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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5337 produtos de "GPCR/Proteína-G"

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  • Cisapride

    CAS:
    <p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>
    Fórmula:C23H29ClFN3O4
    Pureza:99.77%
    Cor e Forma:White To Slightly Biege Powder Solid
    Peso molecular:465.95
  • DPTN dihydrochloride

    CAS:
    <p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>
    Fórmula:C22H20Cl2N4OS
    Pureza:99.95%
    Cor e Forma:Soild
    Peso molecular:459.39
  • LCKLSL hydrochloride


    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Fórmula:C30H58ClN7O8S
    Pureza:98.02% - 99.31%
    Cor e Forma:Solid
    Peso molecular:712.34
  • Tripelennamine hydrochloride

    CAS:
    <p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>
    Fórmula:C16H21N3·HCl
    Pureza:99.54% - 99.81%
    Cor e Forma:White Solid
    Peso molecular:291.82
  • Terlipressin Acetate

    CAS:
    <p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>
    Fórmula:C56H82N16O19S2
    Pureza:98.50% - 99.69%
    Cor e Forma:Solid
    Peso molecular:1347.5
  • Gevotroline

    CAS:
    <p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>
    Fórmula:C19H20FN3
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:309.38
  • Astressin acetate


    <p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>
    Fórmula:C163H273N49O44
    Pureza:96.87%
    Cor e Forma:Solid
    Peso molecular:3623.21
  • ESI-05

    CAS:
    <p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>
    Fórmula:C16H18O2S
    Pureza:97.22%
    Cor e Forma:Solid
    Peso molecular:274.38
  • Dexpramipexole dihydrochloride

    CAS:
    <p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>
    Fórmula:C10H19Cl2N3S
    Pureza:99.75% - 99.88%
    Cor e Forma:Solid
    Peso molecular:284.25
  • Anamorelin

    CAS:
    <p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>
    Fórmula:C31H42N6O3
    Pureza:99.35% - 99.94%
    Cor e Forma:Solid
    Peso molecular:546.7
  • PF-06882961

    CAS:
    <p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>
    Fórmula:C31H30FN5O4
    Pureza:98.06% - 99.54%
    Cor e Forma:Solid
    Peso molecular:555.6
  • Sonepcizumab

    CAS:
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Pureza:SDS-PAGE:95% SEC-HPLC:98.90%
    Cor e Forma:Liquid
    Peso molecular:146.43 kDa
  • Desipramine hydrochloride

    CAS:
    <p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>
    Fórmula:C18H23ClN2
    Pureza:99.58% - 99.94%
    Cor e Forma:White To Off-White Powder
    Peso molecular:302.842
  • Sergliflozin A

    CAS:
    <p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>
    Fórmula:C20H24O7
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:376.4
  • Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49
  • Diphenylpyraline hydrochloride

    CAS:
    <p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>
    Fórmula:C19H23NO·HCl
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:317.85
  • Olanzapine

    CAS:
    <p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>
    Fórmula:C17H20N4S
    Pureza:99.86% - ≥95%
    Cor e Forma:Yellowish Crystalline Powder
    Peso molecular:312.43
  • Bambuterol hydrochloride

    CAS:
    <p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>
    Fórmula:C18H30ClN3O5
    Pureza:99.53% - 99.61%
    Cor e Forma:White Solid
    Peso molecular:403.91
  • Levodropropizine

    CAS:
    <p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>
    Fórmula:C13H20N2O2
    Pureza:99.87% - 99.93%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:236.31
  • Fexofenadine hydrochloride

    CAS:
    <p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>
    Fórmula:C32H40ClNO4
    Pureza:>99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:538.12
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Fórmula:C15H20N2O2·HCl
    Pureza:99.64% - 99.92%
    Cor e Forma:Solid
    Peso molecular:296.79
  • Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Fórmula:C20H22BrFN2O
    Pureza:99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:405.304
  • Acetophenazine dimaleate

    CAS:
    <p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>
    Fórmula:C31H37N3O10S
    Pureza:99.39% - 99.48%
    Cor e Forma:Solid
    Peso molecular:643.71
  • Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Fórmula:C19H21N·HCl
    Pureza:98.54% - 99.98%
    Cor e Forma:Solid
    Peso molecular:299.84
  • Filorexant

    CAS:
    <p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki &lt;3 nM).</p>
    Fórmula:C24H25FN4O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:420.48
  • Indusatumab

