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Proteases/Proteassoma

Proteases/Proteassoma

Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.

Subcategorias de "Proteases/Proteassoma"

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Foram encontrados 977 produtos de "Proteases/Proteassoma"

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  • SFTI-1

    CAS:
    SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.
    Fórmula:C67H104N18O18S2
    Cor e Forma:Solid
    Peso molecular:1513.78

    Ref: TM-TP2622

    10mg
    A consultar
    50mg
    A consultar
  • Tilpisertib fosmecarbil TFA

    CAS:
    Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.
    Fórmula:C37H37ClF3N8O9P
    Cor e Forma:Solid
    Peso molecular:861.16

    Ref: TM-T88817

    10mg
    A consultar
    50mg
    A consultar
  • MMP-9/MMP-13 Inhibitor I

    CAS:
    MMP-9/MMP-13 Inhibitor I is a dual inhibitor of MMP-9 and MMP-13 with IC50 of both 0.9 nM.
    Fórmula:C25H25N3O6S
    Cor e Forma:Solid
    Peso molecular:495.55

    Ref: TM-T37172

    25mg
    740,00€
  • HCV-IN-41

    CAS:
    HCV-IN-41: potent HCV inhibitor; EC50 - 0.006762 nM (1b), 5.183 nM (2a), 1.365 nM (3a), 142.2 nM (4a); hinders RNA replication.
    Fórmula:C48H56N6O8
    Cor e Forma:Solid
    Peso molecular:844.99

    Ref: TM-T74625

    5mg
    A consultar
    50mg
    A consultar
  • VPLSLYSG

    CAS:
    VPLSLYSG, an octapeptide, degraded by MMP-9, MMP-1, MMP-2; potential MMP substrate uses.
    Fórmula:C39H62N8O12
    Cor e Forma:Solid
    Peso molecular:834.96

    Ref: TM-T76618

    5mg
    A consultar
    50mg
    A consultar
  • Obtusifolin-2-O-glucoside

    CAS:
    Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].
    Fórmula:C22H22O10
    Cor e Forma:Solid
    Peso molecular:446.4

    Ref: TM-T75572

    5mg
    A consultar
    50mg
    A consultar
  • GSK2336805

    CAS:
    GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.
    Fórmula:C42H52N8O8
    Cor e Forma:Solid
    Peso molecular:796.91

    Ref: TM-T27461

    25mg
    2.178,00€
    50mg
    2.862,00€
    100mg
    3.870,00€
  • BMS 180742

    CAS:
    BMS 180742 is an exosite inhibitor of thrombin.
    Fórmula:C67H93N11O22
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1404.52

    Ref: TM-T25164

    25mg
    1.369,00€
  • 6-Acetylnimbandiol

    CAS:
    6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.
    Fórmula:C28H34O8
    Cor e Forma:Solid
    Peso molecular:498.56

    Ref: TM-T75506

    5mg
    A consultar
    50mg
    A consultar
  • Radalbuvir

    CAS:
    Radalbuvir (GS-9669) is an investigational antiviral agent for the treatment of hepatitis C virus (HCV) infection as an NS5B inhibitor.
    Fórmula:C30H41NO6S
    Cor e Forma:Solid
    Peso molecular:543.71

    Ref: TM-T34254

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Tiprelestat

    CAS:
    Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.
    Fórmula:C254H416N72O75S10
    Cor e Forma:Solid
    Peso molecular:5999.09

    Ref: TM-T73657

    5mg
    A consultar
    50mg
    A consultar
  • Bortezomib analog


    Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.
    Cor e Forma:Odour Solid

    Ref: TM-T200528

    10mg
    A consultar
    50mg
    A consultar
  • Carboxypeptidase C

    CAS:
    Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.
    Cor e Forma:Solid

    Ref: TM-T76168

    5mg
    A consultar
    50mg
    A consultar
  • Cathepsin L-IN-3

    CAS:
    Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.
    Fórmula:C41H49N7O4S
    Cor e Forma:Solid
    Peso molecular:735.94

    Ref: TM-TP2558

    10mg
    A consultar
    50mg
    A consultar
  • N-CBZ-Phe-Arg-AMC TFA


    N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.
    Fórmula:C35H37F3N6O8
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:726.7

    Ref: TM-T76010

    1mg
    51,00€
    5mg
    99,00€
    10mg
    160,00€
    25mg
    314,00€
    50mg
    498,00€
  • Chymotrypsinogen

    CAS:
    Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .
    Cor e Forma:Solid

