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Proteases/Proteassoma

Proteases/Proteassoma

Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.

Subcategorias de "Proteases/Proteassoma"

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Foram encontrados 1044 produtos de "Proteases/Proteassoma"

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  • BC-05

    CAS:
    <p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>
    Fórmula:C21H29BN2O9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:464.27
  • Tyrosinase-IN-7

    CAS:
    <p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>
    Fórmula:C15H10O5
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:270.24
  • Tanomastat

    CAS:
    <p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>
    Fórmula:C23H19ClO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:410.91
  • HCV-IN-34

    CAS:
    <p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>
    Fórmula:C31H36ClN5
    Cor e Forma:Solid
    Peso molecular:514.1
  • Sortin1

    CAS:
    Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.
    Fórmula:C26H19NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:441.43
  • MDK7677

    CAS:
    <p>MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>
    Fórmula:C12H10N4O3
    Cor e Forma:Solid
    Peso molecular:258.23
  • Furaprofen

    CAS:
    <p>Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.</p>
    Fórmula:C17H14O3
    Pureza:98.49% - 99.52%
    Cor e Forma:Solid
    Peso molecular:266.29
  • Gemigliptin Tartrate(911637-19-9 free base)

    CAS:
    <p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>
    Fórmula:C22H25F8N5O8
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:639.45
  • GEMSA

    CAS:
    <p>GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].</p>
    Fórmula:C7H13N3O4S
    Cor e Forma:Solid
    Peso molecular:235.26
  • Azo-Resveratrol

    CAS:
    <p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>
    Fórmula:C12H10N2O3
    Cor e Forma:Solid
    Peso molecular:230.22
  • (3S,4S)-A2-32-01


    <p>(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .</p>
    Fórmula:C19H27NO2
    Cor e Forma:Solid
    Peso molecular:301.42
  • AK 275

    CAS:
    <p>AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.</p>
    Fórmula:C20H31N3O4
    Cor e Forma:Solid
    Peso molecular:377.48
  • AZD-9684

    CAS:
    <p>AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.</p>
    Fórmula:C10H14N2O2S
    Cor e Forma:Solid
    Peso molecular:226.3
  • ITX-4520

    CAS:
    <p>ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.</p>
    Fórmula:C24H23F2N3OS
    Cor e Forma:Solid
    Peso molecular:439.52
  • MMP-1-IN-1


    <p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>
    Fórmula:C14H17ClN2O3
    Cor e Forma:Solid
    Peso molecular:296.75
  • L 722151

    CAS:
    <p>L 722151 is an FXIIIa inhibitor.</p>
    Fórmula:C8H9ClN2O5S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:344.82
  • SAP2-IN-1

    CAS:
    <p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>
    Fórmula:C34H29NO7
    Cor e Forma:Solid
    Peso molecular:563.6
  • Chymase-IN-1

    CAS:
    <p>Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).</p>
    Fórmula:C20H15ClNO4PS
    Pureza:99.17%
    Cor e Forma:Solid
    Peso molecular:431.83
  • NAAA-IN-2

    CAS:
    <p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>
    Fórmula:C11H13N3O2S
    Cor e Forma:Solid
    Peso molecular:251.3
  • ADAMTS-5-IN-2

    CAS:
    <p>ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.</p>
    Fórmula:C17H15N3OS
    Cor e Forma:Solid
    Peso molecular:309.39
  • TAPI-0

    CAS:
    <p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>
    Fórmula:C24H32N4O5
    Cor e Forma:Solid
    Peso molecular:456.53
  • Safironil

    CAS:
    <p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>
    Fórmula:C15H23N3O4
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:309.36
  • Tyrosinase-IN-10

    CAS:
    <p>Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'</p>
    Fórmula:C16H12O4
    Cor e Forma:Solid
    Peso molecular:268.26
  • Calpain-2-IN-1

    CAS:
    <p>Calpain-2-IN-1 is a selective calpain-2 inhibitor that prolongs ERK activation and thus enhances learning and memory.</p>
    Fórmula:C28H37N3O7
    Cor e Forma:Solid
    Peso molecular:527.61
  • BR351