    CAS:
    <p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>
    Pureza:> 95% - > 95%
    Cor e Forma:Liquid
    Peso molecular:145.18 kDa
  • JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Fórmula:C26H28ClN3O7
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:529.97
  • Erenumab

    CAS:
    <p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>
    Pureza:99.43% (SEC-HPLC) - > 95%
    Cor e Forma:Liquid
    Peso molecular:146.2 kDa
  • Fluoxetine hydrochloride

    CAS:
    <p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>
    Fórmula:C17H19ClF3NO
    Pureza:99.6% - 99.98%
    Cor e Forma:White To Off-White Crystalline Solid White To Off-White Powder
    Peso molecular:345.787
  • Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Fórmula:C34H36Cl2N6O5S·2ClH
    Pureza:99.17% - 99.58%
    Cor e Forma:Soild
    Peso molecular:784.58
  • Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:348.87
  • NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Fórmula:C27H31Cl2N3O3
    Pureza:99.33%
    Cor e Forma:Soild
    Peso molecular:516.46
  • Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Fórmula:C17H18F3NO
    Pureza:99.07% - 99.28%
    Cor e Forma:Solid
    Peso molecular:309.33
  • Promazine hydrochloride

    CAS:
    <p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>
    Fórmula:C17H21ClN2S
    Pureza:99.90%
    Cor e Forma:Solid
    Peso molecular:320.88
  • Blonanserin

    CAS:
    <p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>
    Fórmula:C23H30FN3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:367.5
  • Trazodone hydrochloride

    CAS:
    <p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>
    Fórmula:C19H23Cl2N5O
    Pureza:99.5% - 99.52%
    Cor e Forma:Solid
    Peso molecular:408.33
  • Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Fórmula:C14H15Cl2NS
    Pureza:99.85% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:300.25
  • PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Fórmula:C25H37Cl2N3O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:482.49
  • Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Fórmula:C19H24N2O·HCl
    Pureza:99.84% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:332.87
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Fórmula:C26H27N5O2
    Pureza:99.61%
    Cor e Forma:Light Yellow Solid
    Peso molecular:441.52
  • Adrenalone hydrochloride

    CAS:
    <p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>
    Fórmula:C9H11NO3·HCl
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:217.65
  • Urocortin (rat) acetate


    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Pureza:97.76%
    Cor e Forma:Soild
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Fórmula:C18H29ClN2O4
    Pureza:99.92% - >99.99%
    Cor e Forma:White Or Slightly Off-White Crystalline Powder Solid
    Peso molecular:372.89
  • Prochlorperazine Maleate

    CAS:
    <p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>
    Fórmula:C28H32ClN3O8S
    Pureza:99.78%
    Cor e Forma:Off-White Powder
    Peso molecular:606.09
  • Rimonabant hydrochloride

    CAS:
    <p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>
    Fórmula:C22H22Cl4N4O
    Pureza:98.24% - 99.5%
    Cor e Forma:Off-White To White Crystalline Powder
    Peso molecular:500.25
  • Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Cor e Forma:White Crystal Powder
    Peso molecular:365.86
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Cor e Forma:Solid
    Peso molecular:508.56
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Fórmula:C22H34Cl2N2O2
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:429.42
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Fórmula:C11H9BrO
    Pureza:98.51%
    Cor e Forma:White To Off-White Powder
    Peso molecular:237.09
  • CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Fórmula:C15H18Cl2N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:341.24
  • Chlorprothixene hydrochloride

    CAS:
    <p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>
    Fórmula:C18H18ClNS·HCl
    Pureza:99.76%
    Cor e Forma:White Powder
    Peso molecular:352.32
  • Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Fórmula:C26H35NO7
    Pureza:98.53% - 99.43%
    Cor e Forma:Coa
    Peso molecular:473.57
  • Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Fórmula:C19H31ClF3NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:413.9
  • Pizotifen

