
Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(36 prodotti)
- Cisteina proteasi(110 prodotti)
- DPP-4(20 prodotti)
- Glutaminasi(45 prodotti)
- Proteasi HIV(506 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(54 prodotti)
- Proteasoma(95 prodotti)
- Proteasi serina(55 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 1095 prodotti di "Proteasi/Proteasoma"
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1,10-Phenanthroline Monohydrate [for Biochemical Research]
CAS:Formula:C12H8N2·H2OPurezza:>99.0%(T)Colore e forma:White powder to crystalPeso molecolare:198.23Disodium Dihydrogen Ethylenediaminetetraacetate Dihydrate [for Biochemical Research]
CAS:Formula:C10H14N2Na2O8·2H2OPurezza:>99.0%(T)Colore e forma:White powder to crystalinePeso molecolare:372.24Ethylene Glycol Bis(2-aminoethyl Ether)-N,N,N',N'-tetraacetic Acid [for Biochemical Research]
CAS:Formula:C14H24N2O10Purezza:>95.0%(T)Colore e forma:White to Almost white powder to crystalPeso molecolare:380.35Camostat Mesylate
CAS:Formula:C20H22N4O5·CH4O3SPurezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:494.52MG-132
CAS:Formula:C26H41N3O5Purezza:>95.0%(qNMR)Colore e forma:White to Light yellow powder to crystalPeso molecolare:475.63Limonin
CAS:Formula:C26H30O8Purezza:>95.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:470.52Gabexate Mesylate
CAS:Formula:C16H23N3O4·CH4O3SPurezza:>97.0%(N)Colore e forma:White to Almost white powder to crystalPeso molecolare:417.48Ritonavir
CAS:Formula:C37H48N6O5S2Purezza:>98.0%(HPLC)(N)Colore e forma:White to Almost white powder to crystalinePeso molecolare:720.95Atazanavir
CAS:Formula:C38H52N6O7Purezza:>95.0%(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:704.87Nelfinavir Mesylate
CAS:Formula:C32H45N3O4S·CH4O3SPurezza:>97.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:663.894-(2-Aminoethyl)benzenesulfonyl Fluoride Hydrochloride [for Biochemical Research]
CAS:Formula:C8H10FNO2S·HClPurezza:>99.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:239.692-Iodoacetamide [for Biochemical Research]
CAS:Formula:C2H4INOPurezza:>98.0%(N)Colore e forma:White to Light yellow powder to crystalPeso molecolare:184.96Atazanavir Sulfate
CAS:Formula:C38H52N6O7·H2SO4Purezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:802.94Nafamostat Mesylate
CAS:Formula:C19H17N5O2·2CH4O3SPurezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:539.58Benzylsulfonyl Fluoride [for Biochemical Research]
CAS:Formula:C7H7FO2SPurezza:>98.0%(GC)Colore e forma:White to Almost white powder to crystalPeso molecolare:174.19Islatravir
CAS:Islatravir (MK-8591) is an effective anti-HIV-1 agent.Formula:C12H12FN5O3Purezza:98.77%Colore e forma:SolidPeso molecolare:293.25Ref: TM-T16098
1mg80,00€5mg170,00€10mg259,00€25mg454,00€50mg615,00€100mg827,00€200mg1.111,00€1mL*10mM (DMSO)182,00€N-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Formula:C17H18ClNO3SPurezza:97%Colore e forma:SolidPeso molecolare:351.8477Ref: IN-DA0032JK
5g22,00€10g26,00€1kg229,00€25g30,00€50g40,00€100g59,00€10kgPrezzo su richiesta250g114,00€500g164,00€Levovirin
CAS:<p>Levovirin (L-Ribavirin) is a guanosine nucleoside analog that has immunomodulatory activity and is used in the study of hepatitis C virus infection.</p>Formula:C8H12N4O5Purezza:99.81% - >99.99%Colore e forma:SolidPeso molecolare:244.203-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-, methanesulfonate (1:1)
