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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • [Leu13]-Motilin

    CAS:
    <p>[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinal</p>
    Fórmula:C121H190N34O35
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2681.01
  • Apigenin 6,8-di-C-α-L-arabinopyranoside

    CAS:
    <p>Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.</p>
    Fórmula:C25H26O13
    Cor e Forma:Solid
    Peso molecular:534.47
  • CAY10597

    CAS:
    <p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>
    Fórmula:C20H14ClFN2O5
    Cor e Forma:Solid
    Peso molecular:416.79
  • JPC0323


    <p>JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target properties, acceptable plasma exposure, and adequate</p>
    Fórmula:C22H43NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:385.58
  • Gemeprost

    CAS:
    <p>Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.</p>
    Fórmula:C23H38O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:394.54
  • Leukotriene B5

    CAS:
    <p>LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.</p>
    Fórmula:C20H30O4
    Cor e Forma:Solid
    Peso molecular:334.456
  • 1,2,3-Trilinoelaidoyl-rac-glycerol

    CAS:
    <p>1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.</p>
    Fórmula:C57H98O6
    Cor e Forma:Solid
    Peso molecular:879.405
  • M617

    CAS:
    <p>Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.</p>
    Fórmula:C112H161N29O28
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2361.68
  • 4-Oxo-5-phenylpentanoic aci

    CAS:
    <p>4-Oxo-5-phenylpentanoic aci is a useful organic compound for research related to life sciences. The catalog number is T125056 and the CAS number is 3183-15-1.</p>
    Fórmula:C11H12O3
    Cor e Forma:Solid
    Peso molecular:192.214
  • 5(S),6(R)-11-trans DiHETE

    CAS:
    <p>5(S),6(R)-11-trans DiHETE, a C-11 isomer of 5(S),6(R)-DiHETE, occurs in rat kidneys, formed enzymatically; not a soybean lipoxygenase substrate.</p>
    Fórmula:C20H32O4
    Cor e Forma:Solid
    Peso molecular:336.47
  • Olcegepant hydrochloride

    CAS:
    <p>Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.</p>
    Fórmula:C38H48Br2ClN9O5
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:906.11
  • 17-trifluoromethylphenyl-13,14-dihydro trinor Prostaglandin F2α

    CAS:
    <p>A number of 17-phenyl trinor prostaglandin F2α(17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.1,2,3Of these, the ones</p>
    Fórmula:C24H33F3O5
    Cor e Forma:Solid
    Peso molecular:458.518
  • 16-phenoxy tetranor Prostaglandin F2α isopropyl ester

    CAS:
    <p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>
    Fórmula:C25H36O6
    Cor e Forma:Solid
    Peso molecular:432.557
  • Quinelorane

    CAS:
    <p>Quinelorane is dextrorotary isomer.</p>
    Fórmula:C14H22N4
    Cor e Forma:Solid
    Peso molecular:246.35
  • GR 82334

    CAS:
    <p>Tachykinin NK1 receptor antagonist.</p>
    Fórmula:C69H91N15O16
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1386.57
  • Physalaemin

    CAS:
    <p>Physalaemin is a non-mammalian tachykinin.</p>
    Fórmula:C58H84N14O16S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1265.45
  • SRI-37330

    CAS:
    <p>SRI-37330 inhibits glucagon secretion and function, reduces hepatic glucose production, and reverses hepatic steatosis.</p>
    Fórmula:C16H19F3N4O2S
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:388.41
  • Brain Natriuretic Peptide-45, rat

    CAS:
    <p>BNP-45 (rat) is a circulating form of rat brain natriuretic peptide isolated from rat heart with potent hypotensive and natriuretic potency.</p>
    Fórmula:C213H349N71O65S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:5040.67
  • Endothelin-3, human, mouse, rabbit, rat

    CAS:
    <p>Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.</p>
    Fórmula:C121H168N26O33S4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2643.04
  • ACTH (34-39)

    CAS:
    ACTH (34-39) is an adrenocorticotropic hormone fragment.
    Fórmula:C37H50N6O9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:722.83
  • (D-Trp6)-LHRH free acid

