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UNC2025
CAS:<p>UNC2025 (mrx-6313)(IC50 of 0.74 nM and 0.8 nM) is a potent and orally bioavailable dual MER/FLT3 inhibitor.</p>Formula:C28H40N6OPurity:99.53% - 99.74%Color and Shape:SolidMolecular weight:476.66Cisapride tartrate
CAS:Cisapride tartrate is chemically related to metoclopramide, but unlike metoclopramide, it does not cross the blood-brain barrier or have antidopaminergicFormula:C27H35ClFN3O10Color and Shape:SolidMolecular weight:616.04SLM6031434 (free base)
CAS:SLM6031434 (free base) is an inhibitor of sphingosine kinase type 2 (SphK2). It consists of pedant 1-guanidino-2-phenyloxadiazolylpyrrolidine group.Formula:C22H30F3N5O2Color and Shape:SolidMolecular weight:453.5Aplindore
CAS:<p>Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.</p>Formula:C18H18N2O3Color and Shape:SolidMolecular weight:310.35Fabomotizole dihydrochloride
CAS:<p>Fabomotizole (Afobazole, Obenoxazine, CM346) is a non-sedative anxiolytic with neuroprotective properties, launched in Russia 2000s; exact mechanism unclear.</p>Formula:C15H23Cl2N3O2SColor and Shape:SolidMolecular weight:380.33SB1-F-21
CAS:SB1-F-21 is an UCHL1 inhibitor.Formula:C15H14N4OSColor and Shape:SolidMolecular weight:298.36KDS2010 mesylate
CAS:<p>KDS2010: potent, reversible MAO-B inhibitor with 12,500x selectivity vs. MAO-A; enhances memory in APP/PS1 mice.</p>Formula:C18H21F3N2O4SColor and Shape:SolidMolecular weight:418.43NOSO-95C
CAS:<p>NOSO-95C, an antibacterial, targets bacterial ribosomes, halting translation, and is effective against Enterobacteriaceae in vitro/in vivo.</p>Formula:C54H101N23O12Color and Shape:SolidMolecular weight:1264.53Fadolmidine HCl
CAS:<p>Fadolmidine (MPV-2426) is a potent alpha2-adrenoceptor agonist for spinal analgesia with high affinity across human subtypes and efficacy in vivo.</p>Formula:C13H15ClN2OColor and Shape:SolidMolecular weight:250.72Fadolmidine
CAS:Fadolmidine is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia.Formula:C13H14N2OColor and Shape:SolidMolecular weight:214.26MPV-1306
CAS:MPV-1306 is a metabolite of Dexmedetomidine -- a novel alpha 2-adrenergic receptor agonist.Formula:C13H14N2O2Color and Shape:SolidMolecular weight:230.26Vacquinol-1
CAS:Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma cell death.Formula:C21H21ClN2OPurity:99.92%Color and Shape:SolidMolecular weight:352.86Methasquin
CAS:<p>Methasquin is a folic acid antagonist that has been used in the treatment of experimental leukemia; acts by inhibiting the dihydrofolate reductase in the cell.</p>Formula:C21H22N6O5Color and Shape:SolidMolecular weight:438.44Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52Pyrithione cadmium
CAS:Pyrithione cadmium suppresses tumor growth in vitro and in vivo through inhibition of proteasomal deubiquitinaseFormula:C10H8CdN2O2S2Color and Shape:SolidMolecular weight:364.73Cilengitide hydrochloride
CAS:Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formula:C27H41ClN8O7Color and Shape:SolidMolecular weight:625.12Dersalazine
CAS:<p>Dersalazine, a PAF inhibitor, reduces IL-17 to treat colitis in rodents, potentially aiding ulcerative colitis patients.</p>Formula:C35H32N6O4Purity:99.62%Color and Shape:SolidMolecular weight:600.67IND 1316
CAS:<p>IND 1316 is an activator of AMP-activated protein kinase (AMPK).</p>Formula:C22H17NO3Color and Shape:SolidMolecular weight:343.38EPZ033294
CAS:EPZ033294 has potential anticancer and antiproliferative activity.Formula:C20H22ClN7OPurity:99.95%Color and Shape:SolidMolecular weight:411.89EPZ032597
