PPAR
Os receptores ativados por proliferadores de peroxissomas (PPARs) são um grupo de proteínas receptoras nucleares que funcionam como fatores de transcrição, regulando a expressão de genes envolvidos no metabolismo, particularmente no armazenamento de ácidos graxos e no metabolismo da glicose. Inibidores de PPAR são ferramentas importantes para o estudo de distúrbios metabólicos como diabetes, obesidade e doenças cardiovasculares. Esses inibidores podem modular o metabolismo lipídico, a sensibilidade à insulina e a inflamação, tornando-os valiosos na pesquisa terapêutica. Na CymitQuimica, oferecemos uma gama de inibidores de PPAR para apoiar sua pesquisa em doenças metabólicas, endocrinologia e desenvolvimento de medicamentos.
Foram encontrados 170 produtos de "PPAR"
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β-Amyrone
CAS:beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM.Fórmula:C30H48OPureza:99.55%Cor e Forma:SolidPeso molecular:424.7Fenofibrate
CAS:Fenofibrate (Lipanthyl) is a PPARα agonist. Fenofibrate inhibits cytochrome P450 isoforms. Fenofibrate exhibits antihyperlipidemic activity. Cost-effective and quality-assured.Fórmula:C20H21ClO4Pureza:99.13% - 99.95%Cor e Forma:Crystals From Isopropanol SolidPeso molecular:360.83Mifobate
CAS:Mifobate (SR-202) 是一种有效且特异性的 PPARγ拮抗剂，可选择性抑制噻唑烷二酮 (TZD) 诱导的 PPARγ 转录活性，IC50为140 μM，具有抗肥胖和抗糖尿病作用。Fórmula:C11H17ClO7P2Pureza:99.12%Cor e Forma:SolidPeso molecular:358.655-Aminosalicylic Acid
CAS:5-Aminosalicylic Acid (5-ASA) is a specific PPARγ agonist and also inhibits P21-activated kinase 1 (PAK1) and NF-Κb. High-Quality, Low-Cost!Fórmula:C7H7NO3Pureza:98.88% - 99.49%Cor e Forma:Purplish-Tan Solid PowderPeso molecular:153.14LY518674
CAS:LY518674 (LY-674) decreases triglycerides and increases HDL-C and is used for the treatment of atherosclerosis.Fórmula:C23H27N3O4Pureza:98.87%Cor e Forma:SolidPeso molecular:409.48Ref: TM-T15821
1mg170,00€5mg359,00€10mg533,00€25mg847,00€50mg1.159,00€100mg1.568,00€1mL*10mM (DMSO)398,00€Gemfibrozil
CAS:Gemfibrozil, a fibric acid derivative, stimulates PPARalpha, boosts fatty acid oxidation, LPL, lowers VLDL-C, apoC-III, and raises HDL-C.Fórmula:C15H22O3Pureza:99.53% - 99.88%Cor e Forma:Crystals From Hexane SolidPeso molecular:250.33EHP-101
CAS:EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.Fórmula:C28H35NO3Pureza:98.36%Cor e Forma:SolidPeso molecular:433.58Ref: TM-T13289
1mg107,00€5mg227,00€10mg378,00€25mg620,00€50mg868,00€100mg1.169,00€1mL*10mM (DMSO)250,00€Muraglitazar
CAS:Muraglitazar (BMS-298585) is a PPAR α/γ dual agonist for the treatment of type 2 diabetes and associated dyslipidemia.Fórmula:C29H28N2O7Pureza:99.17%Cor e Forma:SolidPeso molecular:516.54Daidzein
CAS:Daidzein (Isoflavone) is an isoflavone extract from soy, which is an inactive analog of the tyrosine kinase inhibitor genistein.Fórmula:C15H10O4Pureza:98.08%Cor e Forma:SolidPeso molecular:254.24Candesartan
CAS:Candesartan (CV 11974) is an angiotensin II receptor blocker used widely in the therapy of hypertension and heart failure.Fórmula:C24H20N6O3Pureza:98.3% - 99.55%Cor e Forma:Colorless Solid CrystallinePeso molecular:440.47Pioglitazone hydrochloride
