Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(34 produtos)
- Cisteína Protease(96 produtos)
- DPP-4(20 produtos)
- Glutaminase(40 produtos)
- HIV Protease(449 produtos)
- PAI-1(25 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(53 produtos)
- Proteassoma(94 produtos)
- Protease serina(50 produtos)
- p97(14 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1044 produtos de "Proteases/Proteassoma"
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Hepcidin-1 (mouse)
CAS:<p>Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.</p>Fórmula:C111H169N31O35S8Cor e Forma:SolidPeso molecular:2754.24GSK2818713
CAS:<p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>Fórmula:C46H56N8O8Cor e Forma:SolidPeso molecular:849.002PROTAC 20S proteasome subunit β5 degrader 2
<p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>Cor e Forma:Odour SolidLedipasvir D-tartrate
CAS:<p>Ledipasvir D-tartrate (GS-5885 D-tartrate) is an HCV NS5A inhibitor that suppresses viral overphosphorylation and replication</p>Fórmula:C53H60F2N8O12Pureza:99.83%Cor e Forma:SolidPeso molecular:1039.09Ellipyrone B
<p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>Fórmula:C25H38O7Cor e Forma:SolidPeso molecular:450.57Procizumab
<p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Cor e Forma:Odour LiquidBI-1230
CAS:<p>BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.</p>Fórmula:C42H52N6O9SPureza:98%Cor e Forma:SolidPeso molecular:816.96MMP-3 Inhibitor
CAS:<p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>Fórmula:C27H46N10O9SPureza:98.87%Cor e Forma:SolidPeso molecular:686.78HCV-IN-4
CAS:<p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>Fórmula:C52H58FN9O8Pureza:98%Cor e Forma:SolidPeso molecular:956.07Bictegravir Sodium
CAS:<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Fórmula:C21H17F3N3NaO5Pureza:99.97%Cor e Forma:SolidPeso molecular:471.36HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Cor e Forma:Odour SolidPS 915
CAS:<p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>Fórmula:C27H36ClN7O6Pureza:98%Cor e Forma:SolidPeso molecular:590.08Ichorcumab
CAS:<p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Cor e Forma:LiquidKKI-5
CAS:<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Fórmula:C35H55N11O9Pureza:98%Cor e Forma:SolidPeso molecular:773.88Histargin
CAS:<p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>Fórmula:C14H25N7O4Cor e Forma:SolidPeso molecular:355.39Relacatib
CAS:<p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>Fórmula:C27H32N4O6SCor e Forma:SolidPeso molecular:540.64LXE408 fumarate
<p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>Fórmula:C27H22FN7O6Pureza:99.89%Cor e Forma:SoildPeso molecular:559.51Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Cor e Forma:Odour SolidAristololactam IIIa
CAS:<p>Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.</p>Fórmula:C16H9NO4Cor e Forma:SolidPeso molecular:279.25Tiprelestat
CAS:<p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>Fórmula:C254H416N72O75S10Cor e Forma:SolidPeso molecular:5999.09Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)
Fluorogenic substrate for cathepsins D & E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.Cor e Forma:Odour SolidParitaprevir dihydrate
CAS:<p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>Fórmula:C40H47N7O9SCor e Forma:SolidPeso molecular:801.91Lonodelestat TFA
<p>Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.</p>Fórmula:C73H112F3N15O21Cor e Forma:SolidPeso molecular:1592.75Ac-Phe-Gly-pNA
CAS:<p>Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .</p>Fórmula:C19H20N4O5Cor e Forma:SolidPeso molecular:384.39ADAM8-IN-1
CAS:<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Fórmula:C44H44Br4N6O12S2Cor e Forma:SolidPeso molecular:1232.6Sulodexide
CAS:<p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>Cor e Forma:SolidCerpegin
CAS:<p>Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.</p>Fórmula:C10H11NO3Cor e Forma:SolidPeso molecular:193.2Carboxypeptidase C
CAS:<p>Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.</p>Cor e Forma:SolidVAMP
<p>VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.</p>Fórmula:C18H32N4O5SCor e Forma:SolidPeso molecular:416.535Ala-Phe-Pro-pNA TFA
<p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>Cor e Forma:Odour SolidMMP-9-IN-6
CAS:<p>MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.</p>Fórmula:C25H19NO2Pureza:99.75%Cor e Forma:SoildPeso molecular:365.42CTTHWGFTLC, CYCLIC
CAS:<p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>Fórmula:C52H71N13O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1166.33Alisporivir
CAS:<p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>Fórmula:C63H113N11O12Pureza:99.95%Cor e Forma:SolidPeso molecular:1216.64Histatin 5 TFA
Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μMFórmula:C135H196N51F3O35Cor e Forma:SolidPeso molecular:3150.31Chymotrypsinogen
CAS:<p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>Cor e Forma:SolidAcetyl-Calpastatin(184-210)(human) TFA
<p>Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.</p>Fórmula:C144H231F3N36O46SCor e Forma:SolidPeso molecular:3291.65Suc-AAP-Abu-pNA
CAS:<p>Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,</p>Fórmula:C25H34N6O9Cor e Forma:SolidPeso molecular:562.57TR-107
CAS:<p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>Fórmula:C22H19ClN4OCor e Forma:SoildPeso molecular:390.87LMP7/LMP2-IN-1
CAS:<p>LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.</p>Fórmula:C16H27BN4O3Cor e Forma:SoildPeso molecular:334.22Phepropeptin A
CAS:<p>Phepropeptin A is a secondary metabolite produced by microorganisms and acts as a proteasome (proteasome) inhibitor, with an IC50 of 21 μg/mL.</p>Fórmula:C37H58N6O6Cor e Forma:SolidPeso molecular:682.89TWH106
<p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>Cor e Forma:Odour SolidPD150606
CAS:<p>PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.</p>Fórmula:C9H7IO2SPureza:98.19%Cor e Forma:SolidPeso molecular:306.12BMS-767778
CAS:<p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Fórmula:C19H20Cl2N4O2Cor e Forma:SolidPeso molecular:407.29Tyrosinase-IN-34
<p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>Fórmula:C19H14BrClN4OCor e Forma:SolidPeso molecular:429.7Roseltide rT1
CAS:<p>Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.</p>Fórmula:C110H177N31O31S6Cor e Forma:SolidPeso molecular:2622.16α 1(I) Collagen (614-639), human
CAS:<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Fórmula:C134H189N37O39Pureza:98%Cor e Forma:SolidPeso molecular:2942.16MMP-2 Inhibitor-4
<p>MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).</p>Fórmula:C19H23N3O5SCor e Forma:SolidPeso molecular:405.468NVP-DPP728 dihydrochloride
CAS:<p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>Fórmula:C15H20Cl2N6OCor e Forma:SolidPeso molecular:371.27RJS308
<p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>Fórmula:C63H75N13O11SCor e Forma:SolidPeso molecular:1222.42Stevia Powder
<p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>Cor e Forma:Odour SolidPR 39 (porcine) acetate
<p>PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.</p>Pureza:98%Cor e Forma:LiquidPeso molecular:N/A6-Acetylnimbandiol
CAS:<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Fórmula:C28H34O8Cor e Forma:SolidPeso molecular:498.56Zetomipzomib maleate
CAS:<p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>Fórmula:C34H46N4O12Cor e Forma:SolidPeso molecular:702.758Rivulariapeptolides 1185
<p>Rivulariapeptolides 1185 inhibits serine proteases; IC50: chymotrypsin 13.17 nM, elastase 23.59 nM, proteinase K 55.26 nM.</p>Fórmula:C61H87N9O15Cor e Forma:SolidPeso molecular:1186.39L 659286
CAS:<p>L 659286 is one kind of cephalosporin derivative.</p>Fórmula:C17H21N5O7S2Cor e Forma:SolidPeso molecular:471.51Pseudostellarin G
CAS:<p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>Fórmula:C42H56N8O9Cor e Forma:SolidPeso molecular:816.94Rivulariapeptolides 988
<p>Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).</p>Fórmula:C50H68N8O13Cor e Forma:SolidPeso molecular:989.12Ellipyrone A
<p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>Fórmula:C25H34O8Cor e Forma:SolidPeso molecular:462.53CRA-2059
CAS:<p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>Fórmula:C34H46N12O8Pureza:97.68%Cor e Forma:SolidPeso molecular:750.818Emtricitabine S-oxide
CAS:<p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>Fórmula:C8H10FN3O4SPureza:98%Cor e Forma:SolidPeso molecular:263.25Dutogliptin
CAS:<p>Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>Fórmula:C10H20BN3O3Pureza:98%Cor e Forma:SolidPeso molecular:241.10Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS:Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effectFórmula:C47H64N14O10Cor e Forma:SolidPeso molecular:985.1Linagliptin Methyldimer
CAS:<p>Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.</p>Fórmula:C50H56N16O4Pureza:97.23%Cor e Forma:SolidPeso molecular:945.08Fotagliptin
CAS:<p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C17H19FN6OCor e Forma:SolidPeso molecular:342.37E-64d [for Biochemical Research]
CAS:Fórmula:C17H30N2O5Pureza:>95.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:342.44CTS-1027
CAS:<p>CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has > 1,000 fold selectivity over MMP1.</p>Fórmula:C19H20ClNO6SCor e Forma:SolidPeso molecular:425.88Tenofovir hydrate
CAS:<p>Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.</p>Fórmula:C9H16N5O5PPureza:99.63%Cor e Forma:SolidPeso molecular:305.23S-Methylglutathione
