
Apoptose
Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.
Subcategorias de "Apoptose"
- ASK(9 produtos)
- BCL(1 produtos)
- Caspase(154 produtos)
- FOXO1(2 produtos)
- IAP(67 produtos)
- Mdm2(12 produtos)
- PD-1/PD-L1(140 produtos)
- PDK(9 produtos)
- PERK(24 produtos)
- Serina/treonina quinase(19 produtos)
- Survivina(14 produtos)
- TNF(94 produtos)
- c-RET(61 produtos)
- p53(63 produtos)
Exibir 6 mais subcategorias
Foram encontrados 6499 produtos de "Apoptose"
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BMS-1
CAS:BMS-1 is a PD-1/PD-L1 inhibitor and immunomodulator; it targets the CD274 gene product, PD-L1, linked to tumor evasion and higher mortality.
Fórmula:C29H33NO5Pureza:99.40% - 99.81%Cor e Forma:SolidPeso molecular:475.58PFK-158
CAS:PFK-158 is an effective and specific inhibitor PFKFB3.Fórmula:C18H11F3N2OPureza:95.49% - 99.16%Cor e Forma:SolidPeso molecular:328.29Ref: TM-T3105
1mg34,00€2mg46,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg170,00€50mg259,00€100mg409,00€Madecassoside
CAS:Madecassoside (Asiaticoside A) is a pentacyclic triterpene extracted from Centella asitica (L.) with anti-inflammatory, anti-oxidative and anti-aging activitiesFórmula:C48H78O20Pureza:99.46% - 99.85%Cor e Forma:White PowderPeso molecular:975.12Ref: TM-T2813
10mg49,00€1mL*10mM (DMSO)49,00€25mg84,00€50mg120,00€100mg178,00€200mg289,00€500mg485,00€Osthole
CAS:Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Fórmula:C15H16O3Pureza:99.93% - 99.96%Cor e Forma:Fine White PowderPeso molecular:244.298-Prenylnaringenin
CAS:8-Prenylnaringenin is a phytoestrogen with high estrogenic activity,Fórmula:C20H20O5Pureza:98.26% - 99.46%Cor e Forma:SolidPeso molecular:340.37Ref: TM-TN1146
1mg137,00€5mg334,00€1mL*10mM (DMSO)414,00€10mg494,00€25mg782,00€50mg1.054,00€100mg1.414,00€Cilengitide
CAS:Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.Fórmula:C27H40N8O7Pureza:98% - 99.8%Cor e Forma:SolidPeso molecular:588.66Alantolactone
CAS:Alantolactone is a selective inhibitor of STAT3 that induces cancer-associated apoptosis and has antitumor activity.Cost-effective and quality-assured.Fórmula:C15H20O2Pureza:99.02% - 99.66%Cor e Forma:Crystalline PowderPeso molecular:232.32Rabeprazole sodium
CAS:Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.Fórmula:C18H20N3NaO3SPureza:98% - 99.912%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:381.42Y-27632 HCl hydrate
CAS:Y-27632 HCl hydrate is an orally effective, ATP-competitive ROCK1/ROCK2 inhibitor (Ki=220 nM/300 nM) that inhibits caspase-3 and suppresses stem cell apoptosis.Fórmula:C14H25Cl2N3O2Pureza:99.98%Cor e Forma:SolidPeso molecular:338.27BO-264
CAS:BO-264 is a highly potent and orally active inhibitor of transforming acidic coiled-coil 3 (TACC3, IC50 of 188 nM and a Kd of 1.5 nM).Fórmula:C18H19N5O3Pureza:98.03% - 99.81%Cor e Forma:SolidPeso molecular:353.38Mivebresib