    CAS:
    (D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .
    Fórmula:C64H81N17O14
    Peso molecular:1312.43
  • [D-Trp8,Tyr11] Somatostatin

    CAS:
    [D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,
    Fórmula:C76H104N18O20S2
    Peso molecular:1653.88
  • (D-Ala2)-GRF (1-29) amide (human)

    CAS:
    (D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-
    Fórmula:C149H246N44O42S
    Peso molecular:3357.88
  • [Gln8]-C517 (LH-RH), chicken

    CAS:
    [Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.
    Fórmula:C54H71N15O14
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1154.23
  • Glucagon (19-29), human

    CAS:
    Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.
    Fórmula:C61H89N15O18S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1352.53
  • Dp[Tyr(methyl)2,Arg8]-Vasopressin

    CAS:
    <p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>
    Fórmula:C49H70N14O12S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1111.3
  • Galanin-Like Peptide (human)

    CAS:
    <p>Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, body weight, and energy metabolism [1].</p>
    Fórmula:C292H451N83O84S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:6500.28
  • Sulamserod

    CAS:
    <p>Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related</p>
    Fórmula:C19H28ClN3O5S
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:445.96
  • (Iso)-Landipirdine

    CAS:
    <p>(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.</p>
    Fórmula:C18H19FN2O3S
    Pureza:98.50%
    Cor e Forma:Soild
    Peso molecular:362.42
  • [Ala11,D-Leu15]-Orexin B acetate


    <p>[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).</p>
    Fórmula:C122H210N44O37S
    Pureza:98.18%
    Cor e Forma:Solid
    Peso molecular:2917.31
  • Lys-(Des-Arg9,Leu8)-Bradykinin

    CAS:
    <p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>
    Fórmula:C47H75N13O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:998.18
  • Dalcotidine

    CAS:
    <p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>
    Fórmula:C18H29N3O2
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:319.44
  • β-MSH, human

    CAS:
    <p>beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).</p>
    Fórmula:C118H174N34O35S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2660.92
  • LY-426965 hydrochloride

    CAS:
    LY-426965 hydrochloride is a bioactive chemical.
    Fórmula:C28H39ClN2O2
    Cor e Forma:Solid
    Peso molecular:471.07
  • 4-Thiouridine 5′-triphosphate disodium

    CAS:
    <p>4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (</p>
    Fórmula:C9H11N2Na2O14P3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:546.19
  • Petrelintide acetate


    <p>Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.</p>
    Fórmula:C185H305N49O61·xC2H4O2
    Cor e Forma:Solid
    Peso molecular:4191.69 (free base)
  • CRSP-1

    CAS:
    Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.
    Fórmula:C175H294N54O49S5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4098.88
  • 5-HT5AR/5-HT6R ligand-1


    <p>5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.</p>
    Fórmula:C25H30N4O2S
    Cor e Forma:Solid
    Peso molecular:450.6
  • 5-HT6R antagonist 1


    <p>Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability</p>
    Fórmula:C17H22F2N6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.39
  • mPGES-1/sEH-IN-1


    <p>mPGES-1/sEH-IN-1 (compound 1f) is an sEH inhibitor with an IC50 value of 5 μM. It also exhibits antitumor activity by inhibiting mPGES-1, with an IC50 value of 25 µM.</p>
    Fórmula:C20H16F3N3O2
    Cor e Forma:Solid
    Peso molecular:387.355
  • CB2 PET Radioligand 1


    <p>CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.</p>
    Fórmula:C20H19F3N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:388.39
  • BQ-3020 ammonium


    <p>BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2</p>
    Fórmula:C96H140N20O25S·xNH3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2006.32 (free base)
  • TCMCB07 TFA


    <p>TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role in</p>
    Fórmula:C63H87N15O11·xC2HF3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1230.46 (free base)
  • TCMCB07

    CAS:
    <p>TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications in</p>
    Fórmula:C63H87N15O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1230.46
  • Substance P(1-7)

    CAS:
    Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.
    Fórmula:C41H65N13O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:900.04
  • Galanin-Like Peptide (rat)

    CAS:
    <p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>
    Fórmula:C288H461N87O83S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:6502.34
  • pCPA methyl ester hydrochloride

