Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.024 prodotti)
- Recettore dell'adenosina(249 prodotti)
- Recettore adrenergico(3.030 prodotti)
- Recettore della bombesina(35 prodotti)
- Recettore della bradichinina(61 prodotti)
- CXCR(159 prodotti)
- CaSR(34 prodotti)
- Recettore dei cannabinoidi(217 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(443 prodotti)
- Recettore dell'endotelina(86 prodotti)
- Recettore GNRH(84 prodotti)
- GPCR19(33 prodotti)
- GRK(33 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(196 prodotti)
- Proteina Hedgehog/Smoothened(49 prodotti)
- Recettore dell'istamina(385 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(42 prodotti)
- Recettore degli oppioidi(326 prodotti)
- PAFR(14 prodotti)
- PKA(54 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 19 più sottocategorie
Trovati 5981 prodotti di "Proteina G/GPCR"
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Citalopram hydrobromide
CAS:Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFormula:C20H22BrFN2OPurezza:99.81%Colore e forma:White Crystalline PowderPeso molecolare:405.304GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formula:C30H35N3O3Purezza:98.94% - 99.29%Colore e forma:SolidPeso molecolare:485.62Ref: TM-T11463
2mg42,00€5mg62,00€10mg97,00€25mg187,00€50mg305,00€100mg487,00€200mg692,00€1mL*10mM (DMSO)66,00€Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purezza:99.19% - 99.73%Colore e forma:SolidPeso molecolare:395.43Indusatumab
CAS:<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Purezza:> 95% - > 95%Colore e forma:LiquidPeso molecolare:145.18 kDaAnamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Formula:C31H42N6O3Purezza:99.35% - 99.94%Colore e forma:SolidPeso molecolare:546.7Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Formula:C16H21N3·HClPurezza:99.54% - 99.81%Colore e forma:White SolidPeso molecolare:291.82PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C31H30FN5O4Purezza:97.19% - 99.56%Colore e forma:SolidPeso molecolare:555.62-Bromo-6-methoxynaphthalene
CAS:2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formula:C11H9BrOPurezza:98.51%Colore e forma:White To Off-White PowderPeso molecolare:237.09Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Formula:C23H29ClFN3O4Purezza:99.77%Colore e forma:White To Slightly Biege Powder SolidPeso molecolare:465.95Ref: TM-T1291
5mg47,00€10mg59,00€25mg77,00€50mg99,00€100mg135,00€200mg235,00€500mg394,00€1mL*10mM (DMSO)55,00€Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Formula:C19H21N·HClPurezza:98.54% - 99.98%Colore e forma:SolidPeso molecolare:299.84Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Purezza:97.76%Colore e forma:SoildNylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purezza:99.35%Colore e forma:SolidPeso molecolare:335.87Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Formula:C56H82N16O19S2Purezza:98.50% - 99.69%Colore e forma:SolidPeso molecolare:1347.5Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Purezza:SDS-PAGE:95% SEC-HPLC:98.90%Colore e forma:LiquidPeso molecolare:146.43 kDaLafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurezza:98.55%Colore e forma:Yellowish White Crystalline PowderPeso molecolare:431.55Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Formula:C18H26ClN3O3Purezza:99.99% - >99.99%Colore e forma:SolidPeso molecolare:367.87Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formula:C17H28ClNO2Purezza:97.32% - 99.86%Colore e forma:White Crystalline PowderPeso molecolare:313.86Erenumab
CAS:Erenumab: human antibody blocking CGRP receptors to prevent migraines.Purezza:99.43% (SEC-HPLC) - > 95%Colore e forma:LiquidPeso molecolare:146.2 kDaTalastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurezza:99.44% - 99.84%Colore e forma:SolidPeso molecolare:307.39Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormula:C10H13NO4Purezza:98.95% - 99.86%Colore e forma:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecolare:211.21Desipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formula:C18H23ClN2Purezza:99.58% - 99.96%Colore e forma:White To Off-White PowderPeso molecolare:302.842PF-5190457
CAS:PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).Formula:C29H32N6OSPurezza:99.34%Colore e forma:SolidPeso molecolare:512.67Ref: TM-T16508
