Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(34 produtos)
- Cisteína Protease(96 produtos)
- DPP-4(20 produtos)
- Glutaminase(40 produtos)
- HIV Protease(449 produtos)
- PAI-1(25 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(53 produtos)
- Proteassoma(94 produtos)
- Protease serina(50 produtos)
- p97(14 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1044 produtos de "Proteases/Proteassoma"
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Avoralstat
CAS:<p>Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.</p>Fórmula:C28H27N5O5Pureza:99.77%Cor e Forma:SolidPeso molecular:513.54Ref: IN-DA0034HK
5gA consultar10g21,00€1kg124,00€25g25,00€50g25,00€5kg563,00€100g34,00€250g60,00€500g75,00€50kgA consultarFlanvotumab
CAS:<p>Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:145.42 kDaDenagliptin
CAS:<p>Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of</p>Fórmula:C20H18F3N3OPureza:99.12%Cor e Forma:SolidPeso molecular:373.37Anisindione
CAS:<p>Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.</p>Fórmula:C16H12O3Pureza:98.25%Cor e Forma:Pale Yellow Crystals From Acetic Acid Or Ethanol SolidPeso molecular:252.264-(2-Aminoethyl)benzenesulfonyl fluoride, HCl
CAS:Fórmula:C8H11ClFNO2SPureza:98%Cor e Forma:SolidPeso molecular:239.6948(ETHYLENEDINITRILO)TETRAACETIC ACID, TRISODIUM SALT HYDRATE
CAS:Fórmula:C10H18N2NaO9Pureza:97%Cor e Forma:SolidPeso molecular:333.2477(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
CAS:Fórmula:C16H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:308.3728Ref: IN-DA00370Q
1g132,00€5g223,00€10g532,00€25gA consultar50gA consultar100gA consultar10mg29,00€250gA consultar100mg44,00€250mg68,00€N-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Fórmula:C17H18ClNO3SPureza:97%Cor e Forma:SolidPeso molecular:351.8477Ethylenediaminetetraacetic acid disodium salt dihydrate
CAS:Fórmula:C10H18N2Na2O10Pureza:97%Cor e Forma:SolidPeso molecular:372.2369Q-VD-OPH
CAS:<p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>Fórmula:C26H25F2N3O6Pureza:97.8% - 98.95%Cor e Forma:SolidPeso molecular:513.5Ref: IN-DA003O5U
1g542,00€5gA consultar10mg61,00€25mg94,00€50mg148,00€100mg191,00€250mg197,00€500mg333,00€4-Chlorosalicylic acid
CAS:<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Fórmula:C7H5ClO3Pureza:98.59%Cor e Forma:Off-White To Light Beige PowderPeso molecular:172.57BLT-1
CAS:<p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>Fórmula:C12H23N3SPureza:97.97%Cor e Forma:SolidPeso molecular:241.4Elsulfavirine
CAS:<p>Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.</p>Fórmula:C24H17BrCl2FN3O5SPureza:99.66%Cor e Forma:SolidPeso molecular:629.28MK-0608
CAS:<p>MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).</p>Fórmula:C12H16N4O4Pureza:98.48%Cor e Forma:SolidPeso molecular:280.28Fostemsavir Tris
CAS:<p>Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.</p>Fórmula:C29H37N8O11PPureza:99.45%Cor e Forma:SolidPeso molecular:704.62Fenofibric acid
CAS:<p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>Fórmula:C17H15ClO4Pureza:99.36%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:318.75Dolutegravir intermediate-1
CAS:<p>Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.</p>Fórmula:C13H17NO8Pureza:99.52%Cor e Forma:SolidPeso molecular:315.28Ruzasvir
CAS:<p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>Fórmula:C49H55FN10O7SPureza:96.87% - 96.88%Cor e Forma:SolidPeso molecular:947.09Mecarbinate
CAS:<p>Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.</p>Fórmula:C13H15NO3Pureza:99.28%Cor e Forma:Off-White Crystalline PowderPeso molecular:233.26Trelagliptin
CAS:<p>Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.</p>Fórmula:C18H20FN5O2Pureza:98.88%Cor e Forma:SolidPeso molecular:357.38Retagliptin Phosphate
CAS:<p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>Fórmula:C19H21F6N4O7PPureza:98.70%Cor e Forma:SolidPeso molecular:562.36L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Fórmula:C26H41N3O5Pureza:98%Cor e Forma:SolidPeso molecular:475.6208Ref: IN-DA0072SK
1gA consultar5mg68,00€10mg90,00€25mg124,00€50mg168,00€100mg229,00€250mg500,00€500mgA consultarLSP-249
CAS:<p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>Fórmula:C24H22ClN5OPureza:99.51%Cor e Forma:SolidPeso molecular:431.92LDN-27219