CAS:Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties and potential antineoplasticFórmula:C19H20N2O3S·HClPureza:99.64% - >99.99%Cor e Forma:White Crystals Or Crystalline PowderPeso molecular:392.90MA-0204
CAS:MA-0204 is a highly selective and orally available peroxisome proliferator-activated receptor δ (PPARδ) modulator (EC50s: 0.4 nM, 7.9 nM and 10 nM for human,Fórmula:C25H27F3N2O4Pureza:97.8%Cor e Forma:SolidPeso molecular:476.49Ref: TM-T15945
1mg96,00€5mg178,00€10mg301,00€25mg490,00€50mg677,00€100mg900,00€200mg1.206,00€1mL*10mM (DMSO)187,00€Cloxiquine
CAS:Cloxiquine (Dermofongin) is a monohalogenated 8-hydroxyquinoline with activity against bacteria, fungi, and protozoa.Fórmula:C9H6ClNOPureza:99.82% - 99.87%Cor e Forma:Light Yellow CrystalsPeso molecular:179.6Arhalofenate
CAS:Arhalofenate (JNJ 39659100) is a selective partial agonist of peroxisome proliferator-activated receptor PPARγ. It is used for the treatment of type 2 diabetes.Fórmula:C19H17ClF3NO4Pureza:98.97%Cor e Forma:SolidPeso molecular:415.79Ref: TM-T16022
1mg62,00€5mg205,00€10mg359,00€25mg588,00€50mg825,00€100mg1.111,00€200mg1.501,00€1mL*10mM (DMSO)270,00€Pioglitazone
CAS:Pioglitazone (U 72107) is a selective and oral PPARγ agonist with EC50 of 0.93 and 0.99 μM on human and mouse PPARγ, respectively . High-Quality, Low-Cost!Fórmula:C19H20N2O3SPureza:95% - 99.57%Cor e Forma:White PowderPeso molecular:356.44NTP42
CAS:NTP42 is an antagonist of thromboxane A2 (TXA2) receptor(IC50 of 3.278 nM)Fórmula:C25H23F2N3O5SPureza:97.55%Cor e Forma:SolidPeso molecular:515.53Ref: TM-T12268
1mg59,00€2mg86,00€5mg133,00€10mg203,00€25mg344,00€50mg512,00€100mg735,00€1mL*10mM (DMSO)150,00€NSC-87877
CAS:NSC-87877 inhibits Shp2 (IC50=0.318μM), Shp1 (IC50=0.355μM), and DUSP26 phosphatases.Fórmula:C19H13N3O7S2Pureza:97.35%Cor e Forma:SolidPeso molecular:459.45Bezafibrate
CAS:Bezafibrate (BM15075) is an antilipemic agent that lowers CHOLESTEROL and TRIGLYCERIDES.Fórmula:C19H20ClNO4Pureza:99.56% - 99.82%Cor e Forma:SolidPeso molecular:361.82Clofibric acid
CAS:Clofibric acid (Chlorofibrinic acid) is an antilipemic agent that is the biologically active metabolite of CLOFIBRATE.Fórmula:C10H11ClO3Pureza:99.47% - 99.8%Cor e Forma:Pale Yellow SolidPeso molecular:214.65Fenofibric acid
CAS:Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.Fórmula:C17H15ClO4Pureza:99.36%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:318.75Anandamide
CAS:Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but alsoFórmula:C22H37NO2Pureza:95.037% - 99.22%Cor e Forma:Light Yellow OilPeso molecular:347.53Ref: TM-T14046
1mg35,00€2mg48,00€5mg71,00€10mg124,00€25mg234,00€50mg349,00€100mg512,00€200mg713,00€1mL*10mM (DMSO)77,00€Retinoic acid
CAS:Retinoic acid (Tretinoin) binds to and activates RARs, thereby inducing changes in gene expression that lead to inhibition of tumorigenesis.Fórmula:C20H28O2Pureza:97.21% - 99.60%Cor e Forma:Yellow-Orange PowderPeso molecular:300.44Magnolol
CAS:Magnolol (5,5'-Diallyl-2,2'-biphenyldiol) is a dual agonist of RXRα( EC50=10.4 μM) and PPARγ(EC50=17.7 μM). It blocks TNF-α-induced NF-KB activation.Fórmula:C18H18O2Pureza:99.49% - 99.98%Cor e Forma:A Bioactive Compound Found In The Bark Of The Houpu MagnoliaPeso molecular:266.33Rosiglitazone maleate
