Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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Melanotan I
CAS:<p>Melanotan I is a non-specific melanocortin receptor (MCR) agonist, an α-melanocyte-stimulating hormone (α-MSH) analog, which is injected subcutaneously to</p>Formula:C78H111N21O19Purezza:>99.99%Colore e forma:SolidPeso molecolare:1646.85Ambrisentan
CAS:<p>Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.</p>Formula:C22H22N2O4Purezza:99.65% - 99.86%Colore e forma:SolidPeso molecolare:378.42Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Formula:C17H26N4OPurezza:97.1% - 97.76%Colore e forma:OilPeso molecolare:302.41Vazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purezza:98.93%Colore e forma:SolidPeso molecolare:675.3LUN42518 HCl 47142-51-8(free base)
<p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>Formula:C17H20ClN3OPurezza:99.96%Colore e forma:SolidPeso molecolare:317.81Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Formula:C17H20BrNOColore e forma:SolidPeso molecolare:334.25Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Formula:C17H20N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:316.42Dobutamine
CAS:<p>Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.</p>Formula:C18H23NO3Colore e forma:SolidPeso molecolare:301.38Cimetidine hydrochloride
CAS:<p>Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.</p>Formula:C10H17ClN6SColore e forma:SolidPeso molecolare:288.8Montelukast dicyclohexylamine
CAS:<p>Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.</p>Formula:C47H59ClN2O3SColore e forma:SolidPeso molecolare:767.5Men 10376 TFA(135306-85-3,free)
<p>Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4</p>Formula:C59H69F3N12O12Purezza:99.22%Colore e forma:SolidPeso molecolare:1195.25Lidamidine Hydrochloride
CAS:Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formula:C11H17ClN4OColore e forma:SolidPeso molecolare:256.73Sarpogrelate
CAS:<p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>Formula:C24H31NO6Colore e forma:SolidPeso molecolare:429.51Droxidopa hydrochloride
CAS:<p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>Formula:C9H12ClNO5Colore e forma:SolidPeso molecolare:249.65Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormula:C21H32O2Purezza:99.59% - 99.92%Colore e forma:SolidPeso molecolare:316.48Temanogrel
CAS:<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Formula:C24H28N4O4Purezza:99.24%Colore e forma:SolidPeso molecolare:436.5Phentolamine hydrochloride
CAS:<p>Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].</p>Formula:C17H20ClN3OColore e forma:SolidPeso molecolare:317.82AdipoRon hydrochloride
CAS:<p>AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).</p>Formula:C27H29ClN2O3Colore e forma:SolidPeso molecolare:464.99ENMD-1068 HBr
CAS:<p>ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.</p>Formula:C15H30BrN3O2Colore e forma:SolidPeso molecolare:364.32Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Formula:C11H16N2O3Purezza:98%Colore e forma:SolidPeso molecolare:224.26Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Formula:C14H21Cl2F3N6O3Colore e forma:SolidPeso molecolare:449.26Cinaciguat hydrochloride
CAS:<p>Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.</p>Formula:C36H40ClNO5Colore e forma:SolidPeso molecolare:602.17Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Formula:C21H21FO5SPurezza:99.38% - 99.70%Colore e forma:SolidPeso molecolare:404.45Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Formula:C17H18ClN4OColore e forma:SolidPeso molecolare:329.11691GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Formula:C22H21ClN4O4Purezza:99.04%Colore e forma:SolidPeso molecolare:440.88Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Formula:C15H20N8O6Purezza:98%Colore e forma:SolidPeso molecolare:408.37Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Formula:C18H22N2Colore e forma:SolidPeso molecolare:266.38Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Colore e forma:SolidPeso molecolare:349.86BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Formula:C25H28Cl2N2OColore e forma:SolidPeso molecolare:443.41Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurezza:99.99%Colore e forma:Crystalline SolidPeso molecolare:327.90Ajmalicine hydrochloride
CAS:<p>Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.</p>Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89PF3274167
CAS:PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Formula:C19H19ClFN5O3Purezza:99.67% - 99.88%Colore e forma:SolidPeso molecolare:419.84Betazole
CAS:<p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>Formula:C5H9N3Colore e forma:SolidPeso molecolare:111.15Guanabenz hydrochloride
