
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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[Leu13]-Motilin
CAS:<p>[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinal</p>Fórmula:C121H190N34O35Pureza:98%Cor e Forma:SolidPeso molecular:2681.01Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:<p>Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.</p>Fórmula:C25H26O13Cor e Forma:SolidPeso molecular:534.47CAY10597
CAS:<p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>Fórmula:C20H14ClFN2O5Cor e Forma:SolidPeso molecular:416.79JPC0323
<p>JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target properties, acceptable plasma exposure, and adequate</p>Fórmula:C22H43NO4Pureza:98%Cor e Forma:SolidPeso molecular:385.58Gemeprost
CAS:<p>Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.</p>Fórmula:C23H38O5Pureza:98%Cor e Forma:SolidPeso molecular:394.54Leukotriene B5
CAS:<p>LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.4561,2,3-Trilinoelaidoyl-rac-glycerol
CAS:<p>1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.</p>Fórmula:C57H98O6Cor e Forma:SolidPeso molecular:879.405M617
CAS:<p>Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.</p>Fórmula:C112H161N29O28Pureza:98%Cor e Forma:SolidPeso molecular:2361.684-Oxo-5-phenylpentanoic aci
CAS:<p>4-Oxo-5-phenylpentanoic aci is a useful organic compound for research related to life sciences. The catalog number is T125056 and the CAS number is 3183-15-1.</p>Fórmula:C11H12O3Cor e Forma:SolidPeso molecular:192.2145(S),6(R)-11-trans DiHETE
CAS:<p>5(S),6(R)-11-trans DiHETE, a C-11 isomer of 5(S),6(R)-DiHETE, occurs in rat kidneys, formed enzymatically; not a soybean lipoxygenase substrate.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.47Olcegepant hydrochloride
CAS:<p>Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.</p>Fórmula:C38H48Br2ClN9O5Pureza:99.69%Cor e Forma:SolidPeso molecular:906.1117-trifluoromethylphenyl-13,14-dihydro trinor Prostaglandin F2α
CAS:<p>A number of 17-phenyl trinor prostaglandin F2α(17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.1,2,3Of these, the ones</p>Fórmula:C24H33F3O5Cor e Forma:SolidPeso molecular:458.51816-phenoxy tetranor Prostaglandin F2α isopropyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Fórmula:C25H36O6Cor e Forma:SolidPeso molecular:432.557Quinelorane
CAS:<p>Quinelorane is dextrorotary isomer.</p>Fórmula:C14H22N4Cor e Forma:SolidPeso molecular:246.35GR 82334
CAS:<p>Tachykinin NK1 receptor antagonist.</p>Fórmula:C69H91N15O16Pureza:98%Cor e Forma:SolidPeso molecular:1386.57Physalaemin
CAS:<p>Physalaemin is a non-mammalian tachykinin.</p>Fórmula:C58H84N14O16SPureza:98%Cor e Forma:SolidPeso molecular:1265.45SRI-37330
CAS:<p>SRI-37330 inhibits glucagon secretion and function, reduces hepatic glucose production, and reverses hepatic steatosis.</p>Fórmula:C16H19F3N4O2SPureza:99.65%Cor e Forma:SolidPeso molecular:388.41Brain Natriuretic Peptide-45, rat
CAS:<p>BNP-45 (rat) is a circulating form of rat brain natriuretic peptide isolated from rat heart with potent hypotensive and natriuretic potency.</p>Fórmula:C213H349N71O65S3Pureza:98%Cor e Forma:SolidPeso molecular:5040.67Endothelin-3, human, mouse, rabbit, rat
CAS:<p>Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.</p>Fórmula:C121H168N26O33S4Pureza:98%Cor e Forma:SolidPeso molecular:2643.04ACTH (34-39)
CAS:ACTH (34-39) is an adrenocorticotropic hormone fragment.Fórmula:C37H50N6O9Pureza:98%Cor e Forma:SolidPeso molecular:722.83(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Fórmula:C64H81N17O14Peso molecular:1312.43[D-Trp8,Tyr11] Somatostatin
CAS:[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Fórmula:C76H104N18O20S2Peso molecular:1653.88(D-Ala2)-GRF (1-29) amide (human)
CAS:(D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-Fórmula:C149H246N44O42SPeso molecular:3357.88[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Fórmula:C54H71N15O14Pureza:98%Cor e Forma:SolidPeso molecular:1154.23Glucagon (19-29), human
CAS:Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Fórmula:C61H89N15O18SPureza:98%Cor e Forma:SolidPeso molecular:1352.53Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:<p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>Fórmula:C49H70N14O12S2Pureza:98%Cor e Forma:SolidPeso molecular:1111.3Galanin-Like Peptide (human)
CAS:<p>Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, body weight, and energy metabolism [1].</p>Fórmula:C292H451N83O84SPureza:98%Cor e Forma:SolidPeso molecular:6500.28Sulamserod
CAS:<p>Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related</p>Fórmula:C19H28ClN3O5SPureza:98.76%Cor e Forma:SolidPeso molecular:445.96(Iso)-Landipirdine
CAS:<p>(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.</p>Fórmula:C18H19FN2O3SPureza:98.50%Cor e Forma:SoildPeso molecular:362.42[Ala11,D-Leu15]-Orexin B acetate