CAS:Rosiglitazone maleate (BRL 49653) is an oral antidiabetic and potential anticancer agent.Fórmula:C22H23N3O7SPureza:99.33% - 99.51%Cor e Forma:Off-White SolidPeso molecular:473.50Oleoylethanolamide
CAS:Oleoylethanolamide (N-Oleoylethanolamide) is a high affinity endogenous agonist of PPAR-α.Fórmula:C20H39NO2Pureza:99.98%Cor e Forma:SolidPeso molecular:325.53Ref: TM-T12296
2mg35,00€5mg52,00€10mg80,00€25mg145,00€50mg250,00€100mg376,00€200mg550,00€1mL*10mM (DMSO)58,00€GW7647
CAS:GW 7647 is an effective and highly selective PPARα agonist. GW 7647 can reduce the production of nitric oxide in macrophages. Cost-effective and quality-assured.Fórmula:C29H46N2O3SPureza:99.3% - 99.34%Cor e Forma:SolidPeso molecular:502.75MK-0533
CAS:<p>MK-0533 is a novel PPARγ partial agonist for the prevention of vascular endothelial dysfunction (VED) and VED-related cardiovascular disease.</p>Fórmula:C28H24F3NO6Pureza:99.03%Cor e Forma:SoildPeso molecular:527.49Sulotroban
CAS:sulotroban is a TXA2 receptor antagonist that acts synergistically with iloprost to inhibit TXA2-dependent platelet activation.Fórmula:C16H17NO5SPureza:98.86% - 99.98%Cor e Forma:SolidPeso molecular:335.37MCC-555
CAS:MCC-555 (Isaglitazone) is a PPARα and PPARγ agonist exerting antihyperglycemic effects.Fórmula:C21H16FNO3SPureza:99.07% - 99.82%Cor e Forma:SolidPeso molecular:381.42Ref: TM-T21764
5mg66,00€10mg105,00€25mg215,00€50mg356,00€100mg530,00€500mg1.153,00€1mL*10mM (DMSO)73,00€WAY-620472
CAS:WAY-620472 is a PPAR regulator that can be used to alter the lifespan of eukaryotes.Fórmula:C23H21N5OSPureza:98.99%Cor e Forma:SolidPeso molecular:415.51CUDA
CAS:<p>CUDA is an effective soluble cyclohydrolase inhibitor with IC50 of 11.1 nM and 112 nM for mouse sEH and human sEH, respectively.</p>Fórmula:C19H36N2O3Pureza:97.585%Cor e Forma:SolidPeso molecular:340.5PPARγ-IN-3
PPARγ-IN-3 (compound 9ga), a potent and orally active PPARγ inhibitor, effectively reduces triglyceride (TG) accumulation and exhibits low cytotoxicity. Additionally, it prevents excessive body weight gain, lessens fat and liver mass, and decreases lipid accumulation in both the liver and blood. PPARγ-IN-3 holds promise for research into diet-induced obesity.Fórmula:C23H28FN7O3Cor e Forma:SolidPeso molecular:469.51Nuclear Receptor Compound Library
<p>A unique collection of 531 nuclear receptor signaling targeted compounds for high throughput and high content screening;</p>Cor e Forma:Odour SolidBenzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-
CAS:Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)- is a dual PPARα/γ agonist with EC50 of 0.358μM and 1.21μM.Fórmula:C24H23NO5SPureza:99.59%Cor e Forma:SoildPeso molecular:437.51Ref: TM-T63898
1mg185,00€5mg426,00€10mg627,00€25mg938,00€50mg1.320,00€100mg1.786,00€1mL*10mM (DMSO)472,00€Sulotroban potassium
Sulotroban potassium is a small molecule thromboxane A2 receptor (TXA2R) antagonist that can be used to study myocardial infarction and thrombosis.Fórmula:C16H16KNO5SPureza:98.02%Cor e Forma:SoildPeso molecular:373.46Lipid Metabolism Compound Library