CAS:EPZ032597 is a novel selective inhibitor of SMYD2 with an IC50 of 16 nM. EPZ032597 has anticancer activity and prevent and treat pancreatic cancerFormula:C20H23N7OPurity:99.70%Color and Shape:SolidMolecular weight:377.44Grp94-IN-2
CAS:Grp94-IN-2 is a inhibitor of Grp94.Formula:C22H23ClN2O5Color and Shape:SolidMolecular weight:430.88Colterol (free base)
CAS:Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Formula:C12H19NO3Color and Shape:SolidMolecular weight:225.28Soyacerebroside II
CAS:Soyacerebroside II is a Ca2+ ionophore; both I and II inhibit IL-18 in PBMCs and modulate immune responses.Formula:C40H75NO9Purity:98%Color and Shape:SolidMolecular weight:714.02Nizatidine amide
CAS:Nizatidine amide blocks H2 receptors, reducing stomach acid to treat ulcers and GERD.Formula:C11H18N4O3S2Color and Shape:SolidMolecular weight:318.42IACS-4759
CAS:<p>IACS-4759 is a novel potent and selective MTH1 inhibitor with excellent cell permeability and good metabolic stability in microsomes.</p>Formula:C10H17N3O2Color and Shape:SolidMolecular weight:211.26ent-Entecavir
CAS:Ent-Entecavir, an enantiomeric impurity of Entecavir (an oral HBV drug), inhibits HBV replication as a reverse transcriptase inhibitor.Formula:C12H15N5O3Color and Shape:SolidMolecular weight:277.28JTP 103237
CAS:<p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>Formula:C24H29F3N6OColor and Shape:SolidMolecular weight:474.52MS-049 oxalate salt
CAS:MS-049 oxalate salt is a potent and selective inhibitor of protein arginine methyltransferases (PRMTs) PRMT 4 and PRMT6.Formula:C17H26N2O5Color and Shape:SolidMolecular weight:338.4Mps1-IN-1 dihydrochloride
CAS:Mps1-IN-1 dihydrochloride, a potent ATP-competitive inhibitor of Mps1 kinase, exhibits an IC50 of 367 nM.Formula:C28H35Cl2N5O4SColor and Shape:SolidMolecular weight:608.58AEG40730 HCl
CAS:<p>AEG40730: A potent, selective IAP inhibitor, induces cIAP1/2 degradation, reduces RIP1 ubiquitination, and depletes XIAP, c-IAP1.</p>Formula:C52H70Cl2F6N8O8Color and Shape:SolidMolecular weight:1120.0704Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Formula:C9H10N4O4·xC4H10N2Color and Shape:SolidMolecular weight:562.54CDK8-IN-18
CAS:CDK8-IN-18, also known as ZINC584617986, is a potent and selective inhibitor of CDK8, also modulating CDK19.Formula:C18H17N5OColor and Shape:SolidMolecular weight:319.36Methylsilanol ascorbate
CAS:Methylsilanol ascorbate is a silanol analogue and inhibitor of angiotensin-converting enzyme.Formula:C7H12O8SiColor and Shape:SolidMolecular weight:252.25VER-155008
CAS:<p>VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively.</p>Formula:C25H23Cl2N7O4Purity:97.03% - 99.55%Color and Shape:SolidMolecular weight:556.4SG3-179
CAS:SG3-179 is a BET inhibitor.Formula:C28H35ClFN7O3SColor and Shape:SolidMolecular weight:604.14EMD-66684
CAS:EMD-66684 is a non-peptide angiotensin II receptor antagonist.Formula:C28H31ClN8O2Color and Shape:SolidMolecular weight:547.06KFP-H008
CAS:KFP-H008 is a potassium-competitive acid blocker.Formula:C19H18N4O2SColor and Shape:SolidMolecular weight:366.44KSK213
CAS:KSK213: Strongly inhibits C. trachomatis (EC50=60 nM); non-toxic to commensals/host cells at 25 μM.Formula:C28H25N3O2SColor and Shape:SolidMolecular weight:467.58Verubecestat tosylate
CAS:Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.Formula:C25H26N4O4S2Color and Shape:SolidMolecular weight:510.627Chlorpromazine Sulfone Hydrochloride