CAS:Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formula:C8H9Cl3N4Purezza:99.45%Colore e forma:SolidPeso molecolare:267.54Siponimod
CAS:<p>Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.</p>Formula:C29H35F3N2O3Purezza:97.08% - 99.40%Colore e forma:SolidPeso molecolare:516.59CYM-5541
CAS:<p>CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.</p>Formula:C19H28N2O2Purezza:99.74% - 99.76%Colore e forma:SolidPeso molecolare:316.44Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Formula:C20H22ClF3N4OColore e forma:SolidPeso molecolare:426.87Talnetant
CAS:<p>Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.</p>Formula:C25H22N2O2Purezza:97.88%Colore e forma:SolidPeso molecolare:382.45Ganirelix Acetate
CAS:<p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>Formula:C82H117ClN18O15Purezza:96.05%Colore e forma:SolidPeso molecolare:1630.4Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Formula:C129H216N42O42Purezza:98.12%Colore e forma:SolidPeso molecolare:3027.35L-765314
CAS:<p>L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.</p>Formula:C27H34N6O5Purezza:99.73%Colore e forma:SolidPeso molecolare:522.6Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Formula:C19H20N2O3Purezza:99.84% - 99.86%Colore e forma:White PowderPeso molecolare:324.37ESI-09
CAS:ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Formula:C16H15ClN4O2Purezza:97.24% - 99.57%Colore e forma:SolidPeso molecolare:330.77Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purezza:>99.99%Colore e forma:SolidPeso molecolare:1672.92CCG-50014
CAS:<p>CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.</p>Formula:C16H13FN2O2SPurezza:98.53%Colore e forma:SolidPeso molecolare:316.35Xanthotoxol
CAS:<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Formula:C11H6O4Purezza:99.97%Colore e forma:SolidPeso molecolare:202.16TRAP-6
CAS:<p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>Formula:C34H56N10O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:748.87RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Formula:C25H28ClN3O2Purezza:99.74%Colore e forma:SolidPeso molecolare:437.96Diphenhydramine
CAS:<p>Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.</p>Formula:C17H21NOPurezza:98.07%Colore e forma:SolidPeso molecolare:255.35SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Formula:C21H19ClN4O2Purezza:99.75% - ≥98%Colore e forma:SolidPeso molecolare:394.85Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Formula:C22H25ClN2OSPurezza:98.9% - 99.82%Colore e forma:SolidPeso molecolare:400.961-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formula:C6H9N3O2Purezza:99.29%Colore e forma:SolidPeso molecolare:155.15Pimavanserin tartrate
CAS:<p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>Formula:C50H68F2N6O4·C4H6O6Purezza:99.24% - 99.98%Colore e forma:SolidPeso molecolare:1005.2RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Formula:C17H16FN3Purezza:99.32%Colore e forma:SolidPeso molecolare:281.33Ocaperidone
CAS:<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Formula:C24H25FN4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:420.48Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41Ebastine
CAS:<p>Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.</p>Formula:C32H39NO2Purezza:99.65% - 99.93%Colore e forma:White To Off-White PowderPeso molecolare:469.66Pasireotide Acetate
CAS:<p>The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.</p>Formula:C60H70N10O11Purezza:98.64% - 99.92%Colore e forma:SolidPeso molecolare:1107.269-FLUORENOL
CAS:<p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>Formula:C13H10OPurezza:99.98%Colore e forma:Off-White Crystalline PowderPeso molecolare:182.22Ozanimod
CAS:<p>Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.</p>Formula:C23H24N4O3Purezza:98.68% - 99.58%Colore e forma:SolidPeso molecolare:404.46Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formula:C17H25N3O2S·C4H6O5Purezza:99.95%Colore e forma:Pale Yellow SolidPeso molecolare:469.555'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purezza:98.95% - ≥95%Colore e forma:PowderPeso molecolare:308.29Cetrorelix diacetate
CAS:<p>Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.</p>Formula:C74H100ClN17O18Purezza:98.38%Colore e forma:SolidPeso molecolare:1551.17Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purezza:98.97%Colore e forma:SolidPeso molecolare:544.73Adenosine receptor antagonist 4
CAS:<p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>Formula:C10H13N3Purezza:99.63% - 99.65%Colore e forma:Off-White PowderPeso molecolare:175.23Alizapride hydrochloride
CAS:<p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>Formula:C16H21N5O2·HClPurezza:99.35% - 99.48%Colore e forma:CoaPeso molecolare:351.83CYM2503