CAS:Mivebresib (ABBV-075) is a potent BET inhibitor with antitumor effects, disrupting gene expression and MYC, TMPRSS2-ETS proteins.Fórmula:C22H19F2N3O4SPureza:98.74% - 99.32%Cor e Forma:SolidPeso molecular:459.47Ref: TM-T3712
1mg55,00€2mg78,00€5mg92,00€1mL*10mM (DMSO)94,00€10mg150,00€25mg244,00€50mg437,00€100mg625,00€Picropodophyllin
CAS:Picropodophyllin (PPP) is a selective IGF-1R inhibitor with IC50 of 1 nM, not affecting other growth factor receptors.Fórmula:C22H22O8Pureza:98.38% - 99.83%Cor e Forma:SolidPeso molecular:414.41Ref: TM-T6943
5mg64,00€1mL*10mM (DMSO)69,00€10mg88,00€25mg170,00€50mg316,00€100mg535,00€500mg1.121,00€Hispidol
CAS:Hispidol ((Z)-Hispidol) ((Z)-Hispidol) is a potential therapeutic for inflammatory bowel disease; inhibits TNF-α induced adhesion of monocytes to colonFórmula:C15H10O4Pureza:97.86% - 98.45%Cor e Forma:SolidPeso molecular:254.24Ref: TM-T4319
1mg42,00€2mg56,00€1mL*10mM (DMSO)92,00€5mg93,00€10mg137,00€25mg200,00€50mg260,00€100mg409,00€200mg560,00€500mg954,00€ZMC1
CAS:NSC-319726 (ZMC1), a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).Fórmula:C11H14N4SPureza:98.97% - 99.76%Cor e Forma:SolidPeso molecular:234.32Nirogacestat
CAS:Nirogacestat (PF 03084014) is a specific γ-secretase inhibitor (IC50: 6.2 nM, in a cell-free assay).Fórmula:C27H41F2N5OPureza:97.98% - 99.63%Cor e Forma:SolidPeso molecular:489.64Ref: TM-T6935
1mg35,00€5mg78,00€1mL*10mM (DMSO)87,00€10mg117,00€25mg236,00€50mg447,00€100mg675,00€200mg888,00€Bromosporine
CAS:Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.Fórmula:C17H20N6O4SPureza:99.65% - 99.79%Cor e Forma:SolidPeso molecular:404.44Ref: TM-T6255
1mg44,00€2mg57,00€1mL*10mM (DMSO)92,00€5mg93,00€10mg133,00€25mg260,00€50mg416,00€100mg665,00€200mg888,00€Karanjin
CAS:Karanjin, a flavonoid from karanja seeds, boosts GLUT4, AMPK in muscles, and triggers cancer cell apoptosis.Fórmula:C18H12O4Pureza:99.01%Cor e Forma:SolidPeso molecular:292.29Ref: TM-T2S0820
1mg46,00€1mL*10mM (DMSO)94,00€5mg96,00€10mg145,00€25mg259,00€50mg385,00€100mg557,00€200mg790,00€Betulinic acid
CAS:Betulinic acid, a lupane-type triterpene from white birch bark, has antiretroviral, antimalarial, anti-inflammatory, and anticancer properties.Fórmula:C30H48O3Pureza:98.22% - 99.7%Cor e Forma:White Crystalline PowderPeso molecular:456.70Resatorvid
CAS:Resatorvid (TAK-242) inhibits TLR4, with IC50s for IL-6, TNF-R, NO at 1.3, 1.9, 1.8 nM respectively.Fórmula:C15H17ClFNO4SPureza:99.31% - >99.99%Cor e Forma:SolidPeso molecular:361.82Ref: TM-TQ0181
1mg50,00€2mg66,00€5mg90,00€1mL*10mM (DMSO)110,00€10mg156,00€25mg290,00€50mg475,00€100mg763,00€R406 free base
CAS:R406 free base (R406 (free base)) is a potent Syk inhibitor.Fórmula:C22H23FN6O5Pureza:97.64% - 99.11%Cor e Forma:SolidPeso molecular:470.45Ref: TM-T2467
1mg44,00€5mg66,00€1mL*10mM (DMSO)69,00€10mg92,00€25mg177,00€50mg319,00€100mg507,00€500mg1.063,00€
