Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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DOPEXAMINE
CAS:<p>Dopexamine is a dopaminergic agonist</p>Formula:C22H32N2O2Purezza:99.42%Colore e forma:SolidPeso molecolare:356.5Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurezza:99.04%Colore e forma:SolidPeso molecolare:436.95Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Formula:C19H23ClN2Colore e forma:SolidPeso molecolare:314.852Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formula:C4H3F7OPurezza:98%Colore e forma:Less Oil Colorless OilPeso molecolare:200.05RS 100329
CAS:<p>RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).</p>Formula:C20H25F3N4O3Colore e forma:SolidPeso molecolare:426.43Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Formula:C68H90N18O14Purezza:99.92%Colore e forma:SolidPeso molecolare:1383.55Ajmalicine hydrochloride
CAS:<p>Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.</p>Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89BMY-25368
CAS:<p>BMY-25368 is a long-acting antagonist of the H2-receptor.</p>Formula:C19H25N3O3Colore e forma:SolidPeso molecolare:343.42Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Formula:C20H26N2O7SPurezza:99.86% - 99.9%Colore e forma:SolidPeso molecolare:438.49MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurezza:97.69% - 98.15%Colore e forma:SolidPeso molecolare:447.51GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formula:C25H29N5OPurezza:99.2%Colore e forma:SolidPeso molecolare:415.53ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurezza:97.74%Colore e forma:SolidPeso molecolare:527.59[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Formula:C46H62F3N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1018.05Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Formula:C17H18ClN4OColore e forma:SolidPeso molecolare:329.11691[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purezza:97.68%Colore e forma:SolidPeso molecolare:1576.91Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Formula:C23H21F7N4O3Purezza:98% - 99.68%Colore e forma:Off-White To Light Yellow Cyrstalline SolidPeso molecolare:534.43HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Formula:C24H23ClN4O3Purezza:95.73%Colore e forma:SolidPeso molecolare:450.92SB756050
CAS:<p>SB756050 is a specific TGR5 agonist.</p>Formula:C21H28N2O8S2Purezza:98.78% - >99.99%Colore e forma:SolidPeso molecolare:500.59Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Formula:C20H20N2O3Purezza:99.27% - 99.80%Colore e forma:SolidPeso molecolare:336.38Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purezza:99.87% - 99.87%Colore e forma:Yellowish Liquid Liquid LiquidPeso molecolare:136.19Tripelennamine citrate
CAS:<p>Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.</p>Formula:C22H29N3O7Colore e forma:SolidPeso molecolare:447.4883-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Formula:C21H25Cl2NOPurezza:99.03%Colore e forma:SolidPeso molecolare:378.33SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Formula:C10H14ClN3·HClPurezza:99.89%Colore e forma:SolidPeso molecolare:248.15Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Formula:C172H265N43O51Purezza:97.65% - 99.04%Colore e forma:SolidPeso molecolare:3751.25Nonapeptide-1 acetate salt (158563-45-2 free base)
<p>Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)</p>Formula:C63H91N15O11SPurezza:98.26%Colore e forma:SolidPeso molecolare:1266.58Ramosetron
CAS:<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Formula:C17H17N3OPurezza:98.84%Colore e forma:SolidPeso molecolare:279.34LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurezza:99.8%Colore e forma:SolidPeso molecolare:430.94Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68YIL781 hydrochloride
CAS:<p>YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).</p>Formula:C24H29ClFN3O2Colore e forma:SolidPeso molecolare:445.96Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Formula:C25H25Cl2N7OPurezza:99.43%Colore e forma:SolidPeso molecolare:510.42Octreotide Acetate
CAS:<p>Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.</p>Formula:C51H70N10O12S2Purezza:99.03% - 99.87%Colore e forma:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidPeso molecolare:1079.3Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Formula:C28H33ClN2Colore e forma:SolidPeso molecolare:433.03NPS2390
CAS:<p>NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)</p>Formula:C19H21N3OPurezza:97.13%Colore e forma:SolidPeso molecolare:307.39Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Formula:C22H32ClN3O2Colore e forma:SolidPeso molecolare:405.96VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Formula:C13H15ClN4Purezza:99.66%Colore e forma:SolidPeso molecolare:262.74Tavapadon