    Ref: TM-T76157

    5mg
    A consultar
    50mg
    A consultar
  • Tyrosinase-IN-36


    Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.
    Cor e Forma:Odour Solid

    Ref: TM-T200699

    10mg
    A consultar
    50mg
    A consultar
  • Plasma kallikrein-IN-1

    CAS:
    Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.
    Fórmula:C23H25F2N7O
    Cor e Forma:Solid
    Peso molecular:453.498

    Ref: TM-T40312

    5mg
    873,00€
  • TAPI1 acetate


    TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .
    Fórmula:C28H41N5O7
    Pureza:98.82% - 99.94%
    Cor e Forma:Solid
    Peso molecular:559.65

    Ref: TM-T6009L

    1mg
    560,00€
    5mg
    1.198,00€
    10mg
    1.611,00€
    25mg
    2.385,00€
    50mg
    3.222,00€
  • AMG-222

    CAS:
    AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.
    Fórmula:C32H39N9O3
    Cor e Forma:Solid
    Peso molecular:597.71

    Ref: TM-T29970

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • ADAM8-IN-1

    CAS:

    ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.

    Fórmula:C44H44Br4N6O12S2
    Cor e Forma:Solid
    Peso molecular:1232.6

    Ref: TM-T73998

    5mg
    A consultar
    50mg
    A consultar
  • Ellipyrone B


    Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50
    Fórmula:C25H38O7
    Cor e Forma:Solid
    Peso molecular:450.57

    Ref: TM-T75493

    5mg
    A consultar
    50mg
    A consultar
  • Suc-AAP-Abu-pNA

    CAS:
    Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,
    Fórmula:C25H34N6O9
    Cor e Forma:Solid
    Peso molecular:562.57

    Ref: TM-T36351

    1mg
    132,00€
  • Tyrosinase-IN-26


    Tyrosinase-IN-26 (compound 13) is a non-competitive inhibitor of tyrosinase, with an IC50 value of 68.86 µM. It is capable of inhibiting melanin production.
    Fórmula:C25H24N2O6
    Peso molecular:448.16344

    Ref: TM-T209469

    10mg
    A consultar
    50mg
    A consultar
  • HCV-IN-4

    CAS:
    HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.
    Fórmula:C52H58FN9O8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:956.07

    Ref: TM-TP1468

    100mg
    A consultar
    500mg
    A consultar
  • MMP-3 Inhibitor

    CAS:
    MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.
    Fórmula:C27H46N10O9S
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:686.78

    Ref: TM-T37048

    1mg
    77,00€
    5mg
    197,00€
    1mL*10mM (DMSO)
    210,00€
    10mg
    294,00€
    25mg
    497,00€
    50mg
    717,00€
    100mg
    982,00€
    500mg
    1.998,00€
  • CRA-2059 hydrochloride


    CRA-2059 hydrochloride is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].
    Cor e Forma:Solid

    Ref: TM-T38051

    5mg
    315,00€
    10mg
    492,00€
    25mg
    960,00€
  • Tyrosinase-IN-34


    Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.
    Fórmula:C19H14BrClN4O
    Cor e Forma:Solid
    Peso molecular:429.7

    Ref: TM-T89968

    10mg
    A consultar
    50mg
    A consultar
  • Ichorcumab

    CAS:
    Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.
    Cor e Forma:Liquid

    Ref: TM-T9901A-779

    1mg
    A consultar
    5mg
    A consultar
  • Enzyme-IN-1

    CAS:
    Enzyme-IN-1(compound 1)为基于肽的N端亲核试剂(Ntn)水解酶抑制剂,特别针对20S蛋白酶体的糜胰蛋白酶样活性(CT-L)进行抑制,可能展现出抗炎特性。
    Fórmula:C36H50N4O7
    Cor e Forma:Solid
    Peso molecular:650.8

    Ref: TM-T74878

    5mg
    A consultar
    50mg
    A consultar
  • Relacatib

    CAS:
    Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.
    Fórmula:C27H32N4O6S
    Cor e Forma:Solid
    Peso molecular:540.64

    Ref: TM-T40463

    5mg
    1.773,00€
  • LM11


    LM11 is a transglutaminase 2 (TG2) inhibitor that exhibits activity against glioblastoma cells by maintaining TG2 in a cytotoxic conformational state.

