Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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Tofogliflozin (hydrate)
CAS:<p>Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).</p>Formula:C22H28O7Purezza:97.03% - 98.78%Colore e forma:SolidPeso molecolare:404.45MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurezza:99.73%Colore e forma:SolidPeso molecolare:465.52RTICBM-189
CAS:<p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>Formula:C15H14Cl2N2OPurezza:99.96%Colore e forma:SolidPeso molecolare:309.19Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Formula:C14H16N2·HClPurezza:99.74%Colore e forma:SolidPeso molecolare:248.75Bromodiphenhydramine hydrochloride
CAS:<p>Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.</p>Formula:C17H21BrClNOPurezza:97.29%Colore e forma:SolidPeso molecolare:370.71SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurezza:99.61%Colore e forma:SolidPeso molecolare:266.3Triptorelin acetate(57773-63-4 free base)
CAS:<p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>Formula:C66H86N18O15Purezza:99.90%Colore e forma:White PowderPeso molecolare:1371.53SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Formula:C16H20N2O2·HClPurezza:99.64%Colore e forma:SolidPeso molecolare:308.81Myristicin
CAS:<p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>Formula:C11H12O3Purezza:99.828%Colore e forma:LiquidPeso molecolare:192.21Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formula:C40H42ClN5O7Purezza:97.94% - 98.4%Colore e forma:SolidPeso molecolare:740.24Quipazine maleate
CAS:<p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>Formula:C17H19N3O4Colore e forma:SolidPeso molecolare:329.36Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purezza:98% - 99.494%Colore e forma:SolidPeso molecolare:1706.9Naftopidil hydrochloride
CAS:<p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>Formula:C24H29ClN2O3Purezza:99.5%Colore e forma:SolidPeso molecolare:428.95T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Formula:C26H28O11Purezza:99.78%Colore e forma:SolidPeso molecolare:516.49AP1189 acetate
CAS:<p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>Formula:C16H18N6O4Purezza:99.95%Colore e forma:SolidPeso molecolare:358.35R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purezza:99.52%Colore e forma:SolidPeso molecolare:865.93GR 94800 acetate
<p>GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.</p>Formula:C51H65N9O10Purezza:97.86%Colore e forma:SolidPeso molecolare:964.12Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Formula:C21H28N2O2·2ClHPurezza:99.73%Colore e forma:SolidPeso molecolare:413.39ACTH 11-24 acetate(4237-93-8 free base)
CAS:<p>ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.</p>Formula:C79H138N24O18Purezza:>99.99%Colore e forma:SolidPeso molecolare:1712.12Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Formula:C19H20N2Purezza:99.3% - ≥98%Colore e forma:SolidPeso molecolare:276.38[Lys8, Lys9]-Neurotensin (8-13) acetate
<p>[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2</p>Formula:C40H68N8O10Purezza:99.31%Colore e forma:SolidPeso molecolare:821.02PD-168077 maleate
CAS:<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Formula:C24H26N4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:450.49β-CGRP, human acetate
<p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>Formula:C164H271N51O50S3Purezza:99.35%Colore e forma:SolidPeso molecolare:3853.46Bucindolol hydrochloride
CAS:<p>Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.</p>Formula:C22H26ClN3O2Colore e forma:SolidPeso molecolare:399.91Ornipressin Acetate(3397-23-7,free)
CAS:<p>Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent.</p>Formula:C47H67N13O124S2Purezza:>99.99%Colore e forma:SolidPeso molecolare:1102.25S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formula:C31H34N2O4Purezza:99.77%Colore e forma:SolidPeso molecolare:498.61Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Formula:C32H41N5O10Purezza:97.69%Colore e forma:SolidPeso molecolare:655.7Darusentan
CAS:Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteriesFormula:C22H22N2O6Purezza:98.72%Colore e forma:SolidPeso molecolare:410.43L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formula:C18H22Cl4N4Purezza:97.52%Colore e forma:SolidPeso molecolare:436.21Levalbuterol tartrate
CAS:<p>Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.</p>Formula:C17H27NO9Purezza:98.97% - 99.79%Colore e forma:SolidPeso molecolare:389.39ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Formula:C17H11N3O6SPurezza:97.74%Colore e forma:SolidPeso molecolare:385.35Asapiprant