1mg37,00€2mg52,00€5mg79,00€10mg126,00€25mg274,00€50mgPrezzo su richiesta1mL*10mM (DMSO)89,00€Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formula:C17H19ClF3NOPurezza:99.6% - 99.98%Colore e forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecolare:345.787Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purezza:99.16% - 99.86%Colore e forma:SolidPeso molecolare:266.55Sergliflozin A
CAS:Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.Formula:C20H24O7Purezza:99.71%Colore e forma:SolidPeso molecolare:376.4Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurezza:98% - 99.91%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:463.79Indacaterol maleate
CAS:Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.Formula:C28H32N2O7Purezza:99.03% - 99.67%Colore e forma:SolidPeso molecolare:508.56ML-180
CAS:ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .Formula:C20H25ClN4O2Purezza:99.74%Colore e forma:SolidPeso molecolare:388.89Ref: TM-T12075
1mg35,00€2mg52,00€5mg77,00€10mg114,00€25mg207,00€50mg363,00€100mg550,00€1mL*10mM (DMSO)86,00€CD80-IN-3
CAS:CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).Formula:C17H10FN3O3Purezza:98.08%Colore e forma:SolidPeso molecolare:323.28Ref: TM-T10722
1mg80,00€5mg187,00€10mg305,00€25mg494,00€50mg682,00€100mg847,00€1mL*10mM (DMSO)207,00€CYM 50769
CAS:CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).Formula:C24H17ClN2O3Purezza:98% - 99.08%Colore e forma:SolidPeso molecolare:416.86Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormula:C19H25F3N2O6Purezza:99.92% - 99.94%Colore e forma:White Crystalline PowderPeso molecolare:434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purezza:99.282% - 99.76%Colore e forma:Colorless To Pink SolidPeso molecolare:495.53Ref: TM-T1504
5mg35,00€10mg52,00€25mg78,00€50mg96,00€100mg104,00€200mg133,00€1500mg267,00€1mL*10mM (DMSO)38,00€Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Formula:C11H17NO3·5H2O4SPurezza:98.53% - 99.74%Colore e forma:SolidPeso molecolare:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurezza:99.77% - >99.99%Colore e forma:White To Slightly Yellowish Crystalline SolidPeso molecolare:341.88Urapidil hydrochloride
CAS:Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Formula:C20H29N5O3·HClPurezza:99.58%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:423.94Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formula:C21H25N3O2SPurezza:99.14% - 99.63%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:383.51JNJ-18038683
CAS:JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Formula:C26H28ClN3O7Purezza:97.29%Colore e forma:SolidPeso molecolare:529.97Ref: TM-T11720
2mg35,00€5mg50,00€10mg90,00€25mg170,00€50mg259,00€100mg383,00€200mg545,00€1mL*10mM (DMSO)55,00€PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Formula:C25H37Cl2N3O2Purezza:99.68%Colore e forma:SolidPeso molecolare:482.49Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Formula:C31H37N3O10SPurezza:99.39% - 99.48%Colore e forma:SolidPeso molecolare:643.71Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Formula:C24H28N2O3Purezza:99.60% - 99.97%Colore e forma:White Crystalline PowderPeso molecolare:392.49Ifenprodil
CAS:Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.Formula:C21H27NO2Purezza:99.58%Colore e forma:White Crystalline PowderPeso molecolare:325.44Ref: TM-T1186L
1mg73,00€5mg159,00€10mg230,00€25mg378,00€50mg540,00€100mg747,00€200mg1.026,00€1mL*10mM (DMSO)165,00€Granisetron hydrochloride
CAS:Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFormula:C18H25ClN4OPurezza:99.88% - 99.93%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:348.87Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purezza:99.98%Colore e forma:SoildPeso molecolare:231.65Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purezza:99.85%Colore e forma:SolidPeso molecolare:367.5Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Formula:C9H15ClNO5PPurezza:99.84%Colore e forma:SolidPeso molecolare:283.65NF-56-EJ40 hydrochloride
CAS:NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.Formula:C27H31Cl2N3O3Purezza:99.33%Colore e forma:SoildPeso molecolare:516.46Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurezza:98.20% - 99.88%Colore e forma:White Crystalline PowderPeso molecolare:341.43Fluoxetine