    Fórmula:C26H18Cl2N4O5
    Peso molecular:536.06543

    Ref: TM-T209326

    10mg
    A consultar
    50mg
    A consultar
  • Stevia Powder


    Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.
    Cor e Forma:Odour Solid

    Ref: TM-TN8189

    10mg
    A consultar
    50mg
    A consultar
  • 15,16-Dihydrotanshindiol C


    15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.
    Fórmula:C18H18O5
    Cor e Forma:Solid
    Peso molecular:314.337

    Ref: TM-T123985

    1mg
    A consultar
    5mg
    A consultar
  • Lysine 4-nitroanilide

    CAS:
    Lysine 4-nitroanilide is a bioactive chemical.
    Fórmula:C12H18N4O3
    Cor e Forma:Solid
    Peso molecular:266.3

    Ref: TM-T33046

    100mg
    A consultar
    500mg
    A consultar
  • Histatin 5 (TFA)(115966-68-2,free)


    Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM
    Fórmula:C135H196F3N51O35
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3150.32

    Ref: TM-TP1446

    1mg
    159,00€
    5mg
    532,00€
    10mg
    832,00€
    25mg
    1.489,00€
    50mg
    2.247,00€
  • 6,6′-Dihydroxythiobinupharidine

    CAS:
    6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-fold
    Fórmula:C30H42N2O4S
    Cor e Forma:Solid
    Peso molecular:526.73

    Ref: TM-T79978

    5mg
    A consultar
    50mg
    A consultar
  • Ac-PAL-AMC

    CAS:
    Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.
    Fórmula:C26H34N4O6
    Cor e Forma:Solid
    Peso molecular:498.57

    Ref: TM-T37421

    1mg
    241,00€
    5mg
    945,00€
    10mg
    1.665,00€
  • Talabostat

    CAS:
    Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.
    Fórmula:C9H19BN2O3
    Cor e Forma:Solid
    Peso molecular:214.07

    Ref: TM-T37861

    5mg
    100,00€
    10mg
    148,00€
    50mg
    545,00€
  • Pseudostellarin G

    CAS:
    Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.
    Fórmula:C42H56N8O9
    Cor e Forma:Solid
    Peso molecular:816.94

    Ref: TM-TP2861

    10mg
    A consultar
    50mg
    A consultar
  • Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2

    CAS:
    Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect
    Fórmula:C47H64N14O10
    Cor e Forma:Solid
    Peso molecular:985.1

    Ref: TM-T76347

    5mg
    A consultar
    50mg
    A consultar
  • Sadopeptins B


    Sadopeptins B, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].
    Fórmula:C48H69N9O13S
    Cor e Forma:Solid
    Peso molecular:1012.18

    Ref: TM-T75624

    5mg
    A consultar
    50mg
    A consultar
  • 5-epi-Arvestonate A

    CAS:
    5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.
    Fórmula:C16H26O5
    Cor e Forma:Solid
    Peso molecular:298.37

    Ref: TM-T75535

    5mg
    A consultar
    50mg
    A consultar
  • VD2173

    CAS:
    VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.
    Fórmula:C31H45N9O6S
    Cor e Forma:Solid
    Peso molecular:671.81

    Ref: TM-T74390

    5mg
    A consultar
    50mg
    A consultar
  • HCVP-IN-1

    CAS:
    HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.
    Fórmula:C30H34FN5O3
    Cor e Forma:Solid
    Peso molecular:531.632

    Ref: TM-T41002

    5mg
    873,00€
  • NIM811

    CAS:
    NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.
    Fórmula:C62H111N11O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1202.635

    Ref: TM-T12226

    5mg
    A consultar
  • C-telopeptide TFA


    C-telopeptide TFA is a cross-linked peptide of type I collagen, released during bone resorption, and is associated with bone mineral density (BMD).
    Cor e Forma:Odour Solid

    Ref: TM-TP3945

    10mg
    A consultar
    50mg
    A consultar
  • Nostosin G


    Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).
    Fórmula:C25H33N5O6
    Cor e Forma:Solid
    Peso molecular:499.56

    Ref: TM-T75647

    5mg
    A consultar
    50mg
    A consultar
  • Talopeptin

    CAS:
    Talopeptin is a specific thermolysin inhibitor.
    Fórmula:C23H34N3O10P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:543.50

    Ref: TM-T26248

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Cerpegin

    CAS:
    Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.
    Fórmula:C10H11NO3
    Cor e Forma:Solid
    Peso molecular:193.2

    Ref: TM-TN8223

    10mg
    A consultar
    50mg
    A consultar
  • 4-Epianhydrochlortetracycline (hydrochloride)

