GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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SUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Fórmula:C14H15N3O3Pureza:99.38% - 99.38%Cor e Forma:SolidPeso molecular:273.29Ivabradine-d6 hydrochloride
CAS:<p>Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.</p>Fórmula:C27H37ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:511.08Taranabant racemate
CAS:<p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>Fórmula:C27H25ClF3N3O2Pureza:98%Cor e Forma:SolidPeso molecular:515.95BMS-986020 sodium
CAS:<p>BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.</p>Fórmula:C29H25N2NaO5Cor e Forma:SolidPeso molecular:504.51Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Fórmula:C26H27N5O2Pureza:98%Cor e Forma:SolidPeso molecular:449.57Gizzerosine
CAS:<p>Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.</p>Fórmula:C11H20N4O2Cor e Forma:SolidPeso molecular:240.3(+)-Penbutolol
CAS:(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Fórmula:C18H29NO2Cor e Forma:SolidPeso molecular:291.43Apraclonidine hydrochloride
CAS:<p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>Fórmula:C9H11Cl3N4Pureza:99.74%Cor e Forma:SolidPeso molecular:281.57Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H18ClN3SPureza:98%Cor e Forma:White Crystalline PowderPeso molecular:247.79Fluvoxamine
CAS:<p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>Fórmula:C15H21F3N2O2Cor e Forma:SolidPeso molecular:318.33SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Fórmula:C15H15ClN4OPureza:98%Cor e Forma:SolidPeso molecular:302.76GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Fórmula:C15H21N5O5Cor e Forma:SolidPeso molecular:351.36Antazoline phosphate
CAS:<p>Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.</p>Fórmula:C17H22N3O4PPureza:98%Cor e Forma:CoaPeso molecular:363.35Neurotensin(8-13)
CAS:<p>Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>Fórmula:C38H64N12O8Pureza:99.95%Cor e Forma:SolidPeso molecular:816.99Thioridazine
CAS:<p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>Fórmula:C21H26N2S2Cor e Forma:SolidPeso molecular:370.57Bombesin
CAS:<p>Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.</p>Fórmula:C71H110N24O18SCor e Forma:While Lyophilized PowderPeso molecular:1619.85Revdofilimab
CAS:<p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>Pureza:98.80% - 98.80%Cor e Forma:LiquidUCSF924
CAS:<p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>Fórmula:C20H22N2O2Pureza:98%Cor e Forma:SolidPeso molecular:322.4TP-16
CAS:<p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>Fórmula:C24H22FNO4SPureza:98.53% - 99.15%Cor e Forma:SolidPeso molecular:439.5Furprofen
CAS:Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Fórmula:C14H12O4Pureza:98.62% - 99.25%Cor e Forma:SolidPeso molecular:244.24Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Fórmula:C54H69N11O10S2Cor e Forma:SolidPeso molecular:1096.32V-0219
CAS:<p>V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.</p>Fórmula:C20H25F3N4O2Pureza:99.91%Cor e Forma:SoildPeso molecular:410.43Setiptiline maleate
CAS:Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Fórmula:C23H23NO4Pureza:99.94%Cor e Forma:SolidPeso molecular:377.43Timapiprant sodium
CAS:<p>Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.</p>Fórmula:C21H17FN2NaO2Pureza:98%Cor e Forma:SolidPeso molecular:371.367NBI-27914
CAS:<p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>Fórmula:C18H20Cl4N4Pureza:99.47% - 99.64%Cor e Forma:SolidPeso molecular:434.19cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Fórmula:C23H27Cl2F3N2OSPureza:98.07%Cor e Forma:SolidPeso molecular:507.44Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Fórmula:C27H34N4O3Pureza:99.33%Cor e Forma:SolidPeso molecular:462.58Acrivastine D7
CAS:<p>Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.</p>Fórmula:C22H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:355.48YNT-185 dihydrochloride
CAS:<p>Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.</p>Fórmula:C33H39Cl2N5O5SCor e Forma:SolidPeso molecular:688.67SKF-82958 hydrobromide
CAS:<p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>Fórmula:C19H21BrClNO2Pureza:98%Cor e Forma:SolidPeso molecular:410.73WAY-100635
CAS:<p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>Fórmula:C25H34N4O2Pureza:98.972%Cor e Forma:SolidPeso molecular:422.56Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Fórmula:C23H24N2O2Cor e Forma:SolidPeso molecular:360.45SB-408124 Hydrochloride
