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Apoptose

Apoptose

Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.

Subcategorias de "Apoptose"

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Foram encontrados 5618 produtos de "Apoptose"

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  • Acacetin

    CAS:
    <p>Acacetin (5,7-Dihydroxy-4'-methoxyflavone) is an O-methylated flavone found in various plants, shows antinociceptive, anti-inflammatory, and antioxidant</p>
    Fórmula:C16H12O5
    Pureza:96.26% - ≥95%
    Cor e Forma:Pale-Yellow Needles
    Peso molecular:284.26
  • VK3-OCH3

    CAS:
    VK3-OCH3 (2-[(2-Methoxy)ethylthio]-3-methyl-1,4-na) is a selective antitumor agent via heme oxygenase (HO-1) related mechanisms; Vitamine K3 analogue.
    Fórmula:C14H14O3S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:262.32
  • CAY10505

    CAS:
    <p>CAY10505, a form of dehydroxyl of AS-252424, is a PI3Kγ inhibitor (IC50: 33 nM).</p>
    Fórmula:C14H8FNO3S
    Pureza:99.69% - 99.74%
    Cor e Forma:Solid
    Peso molecular:289.28
  • MRS 2578

    CAS:
    MRS2578, an effective P2Y6 receptor antagonist with IC50 of 37 nM, shows insignificant inhibition at P2Y1, P2Y2, P2Y4, and P2Y11 receptors.
    Fórmula:C20H20N6S4
    Pureza:97.58% - 99.73%
    Cor e Forma:White Solid
    Peso molecular:472.67
  • Polyphyllin I

    CAS:
    <p>Polyphyllin D induces apoptosis via the mitochondrial apoptotic pathway as evidenced by decreased Bcl-2 expression levels, disruption of MMP and increased Bax,</p>
    Fórmula:C44H70O16
    Pureza:98% - 99.5%
    Cor e Forma:Solid
    Peso molecular:855.02
  • Epothilone A

    CAS:
    <p>Epothilone A (Epo A) is a microtubule-stabilizing agent with EC0.01 of 2 μM.</p>
    Fórmula:C26H39NO6S
    Pureza:99.89% - 99.92%
    Cor e Forma:Solid
    Peso molecular:493.66
  • Fedratinib hydrochloride hydrate

    CAS:
    <p>Fedratinib hydrochloride hydrate (SAR 302503 hydrochloride hydrate) is a potent, selective, ATP-competitive and orally active JAK2 inhibitor.</p>
    Fórmula:C27H40Cl2N6O4S
    Pureza:98.96% - 99.87%
    Cor e Forma:Solid
    Peso molecular:615.61
  • G5-7

    CAS:
    <p>G5-7 is an oral JAK2 inhibitor targeting EGFR/STAT3 phosphorylation with potential for glioma research.</p>
    Fórmula:C22H19F2NO3
    Pureza:97.3%
    Cor e Forma:Solid
    Peso molecular:383.39
  • Alginic acid

    CAS:
    <p>Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.</p>
    Fórmula:C14H22O13
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:398.317
  • OTS514 hydrochloride

    CAS:
    OTS514 hydrochloride is a highly effective TOPK(T-LAK cell-originated protein kinase) inhibitor (IC50: 2.6 nM).
    Fórmula:C21H20N2O2S·HCl
    Pureza:99.67% - 99.84%
    Cor e Forma:Solid
    Peso molecular:400.92
  • Kynurenic acid sodium

    CAS:
    Kynurenic acid sodium salt is an endogenous tryptophan metabolite. It antagonizes NMDA, glutamate, and α7 nicotinic receptors, and agonizes GPR35.
    Fórmula:C10H6NNaO3
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:211.15
  • MK-886

    CAS:
    MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP).
    Fórmula:C27H34ClNO2S
    Pureza:99.23% - 99.84%
    Cor e Forma:Solid
    Peso molecular:472.08
  • Xanthatin

    CAS:
    Xanthatin exhibits cytotoxic, antibacterial, antifungal properties, may treat NSCLC, and inhibits melanoma by targeting Wnt/β-catenin and angiogenesis.
    Fórmula:C15H18O3
    Pureza:98.48% - 99.96%
    Cor e Forma:Solid
    Peso molecular:246.3
  • CASIN

    CAS:
    CASIN (Pirl1-related Compound 2) is a specific inhibitor of GTPase Cdc42 (IC50: 2 uM).
    Fórmula:C20H22N2O
    Pureza:98.18% - >99.99%
    Cor e Forma:Solid
    Peso molecular:306.4
  • NU 7026

    CAS:
    <p>NU 7026 (DNA-PK Inhibitor II) is an effective DNA-PK inhibitor (IC50: 0.23 μM, in cell-free assays), 60-fold selective for DNA-PK than PI3K and no inhibition</p>
    Fórmula:C17H15NO3
    Pureza:99.51% - >99.99%
    Cor e Forma:Solid
    Peso molecular:281.31
  • 4EGI-1

    CAS:
    <p>4EGI-1, a competitive eIF4E/eIF4 g interaction inhibitor, binds to eIF4E(KD=25 μM).</p>
    Fórmula:C18H12Cl2N4O4S
    Pureza:96.8% - 99.12%
    Cor e Forma:Solid
    Peso molecular:451.28
  • Lithocholic acid

    CAS:
    Lithocholic acid (3α-Hydroxy-5β-cholanic acid) is a toxic secondary bile acid, They were FXR antagonists (IC50=0.7, 1.4 μM). High-Quality, Low-Cost!
    Fórmula:C24H40O3
    Pureza:98% - 99.93%
    Cor e Forma:Hexagonal Leaflets From Alc Prisms From Acetic Acid Powder (Ntp 1992)
    Peso molecular:376.57
  • SKF-96365 hydrochloride

    CAS:
    <p>SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y</p>
    Fórmula:C22H27ClN2O3
    Pureza:99.47% - 99.92%
    Cor e Forma:Solid
    Peso molecular:402.91
  • Xanthohumol

    CAS:
    <p>Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-</p>
    Fórmula:C21H22O5
    Pureza:98.19% - 99.67%
    Cor e Forma:Orange Powder
    Peso molecular:354.4
  • NSC 66811

    CAS:
    <p>NSC 66811 inhibits MDM2-p53 interaction with 120 nM affinity, activating p53 in cancer cells.</p>
    Fórmula:C23H20N2O
    Pureza:96.94%
    Cor e Forma:Solid
    Peso molecular:340.42