CAS:Formula:C33H49N3O7S2Purezza:96%Colore e forma:SolidPeso molecolare:663.8881Benzenemethanesulfonyl fluoride
CAS:Formula:C7H7FO2SPurezza:99%Colore e forma:SolidPeso molecolare:174.1927Ref: IN-DA00I6AP
1g25,00€5g39,00€10g55,00€25g90,00€50g127,00€100g166,00€250g505,00€500gPrezzo su richiestaBestatin hydrochloride
CAS:Formula:C16H25ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:344.8337Ref: IN-DA003O5U
1g542,00€5gPrezzo su richiesta10mg61,00€25mg94,00€50mg148,00€100mg191,00€250mg197,00€500mg333,00€KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Formula:C29H31N5O5SPurezza:99.28%Colore e forma:SolidPeso molecolare:561.65Benzoic acid, 4-[[6-[(aminoiminomethyl)amino]-1-oxohexyl]oxy]-, ethylester, monomethanesulfonate
CAS:Formula:C17H27N3O7SPurezza:98%Colore e forma:SolidPeso molecolare:417.4772Ethylenediaminetetraacetic acid disodium salt dihydrate
CAS:Formula:C10H18N2Na2O10Purezza:97%Colore e forma:SolidPeso molecolare:372.2369Dabigatran ethyl ester hydrochloride
CAS:Dabigatran prevents blood clots, inhibiting NQO2 and thrombin with IC50 0.8 μM.Formula:C27H30ClN7O3Purezza:99.65%Colore e forma:SolidPeso molecolare:536.03DPP-IV-IN-2
CAS:DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Formula:C18H26N4O5Purezza:99.08%Colore e forma:SolidPeso molecolare:378.42(Rac)-Telinavir
CAS:<p>N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.</p>Formula:C33H44N6O5Purezza:99.30%Colore e forma:SolidPeso molecolare:604.74GSK2838232
CAS:<p>GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.</p>Formula:C48H73ClN2O6Purezza:97.97%Colore e forma:SolidPeso molecolare:809.56CL-82198
CAS:CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Formula:C17H22N2O3Purezza:95.91%Colore e forma:SolidPeso molecolare:302.37Ref: TM-T14978
5mg47,00€10mg73,00€25mg153,00€50mg243,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)50,00€Dabigatran etexilate
CAS:Dabigatran etexilate (BIBR 1048) is a thrombin inhibitor, which acts by binding and blocking thrombogenic activity and the prevention of thrombus formation.Formula:C34H41N7O5Purezza:98.19% - 99.98%Colore e forma:White PowderPeso molecolare:627.733-Aminopropionitrile fumarate (2:1)
CAS:3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.Formula:C4H4O4·2C3H6N2Purezza:99.76% - 99.79%Colore e forma:White Crystalline PowderPeso molecolare:256.26Saxagliptin hydrate
CAS:Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).Formula:C18H25N3O2·H2OPurezza:99.52%Colore e forma:SolidPeso molecolare:333.43Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Formula:C19H17NO7Purezza:97.99%Colore e forma:SolidPeso molecolare:371.34Ref: TM-T15574
1mg88,00€2mgPrezzo su richiesta5mg119,00€10mg188,00€25mg393,00€50mg605,00€100mg847,00€200mg1.159,00€1mL*10mM (DMSO)96,00€NBD-556
CAS:NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Formula:C17H24ClN3O2Purezza:99.79%Colore e forma:SolidPeso molecolare:337.84Avoralstat
CAS:Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.Formula:C28H27N5O5Purezza:99.77%Colore e forma:SolidPeso molecolare:513.54DBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Formula:C16H25FN4O2Purezza:99.68%Colore e forma:SolidPeso molecolare:324.39Ref: TM-T15079
1mg50,00€5mg105,00€10mg140,00€25mg226,00€50mg324,00€100mg437,00€200mg605,00€1mL*10mM (DMSO)116,00€HCV-IN-29
CAS:HCV-IN-29 is a hepatitis C virus (HCV) inhibitor.Formula:C26H32Cl4N6Purezza:99.89%Colore e forma:SolidPeso molecolare:570.38Bivalirudin acetate
Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.Formula:C100H142N24O35Purezza:99.84%Colore e forma:SolidPeso molecolare:2240.34PMSF
CAS:PMSF (Phenylmethylsulfonyl fluoride) is an irreversible inhibitor of serine/cysteine protease , preparation of cell lysates. High-Quality, Low-Cost!Formula:C7H7FO2SPurezza:97.75% - 99.88%Colore e forma:White To Cream SolidPeso molecolare:174.19Ref: IN-DA00BBLC
1g57,00€5g128,00€25g262,00€5mg30,00€100gPrezzo su richiesta10mg30,00€50mg30,00€100mg37,00€250mg44,00€Ref: IN-DA0034HK
5gPrezzo su richiesta10g21,00€1kg124,00€25g25,00€50g25,00€5kg563,00€100g34,00€250g60,00€500g75,00€50kgPrezzo su richiestaBenzoic acid, 4-[(aminoiminomethyl)amino]-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate
CAS:Formula:C20H21N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:443.47621,10-Phenanthroline hydrate
CAS:Formula:C12H10N2OPurezza:98%Colore e forma:SolidPeso molecolare:198.22064-(2-Aminoethyl)benzenesulfonyl fluoride, HCl
CAS:Formula:C8H11ClFNO2SPurezza:98%Colore e forma:SolidPeso molecolare:239.6948(ETHYLENEDINITRILO)TETRAACETIC ACID, TRISODIUM SALT HYDRATE
CAS:Formula:C10H18N2NaO9Purezza:97%Colore e forma:SolidPeso molecolare:333.2477(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
CAS:Formula:C16H24N2O4Purezza:98%Colore e forma:SolidPeso molecolare:308.3728Ref: IN-DA00370Q
1g132,00€5g223,00€10g532,00€25gPrezzo su richiesta50gPrezzo su richiesta100gPrezzo su richiesta10mg29,00€250gPrezzo su richiesta50mg34,00€100mg44,00€250mg68,00€Sofosbuvir impurity G
CAS:Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.Formula:C22H29FN3O9PPurezza:98.04%Colore e forma:SolidPeso molecolare:529.45Ref: TM-T12962
1mg1.103,00€5mg2.547,00€10mg3.449,00€25mg5.120,00€50mg6.925,00€1mL*10mM (DMSO)3.202,00€3-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-
CAS:Formula:C32H45N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:567.78242-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Formula:C17H30N2O5Purezza:98%Colore e forma:SolidPeso molecolare:342.4305LSP-249
CAS:LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.Formula:C24H22ClN5OPurezza:99.51%Colore e forma:SolidPeso molecolare:431.924-Chlorosalicylic acid
CAS:<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Formula:C7H5ClO3Purezza:98.59%Colore e forma:Off-White To Light Beige PowderPeso molecolare:172.57Ethylene glycol bis(2-aminoethyl ether)-N,N,N',N'-tetraacetic acid
CAS:Formula:C14H24N2O10Purezza:97%Colore e forma:SolidPeso molecolare:380.3478Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Purezza:> 95%Colore e forma:LiquidPeso molecolare:145.42 kDaFostemsavir Tris
CAS:Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formula:C29H37N8O11PPurezza:99.45%Colore e forma:SolidPeso molecolare:704.62Ref: TM-T10570
1mg57,00€5mg120,00€10mg170,00€25mg283,00€50mg432,00€100mg612,00€1mL*10mM (DMSO)180,00€LDN-27219
CAS:LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.Formula:C20H16N4O2S2Purezza:99.01% - 99.38%Colore e forma:SolidPeso molecolare:408.5Ref: TM-T11831
1mg35,00€5mg66,00€10mg92,00€25mg160,00€50mg234,00€100mg351,00€200mg515,00€1mL*10mM (DMSO)71,00€Retagliptin Phosphate
CAS:Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Formula:C19H21F6N4O7PPurezza:98.70%Colore e forma:SolidPeso molecolare:562.36Ref: TM-T12710
