactive chemical.
    Formula:C21H29N5O7S
    Colore e forma:Solid
    Peso molecolare:495.55
  • 1-(b-D-Xylofuranosyl)-N6-(p-methoxybenzyl) adenine


    1-(β-D-Xylofuranosyl)adenine is a purine analog with antitumor activity, inhibiting DNA synthesis and inducing apoptosis.
    Formula:C18H21N5O5
    Colore e forma:Solid
    Peso molecolare:387.39
  • N1-(2-Methyl)propyl pseudouridine


    N1-(2-Methyl)propyl pseudouridine, a purine analog, targets lymphoid cancer by inhibiting DNA synthesis and inducing apoptosis.
    Formula:C13H20N2O6
    Colore e forma:Solid
    Peso molecolare:300.31
  • 3'-β-C-ethynyl-N6-(m-trifluoromethyl benzyl)adenosine


    3’-Beta-C-ethynyl-N6-(m-trifluoromethyl benzyl)adenosine is an adenosine analog.
    Formula:C20H18F3N5O4
    Colore e forma:Solid
    Peso molecolare:449.38
  • R-BC154 acetate


    R-BC154 acetate: selective α9β1 antagonist, high-affinity integrin probe for α9β1/α4β1 activity study.
    Formula:C56H65N9O14S3
    Colore e forma:Solid
    Peso molecolare:1184.36
  • L-5-Methyluridine

    CAS:
    L-5-Methyluridine, an L-configuration of 5-Methyluridine, is an endogenous methylated nucleoside present in human fluids.
    Formula:C10H14N2O6
    Colore e forma:Solid
    Peso molecolare:258.23
  • DHFR-IN-9


    DHFR-IN-9 (compound 8A), a dihydrofolate reductase (DHFR) inhibitor, impedes purine and thymidylate biosynthesis, pivotal in cell proliferation and growth.
    Formula:C19H16N6S
    Colore e forma:Solid
    Peso molecolare:360.44
  • EFdA-TP tetraammonium


    EFdA-TP tetraammonium is a potent HIV-1 RT inhibitor and DNA synthesis blocker, acting as an ICT or DCT.
    Formula:C12H27N9O12P3
    Colore e forma:Solid
    Peso molecolare:601.31
  • Gly-Arg-Gly-Asp-Ser

    CAS:
    <p>Gly-Arg-Gly-Asp-Ser (GRGDS) GRGDS is a cell binding protein domain derived from the cell-binding region of fibronectin.</p>
    Formula:C17H30N8O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:490.47
  • Pyrindamycin A

    CAS:
    Pyrindamycin A is an antibiotic that inhibits DNA synthesis,and shows antitumor activities against murine leukemia.
    Formula:C26H26ClN3O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:543.95