    CAS:
    <p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.73% - 99.88%
    Cor e Forma:Solid
    Peso molecular:250.12
  • Benzquinamide

    CAS:
    <p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>
    Fórmula:C22H32N2O5
    Pureza:94.86%
    Cor e Forma:Solid
    Peso molecular:404.5
  • V-0219

    CAS:
    <p>V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.</p>
    Fórmula:C20H25F3N4O2
    Pureza:99.91%
    Cor e Forma:Soild
    Peso molecular:410.43
  • Pimozide-d4

    CAS:
    <p>Pimozide D4 is a deuterium labeled Pimozide.</p>
    Fórmula:C28H29F2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:465.57
  • Hydroxyzine D8

    CAS:
    Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
    Fórmula:C21H27ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:382.95
  • TP-16

    CAS:
    <p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>
    Fórmula:C24H22FNO4S
    Pureza:98.53% - 99.15%
    Cor e Forma:Solid
    Peso molecular:439.5
  • Revdofilimab

    CAS:
    <p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>
    Pureza:98.80% - 98.80%
    Cor e Forma:Liquid
  • Eticlopride hydrochloride

    CAS:
    <p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>
    Fórmula:C17H25ClN2O3·HCl
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:377.31
  • Docosahexaenoic acid ethyl ester

    CAS:
    <p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>
    Fórmula:C24H36O2
    Cor e Forma:Solid
    Peso molecular:356.54
  • PD176252

    CAS:
    <p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>
    Fórmula:C32H36N6O5
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:584.67
  • SYL-4

    CAS:
    SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.
    Fórmula:C20H15N3O5S
    Pureza:95.76%
    Cor e Forma:Soild
    Peso molecular:409.42
  • GR79236

    CAS:
    GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
    Fórmula:C15H21N5O5
    Cor e Forma:Solid
    Peso molecular:351.36
  • Lanreotide

    CAS:
    Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.
    Fórmula:C54H69N11O10S2
    Cor e Forma:Solid
    Peso molecular:1096.32
  • L-798106

    CAS:
    L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.
    Fórmula:C27H22BrNO4S
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:536.44
  • Clozapine-d8

    CAS:
    <p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>
    Fórmula:C18H19ClN4
    Cor e Forma:Solid
    Peso molecular:334.87
  • BW 723C86

    CAS:
    <p>BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.</p>
    Fórmula:C16H19ClN2OS
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:322.85
  • Sumatriptan

    CAS:
    <p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>
    Fórmula:C14H21N3O2S
    Pureza:99.93%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:295.4
  • Neurotensin(8-13)

    CAS:
    <p>Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>
    Fórmula:C38H64N12O8
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:816.99
  • Travoprost (Standard)

    CAS:
    Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.
    Fórmula:C26H35F3O6
    Peso molecular:500.55
  • Clencyclohexerol-d10

    CAS:
    <p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>
    Fórmula:C14H20Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:329.29
  • Aramisulpride

    CAS:
    <p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>
    Fórmula:C17H27N3O4S
    Cor e Forma:Solid
    Peso molecular:369.48
  • Scopine hydrochloride

    CAS:
    <p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>
    Fórmula:C8H13NO2·HCl
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:191.66
  • Clothiapine

    CAS:
    Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
    Fórmula:C18H18ClN3S
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:343.87
  • SB-200646A

    CAS:
    SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.
    Fórmula:C15H15ClN4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:302.76
  • MRS-3777 hemioxalate

    CAS:
    <p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>
    Fórmula:C17H19N5OC2H2O4
    Pureza:97.10%
    Cor e Forma:Solid
    Peso molecular:354.39
  • Apraclonidine hydrochloride

    CAS:
    <p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>
    Fórmula:C9H11Cl3N4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:281.57
  • Argipressin

    CAS:
    <p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>
    Fórmula:C46H65N15O12S2
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:1084.23
  • Asenapine hydrochloride

    CAS:
    <p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>
    Fórmula:C17H17Cl2NO
    Cor e Forma:Solid
    Peso molecular:322.23
  • Asenapine

    CAS:
    <p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>
    Fórmula:C17H16ClNO
    Pureza:99.64%
    Cor e Forma:Coa
    Peso molecular:285.77
  • (S)-(+)-Dimethindene maleate

