GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.946 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5360 produtos de "GPCR/Proteína-G"
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Zagociguat
CAS:<p>Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.</p>Fórmula:C16H10F4N6Pureza:99.37%Cor e Forma:SolidPeso molecular:362.28GB-88
CAS:<p>GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.</p>Fórmula:C32H42N4O4Cor e Forma:SolidPeso molecular:546.7SANT 2
CAS:<p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>Fórmula:C26H26ClN3O4Pureza:99.23%Cor e Forma:SolidPeso molecular:479.96YNT-185 dihydrochloride
CAS:<p>Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.</p>Fórmula:C33H39Cl2N5O5SCor e Forma:SolidPeso molecular:688.67Levosalbutamol Hydrochloride
CAS:<p>Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.</p>Fórmula:C13H22ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:275.774,4-Diphenylbutylamine hydrochloride
CAS:<p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>Fórmula:C16H20ClNCor e Forma:SolidPeso molecular:261.79Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Fórmula:C14H22ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:299.80TGR5 Receptor Agonist
CAS:TGR5 is a potent TGR5(GPCR19) agonist.Fórmula:C18H14Cl2N2O2Pureza:99.77% - ≥95%Cor e Forma:SolidPeso molecular:361.22SHU 9119 acetate
<p>SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.</p>Fórmula:C56H75N15O11Pureza:99.8%Cor e Forma:SolidPeso molecular:1134.29Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Fórmula:C29H34O6Pureza:≥98%Cor e Forma:LiquidPeso molecular:478.58TCS 1102
CAS:<p>TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).</p>Fórmula:C27H26N4O2SPureza:99.35% - 99.52%Cor e Forma:SolidPeso molecular:470.59Fluoroclebopride
CAS:<p>Fluoroclebopride is a dopamine (DA) D2 receptor ligand.</p>Fórmula:C20H23ClFN3O2Pureza:99.68% - 99.91%Cor e Forma:SolidPeso molecular:391.872-ATHBI
CAS:<p>2-ATHBI is a S1P lyase inhibitor.</p>Fórmula:C9H14N2O5Pureza:95.00%Cor e Forma:SolidPeso molecular:230.22PD-168077 maleate
CAS:<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Fórmula:C24H26N4O5Pureza:99.13%Cor e Forma:SolidPeso molecular:450.49A-582941 dihydrochloride
CAS:<p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>Fórmula:C17H22Cl2N4Pureza:99.55%Cor e Forma:SolidPeso molecular:353.29Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Cor e Forma:Appearance White Crystalline PowderPeso molecular:264.19Acrivastine
CAS:<p>Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.</p>Fórmula:C22H24N2O2Pureza:99.73% - >99.99%Cor e Forma:SolidPeso molecular:348.449-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Fórmula:C7H9N5Pureza:99.35% - 99.41%Cor e Forma:SolidPeso molecular:163.18Temanogrel
CAS:<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Fórmula:C24H28N4O4Pureza:99.24%Cor e Forma:SolidPeso molecular:436.5LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Cor e Forma:SolidPeso molecular:226.53Protease-Activated Receptor-4 diTFA
<p>Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist</p>Fórmula:C37H48F6N8O11Pureza:98.54%Cor e Forma:SolidPeso molecular:894.812'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Gastrin I (1-14), human
CAS:Gastrin I (1-14), human: a short peptide from the hormone gastrin, which regulates gastric acid secretion.Fórmula:C79H100N16O27Pureza:98.19%Cor e Forma:SolidPeso molecular:1705.738-Cyclopentyl-1,3-dimethylxanthine
CAS:<p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>Fórmula:C12H16N4O2Pureza:98.58% - >99.99%Cor e Forma:SolidPeso molecular:248.28BML-190
CAS:<p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。</p>Fórmula:C23H23ClN2O4Pureza:97.70%Cor e Forma:SolidPeso molecular:426.89Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:236.74Romifidine hydrochloride
CAS:<p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>Fórmula:C9H10BrClFN3Cor e Forma:SolidPeso molecular:294.55Domperidone monomaleate
CAS:<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Fórmula:C26H28ClN5O6Cor e Forma:SolidPeso molecular:541.98Mesdopetam
CAS:Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Fórmula:C12H18FNO3SCor e Forma:SolidPeso molecular:275.34Neuropeptide W-23(human)
CAS:<p>Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2.</p>Fórmula:C119H183N35O28SPureza:98.5%Cor e Forma:SolidPeso molecular:2584.01Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Fórmula:C22H25ClN4O4S2Cor e Forma:SolidPeso molecular:509.04AdipoRon hydrochloride
CAS:<p>AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).</p>Fórmula:C27H29ClN2O3Cor e Forma:SolidPeso molecular:464.99Selexipag