CAS:SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).Fórmula:C19H19ClF2N4OPureza:98%Cor e Forma:SolidPeso molecular:392.83Clencyclohexerol-d10
CAS:<p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:329.29SB-277011 hydrochloride
CAS:<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Fórmula:C28H31ClN4OPureza:98.54%Cor e Forma:SolidPeso molecular:475.03Emedastine Difumarate
CAS:<p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>Fórmula:C25H34N4O9Cor e Forma:SolidPeso molecular:534.56Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Fórmula:C15H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:249.34Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Fórmula:C59H84N16O12Cor e Forma:SolidPeso molecular:1209.4Zaloglanstat
CAS:<p>Zaloglanstat (ISC-27864) is a selective, orally active mPGES-1 inhibitor with an IC50 of 5 nM, analgesic in osteoarthritis and inflammatory arthritis.</p>Fórmula:C21H20ClF3N4O2Pureza:99.97%Cor e Forma:SolidPeso molecular:452.86Virodhamine
CAS:<p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>Fórmula:C22H37NO2Pureza:98%Cor e Forma:SoildPeso molecular:347.53GSK682753A
CAS:GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).Fórmula:C23H21Cl3N2O3Cor e Forma:SolidPeso molecular:479.78Trimethobenzamide
CAS:<p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>Fórmula:C21H28N2O5Cor e Forma:SolidPeso molecular:388.46Paliperidone Palmitate
CAS:<p>Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>Fórmula:C39H57FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:664.89PSB-0739
CAS:<p>PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.</p>Fórmula:C26H17N3Na2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:609.54Nefazodone
CAS:<p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>Fórmula:C25H32ClN5O2Pureza:99.85%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:470.01Endothelin-3 (Rat,Human) (TFA)
<p>Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).</p>Fórmula:C123H169F3N26O35S4·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:2757.07 (free base)Aripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Fórmula:C23H27Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:456.44Cimbuterol-d9
CAS:<p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>Fórmula:C13H10D9N3OPureza:99.22%Cor e Forma:SolidPeso molecular:242.37Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Fórmula:C18H18ClN3SPureza:99.93%Cor e Forma:SolidPeso molecular:343.87Glucagon (1-29), bovine, human, porcine
CAS:Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.Fórmula:C153H225N43O49SPureza:99.56% - 99.56%Cor e Forma:SolidPeso molecular:3482.75ML 00253764
CAS:melanocortin MC4 receptor antagonistFórmula:C18H18BrFN2OCor e Forma:SolidPeso molecular:377.25Pimozide-d4
CAS:<p>Pimozide D4 is a deuterium labeled Pimozide.</p>Fórmula:C28H29F2N3OPureza:98%Cor e Forma:SolidPeso molecular:465.57Docosahexaenoic acid ethyl ester
CAS:<p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>Fórmula:C24H36O2Cor e Forma:SolidPeso molecular:356.54BMS-986224
CAS:<p>BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.</p>Fórmula:C24H23ClN4O6Pureza:98.61% - 99.67%Cor e Forma:SolidPeso molecular:498.92Olanzapine D3
CAS:<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Fórmula:C17H20N4SPureza:98%Cor e Forma:SolidPeso molecular:315.45Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Fórmula:C21H26D6Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:433.45Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Fórmula:C26H27F5N6O3Pureza:98.98% - 98.98%Cor e Forma:SolidPeso molecular:566.52Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Fórmula:C20H21F3N4OPureza:98%Cor e Forma:SolidPeso molecular:394.43(S)-ZINC-3573
CAS:<p>(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.</p>Fórmula:C18H21N5Cor e Forma:SolidPeso molecular:307.401PD176252
CAS:<p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>Fórmula:C32H36N6O5Pureza:99.18%Cor e Forma:SolidPeso molecular:584.67Ziprasidone D8
CAS:<p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>Fórmula:C21H21ClN4OSPureza:98%Cor e Forma:SolidPeso molecular:420.99SB-269970 hydrochloride
CAS:<p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity</p>Fórmula:C18H28N2O3S·HClPureza:98.45%Cor e Forma:SolidPeso molecular:388.95Eticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Cor e Forma:SolidPeso molecular:377.31Dexloxiglumide
CAS:Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.Fórmula:C21H30Cl2N2O5Cor e Forma:SolidPeso molecular:461.38(R)-Praziquantel-d11