    CAS:
    <p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>
    Fórmula:C19H21NS
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:295.44
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79
  • CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Fórmula:C24H17ClN2O3
    Pureza:98% - 99.08%
    Cor e Forma:Solid
    Peso molecular:416.86
  • Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Fórmula:C17H28ClNO2
    Pureza:97.32% - 99.86%
    Cor e Forma:White Crystalline Powder
    Peso molecular:313.86
  • Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Fórmula:C19H21N3O
    Pureza:98.50% - 99.44%
    Cor e Forma:Solid
    Peso molecular:307.39
  • ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Fórmula:C20H25ClN4O2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:388.89
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Fórmula:C19H27N5O4·HCl
    Pureza:99.78%
    Cor e Forma:White To Off-White Solid
    Peso molecular:425.91
  • KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Fórmula:C26H40N4O8
    Pureza:98.46%
    Cor e Forma:Solid
    Peso molecular:536.62
  • Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Fórmula:C21H22CL2N4OS
    Pureza:97.97% - 99.82%
    Cor e Forma:Solid
    Peso molecular:449.4
  • Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Fórmula:C22H29N3O4S
    Pureza:98.55%
    Cor e Forma:Yellowish White Crystalline Powder
    Peso molecular:431.55
  • Silodosin

    CAS:
    <p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>
    Fórmula:C25H32F3N3O4
    Pureza:99.282% - 99.76%
    Cor e Forma:Colorless To Pink Solid
    Peso molecular:495.53
  • Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Fórmula:C16H21N3O2
    Pureza:99.69% - 99.91%
    Cor e Forma:White Or Kind Of White Powder
    Peso molecular:287.36
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51
  • Nylidrin hydrochloride

    CAS:
    <p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells &amp; human basophils.</p>
    Fórmula:C19H26ClNO2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:335.87
  • Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Fórmula:C12H19NO10
    Pureza:99.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:337.28
  • Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65
  • Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Fórmula:C18H26ClN3O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:367.87
  • Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • Salmeterol

    CAS:
    <p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Cor e Forma:Solid
    Peso molecular:415.57
  • Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>
    Fórmula:C28H30N2O8
    Pureza:99.7% - >99.99%
    Cor e Forma:Powder
    Peso molecular:522.55
  • Antazoline hydrochloride

    CAS:
    <p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>
    Fórmula:C17H19N3·HCl
    Pureza:98% - 99.53%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:301.82
  • Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Fórmula:C13H16N4
    Pureza:98.34% - 99.73%
    Cor e Forma:Solid
    Peso molecular:228.29
  • Senktide acetate


    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Fórmula:C42H59N7O13S
    Pureza:98.26%
    Cor e Forma:Solid
    Peso molecular:902.02
  • Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Fórmula:C21H27Cl3N2O3
    Pureza:99.4% - 99.97%
    Cor e Forma:Solid
    Peso molecular:461.81
  • (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Cor e Forma:Soild
    Peso molecular:195.19
  • Ro 10-5824 dihydrochloride

    CAS:
    <p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:353.29
  • AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Fórmula:C17H14O5
    Pureza:97.59%
    Cor e Forma:Solid
    Peso molecular:298.29
  • Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21
  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41
  • Dimenhydrinate

    CAS:
    <p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>
    Fórmula:C24H28ClN5O3
    Pureza:99.57% - 99.77%
    Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Peso molecular:469.96
  • (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Fórmula:C32H30F5N3O5
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:631.59
  • Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Fórmula:C21H16F5N7O3
    Pureza:99.33% - 99.71%
    Cor e Forma:Solid
    Peso molecular:509.39
  • Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Fórmula:C9H15ClNO5P
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:283.65
  • MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Fórmula:C27H25N3O4S2
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:519.64
  • Moxisylyte hydrochloride

    CAS:
    <p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>
    Fórmula:C16H26ClNO3
    Pureza:99.93% - ≥95%
    Cor e Forma:Solid
    Peso molecular:315.84
  • YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74
  • Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Fórmula:C12H9NS
    Pureza:99.95%
    Cor e Forma:Yellow Solid Pellets
    Peso molecular:199.27
  • NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Fórmula:C20H24ClN3O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:357.88
  • Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55
  • Ketanserin

    CAS:
    <p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>
    Fórmula:C22H22FN3O3
    Pureza:99.19% - 99.73%
    Cor e Forma:Solid
    Peso molecular:395.43
  • Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Fórmula:C11H17NO3·5H2O4S
    Pureza:98.53% - 99.74%
    Cor e Forma:Solid
    Peso molecular:260.3
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Fórmula:C21H24ClNO
    Pureza:99.77% - >99.99%
    Cor e Forma:White To Slightly Yellowish Crystalline Solid
    Peso molecular:341.88
  • Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:384.9
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Fórmula:C31H38N2O
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:454.65