CAS:Chlorpromazine Sulfone Hydrochloride: metabolite of anti-psychotic, may inhibit N-methyltransferase.Formula:C17H20Cl2N2O2SColor and Shape:SolidMolecular weight:387.32F-050
CAS:F-050 inhibits platelet aggregation, potentially treating thrombosis in guinea pigs, rabbits, and rats.Formula:C21H20OColor and Shape:SolidMolecular weight:288.38Olcorolimus
CAS:Olcorolimus blocks specific allergen-induced inflammation, reducing eosinophil, lymphocyte infiltration, and IL-4/IL-5 mRNA expression.Formula:C51H81NO12Color and Shape:SolidMolecular weight:900.19Fasudil hydrochloride hydrate
CAS:Fasudil HCl hydrate is a ROCK inhibitor that hinders mature CCM development and lowers portal pressure in cirrhotic rats.Formula:C28H38Cl2N6O5S2Color and Shape:SolidMolecular weight:673.67Delucemine Free Base
CAS:Delucemine Free Base is an NMDA Receptor AntagonistFormula:C16H17F2NColor and Shape:SolidMolecular weight:261.31Verubecestat
CAS:<p>Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.</p>Formula:C17H17F2N5O3SPurity:92.24% - 99.55%Color and Shape:SolidMolecular weight:409.41CVS-1578
CAS:CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Formula:C20H30N6O5SColor and Shape:SolidMolecular weight:466.55GT-2394
CAS:GT-2394 is a histamine H3 receptor agonist.Formula:C14H21N3O2Color and Shape:SolidMolecular weight:263.34GT-2227
CAS:<p>GT-2227 is a histamine H3 receptor antagonist.</p>Formula:C15H24N2Color and Shape:SolidMolecular weight:232.36ATM-1001
CAS:ATM-1001 is an inhibitor of the cancer-associated tropomyosin 3.1 (Tpm3.1), suppressing glucose-stimulated insulin secretion (GSIS) from the pancreatic islets.Formula:C30H36N4OColor and Shape:SolidMolecular weight:468.63Paclitaxel Ceribate
CAS:<p>Paclitaxel Ceribate is a mitotic inhibitor used in cancer chemotherapy.</p>Formula:C51H57NO18Color and Shape:SolidMolecular weight:971.99Pamiparib hydrate
CAS:<p>Pamiparib (BGB-290) is a potent, selective PARP inhibitor that promotes DNA damage and apoptosis in cancer cells.</p>Formula:C16H21FN4O4Color and Shape:SolidMolecular weight:352.36Cyclanoline (free base)
CAS:Cyclanoline (free base) is an acetylcholinesterase inhibitorFormula:C20H24NO4Color and Shape:SolidMolecular weight:342.41PSI-112
CAS:PSI-112 is a fibrinolysis inhibitor.Formula:C35H48N4O3Color and Shape:SolidMolecular weight:572.78Vernolepin
CAS:<p>Vernolepin is a natural reversible plant growth inhibitor.</p>Formula:C15H16O5Color and Shape:SolidMolecular weight:276.28VO-Ohpic trihydrate
CAS:<p>VO-Ohpic trihydrate (VO-Ohpic) is a potent inhibitor of PTEN (phosphatase and tensin homolog) with IC50 of 35 nM.</p>Formula:C12H9N2O8V·3H2O·HPurity:>99.99%Color and Shape:SolidMolecular weight:415.2Zavondemstat
CAS:Zavondemstat (QC8222 free base) is a KDM4 inhibitor with anticancer and antitumor activity for the study of triple-negative and breast cancers.Formula:C26H29N3O3Purity:99.43% - 99.53%Color and Shape:SolidMolecular weight:431.53Acotiamide Methyl Ether
CAS:<p>Acotiamide Methyl Ether is a metabolite enhancing gastric motility, derived from Acotiamide, a drug easing functional dyspepsia symptoms.</p>Formula:C22H32N4O5SColor and Shape:SolidMolecular weight:464.58N-5984 Hydrochloride
CAS:<p>N-5984 Hydrochloride is a beta3-AR agonist.</p>Formula:C20H23Cl2NO5Color and Shape:SolidMolecular weight:428.31Tomivosertib HCl
CAS:Tomivosertib (eFT508) is a MNK1/2 inhibitor that blocks eIF4E phosphorylation, hindering tumor growth and immune signaling.Formula:C17H21ClN6O2Color and Shape:SolidMolecular weight:376.845Pemrametostat succinate
