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Proteases/Proteassoma

Proteases/Proteassoma

Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.

Subcategorias de "Proteases/Proteassoma"

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Foram encontrados 1044 produtos de "Proteases/Proteassoma"

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  • Calpain Inhibitor-1
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    Calpain Inhibitor-1

    CAS:
    <p>Calpain Inhibitor-1, a potent Calpain 1 blocker, has IC50 of 100 nM and Ki of 2.89 μM.</p>
    Fórmula:C19H17FN6O5S
    Cor e Forma:Solid
    Peso molecular:460.44

    Ref: TM-T38931

  • Alisporivir
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    Alisporivir

    CAS:
    <p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>
    Fórmula:C63H113N11O12
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:1216.64

    Ref: TM-T14180

  • midesteine
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    midesteine

    CAS:
    <p>Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.</p>
    Fórmula:C12H13NO3S3
    Pureza:99.52% - 99.98%
    Cor e Forma:Solid
    Peso molecular:315.43

    Ref: TM-T68099

  • PF 00356231
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    PF 00356231

    CAS:
    <p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>
    Fórmula:C25H20N2O3S
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:428.5

    Ref: TM-T60071

  • Sofosbuvir impurity K
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    Sofosbuvir impurity K

    CAS:
    <p>Sofosbuvir impurity K is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Fórmula:C22H29ClN3O9P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:545.91

    Ref: TM-T12966

  • EP 171
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    EP 171

    CAS:
    <p>EP 171 is a potent agonist of TP-receptors.</p>
    Fórmula:C23H29FO5
    Cor e Forma:Solid
    Peso molecular:404.47

    Ref: TM-T27273

  • Nostopeptin B
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    Nostopeptin B

    CAS:
    <p>Nostopeptin B is an inhibitor of elastase.</p>
    Fórmula:C46H70N8O12
    Cor e Forma:Solid
    Peso molecular:927.11

    Ref: TM-T25880

  • Logotipo do CymitQuimica
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    Cepeginterferon alfa-2b

    CAS:
    <p>Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.</p>
    Cor e Forma:Liquid

    Ref: TM-T76943

  • HIV-1 inhibitor-6 
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    HIV-1 inhibitor-6 

    CAS:
    <p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>
    Fórmula:C14H10N4O4S
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:330.32

    Ref: TM-T9854

  • 7-Methoxy obtusifolin
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    7-Methoxy obtusifolin

    CAS:
    <p>7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentration</p>
    Fórmula:C17H14O6
    Cor e Forma:Solid
    Peso molecular:314.29

    Ref: TM-T75613

  • PSI-353661
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    PSI-353661

    CAS:
    <p>PSI-353661 (GS-558093), inhibits HCV's NS5B polymerase; EC90: 8nM (wild-type), 11nM (S282T); active in human hepatocytes.</p>
    Fórmula:C24H32FN6O8P
    Cor e Forma:Solid
    Peso molecular:582.52

    Ref: TM-T74301

  • Logotipo do CymitQuimica
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    Ellipyrone B

    <p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>
    Fórmula:C25H38O7
    Cor e Forma:Solid
    Peso molecular:450.57

    Ref: TM-T75493

  • BPHA
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    BPHA

    CAS:
    <p>BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.</p>
    Fórmula:C21H20N2O4S
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:396.46

    Ref: TM-T36712

  • Obtusifolin-2-O-glucoside
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    Obtusifolin-2-O-glucoside

    CAS:
    <p>Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].</p>
    Fórmula:C22H22O10
    Cor e Forma:Solid
    Peso molecular:446.4

    Ref: TM-T75572

  • AMG-222
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    AMG-222

    CAS:
    <p>AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.</p>
    Fórmula:C32H39N9O3
    Cor e Forma:Solid
    Peso molecular:597.71

    Ref: TM-T29970

  • Logotipo do CymitQuimica
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    Sulodexide

    CAS:
    <p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>
    Cor e Forma:Solid

    Ref: TM-T88323

  • Isoleucylvaline
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    Isoleucylvaline

    CAS:
    <p>Isoleucylvaline is a dipeptide.</p>
    Fórmula:C11H22N2O3
    Cor e Forma:Solid
    Peso molecular:230.30

    Ref: TM-T32214

  • Cajaninstilbene acid
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    Cajaninstilbene acid

    CAS:
    <p>Cajaninstilbene acid is a useful organic compound for research related to life sciences. The catalog number is T124035 and the CAS number is 87402-84-4.</p>
    Fórmula:C21H22O4
    Cor e Forma:Solid
    Peso molecular:338.403

    Ref: TM-T124035

  • Logotipo do CymitQuimica
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    Tyrosinase-IN-36

    <p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>
    Cor e Forma:Odour Solid

    Ref: TM-T200699

  • BMS 180742
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    BMS 180742

    CAS:
    <p>BMS 180742 is an exosite inhibitor of thrombin.</p>
    Fórmula:C67H93N11O22
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1404.52

    Ref: TM-T25164