Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Formula:C23H28ClFN4O2Colore e forma:SolidPeso molecolare:446.95Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Formula:C21H21FO5SPurezza:99.38% - 99.70%Colore e forma:SolidPeso molecolare:404.45Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Formula:C20H24N2OSColore e forma:SolidPeso molecolare:340.48Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Formula:C17H18ClN4OColore e forma:SolidPeso molecolare:329.11691Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Formula:C9H10Cl2N4Colore e forma:SolidPeso molecolare:245.11Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Formula:C23H29NO5SPurezza:98%Colore e forma:SolidPeso molecolare:431.55GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Formula:C22H21ClN4O4Purezza:99.04%Colore e forma:SolidPeso molecolare:440.88S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Formula:C24H26FN3O2Colore e forma:SolidPeso molecolare:407.48PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47Xamoterol
CAS:<p>Xamoterol is a cardiac stimulant.</p>Formula:C16H25N3O5Colore e forma:SolidPeso molecolare:339.39T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Formula:C26H28O11Purezza:99.78%Colore e forma:SolidPeso molecolare:516.49Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Formula:C15H20N8O6Purezza:98%Colore e forma:SolidPeso molecolare:408.37Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Formula:C25H29ClF6N2O3Colore e forma:SolidPeso molecolare:554.95Siponimod hemifumarate
CAS:<p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>Formula:C62H74F6N4O10Colore e forma:SolidPeso molecolare:1149.282Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Formula:C18H22N2Colore e forma:SolidPeso molecolare:266.38Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Colore e forma:SolidPeso molecolare:349.86Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Formula:C15H24N2O4SColore e forma:SolidPeso molecolare:328.43KB-5492 anhydrous
CAS:<p>KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.</p>Formula:C27H34N2O10Colore e forma:SolidPeso molecolare:546.57Tripelennamine citrate
CAS:<p>Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.</p>Formula:C22H29N3O7Colore e forma:SolidPeso molecolare:447.488Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Formula:C19H23ClN2Colore e forma:SolidPeso molecolare:314.852RS 100329
CAS:<p>RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).</p>Formula:C20H25F3N4O3Colore e forma:SolidPeso molecolare:426.43Triprolidine
CAS:<p>Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.</p>Formula:C19H22N2Colore e forma:SolidPeso molecolare:278.39Ajmalicine hydrochloride
CAS:<p>Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.</p>Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formula:C24H29N3O3Colore e forma:SolidPeso molecolare:407.51PF3274167
CAS:PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Formula:C19H19ClFN5O3Purezza:99.67% - 99.88%Colore e forma:SolidPeso molecolare:419.84THIQ
CAS:<p>THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).</p>Formula:C33H41ClN6O2Purezza:98.93%Colore e forma:SolidPeso molecolare:589.17Guanabenz hydrochloride
CAS:<p>Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.</p>Formula:C8H9Cl3N4Purezza:99.45%Colore e forma:SolidPeso molecolare:267.54Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formula:C66H87N17O14Purezza:99.84%Colore e forma:SolidPeso molecolare:1342.5CYM-5541
CAS:<p>CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.</p>Formula:C19H28N2O2Purezza:99.74% - 99.76%Colore e forma:SolidPeso molecolare:316.44SLF1081851 TFA
CAS:<p>SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.</p>Formula:C23H34F3N3O3Colore e forma:SolidPeso molecolare:457.538Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Formula:C21H24Cl2FNO2Colore e forma:SolidPeso molecolare:412.33Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Formula:C20H22ClF3N4OColore e forma:SolidPeso molecolare:426.87Tesmilifene fumarate
CAS:<p>Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。</p>Formula:C23H29NO5Purezza:99.86%Colore e forma:SolidPeso molecolare:399.48Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Formula:C129H216N42O42Purezza:98.12%Colore e forma:SolidPeso molecolare:3027.35L-765314
CAS:<p>L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.</p>Formula:C27H34N6O5Purezza:99.73%Colore e forma:SolidPeso molecolare:522.6Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Formula:C19H20N2O3Purezza:99.84% - 99.86%Colore e forma:White PowderPeso molecolare:324.37ESI-09