CAS:Pemrametostat succinate, an oral PRMT5 inhibitor, strongly curbs tumor growth in vitro and animal studies.Formula:C28H38N6O7Color and Shape:SolidMolecular weight:570.65CJM-061
CAS:<p>CJM-061 is a Wee1 inhibitor.</p>Formula:C28H32N8O4Color and Shape:SolidMolecular weight:544.6Famotine
CAS:Famotidine: H2 blocker that reduces stomach acid, treats ulcers and GERD.Formula:C16H14ClNOColor and Shape:SolidMolecular weight:271.74Olmutinib hydrochloride
CAS:Olmutinib is a third-gen EGFR inhibitor for T790M-positive lung cancer, blocking phosphorylation and tumor pathways. Approved in Korea (2016).Formula:C26H28Cl2N6O2SColor and Shape:SolidMolecular weight:559.51ST-115
CAS:ST-115: potent aminopeptidase P2 inhibitor, reduces bradykinin degradation intravenously, boosting its capillary concentration.Formula:C21H32FN3O5SColor and Shape:SolidMolecular weight:457.56Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Formula:C29H33FN2O4Purity:98.77% - 99.93%Color and Shape:SolidMolecular weight:492.58NPA101.3
CAS:NPA101.3 is a a Second-Generation RET/VEGFR2 Inhibitor. It is a potential clinical candidate for RET-driven cancers.Formula:C29H28N4O4SColor and Shape:SolidMolecular weight:528.62TPP2a bromide
CAS:TPP2a is a mitochondrial thioredoxin reductase (TrxR) inhibitor.Formula:C47H52BrO5PColor and Shape:SolidMolecular weight:807.81HSP-117 dihydrochloride
CAS:HSP-117 dihydrochloride is a novel tachykinin NK1-receptor antagonist.Formula:C23H32Cl2N2OColor and Shape:SolidMolecular weight:423.42BAY-846
CAS:BAY-846: allosteric MEK inhibitor, long-lasting, highly bioavailable, low brain entry, effective in K-Ras A549 model.Formula:C19H13F4IN4O4SColor and Shape:SolidMolecular weight:596.29L-778123 Dihydrochloride
CAS:L-778123 blocks FPTase/GGPTase-I, halts Ki-Ras prenylation, has acceptable toxicity with radiotherapy in advanced pancreatic cancer.Formula:C22H22Cl3N5OColor and Shape:SolidMolecular weight:478.802Nepaprazole sodium dihydrate
CAS:Nepaprazole sodium dihydrate is a proton pump inhibitor potentially for treatment of gastric ulcers.Formula:C18H22N3NaO4SColor and Shape:SolidMolecular weight:399.44CAM 4750
CAS:<p>CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist.</p>Formula:C30H31ClN4O4Color and Shape:SolidMolecular weight:547.05CAM 4515
CAS:CAM 4515 is a nonpeptide tachykinin NK1 receptor antagonist.Formula:C29H27N3O4Color and Shape:SolidMolecular weight:481.54AZ0108
CAS:<p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>Formula:C24H20F4N6O2Color and Shape:SolidMolecular weight:500.45MSD-D
CAS:MSD-D is an inhibitor of voltage-gated K(+) (Kv) channels Kv1.5.Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43Voxtalisib
CAS:Voxtalisib (XL765) (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ with IC50 of 9 nM; also inhibits DNA-PK and mTOR. Phase 1/2.Formula:C13H14N6OPurity:98.21% - 99.69%Color and Shape:SolidMolecular weight:270.29D 22888
CAS:D 22888 is a PDE4 inhibitor.Formula:C16H20N4O2Color and Shape:SolidMolecular weight:300.36MDK80908
CAS:MDK80908 (CAS# 1821380-90-8), a dual PPARα/γ agonist, improves insulin resistance and gluconeogenesis.Formula:C21H43NO2SColor and Shape:SolidMolecular weight:373.64pyimDC
CAS:<p>pyimDC is a novel potent inhibitor of collagen prolyl-4-hydroxylases (CP4H).</p>Formula:C10H7N3O4Color and Shape:SolidMolecular weight:233.18Derazantinib dihydrochloride
CAS:Derazantinib, a multi-kinase inhibitor targeting FGFR, benefits FGFR2-positive iCCA; its dihydrochloride form is a salt variant.Formula:C29H31Cl2FN4OColor and Shape:SolidMolecular weight:541.49ORP-101