CAS:<p>S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.</p>Fórmula:C11H19N3O6SPureza:98%Cor e Forma:SolidPeso molecular:321.35Ilomastat
CAS:Fórmula:C20H28N4O4Pureza:>95.0%(HPLC)(qNMR)Cor e Forma:White to Light yellow powder to crystalPeso molecular:388.47Retagliptin
CAS:<p>Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.</p>Fórmula:C19H18F6N4O3Cor e Forma:SolidPeso molecular:464.36PSI-6206 13C,d3
CAS:<p>PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.</p>Fórmula:C10H13FN2O5Pureza:98%Cor e Forma:SolidPeso molecular:264.23Tripeptide-32
CAS:<p>Tripeptide-32 is a bioactive peptide recognized for its anti-aging properties, commonly utilized as an ingredient in cosmetics [1].</p>Fórmula:C12H22N4O5Pureza:98%Cor e Forma:SolidPeso molecular:302.33MMP-8 Inhibitor I
CAS:<p>MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.</p>Fórmula:C17H18N2O5SCor e Forma:SolidPeso molecular:362.4Glutaminase-IN-3
CAS:<p>Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.</p>Fórmula:C19H19F3N6O2SPureza:98.51%Cor e Forma:SolidPeso molecular:452.45Tilpisertib
CAS:<p>Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).</p>Fórmula:C33H33ClN8OCor e Forma:SolidPeso molecular:593.13Teneligliptin hydrobromide hydrate
CAS:<p>Teneligliptin hydrobromide hydrate: potent, long-lasting DPP-4 inhibitor with ~1 nM IC50.</p>Fórmula:C22H33BrN6O2SCor e Forma:SolidPeso molecular:525.51Sitagliptin fenilalanil
CAS:Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.Fórmula:C25H24F6N6O2Cor e Forma:SolidPeso molecular:554.49PKSI-527
CAS:<p>PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.</p>Fórmula:C25H32ClN3O4Cor e Forma:SolidPeso molecular:473.99H-Arg-4MβNA
CAS:<p>H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.</p>Fórmula:C17H23N5O2Pureza:99.98%Cor e Forma:SolidPeso molecular:329.4BAY-677
CAS:<p>BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.</p>Fórmula:C20H15F3N4O2Cor e Forma:SolidPeso molecular:400.355-Amino-8-hydroxyquinoline
CAS:<p>5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.</p>Fórmula:C9H8N2OPureza:99.69%Cor e Forma:SolidPeso molecular:160.176-Chloro-7-deazapurine-2F-β-D-arabinofuranose
CAS:<p>6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.</p>Fórmula:C11H11ClFN3O3Cor e Forma:SolidPeso molecular:287.67(Arg)9
CAS:<p>(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).</p>Fórmula:C54H110N36O10Cor e Forma:SolidPeso molecular:1423.69Ubenimex Hydrochloride [for Biochemical Research]
CAS:Fórmula:C16H24N2O4·HClPureza:>97.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:344.84Dabigatran ethyl ester
CAS:<p>Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.</p>Fórmula:C27H29N7O3Pureza:99.98%Cor e Forma:SolidPeso molecular:499.56Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Fórmula:C23H27N3O4SPureza:98%Cor e Forma:SolidPeso molecular:441.54Teneligliptin D8
CAS:<p>Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.</p>Fórmula:C22H30N6OSPureza:98%Cor e Forma:SolidPeso molecular:434.63PD-166793
CAS:<p>PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.</p>Fórmula:C17H18BrNO4SPureza:99.86%Cor e Forma:SolidPeso molecular:412.3DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Fórmula:C31H40N4O6Cor e Forma:SolidPeso molecular:564.67Thrombin inhibitor 5
CAS:<p>Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.</p>Fórmula:C11H9FN4O3Pureza:99.58%Cor e Forma:SolidPeso molecular:264.21H-Pro-Lys-OH TFA
<p>H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.</p>Fórmula:C13H22F3N3O5Cor e Forma:SolidPeso molecular:357.332'-β-C-Ethynyladenosine
CAS:<p>2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.</p>Fórmula:C12H13N5O4Cor e Forma:SolidPeso molecular:291.26Sivelestat Sodium Tetrahydrate
CAS:Fórmula:C20H21N2NaO7S·4H2OPureza:>95.0%(T)(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:528.50Urokinase
CAS:<p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>Cor e Forma:SolidPentosan Polysulfate Sodium (W/W 43%)
CAS:<p>Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.</p>Pureza:98%Cor e Forma:SolidPeso molecular:N/AAnguizole
CAS:Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.Fórmula:C17H11ClF2N4O2SCor e Forma:SolidPeso molecular:408.81Pepstatin A
CAS:Fórmula:C34H63N5O9Pureza:>90.0%(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:685.90(-)-Gallocatechin Gallate
CAS:Fórmula:C22H18O11Pureza:>95.0%(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:458.38Tanaproget
CAS:<p>Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.</p>Fórmula:C16H15N3OSPureza:98%Cor e Forma:SolidPeso molecular:297.38Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Fórmula:C10H13N2Na3O8·xH2OPureza:>98.0%(T)Cor e Forma:White to Almost white powder to crystalPeso molecular:358.19 (as Anhydrous)
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