CAS:<p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>Formula:C24H27N3O7SPurezza:99.64%Colore e forma:SolidPeso molecolare:501.55Olcegepant
CAS:<p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>Formula:C38H47Br2N9O5Purezza:96.08% - 97.24%Colore e forma:SolidPeso molecolare:869.65Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formula:C24H30N2O2SPurezza:99.9% - 99.92%Colore e forma:SolidPeso molecolare:410.57Sigma-LIGAND-1 hydrochloride
CAS:<p>Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.</p>Formula:C27H34ClNO4Colore e forma:SolidPeso molecolare:472.02Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formula:C18H15BrF2N4O2Purezza:98.42% - 99.88%Colore e forma:SolidPeso molecolare:437.24GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Formula:C20H20N4O4Purezza:99.92%Colore e forma:SolidPeso molecolare:380.4Netupitant
CAS:<p>Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).</p>Formula:C30H32F6N4OPurezza:99.43%Colore e forma:SolidPeso molecolare:578.59NPS2390
CAS:<p>NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)</p>Formula:C19H21N3OPurezza:97.13%Colore e forma:SolidPeso molecolare:307.39Hypidone hydrochloride
CAS:<p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>Formula:C18H23ClN2O2Purezza:99.82% - 99.93%Colore e forma:SolidPeso molecolare:334.84Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purezza:98.94% - 99.95%Colore e forma:SolidPeso molecolare:373.46Acrivastine
CAS:<p>Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.</p>Formula:C22H24N2O2Purezza:99.73% - >99.99%Colore e forma:SolidPeso molecolare:348.44Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Formula:C17H25N7O4Purezza:99.74%Colore e forma:SolidPeso molecolare:391.42ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purezza:99.12%Colore e forma:SolidPeso molecolare:307.139LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurezza:99.8%Colore e forma:SolidPeso molecolare:430.94Enprofylline
CAS:<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formula:C8H10N4O2Purezza:98.37%Colore e forma:SolidPeso molecolare:194.19Zacopride hydrochloride
CAS:<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Formula:C15H20ClN3O2·HClPurezza:98.32%Colore e forma:SolidPeso molecolare:346.26Cinaciguat
CAS:<p>Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.</p>Formula:C36H39NO5Purezza:98% - 99.18%Colore e forma:SolidPeso molecolare:565.7Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonistFormula:C37H48F6N8O11Purezza:98.54%Colore e forma:SolidPeso molecolare:894.81TRAP-6
CAS:<p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>Formula:C34H56N10O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:748.875-HT1A modulator 2 hydrochloride
CAS:<p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>Formula:C11H16ClNOPurezza:98.5%Colore e forma:SolidPeso molecolare:213.7JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Formula:C14H16ClN3OPurezza:99.83% - 99.96%Colore e forma:SolidPeso molecolare:277.75Haloperidol decanoate
CAS:<p>Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.</p>Formula:C31H41ClFNO3Purezza:99.57% - 99.72%Colore e forma:SolidPeso molecolare:530.11Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:356.44Verucerfont
CAS:<p>Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .</p>Formula:C22H26N6O2Purezza:99.90%Colore e forma:SolidPeso molecolare:406.48Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Formula:C172H265N43O51Purezza:97.65% - 99.04%Colore e forma:SolidPeso molecolare:3751.25PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Formula:C59H80N14O13Purezza:95.3%Colore e forma:SolidPeso molecolare:1193.35Xanthotoxol
CAS:<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Formula:C11H6O4Purezza:99.97%Colore e forma:SolidPeso molecolare:202.16Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurezza:98.64% - 99.97%Colore e forma:SolidPeso molecolare:623.63SBI-115
CAS:<p>SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5</p>Formula:C14H13ClN2O4SPurezza:99.53% - 99.78%Colore e forma:SolidPeso molecolare:340.78Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Formula:C13H16N2O2Purezza:98% - 99.89%Colore e forma:Pale Yellow Leaflets From Benzene SolidPeso molecolare:232.28Taprenepag
CAS:Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).Formula:C24H22N4O5SPurezza:98.89% - 99.15%Colore e forma:SolidPeso molecolare:478.52Benzotript
CAS:<p>Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.</p>Formula:C18H15ClN2O3Purezza:97.82%Colore e forma:SolidPeso molecolare:342.776Obestatin (rat) acetate