    CAS:
    4-Epianhydrochlortetracycline (hydrochloride) can be used in related research in the field of life sciences.
    Fórmula:C22H22Cl2N2O7
    Cor e Forma:Solid
    Peso molecular:497.33

    Ref: TM-T35950

    1mg
    374,00€
  • RXP470

    CAS:
    RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).
    Fórmula:C35H35BrClN4O10P
    Cor e Forma:Solid
    Peso molecular:818

    Ref: TM-T28633

    5mg
    4.626,00€
  • GSK2818713

    CAS:
    GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.
    Fórmula:C46H56N8O8
    Cor e Forma:Solid
    Peso molecular:849.002

    Ref: TM-T38858

    5mg
    922,00€
  • Zetomipzomib maleate

    CAS:
    Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.
    Fórmula:C34H46N4O12
    Cor e Forma:Solid
    Peso molecular:702.758

    Ref: TM-T39653

    5mg
    1.341,00€
  • ZG36


    ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrial
    Cor e Forma:Odour Solid

    Ref: TM-T80737

    5mg
    A consultar
    50mg
    A consultar
  • Acetyl-Calpastatin(184-210)(human) TFA


    Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.
    Fórmula:C144H231F3N36O46S
    Cor e Forma:Solid
    Peso molecular:3291.65

    Ref: TM-T75794

    5mg
    A consultar
    50mg
    A consultar
  • Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2

    CAS:
    Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).
    Fórmula:C49H68N14O12S
    Cor e Forma:Solid
    Peso molecular:1077.22

    Ref: TM-T36360

    1mg
    384,00€
  • Hepcidin-1 (mouse)

    CAS:
    Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.
    Fórmula:C111H169N31O35S8
    Cor e Forma:Solid
    Peso molecular:2754.24

    Ref: TM-T80108

    5mg
    A consultar
    50mg
    A consultar
  • S62798

    CAS:
    S62798 is a highly potent and selective compound that inhibits activated thrombin activatable fibrinolysis inhibitor (TAFIa) with an IC50 value of 6 mM.
    Fórmula:C20H28FN4O4P
    Cor e Forma:Solid
    Peso molecular:438.44

    Ref: TM-T39551

    5mg
    873,00€
  • Fibrinogen-Binding Peptide

    CAS:
    Fibrinogen-binding peptide mimics vitronectin site and activates platelets; thrombin turns it to fibrin.
    Fórmula:C25H39N7O8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:565.62

    Ref: TM-TP1736

    100mg
    A consultar
    500mg
    A consultar
  • Befovacimab

    CAS:
    Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.
    Cor e Forma:Liquid

    Ref: TM-T76921

    5mg
    A consultar
  • MMP-9-IN-6

    CAS:
    MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.
    Fórmula:C25H19NO2
    Pureza:98.96%
    Cor e Forma:Soild
    Peso molecular:365.42

    Ref: TM-T77617

    1mg
    70,00€
    5mg
    138,00€
    10mg
    195,00€
    25mg
    309,00€
    50mg
    408,00€
    100mg
    562,00€
    200mg
    743,00€
  • Sofigatran

    CAS:
    Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.
    Fórmula:C24H44N4O4S
    Cor e Forma:Solid
    Peso molecular:484.7

    Ref: TM-T39310

    5mg
    873,00€
  • GPLGLAGGWGERDGS

    CAS:
    GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.
    Fórmula:C61H93N19O21
    Cor e Forma:Solid
    Peso molecular:1428.51

    Ref: TM-TP3038

    10mg
    A consultar
    50mg
    A consultar
  • TP0597850

    CAS:
    TP0597850, a selective MMP2 inhibitor with an IC50 value of 0.22 nM, demonstrates a prolonged dissociation half-life from MMP2 (t1/2 = 265 minutes) [1].
    Fórmula:C41H57N9O13S
    Cor e Forma:Solid
    Peso molecular:916.01

    Ref: TM-T74714

    5mg
    A consultar
    50mg
    A consultar
  • Sadopeptins A


    Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].
    Fórmula:C49H71N9O13S
    Cor e Forma:Solid
    Peso molecular:1026.21

    Ref: TM-T75623

    5mg
    A consultar
    50mg
    A consultar
  • Activated Protein C (390-404), human

    CAS:
    Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.
    Fórmula:C91H130N22O23
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1900.14

    Ref: TM-TP1628

    100mg
    A consultar
    500mg
    A consultar
  • Sofosbuvir impurity I


    Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Fórmula:C21H27FN3O9P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:515.43

    Ref: TM-T12964

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Ac-PLVE-FMK

    CAS:
    Ac-PLVE-FMK (Ac-Pro-Leu-Val-Glu(OMe)-CH2F), a tetrapeptidyl fluoromethylketone (FMKs), serves as a cathepsin inhibitor. It is utilized in cancer research [1].
    Fórmula:C25H41FN4O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:528.61

    Ref: TM-T78185

    5mg
    A consultar
    50mg
    A consultar
  • GCPII-IN-1

    CAS:

    GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.