<p>[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).</p>Fórmula:C122H210N44O37SPureza:98.18%Cor e Forma:SolidPeso molecular:2917.31Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:<p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>Fórmula:C47H75N13O11Pureza:98%Cor e Forma:SolidPeso molecular:998.18Dalcotidine
CAS:<p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>Fórmula:C18H29N3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:319.44β-MSH, human
CAS:<p>beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).</p>Fórmula:C118H174N34O35SPureza:98%Cor e Forma:SolidPeso molecular:2660.92LY-426965 hydrochloride
CAS:LY-426965 hydrochloride is a bioactive chemical.Fórmula:C28H39ClN2O2Cor e Forma:SolidPeso molecular:471.074-Thiouridine 5′-triphosphate disodium
CAS:<p>4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (</p>Fórmula:C9H11N2Na2O14P3SPureza:98%Cor e Forma:SolidPeso molecular:546.19Petrelintide acetate
<p>Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.</p>Fórmula:C185H305N49O61·xC2H4O2Cor e Forma:SolidPeso molecular:4191.69 (free base)CRSP-1
CAS:Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.Fórmula:C175H294N54O49S5Pureza:98%Cor e Forma:SolidPeso molecular:4098.885-HT5AR/5-HT6R ligand-1
<p>5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.</p>Fórmula:C25H30N4O2SCor e Forma:SolidPeso molecular:450.65-HT6R antagonist 1
<p>Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability</p>Fórmula:C17H22F2N6OPureza:98%Cor e Forma:SolidPeso molecular:364.39mPGES-1/sEH-IN-1
<p>mPGES-1/sEH-IN-1 (compound 1f) is an sEH inhibitor with an IC50 value of 5 μM. It also exhibits antitumor activity by inhibiting mPGES-1, with an IC50 value of 25 µM.</p>Fórmula:C20H16F3N3O2Cor e Forma:SolidPeso molecular:387.355CB2 PET Radioligand 1
<p>CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.</p>Fórmula:C20H19F3N4OPureza:98%Cor e Forma:SolidPeso molecular:388.39BQ-3020 ammonium
<p>BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2</p>Fórmula:C96H140N20O25S·xNH3Pureza:98%Cor e Forma:SolidPeso molecular:2006.32 (free base)TCMCB07 TFA
<p>TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role in</p>Fórmula:C63H87N15O11·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:1230.46 (free base)TCMCB07
CAS:<p>TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications in</p>Fórmula:C63H87N15O11Pureza:98%Cor e Forma:SolidPeso molecular:1230.46Substance P(1-7)
CAS:Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.Fórmula:C41H65N13O10Pureza:98%Cor e Forma:SolidPeso molecular:900.04Galanin-Like Peptide (rat)
CAS:<p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>Fórmula:C288H461N87O83SPureza:98%Cor e Forma:SolidPeso molecular:6502.34pCPA methyl ester hydrochloride
CAS:<p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>Fórmula:C10H13Cl2NO2Pureza:99.73% - 99.88%Cor e Forma:SolidPeso molecular:250.12Benzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Fórmula:C22H32N2O5Pureza:94.86%Cor e Forma:SolidPeso molecular:404.5V-0219
CAS:<p>V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.</p>Fórmula:C20H25F3N4O2Pureza:99.91%Cor e Forma:SoildPeso molecular:410.43Pimozide-d4
CAS:<p>Pimozide D4 is a deuterium labeled Pimozide.</p>Fórmula:C28H29F2N3OPureza:98%Cor e Forma:SolidPeso molecular:465.57Hydroxyzine D8
CAS:Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Fórmula:C21H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:382.95TP-16
CAS:<p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>Fórmula:C24H22FNO4SPureza:98.53% - 99.15%Cor e Forma:SolidPeso molecular:439.5Revdofilimab
CAS:<p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>Pureza:98.80% - 98.80%Cor e Forma:LiquidEticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Cor e Forma:SolidPeso molecular:377.31Docosahexaenoic acid ethyl ester
CAS:<p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>Fórmula:C24H36O2Cor e Forma:SolidPeso molecular:356.54PD176252
CAS:<p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>Fórmula:C32H36N6O5Pureza:99.18%Cor e Forma:SolidPeso molecular:584.67SYL-4
CAS:SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Fórmula:C20H15N3O5SPureza:95.76%Cor e Forma:SoildPeso molecular:409.42GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Fórmula:C15H21N5O5Cor e Forma:SolidPeso molecular:351.36Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Fórmula:C54H69N11O10S2Cor e Forma:SolidPeso molecular:1096.32L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Fórmula:C27H22BrNO4SPureza:98.97%Cor e Forma:SolidPeso molecular:536.44Clozapine-d8
CAS:<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Fórmula:C18H19ClN4Cor e Forma:SolidPeso molecular:334.87BW 723C86
CAS:<p>BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.</p>Fórmula:C16H19ClN2OSPureza:99.35%Cor e Forma:SolidPeso molecular:322.85Sumatriptan
