
Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(38 produtos)
- Cisteína Protease(111 produtos)
- DPP-4(27 produtos)
- Glutaminase(46 produtos)
- HIV Protease(507 produtos)
- PAI-1(26 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(55 produtos)
- Proteassoma(86 produtos)
- Protease serina(54 produtos)
- p97(15 produtos)
Exibir 3 mais subcategorias
Foram encontrados 977 produtos de "Proteases/Proteassoma"
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SFTI-1
CAS:SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.Fórmula:C67H104N18O18S2Cor e Forma:SolidPeso molecular:1513.78Tilpisertib fosmecarbil TFA
CAS:Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.Fórmula:C37H37ClF3N8O9PCor e Forma:SolidPeso molecular:861.16MMP-9/MMP-13 Inhibitor I
CAS:MMP-9/MMP-13 Inhibitor I is a dual inhibitor of MMP-9 and MMP-13 with IC50 of both 0.9 nM.Fórmula:C25H25N3O6SCor e Forma:SolidPeso molecular:495.55HCV-IN-41
CAS:HCV-IN-41: potent HCV inhibitor; EC50 - 0.006762 nM (1b), 5.183 nM (2a), 1.365 nM (3a), 142.2 nM (4a); hinders RNA replication.Fórmula:C48H56N6O8Cor e Forma:SolidPeso molecular:844.99VPLSLYSG
CAS:VPLSLYSG, an octapeptide, degraded by MMP-9, MMP-1, MMP-2; potential MMP substrate uses.Fórmula:C39H62N8O12Cor e Forma:SolidPeso molecular:834.96Obtusifolin-2-O-glucoside
CAS:Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].Fórmula:C22H22O10Cor e Forma:SolidPeso molecular:446.4GSK2336805
CAS:GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.Fórmula:C42H52N8O8Cor e Forma:SolidPeso molecular:796.91BMS 180742
CAS:BMS 180742 is an exosite inhibitor of thrombin.Fórmula:C67H93N11O22Pureza:98%Cor e Forma:SolidPeso molecular:1404.526-Acetylnimbandiol
CAS:6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.Fórmula:C28H34O8Cor e Forma:SolidPeso molecular:498.56Radalbuvir
CAS:Radalbuvir (GS-9669) is an investigational antiviral agent for the treatment of hepatitis C virus (HCV) infection as an NS5B inhibitor.Fórmula:C30H41NO6SCor e Forma:SolidPeso molecular:543.71Tiprelestat
CAS:Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.Fórmula:C254H416N72O75S10Cor e Forma:SolidPeso molecular:5999.09Bortezomib analog
Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.Cor e Forma:Odour SolidCarboxypeptidase C
CAS:Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.Cor e Forma:SolidCathepsin L-IN-3
CAS:Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.Fórmula:C41H49N7O4SCor e Forma:SolidPeso molecular:735.94N-CBZ-Phe-Arg-AMC TFA
N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.Fórmula:C35H37F3N6O8Pureza:99.88%Cor e Forma:SolidPeso molecular:726.7Chymotrypsinogen
CAS:Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .Cor e Forma:SolidTyrosinase-IN-36
Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.Cor e Forma:Odour SolidPlasma kallikrein-IN-1
CAS:Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.Fórmula:C23H25F2N7OCor e Forma:SolidPeso molecular:453.498TAPI1 acetate
TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .Fórmula:C28H41N5O7Pureza:98.82% - 99.94%Cor e Forma:SolidPeso molecular:559.65AMG-222
CAS:AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.Fórmula:C32H39N9O3Cor e Forma:SolidPeso molecular:597.71ADAM8-IN-1
CAS:ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.