    CAS:
    <p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>
    Fórmula:C24H28N2O4
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:408.49
  • GLP-1 receptor agonist 7

    CAS:
    <p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>
    Fórmula:C31H30ClFN4O5
    Cor e Forma:Solid
    Peso molecular:593.05
  • Omidenepag

    CAS:
    Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.
    Fórmula:C23H22N6O4S
    Pureza:99.67% - 99.77%
    Cor e Forma:Solid
    Peso molecular:478.52
  • SLIGRL-NH2

    CAS:
    <p>SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.</p>
    Fórmula:C29H56N10O7
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:656.82
  • Fexofenadine-d6

    CAS:
    <p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>
    Fórmula:C32H39NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:507.69
  • Agomelatine (L(+)-Tartaric acid)

    CAS:
    <p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>
    Fórmula:C19H23NO8
    Cor e Forma:Solid
    Peso molecular:393.39
  • Pramipexole dihydrochloride

    CAS:
    Pramipexole dihydrochloride could be used to treat Parkinson disease.
    Fórmula:C10H18ClN3S
    Pureza:98%
    Cor e Forma:White Crystalline Powder
    Peso molecular:247.79
  • Sumanirole maleate

    CAS:
    <p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>
    Fórmula:C15H17N3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.31
  • ML 00253764

    CAS:
    melanocortin MC4 receptor antagonist
    Fórmula:C18H18BrFN2O
    Cor e Forma:Solid
    Peso molecular:377.25
  • 3-Hydroxy agomelatine

    CAS:
    <p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>
    Fórmula:C15H17NO3
    Cor e Forma:Solid
    Peso molecular:259.3
  • Lysosphingomyelin (d18:1)

    CAS:
    <p>Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.</p>
    Fórmula:C23H49N2O5P
    Cor e Forma:Solid
    Peso molecular:464.628
  • Tegaserod

    CAS:
    Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).
    Fórmula:C16H23N5O
    Pureza:99.20% - 99.89%
    Cor e Forma:Solid
    Peso molecular:301.39
  • LAS101057

    CAS:
    LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
    Fórmula:C18H14FN5O
    Pureza:99.03% - >99.99%
    Cor e Forma:Solid
    Peso molecular:335.34
  • Fedovapagon

    CAS:
    <p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>
    Fórmula:C27H34N4O3
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:462.58
  • Spiroxatrine

    CAS:
    <p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>
    Fórmula:C22H25N3O3
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:379.45
  • SANT 2

    CAS:
    <p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>
    Fórmula:C26H26ClN3O4
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:479.96
  • Calcitonin (salmon)

    CAS:
    <p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>
    Fórmula:C145H240N44O48S2
    Pureza:99.41% - 99.80%
    Cor e Forma:Powder
    Peso molecular:3431.85
  • Bromperidol hydrochloride

    CAS:
    <p>Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.</p>
    Fórmula:C21H24BrClFNO2
    Cor e Forma:Solid
    Peso molecular:456.78
  • Granisetron

    CAS:
    <p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>
    Fórmula:C18H24N4O
    Cor e Forma:Solid
    Peso molecular:312.41
  • Tiotidine

    CAS:
    Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).
    Fórmula:C10H16N8S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:312.42
  • Levomepromazine

    CAS:
    Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.
    Fórmula:C19H24N2OS
    Pureza:99.15%
    Cor e Forma:Solid
    Peso molecular:328.47
  • BMS-986224

    CAS:
    <p>BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.</p>
    Fórmula:C24H23ClN4O6
    Pureza:98.61% - 99.67%
    Cor e Forma:Solid
    Peso molecular:498.92
  • (+)-Penbutolol

    CAS:
    (+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.
    Fórmula:C18H29NO2
    Cor e Forma:Solid
    Peso molecular:291.43
  • Taranabant racemate

    CAS:
    <p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>
    Fórmula:C27H25ClF3N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:515.95
  • 1-Phenylbiguanide HCl

    CAS:
    <p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>
    Fórmula:C8H12ClN5
    Pureza:99.31%
    Cor e Forma:Solid
    Peso molecular:213.67