CAS:<p>LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.</p>Fórmula:C20H16N4O2S2Pureza:99.01% - 99.38%Cor e Forma:SolidPeso molecular:408.5Begelomab
CAS:<p>Begelomab (SAND-26) is a mouse-derived monoclonal antibody targeting DPP-4/CD26. Begelomab can be used to study severe refractory inflammatory myopathies.</p>Pureza:97.8% (SDS-PAGE); 98.3% (SEC-HPLC) - 97.8% (SDS-PAGE); 98.3% (SEC-HPLC)Cor e Forma:LiquidSalicylanilide
CAS:<p>Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.</p>Fórmula:C13H11NO2Pureza:99.55%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:213.233-Deazaadenosine hydrochloride
CAS:<p>3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.</p>Fórmula:C11H15ClN4O4Pureza:98.48%Cor e Forma:SolidPeso molecular:302.71Sitagliptin
CAS:<p>Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.</p>Fórmula:C16H15F6N5OPureza:99.33% - 99.83%Cor e Forma:Yellow GreasePeso molecular:407.31Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Fórmula:C13H19NO4SPureza:98.95% - 99.84%Cor e Forma:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecular:285.36ARP-100
CAS:<p>ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).</p>Fórmula:C17H20N2O5SPureza:97.18%Cor e Forma:SolidPeso molecular:364.42BRD-6929
CAS:<p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>Fórmula:C19H17N3O2SPureza:98.01% - 99.05%Cor e Forma:SolidPeso molecular:351.42Hck-IN-1
CAS:<p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>Fórmula:C16H11ClN6O3SPureza:99.07%Cor e Forma:SolidPeso molecular:402.81Saxagliptin hydrate
CAS:<p>Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).</p>Fórmula:C18H25N3O2·H2OPureza:99.52%Cor e Forma:SolidPeso molecular:333.43PF-3450074
CAS:<p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>Fórmula:C27H27N3O2Pureza:99.92%Cor e Forma:SolidPeso molecular:425.52RAMB4
CAS:<p>RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.</p>Fórmula:C19H13Cl4NOPureza:98.89% - 99.38%Cor e Forma:SolidPeso molecular:413.12NBD-556
CAS:<p>NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.</p>Fórmula:C17H24ClN3O2Pureza:99.79%Cor e Forma:SolidPeso molecular:337.84PMSF
CAS:<p>PMSF (Phenylmethylsulfonyl fluoride) is an irreversible inhibitor of serine/cysteine protease , preparation of cell lysates. High-Quality, Low-Cost!</p>Fórmula:C7H7FO2SPureza:97.75% - 99.88%Cor e Forma:White To Cream SolidPeso molecular:174.193-Aminopropionitrile fumarate (2:1)
CAS:<p>3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.</p>Fórmula:C4H4O4·2C3H6N2Pureza:99.76% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:256.26ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Fórmula:C17H24BF3N2O4Pureza:97.06%Cor e Forma:SolidPeso molecular:388.19Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Fórmula:C12H12FN5O3Pureza:98.77%Cor e Forma:SolidPeso molecular:293.252-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Fórmula:C17H30N2O5Pureza:98%Cor e Forma:SolidPeso molecular:342.4305Sofosbuvir impurity F
CAS:<p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>Fórmula:C34H45FN4O13P2Pureza:98.05%Cor e Forma:SolidPeso molecular:798.69BJJF078
CAS:<p>BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.</p>Fórmula:C27H29N3O6SPureza:98.19%Cor e Forma:SoildPeso molecular:523.6Aprotinin
CAS:<p>Aprotinin (Traskolan) is a broad-spectrum serine protease (BPTI) inhibitor. Aprotinin is an antifibrinolytic agent. Cost-effective and quality-assured.</p>Fórmula:C284H432N84O79S7Pureza:98%Cor e Forma:SolidPeso molecular:6511.51Tenofovir diphosphate TEA
CAS:<p>Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.</p>Fórmula:C9H16N5O10P3·C6H15NPureza:93.45% - 98.51%Cor e Forma:SolidPeso molecular:548.366-Acetylnimbandiol
CAS:<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Fórmula:C28H34O8Cor e Forma:SolidPeso molecular:498.56α 1(I) Collagen (614-639), human
CAS:<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Fórmula:C134H189N37O39Pureza:98%Cor e Forma:SolidPeso molecular:2942.16EP 171
CAS:<p>EP 171 is a potent agonist of TP-receptors.</p>Fórmula:C23H29FO5Cor e Forma:SolidPeso molecular:404.47
![(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FIN%2Fthumb-webp%2FDA00370Q.webp&w=3840&q=75)
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![2-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbony…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FIN%2Fthumb-webp%2FDA0048C1.webp&w=3840&q=75)