Fórmula:C44H44Br4N6O12S2Cor e Forma:SolidPeso molecular:1232.6Ellipyrone B
Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50Fórmula:C25H38O7Cor e Forma:SolidPeso molecular:450.57Suc-AAP-Abu-pNA
CAS:Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Fórmula:C25H34N6O9Cor e Forma:SolidPeso molecular:562.57Tyrosinase-IN-26
Tyrosinase-IN-26 (compound 13) is a non-competitive inhibitor of tyrosinase, with an IC50 value of 68.86 µM. It is capable of inhibiting melanin production.Fórmula:C25H24N2O6Peso molecular:448.16344HCV-IN-4
CAS:HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.Fórmula:C52H58FN9O8Pureza:98%Cor e Forma:SolidPeso molecular:956.07MMP-3 Inhibitor
CAS:MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.Fórmula:C27H46N10O9SPureza:98.87%Cor e Forma:SolidPeso molecular:686.78Ref: TM-T37048
1mg77,00€5mg197,00€1mL*10mM (DMSO)210,00€10mg294,00€25mg497,00€50mg717,00€100mg982,00€500mg1.998,00€CRA-2059 hydrochloride
CRA-2059 hydrochloride is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].Cor e Forma:SolidTyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Fórmula:C19H14BrClN4OCor e Forma:SolidPeso molecular:429.7Ichorcumab
CAS:Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.Cor e Forma:LiquidEnzyme-IN-1
CAS:Enzyme-IN-1(compound 1)为基于肽的N端亲核试剂(Ntn)水解酶抑制剂,特别针对20S蛋白酶体的糜胰蛋白酶样活性(CT-L)进行抑制,可能展现出抗炎特性。Fórmula:C36H50N4O7Cor e Forma:SolidPeso molecular:650.8Relacatib
CAS:Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.Fórmula:C27H32N4O6SCor e Forma:SolidPeso molecular:540.64LM11
LM11 is a transglutaminase 2 (TG2) inhibitor that exhibits activity against glioblastoma cells by maintaining TG2 in a cytotoxic conformational state.
Fórmula:C26H18Cl2N4O5Peso molecular:536.06543Stevia Powder
Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.Cor e Forma:Odour Solid15,16-Dihydrotanshindiol C
15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.Fórmula:C18H18O5Cor e Forma:SolidPeso molecular:314.337Lysine 4-nitroanilide
CAS:Lysine 4-nitroanilide is a bioactive chemical.Fórmula:C12H18N4O3Cor e Forma:SolidPeso molecular:266.3Histatin 5 (TFA)(115966-68-2,free)
Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μMFórmula:C135H196F3N51O35Pureza:98%Cor e Forma:SolidPeso molecular:3150.326,6′-Dihydroxythiobinupharidine
CAS:6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-foldFórmula:C30H42N2O4SCor e Forma:SolidPeso molecular:526.73Ac-PAL-AMC
CAS:Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.Fórmula:C26H34N4O6Cor e Forma:SolidPeso molecular:498.57Talabostat
CAS:Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.Fórmula:C9H19BN2O3Cor e Forma:SolidPeso molecular:214.07Pseudostellarin G
CAS:Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.Fórmula:C42H56N8O9Cor e Forma:SolidPeso molecular:816.94Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS:Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effectFórmula:C47H64N14O10Cor e Forma:SolidPeso molecular:985.1Sadopeptins B
Sadopeptins B, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].Fórmula:C48H69N9O13SCor e Forma:SolidPeso molecular:1012.185-epi-Arvestonate A
CAS:5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.Fórmula:C16H26O5Cor e Forma:SolidPeso molecular:298.37VD2173
CAS:VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.Fórmula:C31H45N9O6SCor e Forma:SolidPeso molecular:671.81HCVP-IN-1
CAS:HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.Fórmula:C30H34FN5O3Cor e Forma:SolidPeso molecular:531.632NIM811
CAS:NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.Fórmula:C62H111N11O12Pureza:98%Cor e Forma:SolidPeso molecular:1202.635C-telopeptide TFA
C-telopeptide TFA is a cross-linked peptide of type I collagen, released during bone resorption, and is associated with bone mineral density (BMD).Cor e Forma:Odour SolidNostosin G
Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).Fórmula:C25H33N5O6Cor e Forma:SolidPeso molecular:499.56Talopeptin