CAS:<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Fórmula:C14H21N3O2SPureza:99.93%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.4Neurotensin(8-13)
CAS:<p>Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>Fórmula:C38H64N12O8Pureza:99.95%Cor e Forma:SolidPeso molecular:816.99Travoprost (Standard)
CAS:Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Fórmula:C26H35F3O6Peso molecular:500.55Clencyclohexerol-d10
CAS:<p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:329.29Aramisulpride
CAS:<p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>Fórmula:C17H27N3O4SCor e Forma:SolidPeso molecular:369.48Scopine hydrochloride
CAS:<p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>Fórmula:C8H13NO2·HClPureza:98%Cor e Forma:White PowderPeso molecular:191.66Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Fórmula:C18H18ClN3SPureza:99.93%Cor e Forma:SolidPeso molecular:343.87SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Fórmula:C15H15ClN4OPureza:98%Cor e Forma:SolidPeso molecular:302.76MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Fórmula:C17H19N5OC2H2O4Pureza:97.10%Cor e Forma:SolidPeso molecular:354.39Apraclonidine hydrochloride
CAS:<p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>Fórmula:C9H11Cl3N4Pureza:99.74%Cor e Forma:SolidPeso molecular:281.57Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Fórmula:C46H65N15O12S2Pureza:98%Cor e Forma:White PowderPeso molecular:1084.23Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Fórmula:C17H17Cl2NOCor e Forma:SolidPeso molecular:322.23Asenapine
CAS:<p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>Fórmula:C17H16ClNOPureza:99.64%Cor e Forma:CoaPeso molecular:285.77(S)-(+)-Dimethindene maleate
CAS:<p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>Fórmula:C24H28N2O4Pureza:99.94%Cor e Forma:SolidPeso molecular:408.49GLP-1 receptor agonist 7
CAS:<p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>Fórmula:C31H30ClFN4O5Cor e Forma:SolidPeso molecular:593.05Omidenepag
CAS:Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Fórmula:C23H22N6O4SPureza:99.67% - 99.77%Cor e Forma:SolidPeso molecular:478.52SLIGRL-NH2
CAS:<p>SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.</p>Fórmula:C29H56N10O7Pureza:98.29%Cor e Forma:SolidPeso molecular:656.82Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Fórmula:C32H39NO4Pureza:98%Cor e Forma:SolidPeso molecular:507.69Agomelatine (L(+)-Tartaric acid)
CAS:<p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>Fórmula:C19H23NO8Cor e Forma:SolidPeso molecular:393.39Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H18ClN3SPureza:98%Cor e Forma:White Crystalline PowderPeso molecular:247.79Sumanirole maleate
CAS:<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Fórmula:C15H17N3O5Pureza:98%Cor e Forma:SolidPeso molecular:319.31ML 00253764
CAS:melanocortin MC4 receptor antagonistFórmula:C18H18BrFN2OCor e Forma:SolidPeso molecular:377.253-Hydroxy agomelatine
CAS:<p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>Fórmula:C15H17NO3Cor e Forma:SolidPeso molecular:259.3Lysosphingomyelin (d18:1)
CAS:<p>Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.</p>Fórmula:C23H49N2O5PCor e Forma:SolidPeso molecular:464.628Tegaserod
CAS:Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Fórmula:C16H23N5OPureza:99.20% - 99.89%Cor e Forma:SolidPeso molecular:301.39LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:335.34Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Fórmula:C27H34N4O3Pureza:99.33%Cor e Forma:SolidPeso molecular:462.58Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Fórmula:C22H25N3O3Pureza:99.94%Cor e Forma:SolidPeso molecular:379.45SANT 2
CAS:<p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>Fórmula:C26H26ClN3O4Pureza:99.23%Cor e Forma:SolidPeso molecular:479.96Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Fórmula:C145H240N44O48S2Pureza:99.41% - 99.80%Cor e Forma:PowderPeso molecular:3431.85Bromperidol hydrochloride
CAS:<p>Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.</p>Fórmula:C21H24BrClFNO2Cor e Forma:SolidPeso molecular:456.78Granisetron
CAS:<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Fórmula:C10H16N8S2Pureza:98%Cor e Forma:SolidPeso molecular:312.42Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Fórmula:C19H24N2OSPureza:99.15%Cor e Forma:SolidPeso molecular:328.47BMS-986224
CAS:<p>BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.</p>Fórmula:C24H23ClN4O6Pureza:98.61% - 99.67%Cor e Forma:SolidPeso molecular:498.92(+)-Penbutolol
CAS:(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Fórmula:C18H29NO2Cor e Forma:SolidPeso molecular:291.43Taranabant racemate
CAS:<p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>Fórmula:C27H25ClF3N3O2Pureza:98%Cor e Forma:SolidPeso molecular:515.951-Phenylbiguanide HCl
CAS:<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Fórmula:C8H12ClN5Pureza:99.31%Cor e Forma:SolidPeso molecular:213.67