CAS:<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Formula:C19H16F3N3O3Purezza:99.33% - 99.8%Colore e forma:SolidPeso molecolare:391.34GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Formula:C20H20N4O4Purezza:99.92%Colore e forma:SolidPeso molecolare:380.4γ-Mangostin
CAS:<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Formula:C23H24O6Purezza:98.55% - 99.08%Colore e forma:SolidPeso molecolare:396.43Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Formula:C37H56F7N6O16PPurezza:98% - 99.03%Colore e forma:SolidPeso molecolare:1004.83Atrasentan
CAS:Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.Formula:C29H38N2O6Purezza:97.65% - 99.08%Colore e forma:SolidPeso molecolare:510.62ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Formula:C29H29ClN4O2Purezza:99.88%Colore e forma:SolidPeso molecolare:501.02Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purezza:97.41%Colore e forma:SolidPeso molecolare:244.38Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Formula:C29H33FN2O4Purezza:98.77% - 99.93%Colore e forma:SolidPeso molecolare:492.58γ-L-Glutamyl-L-alanine
CAS:<p>γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).</p>Formula:C8H14N2O5Purezza:99.49%Colore e forma:SolidPeso molecolare:218.21Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Formula:C26H29N5O3SPurezza:99.49% - 99.843%Colore e forma:SolidPeso molecolare:491.61Darbufelone mesylate
CAS:Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formula:C19H28N2O5S2Purezza:96.81% - 99.92%Colore e forma:SolidPeso molecolare:428.57Darusentan
CAS:Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteriesFormula:C22H22N2O6Purezza:98.72%Colore e forma:SolidPeso molecolare:410.43Rimcazole dihydrochloride
CAS:<p>Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.</p>Formula:C21H28ClN3Purezza:99.63%Colore e forma:SolidPeso molecolare:357.92UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formula:C52H68N10O14S2Purezza:99.78%Colore e forma:SolidPeso molecolare:1121.29Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Formula:C16H22FNOPurezza:98.84%Colore e forma:SolidPeso molecolare:263.35Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurezza:97.25% - 97.36%Colore e forma:SolidPeso molecolare:321.34Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Formula:C18H22ClNOPurezza:99.44% - 99.85%Colore e forma:SolidPeso molecolare:303.83Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurezza:99.99%Colore e forma:Crystalline SolidPeso molecolare:327.90EST64454 Maleic acid salt
CAS:<p>EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.</p>Formula:C22H26F2N4O6Purezza:97.54%Colore e forma:SolidPeso molecolare:480.46Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Formula:C19H26N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:406.5Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C13H16N2·HClPurezza:99.94% - 99.94%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:236.74Vorapaxar sulfate
CAS:<p>Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.</p>Formula:C29H35FN2O8SPurezza:99.9% - >99.99%Colore e forma:SolidPeso molecolare:590.66cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Formula:C16H14O2Purezza:98.15%Colore e forma:SolidPeso molecolare:238.2812Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formula:C41H52N4O4SPurezza:97.87%Colore e forma:SolidPeso molecolare:696.94Naftopidil hydrochloride
CAS:<p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>Formula:C24H29ClN2O3Purezza:99.5%Colore e forma:SolidPeso molecolare:428.95Opromazine hydrochloride
CAS:<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Formula:C17H20Cl2N2OSPurezza:98.03%Colore e forma:SolidPeso molecolare:371.32Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purezza:98% - 99.494%Colore e forma:SolidPeso molecolare:1706.9AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formula:C17H21N5O2SPurezza:99.81%Colore e forma:SolidPeso molecolare:359.45Zafirlukast
CAS:<p>Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and anti-inflammatory effects. Cost-effective and quality-assured.</p>Formula:C31H33N3O6SPurezza:99% - 99.83%Colore e forma:SolidPeso molecolare:575.68Fenoprofen Calcium
CAS:<p>Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.</p>Formula:C30H26CaO6Purezza:99.24% - 99.66%Colore e forma:SolidPeso molecolare:522.6Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:1024.18Neuropeptide W-23(human)
CAS:<p>Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2.</p>Formula:C119H183N35O28SPurezza:98.5%Colore e forma:SolidPeso molecolare:2584.01FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Formula:C23H25Cl2N3OSPurezza:99.62%Colore e forma:SolidPeso molecolare:462.44RTICBM-189