<p>Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).</p>Formula:C114H174N34O31Purezza:99.05%Colore e forma:SolidPeso molecolare:2516.81[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Formula:C46H62F3N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1018.05MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurezza:97.69% - 98.15%Colore e forma:SolidPeso molecolare:447.51TCS-OX2-29
CAS:TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formula:C23H31N3O3Purezza:99.81%Colore e forma:SolidPeso molecolare:397.51Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Formula:C19H17ClFN5SPurezza:97.79% - 98.07%Colore e forma:SolidPeso molecolare:401.89Serotonin
CAS:<p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>Formula:C10H12N2OPurezza:97.47% - 99.92%Colore e forma:SolidPeso molecolare:176.22RS-127445 hydrochloride
CAS:<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Formula:C17H17ClFN3Purezza:99.48%Colore e forma:SolidPeso molecolare:317.79ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purezza:98.24%Colore e forma:SolidPeso molecolare:3140.5Abaperidone Hydrochloride
CAS:<p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>Formula:C25H26ClFN2O5Colore e forma:SolidPeso molecolare:488.94Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purezza:>99.99%Colore e forma:SolidPeso molecolare:1672.92ESI-09
CAS:ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Formula:C16H15ClN4O2Purezza:97.24% - 99.57%Colore e forma:SolidPeso molecolare:330.77Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formula:C41H52N4O4SPurezza:97.87%Colore e forma:SolidPeso molecolare:696.949-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Formula:C7H9N5Purezza:99.35% - 99.41%Colore e forma:SolidPeso molecolare:163.18Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formula:C32H34N4O5SPurezza:98.26% - 99.43%Colore e forma:SolidPeso molecolare:586.7TS-011
CAS:<p>N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.</p>Formula:C11H14ClN3O2Purezza:99.48%Colore e forma:SolidPeso molecolare:255.7Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Formula:C19H20N2O3Purezza:99.84% - 99.86%Colore e forma:White PowderPeso molecolare:324.37Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purezza:99.12%Colore e forma:SolidPeso molecolare:184.067Spexin acetate(1370290-58-6 free base)
<p>Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.</p>Formula:C76H117N19O22SPurezza:95.43%Colore e forma:SolidPeso molecolare:1680.94Metadoxine
CAS:<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Formula:C8H11NO3·C5H7NO3Purezza:99.19%Colore e forma:Off-White PowderPeso molecolare:298.292-ATHBI
CAS:<p>2-ATHBI is a S1P lyase inhibitor.</p>Formula:C9H14N2O5Purezza:95.00%Colore e forma:SolidPeso molecolare:230.22Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Formula:C21H35ClN2O5Purezza:99.33%Colore e forma:SolidPeso molecolare:430.97S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Formula:C24H26FN3O2Colore e forma:SolidPeso molecolare:407.48BAR501
CAS:<p>BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。</p>Formula:C26H46O3Purezza:99.29% - 99.68%Colore e forma:SolidPeso molecolare:406.64BML-190
CAS:<p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。</p>Formula:C23H23ClN2O4Purezza:97.70%Colore e forma:SolidPeso molecolare:426.89PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Formula:C23H31ClN2O2Purezza:99.71%Colore e forma:SolidPeso molecolare:402.96VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Formula:C15H19N5Purezza:99.44% - 99.57%Colore e forma:SolidPeso molecolare:269.34Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Formula:C23H31ClN4O2SPurezza:99.37%Colore e forma:White SolidPeso molecolare:463Exendin-4 acetate
CAS:<p>Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).</p>Formula:C186H286N50O62SPurezza:98.48% - 99.78%Colore e forma:SolidPeso molecolare:4247(±)-Ibipinabant
CAS:<p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>Formula:C23H20Cl2N4O2SPurezza:99.28% - 99.83%Colore e forma:SolidPeso molecolare:487.4Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:1024.18Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formula:C23H30N4O2SPurezza:99.23%Colore e forma:White PowderPeso molecolare:426.57Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Formula:C15H24ClNO3Purezza:99.46%Colore e forma:SolidPeso molecolare:301.81Men 10376 TFA(135306-85-3,free)
<p>Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4</p>Formula:C59H69F3N12O12Purezza:99.22%Colore e forma:SolidPeso molecolare:1195.25TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formula:C27H26N4O2SPurezza:99.35% - 99.52%Colore e forma:SolidPeso molecolare:470.59
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