CAS:Talopeptin is a specific thermolysin inhibitor.Fórmula:C23H34N3O10PPureza:98%Cor e Forma:SolidPeso molecular:543.50Cerpegin
CAS:Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.Fórmula:C10H11NO3Cor e Forma:SolidPeso molecular:193.24-Epianhydrochlortetracycline (hydrochloride)
CAS:4-Epianhydrochlortetracycline (hydrochloride) can be used in related research in the field of life sciences.Fórmula:C22H22Cl2N2O7Cor e Forma:SolidPeso molecular:497.33RXP470
CAS:RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).Fórmula:C35H35BrClN4O10PCor e Forma:SolidPeso molecular:818GSK2818713
CAS:GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.Fórmula:C46H56N8O8Cor e Forma:SolidPeso molecular:849.002Zetomipzomib maleate
CAS:Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.Fórmula:C34H46N4O12Cor e Forma:SolidPeso molecular:702.758ZG36
ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrialCor e Forma:Odour SolidAcetyl-Calpastatin(184-210)(human) TFA
Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.Fórmula:C144H231F3N36O46SCor e Forma:SolidPeso molecular:3291.65Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2
CAS:Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).Fórmula:C49H68N14O12SCor e Forma:SolidPeso molecular:1077.22Hepcidin-1 (mouse)
CAS:Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.Fórmula:C111H169N31O35S8Cor e Forma:SolidPeso molecular:2754.24S62798
CAS:S62798 is a highly potent and selective compound that inhibits activated thrombin activatable fibrinolysis inhibitor (TAFIa) with an IC50 value of 6 mM.Fórmula:C20H28FN4O4PCor e Forma:SolidPeso molecular:438.44Fibrinogen-Binding Peptide
CAS:Fibrinogen-binding peptide mimics vitronectin site and activates platelets; thrombin turns it to fibrin.Fórmula:C25H39N7O8Pureza:98%Cor e Forma:SolidPeso molecular:565.62Befovacimab
CAS:Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.Cor e Forma:LiquidMMP-9-IN-6
CAS:MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.Fórmula:C25H19NO2Pureza:98.96%Cor e Forma:SoildPeso molecular:365.42Sofigatran
CAS:Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.Fórmula:C24H44N4O4SCor e Forma:SolidPeso molecular:484.7GPLGLAGGWGERDGS
CAS:GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.Fórmula:C61H93N19O21Cor e Forma:SolidPeso molecular:1428.51TP0597850
CAS:TP0597850, a selective MMP2 inhibitor with an IC50 value of 0.22 nM, demonstrates a prolonged dissociation half-life from MMP2 (t1/2 = 265 minutes) [1].Fórmula:C41H57N9O13SCor e Forma:SolidPeso molecular:916.01Sadopeptins A
Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].Fórmula:C49H71N9O13SCor e Forma:SolidPeso molecular:1026.21Activated Protein C (390-404), human
CAS:Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.Fórmula:C91H130N22O23Pureza:98%Cor e Forma:SolidPeso molecular:1900.14Sofosbuvir impurity I
Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Fórmula:C21H27FN3O9PPureza:98%Cor e Forma:SolidPeso molecular:515.43Ac-PLVE-FMK
CAS:Ac-PLVE-FMK (Ac-Pro-Leu-Val-Glu(OMe)-CH2F), a tetrapeptidyl fluoromethylketone (FMKs), serves as a cathepsin inhibitor. It is utilized in cancer research [1].Fórmula:C25H41FN4O7Pureza:98%Cor e Forma:SolidPeso molecular:528.61GCPII-IN-1
CAS:GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.
Fórmula:C12H21N3O7Cor e Forma:SolidPeso molecular:319.314Chetoseminudin B
CAS:Chetoseminudin B exhibits inhibitory activity against mushroom tyrosinase, with an IC 50 value of 31.7 μM [1].Fórmula:C17H21N3O3S2Cor e Forma:SolidPeso molecular:379.5N-CBZ-Phe-Arg-AMC
CAS:Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.Fórmula:C33H36N6O6Pureza:98%Cor e Forma:White To Off-White PowderPeso molecular:612.68PM 102
CAS:Peptide that reverses the anticoagulant effect of heparin. Potently binds heparin (Kd = 36 nM in vitro).Fórmula:C235H425N111O64Pureza:98%Cor e Forma:SolidPeso molecular:5830Ellipyrone A
Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).Fórmula:C25H34O8Cor e Forma:SolidPeso molecular:462.53Dutogliptin