    CAS:
    <p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>
    Fórmula:C20H25FN2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:424.49
  • Adafosbuvir PM

    CAS:
    <p>Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.</p>
    Fórmula:C10H13FN2O6
    Pureza:97.08%
    Cor e Forma:Solid
    Peso molecular:276.22
  • HCV-IN-35

    CAS:
    <p>HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.</p>
    Fórmula:C30H36ClN5
    Cor e Forma:Solid
    Peso molecular:502.09
  • Calpain Inhibitor XI

    CAS:
    <p>Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.</p>
    Fórmula:C26H40N4O6
    Cor e Forma:Solid
    Peso molecular:504.62
  • AM 4299 B

    CAS:
    <p>AM 4299 B is a novel inhibitor of a thiol protease.</p>
    Fórmula:C16H27N3O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.4
  • MDL 27399

    CAS:
    <p>MDL 27399 suppresses human neutrophil cathepsin G.</p>
    Fórmula:C26H36N4O8
    Cor e Forma:Solid
    Peso molecular:532.59
  • α-Glucosidase-IN-5

    CAS:
    <p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>
    Fórmula:C15H13NO3
    Cor e Forma:Solid
    Peso molecular:255.27
  • BMS-363131

    CAS:
    <p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of &lt;1.7 nM.</p>
    Fórmula:C28H40N6O5
    Pureza:97.99%
    Cor e Forma:Solid
    Peso molecular:540.65
  • CAA0225

    CAS:
    <p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>
    Fórmula:C28H29N3O5
    Cor e Forma:Solid
    Peso molecular:487.55
  • Immunoproteasome inhibitor 1

    CAS:
    <p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>
    Fórmula:C20H26N2O4
    Cor e Forma:Solid
    Peso molecular:358.43
  • JO146

    CAS:
    <p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。</p>
    Fórmula:C31H44N3O7P
    Cor e Forma:Solid
    Peso molecular:601.67
  • L-873724

    CAS:
    <p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>
    Fórmula:C23H26F3N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.53
  • (R)-ND-336

    CAS:
    <p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>
    Fórmula:C16H18ClNO3S2
    Cor e Forma:Solid
    Peso molecular:371.89
  • OM-189

    CAS:
    <p>OM-189 is a selective inhibitor of synthetic thrombin.</p>
    Fórmula:C24H36N6O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:488.65
  • Tyrosinase-IN-1

    CAS:
    <p>Tyrosinase-IN-1: potent inhibitor for skin-whitening &amp; food preservation with uses in cosmetics &amp; medicine.</p>
    Fórmula:C10H9N3O2S2
    Cor e Forma:Solid
    Peso molecular:267.33
  • CA 074

    CAS:
    <p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>
    Fórmula:C18H29N3O6
    Pureza:97.80%
    Cor e Forma:Solid
    Peso molecular:383.44
  • XMU-MP-2

    CAS:
    <p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>
    Fórmula:C32H33F3N8O2
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:618.65
  • MMP-2/9-IN-1

    CAS:
    <p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>
    Fórmula:C14H16IN7S
    Cor e Forma:Solid
    Peso molecular:441.29
  • GLS1 Inhibitor-3

    CAS:
    <p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>
    Fórmula:C30H32N10O2S
    Cor e Forma:Solid
    Peso molecular:596.71
  • HCV-IN-36

    CAS:
    <p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>
    Fórmula:C30H36ClN5
    Cor e Forma:Solid
    Peso molecular:502.09
  • 2',5-Difluoro-2'-deoxycytidine

    CAS:
    <p>2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.</p>
    Fórmula:C9H11F2N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:263.2
  • BRD-8899

    CAS:
    <p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>
    Fórmula:C17H22N4O3S
    Cor e Forma:Solid
    Peso molecular:362.45
  • Calpain Inhibitor XII

    CAS:
    <p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>
    Fórmula:C26H34N4O5
    Cor e Forma:Solid
    Peso molecular:482.57
  • Tyrosinase-IN-5

    CAS:
    <p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>
    Fórmula:C18H13N3O6
    Cor e Forma:Solid
    Peso molecular:367.31
  • Elasnin