CAS:<p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:323.47Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Fórmula:C21H23ClFNO2Pureza:98%Cor e Forma:SolidPeso molecular:379.89MK-761 TFA
<p>MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.</p>Fórmula:C15H20F3N3O4Cor e Forma:SolidPeso molecular:363.332Terlipressin
CAS:<p>Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.</p>Fórmula:C52H74N16O15S2Pureza:98%Cor e Forma:SolidPeso molecular:1227.37R121919
CAS:<p>R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.</p>Fórmula:C22H32N6Pureza:99.75%Cor e Forma:SolidPeso molecular:380.53Clomipramine D3 hydrochloride
CAS:<p>Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).</p>Fórmula:C19H24Cl2N2Cor e Forma:SolidPeso molecular:354.33LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:335.34Sumanirole maleate
CAS:<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Fórmula:C15H17N3O5Pureza:98%Cor e Forma:SolidPeso molecular:319.31Omidenepag
CAS:Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Fórmula:C23H22N6O4SPureza:99.67% - 99.77%Cor e Forma:SolidPeso molecular:478.52Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Fórmula:C10H16N8S2Pureza:98%Cor e Forma:SolidPeso molecular:312.42rac-Propranolol-d7
CAS:Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Fórmula:C16H14D7NO2Cor e Forma:SolidPeso molecular:266.39Clorprenaline
CAS:<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Fórmula:C11H16ClNOPureza:98.9%Cor e Forma:SolidPeso molecular:213.7Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Fórmula:C27H40N8O6Cor e Forma:SolidPeso molecular:572.66β2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Fórmula:C36H49ClN4O7SCor e Forma:SolidPeso molecular:717.31SAR247799
CAS:<p>SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.</p>Fórmula:C21H16ClN3O5Cor e Forma:SolidPeso molecular:425.82GB-88
CAS:GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Fórmula:C32H42N4O4Cor e Forma:SolidPeso molecular:546.7GLP-1 receptor agonist 7
CAS:<p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>Fórmula:C31H30ClFN4O5Cor e Forma:SolidPeso molecular:593.05Diacetolol D7
CAS:<p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>Fórmula:C16H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:315.42Levosalbutamol Hydrochloride
CAS:<p>Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.</p>Fórmula:C13H22ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:275.774-Hydroxyatomoxetine D3
CAS:<p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>Fórmula:C17H21NO2Pureza:98%Cor e Forma:SolidPeso molecular:274.37Ceralifimod
CAS:Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Fórmula:C27H33NO4Cor e Forma:SolidPeso molecular:435.56Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Fórmula:C25H29N3O6SPureza:98%Cor e Forma:White SolidPeso molecular:503.61Doxazosin D8
CAS:Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Fórmula:C23H25N5O5Pureza:98%Cor e Forma:SolidPeso molecular:459.52Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOCor e Forma:SolidPeso molecular:281.39Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Fórmula:C16H18N4O2Pureza:98%Cor e Forma:SolidPeso molecular:306.39Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Fórmula:C20H22Cl2N2O4Cor e Forma:SolidPeso molecular:425.31Nadolol-d9
CAS:<p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>Fórmula:C17H27NO4Pureza:98%Cor e Forma:SolidPeso molecular:318.46Brombuterol hydrochloride
CAS:<p>Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.</p>Fórmula:C12H19Br2ClN2OCor e Forma:SolidPeso molecular:402.56Methyldopate
CAS:<p>Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.</p>Fórmula:C12H17NO4Cor e Forma:SolidPeso molecular:239.27ML224
CAS:<p>ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.</p>Fórmula:C31H31N3O5Pureza:99.14%Cor e Forma:SolidPeso molecular:525.59Zilpaterol-d7
CAS:<p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>Fórmula:C14H12D7N3O2Cor e Forma:SolidPeso molecular:268.36Scopine hydrochloride
CAS:<p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>Fórmula:C8H13NO2·HClPureza:98%Cor e Forma:White PowderPeso molecular:191.66Mozavaptan hydrochloride
CAS:<p>Mozavaptan is a vasopressin receptor antagonist.</p>Fórmula:C27H30ClN3O2Cor e Forma:SolidPeso molecular:464Granisetron
CAS:<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41Ipragliflozin (L-Proline)
CAS:Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.Fórmula:C26H30FNO7SCor e Forma:SolidPeso molecular:519.58TFLLR-NH2(TFA)
CAS:TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Fórmula:C33H54F3N9O8Pureza:98%Cor e Forma:SolidPeso molecular:761.83