CAS:<p>ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.</p>Formula:C16H15ClN4O2Purezza:97.24% - 99.57%Colore e forma:SolidPeso molecolare:330.77Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purezza:>99.99%Colore e forma:SolidPeso molecolare:1672.92TCS-OX2-29
CAS:<p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.</p>Formula:C23H31N3O3Purezza:99.81%Colore e forma:SolidPeso molecolare:397.51CCG-50014
CAS:<p>CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.</p>Formula:C16H13FN2O2SPurezza:98.53%Colore e forma:SolidPeso molecolare:316.35Xanthotoxol
CAS:<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Formula:C11H6O4Purezza:99.97%Colore e forma:SolidPeso molecolare:202.16TRAP-6
CAS:<p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>Formula:C34H56N10O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:748.87Netupitant
CAS:<p>Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).</p>Formula:C30H32F6N4OPurezza:99.43%Colore e forma:SolidPeso molecolare:578.59β-CGRP, human acetate
<p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>Formula:C164H271N51O50S3Purezza:99.35%Colore e forma:SolidPeso molecolare:3853.46Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formula:C40H42ClN5O7Purezza:97.94% - 98.4%Colore e forma:SolidPeso molecolare:740.24SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Formula:C21H19ClN4O2Purezza:99.75% - ≥98%Colore e forma:SolidPeso molecolare:394.85AnaMorelin hydrochloride
CAS:<p>AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).</p>Formula:C31H43ClN6O3Purezza:99.18% - ≥98%Colore e forma:SolidPeso molecolare:583.16Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Formula:C22H25ClN2OSPurezza:98.9% - 99.82%Colore e forma:SolidPeso molecolare:400.961-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formula:C6H9N3O2Purezza:99.29%Colore e forma:SolidPeso molecolare:155.15Gadolinium chloride
CAS:<p>Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist</p>Formula:Cl3GdPurezza:98%Colore e forma:White Crystalline SolidPeso molecolare:263.61Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41Propionylpromazine hydrochloride
CAS:<p>Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.</p>Formula:C20H25ClN2OSPurezza:99.17%Colore e forma:SolidPeso molecolare:376.94H2L 5765834
CAS:<p>H2L 5765834 is a lysophosphatidic acid receptors antagonist</p>Formula:C21H12N2O7Purezza:98.25% - 99.47%Colore e forma:SolidPeso molecolare:404.33Ebastine
CAS:<p>Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.</p>Formula:C32H39NO2Purezza:99.65% - 99.93%Colore e forma:White To Off-White PowderPeso molecolare:469.66Paltusotine
CAS:<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Formula:C27H22F2N4OPurezza:99.91%Colore e forma:SolidPeso molecolare:456.499-FLUORENOL
CAS:<p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>Formula:C13H10OPurezza:99.98%Colore e forma:Off-White Crystalline PowderPeso molecolare:182.22Pitolisant hydrochloride
CAS:<p>Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).</p>Formula:C17H27Cl2NOPurezza:99.72% - 99.91%Colore e forma:SolidPeso molecolare:332.31Ozanimod
CAS:<p>Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.</p>Formula:C23H24N4O3Purezza:98.68% - 99.58%Colore e forma:SolidPeso molecolare:404.465'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purezza:98.95% - ≥95%Colore e forma:PowderPeso molecolare:308.29ELA-14(human) acetate
<p>ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.</p>Formula:C77H123N25O19S2Purezza:97.2%Colore e forma:SolidPeso molecolare:1767.09Cetrorelix diacetate
CAS:<p>Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.</p>Formula:C74H100ClN17O18Purezza:98.38%Colore e forma:SolidPeso molecolare:1551.17Adenosine receptor antagonist 4
CAS:<p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>Formula:C10H13N3Purezza:99.63% - 99.65%Colore e forma:Off-White PowderPeso molecolare:175.23Dapiprazole Hydrochloride
CAS:<p>Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.</p>Formula:C19H28ClN5Purezza:99.75% - 99.93%Colore e forma:SolidPeso molecolare:361.92ONO-AE3-208
CAS:<p>ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.</p>Formula:C24H21FN2O3Purezza:98.04% - 99.55%Colore e forma:SolidPeso molecolare:404.43Harmine hydrochloride
CAS:<p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>Formula:C13H13ClN2OPurezza:99.61% - >99.99%Colore e forma:Yellow To Slightly Green Crystalline PowderPeso molecolare:248.71Alizapride hydrochloride
CAS:<p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>Formula:C16H21N5O2·HClPurezza:99.35% - 99.48%Colore e forma:CoaPeso molecolare:351.83CYM2503
CAS:<p>CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.</p>Formula:C45H55N5O7Purezza:97.04%Colore e forma:SolidPeso molecolare:777.95CYM50358