CAS:ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.Formula:C60H84N2O8Color and Shape:SolidMolecular weight:961.32LYRM03
CAS:LYRM03, a ubenimex derivative and aminopeptidase inhibitor, suppresses TLR4 to treat LPS-induced ALI in mice.Formula:C21H33N3O5Color and Shape:SolidMolecular weight:407.510-Oxononadecanedioic acid
CAS:10-Oxononadecanedioic acid: a long-chain linker with two carboxylic ends, forms stable amides with amines using activators like EDC/HATU.Formula:C19H34O5Color and Shape:SolidMolecular weight:342.47Fipravirimat
CAS:Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.Formula:C43H67FN2O4SColor and Shape:SolidMolecular weight:727.07CDK8-IN-4k
CAS:<p>CDK8-IN-4k is a potent and highly selective CDK8 inhibitor, with no apparent potential for time-dependent CYP3A4 inhibition.</p>Formula:C24H23F2N5OColor and Shape:SolidMolecular weight:435.47PomCapstafin
CAS:PomCapstafin is a prodrug of Capstafin, acting as a potent, selective STAT5b inhibitor.Formula:C41H69NO17P2Color and Shape:SolidMolecular weight:909.93Vps34-IN-1
CAS:Vps34-IN-1: potent, selective Vps34 inhibitor, 25 nM IC50, spares class I/II PI3Ks.Formula:C21H24ClN7OPurity:97.04%Color and Shape:SolidMolecular weight:425.91Capstafin
CAS:Capstafin is a highly potent and selective inhibitor of STAT5b.Formula:C17H29NO9P2Color and Shape:SolidMolecular weight:453.36MeTC7
CAS:<p>MeTC7 is a VDR antagonist with antitumor activity that inhibits PD-L1 and may inhibit the growth of xenografts and transgenic tumors in vivo.</p>Formula:C32H48BrN3O4Purity:99.69%Color and Shape:SolidMolecular weight:618.65Miransertib mesylate
CAS:Miransertib mesylate inhibits AKT non-competitively, potentially reducing tumor growth and triggering apoptosis.Formula:C29H32N6O6S2Color and Shape:SolidMolecular weight:624.73Pipoxolan hydrochloride
CAS:<p>Pipoxolan is an antispasmodic treating GI tract, gallbladder, urogenital, and menstrual cramps, with emerging anticancer properties.</p>Formula:C22H26ClNO3Color and Shape:SolidMolecular weight:387.9041-Hydroxyvaldecoxib
CAS:1-Hydroxyvaldecoxib is a COX-2 inhibitor.Formula:C16H14N2O4SColor and Shape:SolidMolecular weight:330.36Fenoldopam hydrochloride
CAS:<p>Fenoldopam HCl: D1 dopamine receptor agonist, vasodilator, doesn't cross blood-brain barrier, α2-adrenoceptor antagonist.</p>Formula:C16H17Cl2NO3Color and Shape:SolidMolecular weight:342.22K-5a2
CAS:K-5a2 is a novel human immunodeficiency virus type 1 (HIV-1) non-nucleoside reverse transcriptase inhibitor (NNRTI).Formula:C27H28N6O3S2Color and Shape:SolidMolecular weight:548.68GGTI-297
CAS:GGTI-297 is a potent, cell-permeable, and selective peptidomimetic inhibitor of GGTase I compared to Farnesyl Transferase (FTase).Formula:C26H31N3O3SColor and Shape:SolidMolecular weight:465.61UniPR1331
CAS:UniPR1331 is a novel selective antagonist of the Eph-ephrin system.Formula:C35H48N2O4Color and Shape:SolidMolecular weight:560.77VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Formula:C19H16ClN5O6SPurity:98.99% - 99.22%Color and Shape:SolidMolecular weight:477.88PF-06427878
CAS:<p>PF-06427878 is an orally active, potent and selective diacylglycerol acyltransferase 2 inhibitor.</p>Formula:C26H28N4O5Color and Shape:SolidMolecular weight:476.52Berotralstat HCl
CAS:<p>Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.</p>Formula:C30H28Cl2F4N6OColor and Shape:SolidMolecular weight:635.4886GPA512
CAS:<p>GPA512 is a prodrug of aliellalactone, inhibiting STAT3 and preventing the transcription of STAT3 regulated genes.</p>Formula:C17H25NO6SColor and Shape:SolidMolecular weight:371.45