    CAS:
    <p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>
    Fórmula:C24H40O4
    Cor e Forma:Solid
    Peso molecular:392.57
  • Gü1303

    CAS:
    <p>Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).</p>
    Fórmula:C20H22N4O3
    Cor e Forma:Solid
    Peso molecular:366.41
  • ABT-770

    CAS:
    <p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>
    Fórmula:C22H22F3N3O6
    Cor e Forma:Solid
    Peso molecular:481.42
  • ASPER-29

    CAS:
    <p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>
    Fórmula:C31H29BrN2O5S
    Cor e Forma:Solid
    Peso molecular:621.54
  • CAY10704

    CAS:
    <p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>
    Fórmula:C18H20Cl2N2
    Cor e Forma:Solid
    Peso molecular:335.27
  • DPP-4-IN-1

    CAS:
    <p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>
    Fórmula:C19H19ClN6
    Cor e Forma:Solid
    Peso molecular:366.85
  • AA10 TG2 inhibitor

    CAS:
    <p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>
    Fórmula:C32H36N4O5
    Cor e Forma:Solid
    Peso molecular:556.65
  • Antiviral agent 30

    CAS:
    <p>Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].</p>
    Fórmula:C21H32N2O3S
    Cor e Forma:Solid
    Peso molecular:392.56
  • BAY8040

    CAS:
    <p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>
    Fórmula:C21H16F3N5O2
    Cor e Forma:Solid
    Peso molecular:427.38
  • PK44 phosphate

    CAS:
    <p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>
    Fórmula:C17H19F5N7O5P
    Cor e Forma:Solid
    Peso molecular:527.349
  • BrBzGCp2

    CAS:
    <p>BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.</p>
    Fórmula:C27H38BrN3O6S
    Pureza:98.68% - 98.68%
    Cor e Forma:Solid
    Peso molecular:612.58
  • ACH-806

    CAS:
    <p>ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.</p>
    Fórmula:C19H20F3N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:411.44
  • VEL-0230

    CAS:
    <p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>
    Fórmula:C14H24NNaO5
    Cor e Forma:Solid
    Peso molecular:309.33
  • AZD5248

    CAS:
    <p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>
    Fórmula:C22H22N4O2
    Cor e Forma:Solid
    Peso molecular:374.44
  • A-933548

    CAS:
    <p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>
    Fórmula:C25H21N5O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:439.47
  • Alicapistat

    CAS:
    <p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>
    Fórmula:C25H27N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.5
  • SP-Chymostatin B

    CAS:
    <p>SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.</p>
    Fórmula:C30H41N7O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:595.69
  • DPP-IV-IN-1

    CAS:
    <p>DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).</p>
    Fórmula:C11H18FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:243.28
  • Tyrosinase-IN-6

    CAS:
    <p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>
    Fórmula:C24H31N3O2
    Cor e Forma:Solid
    Peso molecular:393.52
  • Anticancer agent 82

    CAS:
    <p>Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.</p>
    Fórmula:C19H18Cl2N4O
    Cor e Forma:Solid
    Peso molecular:389.28
  • MK-2048

    CAS:
    <p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>
    Fórmula:C21H21ClFN5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:461.87
  • Tyrosinase-IN-3

    CAS:
    <p>Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.</p>
    Fórmula:C21H23NO5
    Cor e Forma:Solid
    Peso molecular:369.41
  • Gü2602

    CAS:
    <p>Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for mature</p>
    Fórmula:C16H22N4O3
    Cor e Forma:Solid
    Peso molecular:318.37
  • VA4 TG2 inhibitor

    CAS:
    <p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>
    Fórmula:C33H41N5O6S
    Cor e Forma:Solid
    Peso molecular:635.77
  • Gosogliptin

    CAS:
    <p>Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.</p>
    Fórmula:C17H24F2N6O
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:366.41
  • HCV-IN-33

    CAS:
    <p>HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.</p>
    Fórmula:C31H36ClN5
    Cor e Forma:Solid
    Peso molecular:514.1
  • JNJ-10329670

    CAS:
    <p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>
    Fórmula:C30H34ClF3N6O3S
    Cor e Forma:Solid
    Peso molecular:651.14
  • (Rac)-Tanomastat