CAS:<p>N-(4-(aminomethyl)-2,6-dimethylphenyl)-5 is a potent, selective antagonist of the sphingosine-1-phosphate receptor 4 (S1P4).</p>Formula:C20H18Cl2N2O2Purezza:98.05% - 99.76%Colore e forma:SolidPeso molecolare:389.28SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurezza:98.94%Colore e forma:SolidPeso molecolare:446.35Glucagon (19-29), human acetate
<p>Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.</p>Formula:C63H93N15O20SPurezza:98.11%Colore e forma:SolidPeso molecolare:1412.57ABT-724
CAS:<p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>Formula:C17H19N5Purezza:99.73%Colore e forma:SolidPeso molecolare:293.37HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Formula:C27H33F3N4O9Purezza:99.51%Colore e forma:SolidPeso molecolare:614.57Tropisetron
CAS:<p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>Formula:C17H20N2O2Purezza:99.68%Colore e forma:White SolidPeso molecolare:284.35Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purezza:99.11%Colore e forma:SolidPeso molecolare:306.12Riociguat
CAS:<p>Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterial</p>Formula:C20H19FN8O2Purezza:99.28% - 99.95%Colore e forma:SolidPeso molecolare:422.42Etrasimod
CAS:<p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>Formula:C26H26F3NO3Purezza:98.52% - 99.73%Colore e forma:SolidPeso molecolare:457.48CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Formula:C58H69F3N12O16S2Purezza:99.7%Colore e forma:SolidPeso molecolare:1311.36Cinacalcet hydrochloride
CAS:<p>Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-</p>Formula:C22H23ClF3NPurezza:99.96% - >99.99%Colore e forma:Off-White To Tan SolidPeso molecolare:393.87Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Formula:C25H34FN3O2Purezza:97.84% - 99.69%Colore e forma:Pale Yellow To Pale Orange SolidPeso molecolare:427.55JNJ-10229570
CAS:<p>JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland</p>Formula:C22H19N3O2SPurezza:98.41%Colore e forma:SolidPeso molecolare:389.47NGB 2904
CAS:<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Formula:C28H29Cl2N3OPurezza:98.79%Colore e forma:SolidPeso molecolare:494.46RO1138452
CAS:<p>RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).</p>Formula:C19H23N3OPurezza:97.01% - 99.34%Colore e forma:SolidPeso molecolare:309.41Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Formula:C21H25ClN2O3Purezza:99.75%Colore e forma:SolidPeso molecolare:388.89Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Formula:C18H19N3O·HClPurezza:99.78%Colore e forma:White PowderPeso molecolare:329.82Mesdopetam hemitartrate
CAS:<p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>Formula:C28H42F2N2O12S2Purezza:99.98%Colore e forma:SolidPeso molecolare:700.77Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Formula:C14H20F6N4O7Purezza:98.18%Colore e forma:SolidPeso molecolare:470.32β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurezza:99.64%Colore e forma:SolidPeso molecolare:2720.97MHP
CAS:<p>MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.</p>Formula:C16H23NO4Purezza:98.58%Colore e forma:SolidPeso molecolare:293.36ML401
CAS:<p>ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .</p>Formula:C20H20BrClN2OPurezza:99.13%Colore e forma:SolidPeso molecolare:419.74Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Formula:C21H20O9Purezza:98.90% - 99.21%Colore e forma:Yellow Brown Fine PowderPeso molecolare:416.38ML-031
CAS:<p>ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.</p>Formula:C19H20N2O3Purezza:99.21%Colore e forma:SolidPeso molecolare:324.37JNJ-31020028
CAS:<p>JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).</p>Formula:C34H36FN5O2Purezza:95.92% - 99.65%Colore e forma:SolidPeso molecolare:565.68Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Formula:C40H55N7O11SPurezza:99.84% - >99.99%Colore e forma:White PowderPeso molecolare:841.97Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.97Terutroban
CAS:<p>Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.</p>Formula:C20H22ClNO4SPurezza:99.53%Colore e forma:SolidPeso molecolare:407.91Tetrahydrozoline hydrochloride
CAS:<p>Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.</p>Formula:C13H16N2·HClPurezza:99.90%Colore e forma:Off-White SolidPeso molecolare:236.74PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formula:C21H29Cl2N3O4SPurezza:98.5%Colore e forma:SolidPeso molecolare:490.44Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Formula:C25H26Cl3N7OPurezza:99.79% - ≥95%Colore e forma:SolidPeso molecolare:546.88Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Formula:C21H30N4O4Purezza:99.52%Colore e forma:SolidPeso molecolare:402.49JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Formula:C20H34Cl2N2OPurezza:99.51%Colore e forma:SolidPeso molecolare:389.4