1mg35,00€2mg44,00€5mg64,00€10mg93,00€25mg170,00€50mg259,00€100mgPrezzo su richiesta1mL*10mM (DMSO)84,00€Anisindione
CAS:Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.Formula:C16H12O3Purezza:98.25%Colore e forma:Pale Yellow Crystals From Acetic Acid Or Ethanol SolidPeso molecolare:252.26Aprotinin
CAS:<p>Aprotinin (Traskolan) is a broad-spectrum serine protease (BPTI) inhibitor. Aprotinin is an antifibrinolytic agent. Cost-effective and quality-assured.</p>Formula:C284H432N84O79S7Purezza:98%Colore e forma:SolidPeso molecolare:6511.51Sitagliptin
CAS:Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.Formula:C16H15F6N5OPurezza:99.33% - 99.83%Colore e forma:Yellow GreasePeso molecolare:407.31Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Formula:C49H55FN10O7SPurezza:96.87% - 99.93%Colore e forma:SolidPeso molecolare:947.09BJJF078
CAS:BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Formula:C27H29N3O6SPurezza:99.56%Colore e forma:SoildPeso molecolare:523.6Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Formula:C13H17NO8Purezza:99.52%Colore e forma:SolidPeso molecolare:315.28L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Formula:C26H41N3O5Purezza:98%Colore e forma:SolidPeso molecolare:475.6208Ref: IN-DA0072SK
1gPrezzo su richiesta5mg68,00€10mg90,00€25mg124,00€50mg168,00€100mg229,00€250mg500,00€500mgPrezzo su richiestaElsulfavirine
CAS:Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.Formula:C24H17BrCl2FN3O5SPurezza:99.66%Colore e forma:SolidPeso molecolare:629.28Ref: TM-T15210
1mg72,00€5mg156,00€10mg243,00€25mg487,00€50mg730,00€100mg1.026,00€1mL*10mM (DMSO)210,00€BLT-1
CAS:<p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>Formula:C12H23N3SPurezza:97.97%Colore e forma:SolidPeso molecolare:241.4MK-0608
CAS:MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).Formula:C12H16N4O4Purezza:98.48%Colore e forma:SolidPeso molecolare:280.28Ref: TM-T16088
1mg48,00€2mg63,00€5mg92,00€10mg140,00€25mg264,00€50mg434,00€100mg697,00€1mL*10mM (DMSO)97,00€Begelomab
CAS:Begelomab (SAND-26) is a mouse-derived monoclonal antibody targeting DPP-4/CD26. Begelomab can be used to study severe refractory inflammatory myopathies.Purezza:97.8% (SDS-PAGE); 98.3% (SEC-HPLC) - 97.8% (SDS-PAGE); 98.3% (SEC-HPLC)Colore e forma:LiquidSalicylanilide
CAS:<p>Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.</p>Formula:C13H11NO2Purezza:99.55%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:213.23BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formula:C19H17N3O2SPurezza:98.01% - 99.05%Colore e forma:SolidPeso molecolare:351.42Ref: TM-T10603
5mg50,00€10mg90,00€25mg170,00€50mg305,00€100mg442,00€200mg620,00€1mL*10mM (DMSO)51,00€Gly-Pro-pNA hydrochloride
CAS:<p>Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase</p>Formula:C13H17ClN4O4Purezza:99.84%Colore e forma:SolidPeso molecolare:328.75ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Formula:C17H20N2O5SPurezza:97.18%Colore e forma:SolidPeso molecolare:364.42Probenecid
CAS:Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.Formula:C13H19NO4SPurezza:98.95% - 99.84%Colore e forma:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecolare:285.36Mecarbinate
CAS:Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.Formula:C13H15NO3Purezza:99.28%Colore e forma:Off-White Crystalline PowderPeso molecolare:233.26(Rac)-Telmesteine