    CAS:
    <p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>
    Fórmula:C23H19ClO3S
    Cor e Forma:Solid
    Peso molecular:410.91
  • GSK2793660 HCl

    CAS:
    <p>GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.</p>
    Fórmula:C22H32ClN3O3
    Cor e Forma:Solid
    Peso molecular:421.96
  • Cysteine Protease inhibitor

    CAS:
    <p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>
    Fórmula:C18H14N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:302.33
  • Cysteine Protease inhibitor hydrochloride

    CAS:
    <p>Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.</p>
    Fórmula:C18H15ClN4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:338.79
  • Kallikrein 5-IN-2

    CAS:
    <p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation &amp; itching.</p>
    Fórmula:C23H22N6O
    Cor e Forma:Solid
    Peso molecular:398.46
  • BI-L 45XX

    CAS:
    <p>BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.</p>
    Fórmula:C10H9F3N2O2S
    Cor e Forma:Solid
    Peso molecular:278.25
  • Tec-IN-21

    CAS:
    <p>Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).</p>
    Fórmula:C16H15ClN4O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:362.83
  • Sheng Gelieting

    CAS:
    <p>CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.</p>
    Fórmula:C17H16F6N4O
    Cor e Forma:Solid
    Peso molecular:406.33
  • CP-471474

    CAS:
    <p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>
    Fórmula:C16H17FN2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:368.38
  • Tyrphostin 47

    CAS:
    <p>Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.</p>
    Fórmula:C10H8N2O2S
    Cor e Forma:Solid
    Peso molecular:220.25
  • Elastase-IN-1

    CAS:
    <p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>
    Fórmula:C17H12N4O3
    Cor e Forma:Solid
    Peso molecular:320.3
  • SJA6017

    CAS:
    <p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>
    Fórmula:C17H25FN2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:372.45
  • Plasma kallikrein-IN-3

    CAS:
    <p>Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.</p>
    Fórmula:C20H23N5O2
    Cor e Forma:Solid
    Peso molecular:365.43
  • HIV-1 integrase inhibitor 8

    CAS:
    <p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>
    Fórmula:C21H24O2
    Pureza:98.91%
    Cor e Forma:Solid
    Peso molecular:308.41
  • Tyrosinase-IN-2

    CAS:
    <p>Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.</p>
    Fórmula:C8H8N4O2S
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:224.24
  • BILB-1941

    CAS:
    <p>BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.</p>
    Fórmula:C34H34N4O4
    Pureza:99.51% - 99.65%
    Cor e Forma:Solid
    Peso molecular:562.66
  • CP-544439

    CAS:
    <p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>
    Fórmula:C18H19FN2O6S
    Pureza:95.02% - 98.66%
    Cor e Forma:Solid
    Peso molecular:410.42
  • BMS-929075

    CAS:
    <p>BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic</p>
    Fórmula:C31H24F2N4O3
    Pureza:98.44% - 99.94%
    Cor e Forma:Solid
    Peso molecular:538.54
  • Emivirine

    CAS:
    <p>Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.</p>
    Fórmula:C17H22N2O3
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:302.37
  • AGPS-IN-2i

    CAS:
    AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.
    Fórmula:C18H17F2N3O2
    Pureza:98.92%
    Cor e Forma:Solid
    Peso molecular:345.34
  • TS-021

    CAS:
    <p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>
    Fórmula:C17H24FN3O5S
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:401.45
  • GSK-364735

    CAS:
    <p>GSK-364735 is an HIV-1 IN inhibitor.</p>
    Fórmula:C19H18FN3O4
    Pureza:97.73%
    Cor e Forma:Solid
    Peso molecular:371.36
  • 2'-C-Methyladenosine

    CAS:
    <p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>
    Fórmula:C11H15N5O4
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:281.27
  • Isatoribine

    CAS:
    <p>Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.</p>
    Fórmula:C10H12N4O6S
    Pureza:98.99% - 99.75%
    Cor e Forma:Solid
    Peso molecular:316.29
  • JNJ-10311795

    CAS:
    <p>JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.</p>
    Fórmula:C40H35N2O6P
    Pureza:97.43%
    Cor e Forma:Solid
    Peso molecular:670.69