CAS:Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.Formula:C17H18F3NOPurezza:99.07% - 99.28%Colore e forma:SolidPeso molecolare:309.33Astressin acetate
Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the clonedFormula:C163H273N49O44Purezza:96.87%Colore e forma:SolidPeso molecolare:3623.21Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Formula:C19H23NO·HClPurezza:98.72%Colore e forma:SolidPeso molecolare:317.85Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurezza:99.76%Colore e forma:White PowderPeso molecolare:352.32Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Formula:C28H30N2O8Purezza:99.7% - >99.99%Colore e forma:PowderPeso molecolare:522.55Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurezza:99.86% - ≥95%Colore e forma:Yellowish Crystalline PowderPeso molecolare:312.43CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H18Cl2N4OPurezza:99.5%Colore e forma:SolidPeso molecolare:341.24Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Formula:C19H23Cl2N5OPurezza:99.5% - 99.52%Colore e forma:SolidPeso molecolare:408.33MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Formula:C24H26F3N3O4Purezza:99.98%Colore e forma:SolidPeso molecolare:477.48Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFormula:C17H19N3·HClPurezza:98% - 99.53%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:301.82Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.Formula:C22H29ClN2O2Purezza:99.98%Colore e forma:SolidPeso molecolare:388.93Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purezza:99.43% - 99.62%Colore e forma:Colourless Flake Crystalline SolidPeso molecolare:448.39YNT-185
CAS:YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,Formula:C33H37N5O5SPurezza:99.67%Colore e forma:SolidPeso molecolare:615.74Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formula:C26H35NO7Purezza:98.53% - 99.43%Colore e forma:CoaPeso molecolare:473.57KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Formula:C26H40N4O8Purezza:98.46%Colore e forma:SolidPeso molecolare:536.62Ref: TM-T15656
1mg109,00€2mg158,00€5mg260,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€1mL*10mM (DMSO)305,00€(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purezza:97.82%Colore e forma:SoildPeso molecolare:195.19Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formula:C14H15Cl2NSPurezza:99.85% - >99.99%Colore e forma:White PowderPeso molecolare:300.25Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formula:C16H21N3O2Purezza:99.69% - 99.91%Colore e forma:White Or Kind Of White PowderPeso molecolare:287.36Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purezza:97.59%Colore e forma:SolidPeso molecolare:298.29Ref: TM-T14148
1mg35,00€5mg66,00€10mg96,00€25mg168,00€50mg264,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)71,00€Phenothiazine
CAS:Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.Formula:C12H9NSPurezza:99.95%Colore e forma:Yellow Solid PelletsPeso molecolare:199.27Noradrenaline bitartrate
CAS:Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.Formula:C12H19NO10Purezza:99.53% - >99.99%Colore e forma:SolidPeso molecolare:337.28ESI-05
CAS:ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.Formula:C16H18O2SPurezza:97.22%Colore e forma:SolidPeso molecolare:274.38Timonacic
CAS:Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.Formula:C4H7NO2SPurezza:99.99%Colore e forma:SolidPeso molecolare:133.17Centanafadine hydrochloride
CAS:Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).Formula:C15H16ClNPurezza:99.65%Colore e forma:SolidPeso molecolare:245.75Ref: TM-T10758L
1mg59,00€5mg126,00€10mg202,00€25mg406,00€50mg653,00€100mg1.026,00€200mg1.378,00€500mg2.052,00€1mL*10mM (DMSO)140,00€Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormula:C10H17Cl2N3SPurezza:99.89%Colore e forma:Light Yellow SolidPeso molecolare:282.23Ref: TM-T14490
2mg35,00€5mg52,00€10mg80,00€25mg144,00€50mg225,00€100mg359,00€200mg532,00€1mL*10mM (DMSO)52,00€LCKLSL hydrochloride
LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.Formula:C30H58ClN7O8SPurezza:98.02% - 99.31%Colore e forma:SolidPeso molecolare:712.34(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Formula:C32H30F5N3O5Purezza:99.08%Colore e forma:SolidPeso molecolare:631.59Ref: TM-T11174
5mg52,00€10mg80,00€25mg144,00€50mg205,00€100mg324,00€200mg477,00€1mL*10mM (DMSO)73,00€Ezlopitant
CAS:Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.Formula:C31H38N2OPurezza:97.49%Colore e forma:SolidPeso molecolare:454.65Tetrahydrozoline
CAS:Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.Formula:C13H16N2Purezza:97.85% - 99.77%Colore e forma:SolidPeso molecolare:200.28RS102895 hydrochloride
CAS:RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).Formula:C21H22ClF3N2O2Purezza:98.95%Colore e forma:SolidPeso molecolare:426.86Filorexant
CAS:Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).Formula:C24H25FN4O2Purezza:98.88%Colore e forma:SolidPeso molecolare:420.48Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Formula:C13H20N2O2Purezza:99.87% - 99.93%Colore e forma:White Or Off White Crystalline PowderPeso molecolare:236.31Palonosetron hydrochloride
CAS:Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Formula:C19H24N2O·HClPurezza:99.84% - 99.92%Colore e forma:White SolidPeso molecolare:332.87Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purezza:99.79%Colore e forma:SolidPeso molecolare:353.29Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Formula:C16H26ClNO3Purezza:99.94% - ≥95%Colore e forma:SolidPeso molecolare:315.84Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormula:C21H22CL2N4OSPurezza:97.97% - 99.82%Colore e forma:SolidPeso molecolare:449.4Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Formula:C26H27N5O2Purezza:99.61%Colore e forma:Light Yellow SolidPeso molecolare:441.52Dopexamine hydrochloride
CAS:Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.Formula:C22H34Cl2N2O2Purezza:98.55%Colore e forma:SolidPeso molecolare:429.42Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Formula:C24H28ClN5O3Purezza:99.57% - 99.77%Colore e forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecolare:469.96Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurezza:99.94%Colore e forma:SolidPeso molecolare:217.65Azasetron hydrochloride
CAS:Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.Formula:C17H20ClN3O3·HClPurezza:99.50%Colore e forma:SolidPeso molecolare:386.27Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurezza:99.90%Colore e forma:SolidPeso molecolare:320.88Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Formula:C18H29ClN2O4Purezza:99.92% - >99.99%Colore e forma:White Or Slightly Off-White Crystalline Powder SolidPeso molecolare:372.89Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Formula:C19H21NSPurezza:99.93%Colore e forma:SolidPeso molecolare:295.44Linaclotide
CAS:Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.Formula:C59H79N15O21S6Purezza:97.93% - 98.71%Colore e forma:SolidPeso molecolare:1526.74Ref: TM-T11852
1mg49,00€5mg104,00€10mg187,00€25mg329,00€50mg490,00€100mg700,00€200mg938,00€1mL*10mM (DMSO)269,00€MP-A08
CAS:MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.Formula:C27H25N3O4S2Purezza:97.44%Colore e forma:SolidPeso molecolare:519.64Fenspiride hydrochloride
CAS:Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.Formula:C15H20N2O2·HClPurezza:99.64% - 99.92%Colore e forma:SolidPeso molecolare:296.79Leronlimab
CAS:Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.Purezza:SDS-PAGE:95.0%;SEC-HPLC:99.6%Colore e forma:LiquidPeso molecolare:146.66 kDaCetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purezza:99.4% - 99.97%Colore e forma:SolidPeso molecolare:461.81Olinciguat
CAS:Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.Formula:C21H16F5N7O3Purezza:99.33% - 99.71%Colore e forma:SolidPeso molecolare:509.39Ref: TM-T16383
1mg178,00€5mg454,00€10mg655,00€25mg1.026,00€50mg1.406,00€100mg1.863,00€1mL*10mM (DMSO)502,00€Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purezza:99.49%Colore e forma:SolidPeso molecolare:384.9EMPA
CAS:EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nMFormula:C23H26N4O4SPurezza:99.11%Colore e forma:SolidPeso molecolare:454.54Ref: TM-T11186
1mg49,00€2mg69,00€5mg92,00€10mg142,00€25mg250,00€50mg375,00€100mg563,00€200mg795,00€1mL*10mM (DMSO)104,00€