CAS:Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.Fórmula:C10H20BN3O3Pureza:98%Cor e Forma:SolidPeso molecular:241.10Micropeptin 478A
CAS:Micropeptin 478A is a plasmin inhibitor from the Cyanobacterium Microcystis aeruginosa.Fórmula:C40H62ClN9O15SPureza:98%Cor e Forma:SolidPeso molecular:976.49Acetyl-Calpastatin(184-210)(human)
CAS:Calpain inhibitor, Ki 0.2 nM for calpain I/II, doesn't affect papain/trypsin/cat L. Raises Aβ42, Aβ40 secretion & Aβ42/Aβ40 ratio.Fórmula:C142H230N36O44SPureza:98%Cor e Forma:SolidPeso molecular:3177.65Talabostat isomer mesylate
Talabostat isomer mesylate, a PT100/Val-boroPro variant, is a potent oral DPP-IV inhibitor (Ki: 0.18 nM).Fórmula:C10H23BN2O6SPureza:98%Cor e Forma:SolidPeso molecular:310.18FFAGLDD
"FFAGLDD: MMP9 peptide for controlled DOX delivery inside cells."Fórmula:C37H49N7O12Pureza:98%Cor e Forma:SolidPeso molecular:783.82Aristololactam IIIa
CAS:Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.Fórmula:C16H9NO4Cor e Forma:SolidPeso molecular:279.25AP-C2
CAS:AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.Fórmula:C18H16N4SPureza:99.99%Cor e Forma:SoildPeso molecular:320.41Leptosin D
CAS:Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)Fórmula:C25H24N4O3S2Cor e Forma:SolidPeso molecular:492.61C-telopeptide
CAS:C-telopeptide from type I collagen is released during bone resorption; it correlates with bone mineral density.Fórmula:C34H56N14O13Pureza:98%Cor e Forma:SolidPeso molecular:868.9Alisporivir
CAS:Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.Fórmula:C63H113N11O12Pureza:99.95%Cor e Forma:SolidPeso molecular:1216.64NS5A-IN-1
NS5A-IN-1 is a proagent of the HCV NS5A inhibitor Pibrentasvir (ABT-530).Fórmula:C72H86F5N10O14PCor e Forma:SolidPeso molecular:1441.48(-)-Taxifolin
CAS:(-)-Taxifolin, less active enantiomer with anti-tyrosinase, collagenase inhibition (IC50 = 193.3 μM), antifibrotic, antioxidant properties.Fórmula:C15H12O7Cor e Forma:SolidPeso molecular:304.25JC-10
CAS:JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.Fórmula:C25H29Cl2IN4Pureza:95%Cor e Forma:SolidPeso molecular:583.34Paritaprevir dihydrate
CAS:Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.Fórmula:C40H47N7O9SCor e Forma:SolidPeso molecular:801.91Linagliptin Methyldimer
CAS:Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.Fórmula:C50H56N16O4Pureza:99.91%Cor e Forma:SolidPeso molecular:945.08FFAGLDD TFA
FFAGLDD TFA: MMP9 peptide for controlled DOX delivery to cytoplasm.Fórmula:C39H50F3N7O14Pureza:98%Cor e Forma:SolidPeso molecular:897.85Mipomersen
CAS:Mipomersen (ISIS 301012) is an antisense oligo that inhibits apoB, has anti-HCV properties, and is researched for HoFH.Cor e Forma:SolidPeso molecular:7177AR-H067637
CAS:AR-H067637 is a fast-acting, reversible thrombin inhibitor with K(i) 2-4 nM; it also reduces clot-bound thrombin and platelet activation/aggregation.Fórmula:C21H21ClF2N4O4Cor e Forma:SolidPeso molecular:466.87Procizumab
Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.Cor e Forma:Odour LiquidRivulariapeptolides 1121
Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).Fórmula:C56H83N9O15Cor e Forma:SolidPeso molecular:1122.31Ac-DEMEEC-OH
CAS:Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.Fórmula:C29H44N6O16S2Cor e Forma:SolidPeso molecular:796.82PPACK II
CAS:PPACK II is an irreversible and specific glandular and plasma kallikreins inhibitor [1] .Fórmula:C25H33ClN6O3Cor e Forma:SolidPeso molecular:501.02Rivulariapeptolides 988
Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).Fórmula:C50H68N8O13Cor e Forma:SolidPeso molecular:989.12Nitidanin
Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.Fórmula:C21H24O8Cor e Forma:SolidPeso molecular:404.415Sofosbuvir impurity A
CAS:Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.Fórmula:C22H29FN3O9PPureza:98%Cor e Forma:SolidPeso molecular:529.45AL-611
CAS:AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).
Fórmula:C25H33F2N6O8PCor e Forma:SolidPeso molecular:614.544