<p>A unique collection of 492 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS).</p>Cor e Forma:Odour SolidAnti-osteoporosis agent-10
Anti-osteoporosis agent-10 is an inhibitor of osteoporosis that suppresses the formation of osteoclasts with an IC50 of 0.042 μM. It also exhibits antagonistic activity towards PPARγ, with an EC50 value of 0.75 μM.Cor e Forma:Odour SolidAnti-obesity agent 1
<p>Compound 4 (Anti-obesity agent 1) demonstrates potential for enhanced lipolysis, highlighting its anti-obesity characteristics.</p>Fórmula:C21H22N2O6Cor e Forma:SolidPeso molecular:398.409SP4f
SP4f, an activator of PPAR-γ, exhibits an EC50 value of 826 nM in HK-2 cells.Pureza:98%Cor e Forma:Odour SolidSP4e
SP4e is a PPAR-γ activator.SP4e was effective in decreasing blood glucose, total cholesterol, triglycerides and LDL levels and increasing HDL levels.Fórmula:C22H17ClN2O2S2Pureza:99.79%Cor e Forma:SoildPeso molecular:440.97(±)-CBCQ
CAS:(±)-CBCQ, an oxidation product of cannabidiol, exhibits an EC50 value of 14.7 μM for the activation of peroxisome proliferator-activated receptor γ (PPAR-γ).Fórmula:C21H28O3Cor e Forma:SolidPeso molecular:328.45E0924G
CAS:E0924G is an orally active PPARδ agonist with an EC50 of 2.82 μM. It enhances the upregulation of osteoprotegerin (OPG) expression, with an EC50 of 0.29 μM. E0924G reduces RANKL-induced osteoclast differentiation and inhibits F-actin ring formation in RAW264.7 macrophages. Additionally, E0924G modulates bone density and bone loss in models of ovariectomy (OVX) and age-related osteoporosis.Fórmula:C12H12N2O3Cor e Forma:SolidPeso molecular:232.24PPARγ agonist 15
PPARγ agonist15 (Compound 7c) functions as an agonist of PPARγ, inhibiting the expression of α-amylase (HPA) and α-glucosidase (HLAG) with IC50 values of 28.35 µM and 26.21 µM, respectively. It enhances glucose uptake in L6 myotubes and improves glucose homeostasis, insulin sensitivity, and lipid metabolism in a rat model of Streptozotocin-induced diabetes.Fórmula:C21H16N4O3S2Cor e Forma:SolidPeso molecular:436.51PPARγ agonist 16
CAS:PPARγ agonist16 (Compound 4G) is a PPARγ agonist that competitively binds to the ligand-binding domain (LBD) of PPARγ with an IC50 of 1790 nM. It reduces ear swelling in mouse models and exhibits antihyperglycemic activity in mice with Streptozotocin-induced diabetes.Fórmula:C19H14BrNO4SCor e Forma:SolidPeso molecular:432.29Mavodelpar free acid hydrochloride
<p>Mavodelpar free acid hydrochloride (Pparδ agonist HCl) is a potent PPARδ agonist.</p>Fórmula:C31H31ClFNO5Pureza:98.13%Cor e Forma:SoildPeso molecular:552.03PPAR agonist 6
PPAR agonist6 (compound 5a) acts as an agonist for PPAR, exhibiting EC50 values of 3.6 μM and 2.6 μM for PPARα and PPARβ/δ respectively. Additionally, PPAR agonist6 inhibits the transactivation of a TNFα-dependent NF-κB-driven reporter gene in L929 cells [1].Cor e Forma:Odour Solid8-iso Prostaglandin F1β
CAS:8-iso Prostaglandin F1β,inducet vasoconstrictor effects in (PA), (PV) and (MA) through the activation of TXA2R, tyrosine kinase and Rho kinase.Fórmula:C20H36O5Cor e Forma:SolidPeso molecular:356.58-iso Prostaglandin F1α