CAS:<p>Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.</p>Fórmula:C26H32N4O4SPureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:496.62Sultopride hydrochloride
CAS:<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Fórmula:C17H27ClN2O4SPureza:≥95%Cor e Forma:White Or Yellowish PowderPeso molecular:390.93Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Fórmula:C10H17N3S·2HCl·H2OPureza:99.68%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:302.26Pancreatic Polypeptide, rat acetate
<p>Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.</p>Pureza:97.53%Cor e Forma:SolidPeso molecular:N/AVanoxerine dihydrochloride
CAS:<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Fórmula:C28H34Cl2F2N2OPureza:98.16% - 98.35%Cor e Forma:White SolidPeso molecular:523.49ENMD-1068 HBr
CAS:<p>ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.</p>Fórmula:C15H30BrN3O2Cor e Forma:SolidPeso molecular:364.32PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Fórmula:C26H32O4Pureza:98.53%Cor e Forma:SolidPeso molecular:408.53Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Fórmula:C23H29Cl2N3O3Cor e Forma:SolidPeso molecular:466.4Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Cor e Forma:SolidPeso molecular:224.26LY255283
CAS:<p>LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.</p>Fórmula:C19H28N4O3Pureza:99.18%Cor e Forma:SolidPeso molecular:360.45Fipamezole HCl
CAS:<p>Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.</p>Fórmula:C14H16ClFN2Cor e Forma:SolidPeso molecular:266.74Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Fórmula:C32H41N5O10Pureza:97.69%Cor e Forma:SolidPeso molecular:655.7Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Fórmula:C32H29F5N3NaO5Pureza:99.71%Cor e Forma:SolidPeso molecular:653.57(R)-Propranolol hydrochloride
CAS:<p>(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.</p>Fórmula:C16H22ClNO2Pureza:98.63% - 99.01%Cor e Forma:SolidPeso molecular:295.8Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Fórmula:C14H21Cl2F3N6O3Cor e Forma:SolidPeso molecular:449.26Harmine
CAS:<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Fórmula:C13H12N2OPureza:98.29% - 99.92%Cor e Forma:Off-White SolidPeso molecular:212.25Detomidine hydrochloride
CAS:<p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71Cinaciguat hydrochloride
CAS:<p>Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.</p>Fórmula:C36H40ClNO5Cor e Forma:SolidPeso molecular:602.17Amylin, amide, rat acetate(124447-81-0,free base)
<p>Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.</p>Fórmula:C169H276N52O55S2Pureza:98.93%Cor e Forma:SolidPeso molecular:3980.45CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Fórmula:C16H11N3OPureza:99.81%Cor e Forma:SolidPeso molecular:261.28Bucindolol hydrochloride
CAS:<p>Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.</p>Fórmula:C22H26ClN3O2Cor e Forma:SolidPeso molecular:399.91GR 125743
CAS:<p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Fórmula:C17H18ClN3OPureza:99.95%Cor e Forma:SolidPeso molecular:315.8Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Fórmula:C21H21FO5SPureza:99.38% - 99.70%Cor e Forma:SolidPeso molecular:404.45Donitriptan Mesylate
CAS:<p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>Fórmula:C24H29N5O5SCor e Forma:SolidPeso molecular:499.58Montelukast
CAS:<p>Montelukast (Singular), oral asthma med, linked to rare liver injury.</p>Fórmula:C35H36ClNO3SPureza:98.56% - >99.99%Cor e Forma:SolidPeso molecular:586.18LP-211
CAS:<p>LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.</p>Fórmula:C30H34N4OPureza:98.65%Cor e Forma:SolidPeso molecular:466.623-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Fórmula:C21H25Cl2NOPureza:99.03%Cor e Forma:SolidPeso molecular:378.33Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Fórmula:C37H56F7N6O16PPureza:98% - 99.03%Cor e Forma:SolidPeso molecular:1004.83Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Fórmula:C24H27ClO6Pureza:97.37%Cor e Forma:SolidPeso molecular:446.92Substance P (7-11)
CAS:<p>Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .</p>Fórmula:C31H44N6O5SPureza:98.39%Cor e Forma:SolidPeso molecular:612.78LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Fórmula:C21H22FN3OPureza:99.32%Cor e Forma:SolidPeso molecular:351.42Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44Trazodone
CAS:<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Fórmula:C19H22ClN5OPureza:99.79% - 99.92%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:371.86Midaglizole
