
Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(49 produtos)
- Cisteína Protease(119 produtos)
- DPP-4(26 produtos)
- Glutaminase(46 produtos)
- HIV Protease(486 produtos)
- PAI-1(29 produtos)
- Inibidores de Protease(49 produtos)
- Receptor activado por protease(57 produtos)
- Proteassoma(91 produtos)
- Protease serina(66 produtos)
- p97(15 produtos)
Exibir 3 mais subcategorias
Foram encontrados 922 produtos para "Proteases/Proteassoma".
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Atazanavir Sulfate
CAS:Fórmula:C38H52N6O7·H2SO4Pureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:802.94Gabexate Mesylate
CAS:Fórmula:C16H23N3O4·CH4O3SPureza:>97.0%(N)Cor e Forma:White to Almost white powder to crystalPeso molecular:417.48Atazanavir
CAS:Fórmula:C38H52N6O7Pureza:>95.0%(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:704.874-(2-Aminoethyl)benzenesulfonyl Fluoride Hydrochloride [for Biochemical Research]
CAS:Fórmula:C8H10FNO2S·HClPureza:>99.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:239.692-Iodoacetamide [for Biochemical Research]
CAS:Fórmula:C2H4INOPureza:>98.0%(N)Cor e Forma:White to Light yellow powder to crystalPeso molecular:184.96Ritonavir
CAS:Fórmula:C37H48N6O5S2Pureza:>98.0%(HPLC)(N)Cor e Forma:White to Almost white powder to crystalinePeso molecular:720.95Benzamidine Hydrochloride [for Biochemical Research]
CAS:Fórmula:C7H8N2·HClPureza:>95.0%(T)(N)Cor e Forma:White to Almost white powder to crystalPeso molecular:156.61Disodium Dihydrogen Ethylenediaminetetraacetate Dihydrate [for Biochemical Research]
CAS:Fórmula:C10H14N2Na2O8·2H2OPureza:>99.0%(T)Cor e Forma:White powder to crystalinePeso molecular:372.24Ethylene Glycol Bis(2-aminoethyl Ether)-N,N,N',N'-tetraacetic Acid [for Biochemical Research]
CAS:Fórmula:C14H24N2O10Pureza:>95.0%(T)Cor e Forma:White to Almost white powder to crystalPeso molecular:380.35Benzylsulfonyl Fluoride [for Biochemical Research]
CAS:Fórmula:C7H7FO2SPureza:>98.0%(GC)Cor e Forma:White to Almost white powder to crystalPeso molecular:174.19Nafamostat Mesylate
CAS:Fórmula:C19H17N5O2·2CH4O3SPureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:539.58Camostat Mesylate
CAS:Fórmula:C20H22N4O5·CH4O3SPureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:494.52Limonin
CAS:Fórmula:C26H30O8Pureza:>95.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:470.521,10-Phenanthroline Monohydrate [for Biochemical Research]
CAS:Fórmula:C12H8N2·H2OPureza:>99.0%(T)Cor e Forma:White powder to crystalPeso molecular:198.23Dabigatran ethyl ester hydrochloride
CAS:Dabigatran prevents blood clots, inhibiting NQO2 and thrombin with IC50 0.8 μM.Fórmula:C27H30ClN7O3Pureza:99.65%Cor e Forma:White SolidPeso molecular:536.03HCV-IN-29
CAS:HCV-IN-29 is a hepatitis C virus (HCV) inhibitor.Fórmula:C26H32Cl4N6Pureza:99.89%Cor e Forma:Yellow SolidPeso molecular:570.38(Rac)-Telinavir
CAS:N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.
Fórmula:C33H44N6O5Pureza:99.30%Cor e Forma:SolidPeso molecular:604.74Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Fórmula:C19H17NO7Pureza:97.99%Cor e Forma:SolidPeso molecular:371.34Ref: TM-T15574
1mg84,00€2mg89,00€1mL*10mM (DMSO)90,00€5mg113,00€10mg178,00€25mg371,00€50mg573,00€100mg802,00€200mg1.099,00€CL-82198
CAS:CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Fórmula:C17H22N2O3Pureza:95.91%Cor e Forma:SolidPeso molecular:302.37Ref: TM-T14978
5mg44,00€1mL*10mM (DMSO)48,00€10mg70,00€25mg144,00€50mg230,00€100mg358,00€200mg523,00€500mg822,00€L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Fórmula:C26H41N3O5Pureza:98%Cor e Forma:SolidPeso molecular:475.6208(Rac)-Telmesteine
CAS:(Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) is an inhibitor of protease and is thus a suitable enzyme stabilizer.Fórmula:C7H11NO4SPureza:99.91%Cor e Forma:SolidPeso molecular:205.23RA190
CAS:RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.Fórmula:C28H23Cl5N2O2Pureza:97.7%Cor e Forma:SolidPeso molecular:596.76Ref: TM-T13858
1mg54,00€5mg109,00€1mL*10mM (DMSO)142,00€10mg159,00€25mg233,00€50mg414,00€100mg608,00€Saxagliptin hydrate
CAS:Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).Fórmula:C18H25N3O2·H2OPureza:99.52%Cor e Forma:SolidPeso molecular:333.43PMSF