CAS:<p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>Formula:C15H14Cl2N2OPurezza:99.96%Colore e forma:SolidPeso molecolare:309.19Gastrin I (1-14), human
CAS:Gastrin I (1-14), human: a short peptide from the hormone gastrin, which regulates gastric acid secretion.Formula:C79H100N16O27Purezza:98.19%Colore e forma:SolidPeso molecolare:1705.73Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Formula:C20H20FNO3S·HClPurezza:99.39% - 99.79%Colore e forma:SolidPeso molecolare:409.9AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Formula:C23H31ClN2O2Purezza:99.71%Colore e forma:SolidPeso molecolare:402.96Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Formula:C20H24N2OSColore e forma:SolidPeso molecolare:340.48Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Formula:C21H35ClN2O5Purezza:99.33%Colore e forma:SolidPeso molecolare:430.97Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Formula:C5H15ClNO4PPurezza:99.481% - 99.85%Colore e forma:SolidPeso molecolare:219.6Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:356.44Spexin acetate(1370290-58-6 free base)
<p>Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.</p>Formula:C76H117N19O22SPurezza:95.43%Colore e forma:SolidPeso molecolare:1680.94Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Formula:C40H67N7O10Purezza:99.95%Colore e forma:SolidPeso molecolare:805.9Dobutamine tartrate
CAS:<p>Dobutamine tartrate is a cardiotonic.</p>Formula:C22H29NO9Colore e forma:SolidPeso molecolare:451.472Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purezza:99.89%Colore e forma:SolidPeso molecolare:239.27Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Formula:C15H24ClNO2Purezza:99.79%Colore e forma:SolidPeso molecolare:285.81Fluorogestone acetate
CAS:<p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>Formula:C23H31FO5Purezza:99.47%Colore e forma:CoaPeso molecolare:406.49Enprofylline
CAS:<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formula:C8H10N4O2Purezza:98.37%Colore e forma:SolidPeso molecolare:194.19Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Formula:C25H37NO4Purezza:98% - >99.99%Colore e forma:Crystalline SolidPeso molecolare:415.57Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purezza:98.94% - 99.95%Colore e forma:SolidPeso molecolare:373.46Obestatin (rat) acetate
<p>Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).</p>Formula:C114H174N34O31Purezza:99.05%Colore e forma:SolidPeso molecolare:2516.81Sigma-LIGAND-1 hydrochloride
CAS:<p>Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.</p>Formula:C27H34ClNO4Colore e forma:SolidPeso molecolare:472.02Olcegepant
CAS:<p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>Formula:C38H47Br2N9O5Purezza:96.08% - 97.24%Colore e forma:SolidPeso molecolare:869.65Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurezza:98.64% - 99.97%Colore e forma:SolidPeso molecolare:623.63KB-5492 anhydrous
CAS:<p>KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.</p>Formula:C27H34N2O10Colore e forma:SolidPeso molecolare:546.57TRAP-6 amide acetate
<p>TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].</p>Formula:C36H61N11O10Purezza:98.55%Colore e forma:SolidPeso molecolare:807.94Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Formula:C14H22ClNO2Purezza:97.63%Colore e forma:SolidPeso molecolare:271.78Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formula:C32H29F5N3NaO5Purezza:99.71%Colore e forma:SolidPeso molecolare:653.57Quipazine maleate
CAS:<p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>Formula:C17H19N3O4Colore e forma:SolidPeso molecolare:329.36Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purezza:98.25%Colore e forma:SolidPeso molecolare:233.18Carbazochrome
CAS:<p>Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.</p>Formula:C10H12N4O3Purezza:98.36%Colore e forma:Nacarat Crystalline PowderPeso molecolare:236.23Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formula:C24H30N2O2SPurezza:99.9% - 99.92%Colore e forma:SolidPeso molecolare:410.57Fluoroclebopride
CAS:Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Formula:C20H23ClFN3O2Purezza:99.68% - 99.91%Colore e forma:SolidPeso molecolare:391.87Ornipressin Acetate(3397-23-7,free)
CAS:<p>Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent.</p>Formula:C47H67N13O124S2Purezza:>99.99%Colore e forma:SolidPeso molecolare:1102.25Cloprostenol sodium salt
CAS:<p>Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.</p>Formula:C22H28ClNaO6Purezza:97.17% - 98.47%Colore e forma:White To Almost White Hygroscopic PowderPeso molecolare:446.9
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