CAS:<p>CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.</p>Formula:C45H55N5O7Purezza:97.04%Colore e forma:SolidPeso molecolare:777.95SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurezza:98.94%Colore e forma:SolidPeso molecolare:446.35Glucagon (19-29), human acetate
<p>Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.</p>Formula:C63H93N15O20SPurezza:98.11%Colore e forma:SolidPeso molecolare:1412.57HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Formula:C27H33F3N4O9Purezza:99.51%Colore e forma:SolidPeso molecolare:614.57Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Formula:C27H29N3O2Purezza:98.98% - 99.12%Colore e forma:SolidPeso molecolare:427.54Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purezza:99.11%Colore e forma:SolidPeso molecolare:306.12Etrasimod
CAS:<p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>Formula:C26H26F3NO3Purezza:98.52% - 99.73%Colore e forma:SolidPeso molecolare:457.48CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Formula:C58H69F3N12O16S2Purezza:99.7%Colore e forma:SolidPeso molecolare:1311.36Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Formula:C25H34FN3O2Purezza:97.84% - 99.69%Colore e forma:Pale Yellow To Pale Orange SolidPeso molecolare:427.55JNJ-10229570
CAS:<p>JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland</p>Formula:C22H19N3O2SPurezza:98.41%Colore e forma:SolidPeso molecolare:389.47NGB 2904
CAS:<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Formula:C28H29Cl2N3OPurezza:98.79%Colore e forma:SolidPeso molecolare:494.46Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Formula:C21H25ClN2O3Purezza:99.75%Colore e forma:SolidPeso molecolare:388.89Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Formula:C18H19N3O·HClPurezza:99.78%Colore e forma:White PowderPeso molecolare:329.82Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Formula:C28H42F2N2O12S2Purezza:99.98%Colore e forma:SolidPeso molecolare:700.77β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurezza:99.64%Colore e forma:SolidPeso molecolare:2720.97L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Formula:C18H20Cl2N4Purezza:97.36%Colore e forma:SolidPeso molecolare:363.28Rimegepant
CAS:<p>View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.</p>Formula:C28H28F2N6O3Purezza:99.1% - 99.99%Colore e forma:SolidPeso molecolare:534.56Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Formula:C19H16F2N8O2Purezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:426.38Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Formula:C40H55N7O11SPurezza:99.84% - >99.99%Colore e forma:White PowderPeso molecolare:841.97Terutroban
CAS:<p>Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.</p>Formula:C20H22ClNO4SPurezza:99.53%Colore e forma:SolidPeso molecolare:407.91Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Formula:C19H26ClNOSPurezza:99.53% - 99.56%Colore e forma:Almost White To White Crystalline PowderPeso molecolare:351.93PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formula:C21H29Cl2N3O4SPurezza:98.5%Colore e forma:SolidPeso molecolare:490.44Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Formula:C25H26Cl3N7OPurezza:99.79% - ≥95%Colore e forma:SolidPeso molecolare:546.88Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Formula:C21H30N4O4Purezza:99.52%Colore e forma:SolidPeso molecolare:402.49Bombesin acetate(31362-50-2 free base)
CAS:<p>Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).</p>Formula:C73H114N24O20SPurezza:98.44%Colore e forma:SolidPeso molecolare:1679.92CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purezza:99.08% - 99.76%Colore e forma:SolidPeso molecolare:751.67Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Formula:C19H25NOSPurezza:98.08% - 99.59%Colore e forma:SolidPeso molecolare:315.47ICI 118,551 hydrochloride
CAS:<p>ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3</p>Formula:C17H28ClNO2Purezza:99.296% - 99.76%Colore e forma:SolidPeso molecolare:313.86A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurezza:99.94%Colore e forma:SolidPeso molecolare:310.45Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Formula:C28H37N3O3Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:463.61ML 154
CAS:<p>ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.</p>Formula:C29H26BrN2PSPurezza:99.53%Colore e forma:SolidPeso molecolare:545.47MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Formula:C8H11ClN4·HClPurezza:99.88%Colore e forma:SolidPeso molecolare:235.12Melitracen
CAS:<p>Melitracen is a tricyclic antidepressant.</p>Formula:C21H25NColore e forma:SolidPeso molecolare:291.43Ipsapirone hydrochloride
CAS:<p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>Formula:C19H24ClN5O3SColore e forma:SolidPeso molecolare:437.94