CAS:PMSF (Phenylmethylsulfonyl fluoride) is an irreversible inhibitor of serine/cysteine protease , preparation of cell lysates. High-Quality, Low-Cost!Fórmula:C7H7FO2SPureza:97.75% - 99.88%Cor e Forma:White SolidPeso molecular:174.19DBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Fórmula:C16H25FN4O2Pureza:99.68%Cor e Forma:SolidPeso molecular:324.39Ref: TM-T15079
1mg48,00€5mg100,00€1mL*10mM (DMSO)110,00€10mg133,00€25mg215,00€50mg306,00€100mg414,00€200mg573,00€BAY-85-8501
CAS:BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Fórmula:C22H17F3N4O3SPureza:99.16%Cor e Forma:SolidPeso molecular:474.46Ref: TM-T12613L
1mg92,00€2mg122,00€5mg200,00€1mL*10mM (DMSO)208,00€10mg298,00€25mg535,00€50mg750,00€100mg1.035,00€Bivalirudin acetate
Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.Fórmula:C100H142N24O35Pureza:99.84%Cor e Forma:SolidPeso molecular:2240.34Anisindione
CAS:Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.Fórmula:C16H12O3Pureza:98.25%Cor e Forma:White SolidPeso molecular:252.26RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Fórmula:C19H13Cl4NOPureza:98.89% - 99.38%Cor e Forma:Yellow SolidPeso molecular:413.12LDN-27219
CAS:LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.Fórmula:C20H16N4O2S2Pureza:99.01% - 99.38%Cor e Forma:SolidPeso molecular:408.5Ref: TM-T11831
1mg34,00€5mg63,00€1mL*10mM (DMSO)67,00€10mg96,00€25mg152,00€50mg221,00€100mg334,00€200mg489,00€Trelagliptin
CAS:Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.Fórmula:C18H20FN5O2Pureza:98.88%Cor e Forma:SolidPeso molecular:357.38Gly-Pro-pNA hydrochloride
CAS:Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidaseFórmula:C13H17ClN4O4Pureza:99.84%Cor e Forma:SolidPeso molecular:328.75Retagliptin Phosphate
CAS:Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Fórmula:C19H21F6N4O7PPureza:98.70%Cor e Forma:SolidPeso molecular:562.36Ref: TM-T12710
100mgA consultar1mg34,00€2mg42,00€5mg60,00€1mL*10mM (DMSO)79,00€10mg87,00€25mg161,00€50mg245,00€ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Fórmula:C17H20N2O5SPureza:97.18%Cor e Forma:White SolidPeso molecular:364.42BJJF078
CAS:BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Fórmula:C27H29N3O6SPureza:99.56%Cor e Forma:SoildPeso molecular:523.6LSP-249
CAS:LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.Fórmula:C24H22ClN5OPureza:99.51%Cor e Forma:SolidPeso molecular:431.92midesteine
CAS:Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.Fórmula:C12H13NO3S3Pureza:99.87% - 99.98%Cor e Forma:SolidPeso molecular:315.43Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Fórmula:C49H55FN10O7SPureza:96.87% - 99.93%Cor e Forma:SolidPeso molecular:947.092-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Fórmula:C17H30N2O5Pureza:98%Cor e Forma:SolidPeso molecular:342.4305ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Fórmula:C17H24BF3N2O4Pureza:97.06%Cor e Forma:SolidPeso molecular:388.19Ref: TM-T12079
1mg109,00€2mg158,00€5mg259,00€1mL*10mM (DMSO)285,00€10mg409,00€25mg677,00€50mg954,00€100mg1.288,00€200mg1.728,00€BLT-1
CAS:BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.Fórmula:C12H23N3SPureza:97.97%Cor e Forma:White SolidPeso molecular:241.4Ref: TM-T14667
1mg43,00€2mg56,00€1mL*10mM (DMSO)90,00€5mg93,00€10mg152,00€25mg259,00€50mg409,00€100mg592,00€Mecarbinate
CAS:Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.Fórmula:C13H15NO3Pureza:99.28%Cor e Forma:Off-White Crystalline PowderPeso molecular:233.26Dabigatran etexilate
CAS:Dabigatran etexilate (BIBR 1048) is a thrombin inhibitor, which acts by binding and blocking thrombogenic activity and the prevention of thrombus formation.Fórmula:C34H41N7O5Pureza:98.19% - 99.98%Cor e Forma:White SolidPeso molecular:627.733-Aminopropionitrile fumarate (2:1)
CAS:3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.Fórmula:C4H4O4·2C3H6N2Pureza:99.76% - 99.79%Cor e Forma:White Crystalline PowderPeso molecular:256.26DPP-IV-IN-2
CAS:DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Fórmula:C18H26N4O5Pureza:99.08% - 99.51%Cor e Forma:White SolidPeso molecular:378.42Avoralstat
CAS:Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.Fórmula:C28H27N5O5Pureza:99.77%Cor e Forma:SolidPeso molecular:513.54IMAB027
CAS:Naratuximab (Anti-TSPAN26/CD37 Reference Antibody) is a humanized monoclonal antibody against CD37 that can be used to synthesize ADC compounds.Pureza:97.7% (SDS-PAGE); 97.5% (SEC-HPLC) - 97.7% (SDS-PAGE); 97.5% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:144.42 kDa