CAS:8-iso Prostaglandin F1α induces vasoconstrictor effects in (PA),(PV) and (MA) through activation of TXA2R, tyrosine kinases and Rho kinases.Fórmula:C20H36O5Cor e Forma:SolidPeso molecular:356.5CC618
CAS:CC618 is a selective PPARβ/δ antagonist with an IC50 of 10.0 μM.Fórmula:C20H15F6N3O3S2Pureza:99.94%Cor e Forma:SolidPeso molecular:523.47Ref: TM-T9767
1mg115,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)314,00€AZD-9574
CAS:AZD-9574 is a selective inhibitor of PARP1 at the sites of SSBs.Fórmula:C21H22F2N6O2Pureza:98.46% - 99.39%Cor e Forma:SolidPeso molecular:428.44GW590735
CAS:GW590735: PPARα agonist, EC50=4 nM, >500x selective over PPARδ/γ, for dyslipidemia research.Fórmula:C23H21F3N2O4SPureza:99.53%Cor e Forma:SolidPeso molecular:478.48Ref: TM-T9766
1mg95,00€5mg202,00€10mg298,00€25mg507,00€50mg730,00€100mg1.026,00€1mL*10mM (DMSO)213,00€GQ-16
CAS:GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.Fórmula:C19H16BrNO3SPureza:99.84%Cor e Forma:SolidPeso molecular:418.3Ref: TM-T21955
10mg39,00€25mg80,00€50mg116,00€100mg187,00€200mg280,00€500mg449,00€1mL*10mM (DMSO)35,00€Balaglitazone
CAS:Balaglitazone is a PPARγ agonist that regulates blood glucose and is used in studies of heart failure and myocardial infarction.Fórmula:C20H17N3O4SPureza:99.74%Cor e Forma:SolidPeso molecular:395.43CP-868388 free base
CAS:CP-868388 free base (CP-868388) is a PPARα agonist with hypolipidemic and anti-inflammatory activity and is used in the study of dyslipidemia.Fórmula:C26H33NO5Pureza:99.84%Cor e Forma:SolidPeso molecular:439.54PPAR α/PPARA Protein, Mouse, Recombinant (His)
PPAR alpha/PPARA Protein, Mouse, Recombinant (His) is expressed in E.Cor e Forma:Lyophilized PowderPeso molecular:31.49 kDa (predicted)Ref: TM-TMPY-06837
5µg115,00€10µg184,00€20µg305,00€50µg608,00€100µg1.074,00€200µg1.813,00€500µg4.440,00€PPAR α/PPARA Protein, Human, Recombinant (His)
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E.Cor e Forma:Lyophilized PowderPeso molecular:31.36 kDa (predicted)Ref: TM-TMPY-06830
5µg116,00€10µg187,00€20µg305,00€50µg608,00€100µg1.063,00€200µg1.794,00€500µg3.832,00€SR 16832
CAS:SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.Fórmula:C17H12ClN3O4Pureza:99.6%Cor e Forma:SolidPeso molecular:357.75GW0742
CAS:GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).Fórmula:C21H17F4NO3S2Pureza:99.75% - 99.85%Cor e Forma:SolidPeso molecular:471.49CDDO-Im
CAS:CDDO-Im (TP-235) is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).Fórmula:C34H43N3O3Pureza:98.3% - 99.61%Cor e Forma:SolidPeso molecular:541.72Ref: TM-TQ0120
1mg34,00€5mg74,00€10mg105,00€25mg200,00€50mg319,00€100mg485,00€500mg1.035,00€1mL*10mM (DMSO)89,00€Angeloylgomisin H
CAS:Angeloylgomisin H shows moderate cytotoxic activities with IC50 values ranging from 100 to 200 ug/mL against MCF7, HEK293 and CAL27 cell lines.Fórmula:C28H36O8Pureza:99.84% - 99.95%Cor e Forma:SolidPeso molecular:500.58Ref: TM-TN1018
1mg55,00€5mg117,00€10mg182,00€25mg306,00€50mg444,00€100mg610,00€1mL*10mM (DMSO)158,00€Cinnamyl alcohol