    Fórmula:C12H21N3O7
    Cor e Forma:Solid
    Peso molecular:319.314

    Ref: TM-T38420

    5mg
    922,00€
  • Chetoseminudin B

    CAS:
    Chetoseminudin B exhibits inhibitory activity against mushroom tyrosinase, with an IC 50 value of 31.7 μM [1].
    Fórmula:C17H21N3O3S2
    Cor e Forma:Solid
    Peso molecular:379.5

    Ref: TM-T75471

    5mg
    A consultar
    50mg
    A consultar
  • N-CBZ-Phe-Arg-AMC

    CAS:
    Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.
    Fórmula:C33H36N6O6
    Pureza:98%
    Cor e Forma:White To Off-White Powder
    Peso molecular:612.68

    Ref: TM-TP1013

    100mg
    A consultar
    500mg
    A consultar
  • PM 102

    CAS:
    Peptide that reverses the anticoagulant effect of heparin. Potently binds heparin (Kd = 36 nM in vitro).
    Fórmula:C235H425N111O64
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:5830

    Ref: TM-TP1959

    1mg
    284,00€
  • Ellipyrone A


    Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).
    Fórmula:C25H34O8
    Cor e Forma:Solid
    Peso molecular:462.53

    Ref: TM-T75492

    5mg
    A consultar
    50mg
    A consultar
  • Dutogliptin

    CAS:
    Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.
    Fórmula:C10H20BN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:241.10

    Ref: TM-T11128

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Micropeptin 478A

    CAS:
    Micropeptin 478A is a plasmin inhibitor from the Cyanobacterium Microcystis aeruginosa.
    Fórmula:C40H62ClN9O15S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:976.49

    Ref: TM-T25810

    25mg
    1.369,00€
  • Acetyl-Calpastatin(184-210)(human)

    CAS:
    Calpain inhibitor, Ki 0.2 nM for calpain I/II, doesn't affect papain/trypsin/cat L. Raises Aβ42, Aβ40 secretion & Aβ42/Aβ40 ratio.
    Fórmula:C142H230N36O44S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3177.65

    Ref: TM-TP2056

    1mg
    1.378,00€
  • Talabostat isomer mesylate


    Talabostat isomer mesylate, a PT100/Val-boroPro variant, is a potent oral DPP-IV inhibitor (Ki: 0.18 nM).
    Fórmula:C10H23BN2O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:310.18

    Ref: TM-T13069

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • FFAGLDD


    "FFAGLDD: MMP9 peptide for controlled DOX delivery inside cells."
    Fórmula:C37H49N7O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:783.82

    Ref: TM-TP1545

    2mg
    71,00€
    5mg
    92,00€
    10mg
    131,00€
    25mg
    229,00€
    50mg
    343,00€
    100mg
    517,00€
  • Aristololactam IIIa

    CAS:
    Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.
    Fórmula:C16H9NO4
    Cor e Forma:Solid
    Peso molecular:279.25

    Ref: TM-T75619

    5mg
    A consultar
    50mg
    A consultar
  • AP-C2

    CAS:
    AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.
    Fórmula:C18H16N4S
    Pureza:99.99%
    Cor e Forma:Soild
    Peso molecular:320.41

    Ref: TM-T77570

    2mg
    38,00€
    5mg
    59,00€
    10mg
    82,00€
    25mg
    148,00€
    50mg
    245,00€
    100mg
    427,00€
    200mg
    577,00€
  • Leptosin D

    CAS:
    Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)
    Fórmula:C25H24N4O3S2
    Cor e Forma:Solid
    Peso molecular:492.61

    Ref: TM-T75472

    5mg
    A consultar
    50mg
    A consultar
  • C-telopeptide

    CAS:
    C-telopeptide from type I collagen is released during bone resorption; it correlates with bone mineral density.
    Fórmula:C34H56N14O13
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:868.9

    Ref: TM-TP1779

    1mg
    109,00€
    5mg
    424,00€
    10mg
    720,00€
  • Alisporivir

    CAS:
    Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.
    Fórmula:C63H113N11O12
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:1216.64