CAS:<p>(Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) is an inhibitor of protease and is thus a suitable enzyme stabilizer.</p>Formula:C7H11NO4SPurezza:99.91%Colore e forma:SolidPeso molecolare:205.23PF-3450074
CAS:PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Formula:C27H27N3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:425.52RA190
CAS:RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.Formula:C28H23Cl5N2O2Purezza:97.7%Colore e forma:SolidPeso molecolare:596.76Ref: TM-T13858
1mg57,00€5mg115,00€10mg168,00€25mg245,00€50mg437,00€100mg642,00€1mL*10mM (DMSO)150,00€ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Formula:C17H24BF3N2O4Purezza:97.06%Colore e forma:SolidPeso molecolare:388.19Ref: TM-T12079
1mg115,00€2mg166,00€5mg274,00€10mg432,00€25mg715,00€50mg1.008,00€100mg1.359,00€200mg1.825,00€1mL*10mM (DMSO)301,00€BAY-85-8501
CAS:BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Formula:C22H17F3N4O3SPurezza:99.16%Colore e forma:SolidPeso molecolare:474.46Ref: TM-T12613L
1mg96,00€2mg128,00€5mg212,00€10mg314,00€25mg565,00€50mg792,00€100mg1.093,00€1mL*10mM (DMSO)220,00€Sofosbuvir impurity F
CAS:Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNAFormula:C34H45FN4O13P2Purezza:98.05%Colore e forma:SolidPeso molecolare:798.69RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Formula:C19H13Cl4NOPurezza:98.89% - 99.38%Colore e forma:SolidPeso molecolare:413.12Trelagliptin
CAS:Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.Formula:C18H20FN5O2Purezza:98.88%Colore e forma:SolidPeso molecolare:357.383-Deazaadenosine hydrochloride
CAS:3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.Formula:C11H15ClN4O4Purezza:98.48%Colore e forma:SolidPeso molecolare:302.71Ref: TM-T10111
1mg126,00€5mg216,00€10mg374,00€25mg620,00€50mg868,00€100mg1.169,00€1mL*10mM (DMSO)149,00€Sofosbuvir impurity J
CAS:Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H30FN4O8PPurezza:98%Colore e forma:SolidPeso molecolare:528.47BPHA
CAS:BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.Formula:C21H20N2O4SPurezza:99.44%Colore e forma:SolidPeso molecolare:396.46Ref: TM-T36712
1mg170,00€5mg467,00€10mg655,00€25mg1.008,00€50mg1.378,00€100mg1.833,00€200mg2.452,00€1mL*10mM (DMSO)465,00€HCV-IN-4
CAS:HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.Formula:C52H58FN9O8Purezza:98%Colore e forma:SolidPeso molecolare:956.07ADAM8-IN-1
CAS:<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Formula:C44H44Br4N6O12S2Colore e forma:SolidPeso molecolare:1232.6HIV-1 protease-IN-14
HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.Colore e forma:Odour SolidMMP-3 Inhibitor
CAS:MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.Formula:C27H46N10O9SPurezza:98.87%Colore e forma:SolidPeso molecolare:686.78Ref: TM-T37048
1mg81,00€5mg208,00€10mg309,00€25mg525,00€50mg757,00€100mg1.035,00€500mg2.110,00€1mL*10mM (DMSO)221,00€PS 915
CAS:PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.Formula:C27H36ClN7O6Purezza:98%Colore e forma:SolidPeso molecolare:590.08Neutrophil elastase inhibitor 4
Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.Formula:C20H21N3O5Colore e forma:SolidPeso molecolare:383.4PROTAC 20S proteasome subunit β5 degrader 2
PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.Colore e forma:Odour SolidBMS-767778
CAS:BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.Formula:C19H20Cl2N4O2Colore e forma:SolidPeso molecolare:407.29