CAS:Cinnamyl alcohol (Styryl Carbinol) readily autoxidizes upon air exposure, and forms strong sensitizers as determined by the local lymph node assay.Fórmula:C9H10OPureza:99.00%Cor e Forma:Colourless LiquidPeso molecular:134.18SC-236
CAS:SC-236 (Sc 236) is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 μM and 17.8 μM for COX-2 and COX-1, respectively).Fórmula:C16H11ClF3N3O2SPureza:99.74%Cor e Forma:SolidPeso molecular:401.79Clofibrate
CAS:Clofibrate (Clofibrato) is an aryloxyisobutyric acid derivate with antihyperlipidemic activity.Fórmula:C12H15ClO3Pureza:98.77%Cor e Forma:Oil LiquidPeso molecular:242.70Raspberry ketone
CAS:1.Fórmula:C10H12O2Pureza:99.84% - 99.89%Cor e Forma:White Solid CrystallinePeso molecular:164.2Fisetin
CAS:Fisetin belongs to a group of natural flavonols with anti-inflammatory, antioxidant, anti-tumor, anti-aging and neuroprotective effects. Cost effective and quality assured.Fórmula:C15H10O6Pureza:94.14% - 99.05%Cor e Forma:Yellow To Brown Crystalline PowderPeso molecular:286.24Ginsenoside Rh1
CAS:Ginsenoside Rh1 (Sanchinoside B2) , one of the main constituents of Panax ginseng, exhibits anti-inflammatory effect.Fórmula:C36H62O9Pureza:99% - 99.64%Cor e Forma:SolidPeso molecular:638.87Alpinetin
CAS:Alpinetin: antibacterial, anti-inflammatory, boosts HepG2 sensitivity to CDDP, fights hepatoma/pancreatic cancer, inhibits cell growth & activates caspases.Fórmula:C16H14O4Pureza:98.39%Cor e Forma:SolidPeso molecular:270.28Oleuropein
CAS:Oleuropein is an antioxidant polyphenol isolated from olive leaf.Fórmula:C25H32O13Pureza:98% - 99.95%Cor e Forma:Brown PowderPeso molecular:540.51EPI-001
CAS:EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.Fórmula:C21H27ClO5Pureza:99% - 99.67%Cor e Forma:SolidPeso molecular:394.89Ref: TM-T6829
2mg35,00€5mg50,00€10mg77,00€25mg127,00€50mg202,00€100mg303,00€200mg449,00€1mL*10mM (DMSO)51,00€Glabridin
CAS:Glabridin aids in diabetes by reducing inflammation and glucose levels and may prevent liver cancer spread.Fórmula:C20H20O4Pureza:99.78% - 99.99%Cor e Forma:Light Yellow Powder Insoluble In WaterPeso molecular:324.37Convallatoxin
CAS:Convallatoxin is a natural product.Fórmula:C29H42O10Pureza:99.27% - 99.53%Cor e Forma:Prisms From Methanol + Ether SolidPeso molecular:550.64Elafibranor
CAS:Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) withFórmula:C22H24O4SPureza:98.42% - 98.78%Cor e Forma:SolidPeso molecular:384.49Ref: TM-T4408
2mg35,00€5mg52,00€10mg70,00€25mg110,00€50mg177,00€100mg283,00€200mg426,00€1mL*10mM (DMSO)57,00€Methyl oleanonate
CAS:3-Oxoolean-12-en-28-oic acid methyl ester is a triterpenoid PPARγ agonist isolated from Pistacia with anticancer properties.Fórmula:C31H48O3Pureza:98.99%Cor e Forma:SolidPeso molecular:468.71Gypenoside XLIX
CAS:Extracted from whole herb of Gynostemsma pentaphyllum(Thunb.)Mak.;Store the product in sealed, cool and dry conditionFórmula:C52H86O21Pureza:97.05% - 99.78%Cor e Forma:SolidPeso molecular:1047.23NPC 15199
CAS:<p>NPC 15199 (FMOC-L-Leucine) is an anti-inflammatory agent.</p>Fórmula:C21H23NO4Pureza:99.93% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:353.41AMG131
CAS:AMG131 (CHS 131) , is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, which can be used forFórmula:C21H12Cl4N2O3SPureza:99.37%Cor e Forma:SolidPeso molecular:514.21MK-886