    Ref: TM-T14180

    1mg
    177,00€
    5mg
    447,00€
    10mg
    650,00€
  • NS5A-IN-1


    NS5A-IN-1 is a proagent of the HCV NS5A inhibitor Pibrentasvir (ABT-530).
    Fórmula:C72H86F5N10O14P
    Cor e Forma:Solid
    Peso molecular:1441.48

    Ref: TM-T74403

    5mg
    A consultar
    50mg
    A consultar
  • (-)-Taxifolin

    CAS:
    (-)-Taxifolin, less active enantiomer with anti-tyrosinase, collagenase inhibition (IC50 = 193.3 μM), antifibrotic, antioxidant properties.
    Fórmula:C15H12O7
    Cor e Forma:Solid
    Peso molecular:304.25

    Ref: TM-T38497

    25mg
    1.369,00€
  • JC-10

    CAS:
    JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.
    Fórmula:C25H29Cl2IN4
    Pureza:95%
    Cor e Forma:Solid
    Peso molecular:583.34

    Ref: TM-TD0056

    1mg
    118,00€
  • Paritaprevir dihydrate

    CAS:
    Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.
    Fórmula:C40H47N7O9S
    Cor e Forma:Solid
    Peso molecular:801.91

    Ref: TM-T73898

    5mg
    A consultar
    50mg
    A consultar
  • Linagliptin Methyldimer

    CAS:
    Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
    Fórmula:C50H56N16O4
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:945.08

    Ref: TM-T67852

    1mg
    109,00€
    2mg
    158,00€
    5mg
    260,00€
    10mg
    385,00€
    25mg
    628,00€
    50mg
    872,00€
    100mg
    1.153,00€
  • FFAGLDD TFA


    FFAGLDD TFA: MMP9 peptide for controlled DOX delivery to cytoplasm.
    Fórmula:C39H50F3N7O14
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:897.85

    Ref: TM-TP1498

    100mg
    A consultar
    500mg
    A consultar
  • Mipomersen

    CAS:
    Mipomersen (ISIS 301012) is an antisense oligo that inhibits apoB, has anti-HCV properties, and is researched for HoFH.
    Cor e Forma:Solid
    Peso molecular:7177

    Ref: TM-T74720

    5mg
    A consultar
    50mg
    A consultar
  • AR-H067637

    CAS:
    AR-H067637 is a fast-acting, reversible thrombin inhibitor with K(i) 2-4 nM; it also reduces clot-bound thrombin and platelet activation/aggregation.
    Fórmula:C21H21ClF2N4O4
    Cor e Forma:Solid
    Peso molecular:466.87

    Ref: TM-T26657

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Procizumab


    Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.
    Cor e Forma:Odour Liquid

    Ref: TM-T9901A-771

    1mg
    A consultar
    5mg
    A consultar
  • Rivulariapeptolides 1121


    Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).
    Fórmula:C56H83N9O15
    Cor e Forma:Solid
    Peso molecular:1122.31

    Ref: TM-T75650

    5mg
    A consultar
    50mg
    A consultar
  • Ac-DEMEEC-OH

    CAS:
    Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.
    Fórmula:C29H44N6O16S2
    Cor e Forma:Solid
    Peso molecular:796.82

    Ref: TM-TP2848

    10mg
    A consultar
    50mg
    A consultar
  • PPACK II

    CAS:
    PPACK II is an irreversible and specific glandular and plasma kallikreins inhibitor [1] .
    Fórmula:C25H33ClN6O3
    Cor e Forma:Solid
    Peso molecular:501.02

    Ref: TM-T73863

    5mg
    A consultar
    50mg
    A consultar
  • Rivulariapeptolides 988


    Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).
    Fórmula:C50H68N8O13
    Cor e Forma:Solid
    Peso molecular:989.12

    Ref: TM-T75651

    5mg
    A consultar
    50mg
    A consultar
  • Nitidanin


    Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.
    Fórmula:C21H24O8
    Cor e Forma:Solid
    Peso molecular:404.415

    Ref: TM-T125599

    1mg
    A consultar
    5mg
    A consultar
  • Sofosbuvir impurity A

    CAS:
    Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.
    Fórmula:C22H29FN3O9P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:529.45

    Ref: TM-T12956

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • AL-611

    CAS:

    AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).

    Fórmula:C25H33F2N6O8P
    Cor e Forma:Solid
    Peso molecular:614.544

    Ref: TM-T39082

    5mg
    922,00€