CAS:<p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>Fórmula:C16H17N3Cor e Forma:SolidPeso molecular:251.33Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Cor e Forma:White SolidPeso molecular:238.24BAR 501 impurity
CAS:<p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>Fórmula:C26H46O3Pureza:98.78%Cor e Forma:SolidPeso molecular:406.64Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Fórmula:C25H37NO4Pureza:98% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:415.57Pranlukast hemihydrate
CAS:<p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>Fórmula:C27H23N5O40·5H2OPureza:99.28%Cor e Forma:SolidPeso molecular:490.52Zatebradine
CAS:<p>Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).</p>Fórmula:C26H36N2O5Pureza:98%Cor e Forma:SolidPeso molecular:456.57BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Fórmula:C59H83N13O14S2Pureza:99.7%Cor e Forma:SolidPeso molecular:1262.5S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Cor e Forma:SolidPeso molecular:407.48(±)-Ibipinabant
CAS:<p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>Fórmula:C23H20Cl2N4O2SPureza:99.28% - 99.83%Cor e Forma:SolidPeso molecular:487.4OS-3-106
CAS:<p>OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.</p>Fórmula:C25H30N4O2SPureza:99.4% - 99.57%Cor e Forma:SolidPeso molecular:450.6Xamoterol
CAS:<p>Xamoterol is a cardiac stimulant.</p>Fórmula:C16H25N3O5Cor e Forma:SolidPeso molecular:339.39RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Fórmula:C67H109N19O19Pureza:99.87%Cor e Forma:SolidPeso molecular:1484.71Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Fórmula:C15H20N8O6Pureza:98%Cor e Forma:SolidPeso molecular:408.37Dasotraline
CAS:<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Fórmula:C16H15Cl2NCor e Forma:SolidPeso molecular:292.2[Pyr1]-Apelin-13
CAS:<p>[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.</p>Fórmula:C69H108N22O16SPureza:99.71%Cor e Forma:SolidPeso molecular:1533.8Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Fórmula:C21H27ClN2O5Pureza:99.11%Cor e Forma:SolidPeso molecular:422.9AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Fórmula:C15H11ClFN5Pureza:99.15% - 99.90%Cor e Forma:SolidPeso molecular:315.73Epinastine
CAS:<p>Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.</p>Fórmula:C16H15N3Pureza:99.94%Cor e Forma:SolidPeso molecular:249.31Blarcamesine hydrochloride
CAS:Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).Fórmula:C19H24ClNOPureza:99.57% - 99.9%Cor e Forma:SolidPeso molecular:317.85CCG215022
CAS:<p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>Fórmula:C26H22FN7O3Pureza:97.63% - 99.69%Cor e Forma:SolidPeso molecular:499.5A-836339
CAS:<p>A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.</p>Fórmula:C16H26N2O2SPureza:99.94%Cor e Forma:SolidPeso molecular:310.45BQ-123
CAS:<p>BQ-123 is a selective endothelin A receptor (ETA) antagonist with IC50 of 7.3 nM. Phase 2.</p>Fórmula:C31H42N6O7Pureza:99.22% - ≥95%Cor e Forma:SolidPeso molecular:610.7R 396 acetate
<p>R 396 acetate is an NK-2 Tachykinin Receptor <br>Antagonist.</p>Fórmula:C41H55N9O12Pureza:99.52%Cor e Forma:SolidPeso molecular:865.93Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Fórmula:C20H22N2O4Pureza:98.46%Cor e Forma:SolidPeso molecular:354.4Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Fórmula:C20H20FNO3S·HClPureza:99.39% - 99.79%Cor e Forma:SolidPeso molecular:409.9Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Fórmula:C19H21Cl2N3Pureza:>99.99%Cor e Forma:SolidPeso molecular:362.31-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Fórmula:C13H13NO5Pureza:99.55%Cor e Forma:SolidPeso molecular:263.25DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Fórmula:C16H24N4O2Pureza:99.23% - 99.93%Cor e Forma:White SolidPeso molecular:304.39Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Fórmula:C25H29ClF6N2O3Cor e Forma:SolidPeso molecular:554.95Decynium 22
CAS:<p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>Fórmula:C23H23IN2Pureza:99.92%Cor e Forma:Dark Red CrystalsPeso molecular:454.35Glucagon-like peptide 1 (1-37), human acetate
<p>Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.</p>Pureza:98%Cor e Forma:LiquidPeso molecular:N/APoloxamer 407
CAS:<p>Poloxamer 407 is a nonionic surfactant.</p>Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:7700(Average)Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Fórmula:C40H67N7O10Pureza:99.95%Cor e Forma:SolidPeso molecular:805.9Oxyntomodulin acetate
<p>Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].</p>Pureza:99.24%Cor e Forma:LiquidPeso molecular:N/A
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