CAS:MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP).Fórmula:C27H34ClNO2SPureza:99.23% - 99.84%Cor e Forma:SolidPeso molecular:472.08Ref: TM-T6893
1mg35,00€5mg70,00€10mg111,00€25mg216,00€50mg354,00€100mg540,00€200mg772,00€1mL*10mM (DMSO)72,00€BMS-687453
CAS:BMS-687453 is a potent and selective PPAR alpha agonist, with an EC(50) of 10 nM for human PPARalpha and approximately 410-fold selectivity vs human PPARgammaFórmula:C22H21ClN2O6Pureza:99.4%Cor e Forma:SolidPeso molecular:444.86Ref: TM-T5532
1mg44,00€2mg57,00€5mg93,00€10mg137,00€25mg268,00€50mg409,00€100mg620,00€1mL*10mM (DMSO)92,00€Oroxin A
CAS:Oroxin A (Baicalein 7-O-glucoside) has antitussive and expectorant effects.Fórmula:C21H20O10Pureza:98.05% - 99.74%Cor e Forma:SolidPeso molecular:432.38Ref: TM-T5S0788
1mg43,00€5mg87,00€10mg135,00€25mg221,00€50mg349,00€100mg507,00€200mg720,00€1mL*10mM (DMSO)95,00€G3335 Acetate
G3335 Acetate was discovered to be a novel PPARgamma antagonist.Fórmula:C18H23N3O7Pureza:99.75%Cor e Forma:SolidPeso molecular:393.39Ref: TM-T21598L
5mg55,00€10mg82,00€25mg126,00€50mg182,00€100mg273,00€200mg409,00€500mg677,00€1mL*10mM (DMSO)79,00€LJ570
CAS:LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)Fórmula:C27H22O3Pureza:99.64%Cor e Forma:SolidPeso molecular:394.46Ref: TM-T8374
1mg138,00€2mg202,00€5mg311,00€10mg445,00€25mg680,00€50mg888,00€100mg1.234,00€500mg2.475,00€1mL*10mM (DMSO)334,00€Ciprofibrate
CAS:Ciprofibrate (Win35833) is a fibrate derivative with antilipidemic activity.Fórmula:C13H14Cl2O3Pureza:99.63% - >99.99%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:289.15L-165041
CAS:L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = 9 nM, EC50 = ~500 nM ,respectively)Fórmula:C22H26O7Pureza:97.97%Cor e Forma:SolidPeso molecular:402.44GSK0660
CAS:GSK0660 is an antagonist and inverse agonist of PPARβ/δ.Fórmula:C19H18N2O5S2Pureza:99.26% - ≥95%Cor e Forma:SolidPeso molecular:418.49Ref: TM-T2674
2mg44,00€5mg65,00€10mg99,00€25mg175,00€50mg349,00€100mg520,00€500mg1.134,00€1mL*10mM (DMSO)65,00€OPHIOPOGONIN D
CAS:Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.Fórmula:C44H70O16Pureza:99.46% - ≥95%Cor e Forma:SolidPeso molecular:855.02XMD8-87
CAS:XMD8-87 (ACK1-B19), a TNK2 inhibitor, strongly blocks TNK2 phosphorylation and mutations in tumors.Fórmula:C24H27N7O2Pureza:98.05% - 99.89%Cor e Forma:SolidPeso molecular:445.52Ref: TM-T3709
2mg47,00€5mg73,00€10mg103,00€25mg188,00€50mg306,00€100mg507,00€500mg1.225,00€1mL*10mM (DMSO)88,00€GW 501516
CAS:GW 501516 (Endurobol) is a effective and highly specifc PPARβ/δ agonist (EC50: 1 nM), with 1000-fold selectivity over hPPARα/γ.Fórmula:C21H18F3NO3S2Pureza:98.91% - 99.64%Cor e Forma:White SolidPeso molecular:453.50XMD16-5
CAS:XMD16-5 blocks TNK2, linked to advanced lung/prostate cancers and breast cancer metastasis in mice; disrupts signaling in several tumors.Fórmula:C23H24N6O2Pureza:98.89% - 99.98%Cor e Forma:SolidPeso molecular:416.48Ref: TM-T3710
1mg44,00€2mg56,00€5mg90,00€10mg144,00€25mg225,00€50mg415,00€100mg615,00€500mg1.311,00€1mL*10mM (DMSO)90,00€Astaxanthin
CAS:<p>Astaxanthin, a keto-carotenoid and xanthophyll, offers antioxidant benefits, present in red aquatic species, and used as a colorant in animal feed.</p>Fórmula:C40H52O4Pureza:95.1% - 99.79%Cor e Forma:Needles From Acetone/Light Petroleum SolidPeso molecular:596.84Agrimol B
CAS:1. Agrimol B is a main active ingredient isolated from Agrimonia pilosa Ledeb.Fórmula:C37H46O12Pureza:99.06% - ≥95%Cor e Forma:SolidPeso molecular:682.75(E/Z)-Elafibranor
CAS:<p>GFT505 (Elafibranor) (Elafibranor) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.</p>Fórmula:C22H24O4SPureza:98.36%Cor e Forma:SolidPeso molecular:384.49Avicularin
CAS:Avicularin reduces inflammation via ERK pathway in RAW 264.7 cells and hinders lipid buildup in adipocytes by limiting glucose uptake and fatty acid synthesis.Fórmula:C20H18O11Pureza:97.02% - 99.94%Cor e Forma:White PowderPeso molecular:434.35Ref: TM-T6S0117
1mg58,00€5mg97,00€10mg160,00€25mg283,00€50mg418,00€100mg615,00€200mg878,00€1mL*10mM (DMSO)111,00€Bilobetin
CAS:Bilobetin ameliorates insulin resistance by PKA-mediated phosphorylation of PPARα in rats fed a high-fat diet.Fórmula:C31H20O10Pureza:97.74% - 99.69%Cor e Forma:SolidPeso molecular:552.48Ref: TM-T4S2128
1mg47,00€2mg70,00€5mg144,00€10mg250,00€25mg424,00€50mg613,00€100mg843,00€1mL*10mM (DMSO)187,00€Choline Fenofibrate
CAS:<p>Choline Fenofibrate (Trilipix) is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and prodrug with antihyperlipidemic</p>Fórmula:C22H28ClNO5Pureza:98.82%Cor e Forma:SolidPeso molecular:421.91Pirinixic Acid
CAS:Pirinixic Acid (NSC 310038) is a synthetic thiacetic acid derivative used in biomedical research, a peroxisome proliferator that activates specific PPAR.Fórmula:C14H14ClN3O2SPureza:98.27% - 99.92%Cor e Forma:SolidPeso molecular:323.8Ref: TM-T2269
1g350,00€10mg48,00€25mg64,00€50mg79,00€100mg105,00€200mg148,00€500mg236,00€1mL*10mM (DMSO)47,00€Adelmidrol
CAS:Adelmidrol is an anti-inflammatory ethanolamide derivative of azelaic acid.Fórmula:C13H26N2O4Pureza:99.35% - 99.73%Cor e Forma:SolidPeso molecular:274.36Rosiglitazone hydrochloride
CAS:Rosiglitazone hydrochloride (BRL-49653 HCl) is a blood glucose-lowering drugs, stimulating insulin secretion by binding to the PPAR receptors in fat cells.Fórmula:C18H19N3O3S·HClPureza:99.63% - 99.79%Cor e Forma:SolidPeso molecular:393.89GW1929
CAS:<p>GW1929 is a potent PPAR-γ agonist (pKi: 8.84 for human PPAR-γ; pEC50s of 8.56 and 8.27 for human and murine PPAR-γ).</p>Fórmula:C30H29N3O4Pureza:98.1% - 98.21%Cor e Forma:SolidPeso molecular:495.57GSK3787
CAS:GSK3787 is a specific and irreversible PPARδ inhibitor（pIC50= 6.6）.Fórmula:C15H12ClF3N2O3SPureza:98% - 99.56%Cor e Forma:SolidPeso molecular:392.78Ref: TM-T1941
5mg55,00€10mg87,00€25mg173,00€50mg309,00€100mg520,00€500mg1.111,00€1mL*10mM (DMSO)55,00€Bocidelpar
CAS:Bocidelpar is a modulator of PPARδ with an EC50 of 7.80 nM and improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy muscle cells.Fórmula:C25H27F3N2O3Pureza:97.77%Cor e Forma:SolidPeso molecular:460.49Ref: TM-T39516
1mg114,00€5mg260,00€10mg389,00€25mg703,00€50mg1.054,00€100mg1.468,00€1mL*10mM (DMSO)264,00€
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