GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.946 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5360 produtos de "GPCR/Proteína-G"
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Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:White SolidPeso molecular:506.47RO 46-8443
CAS:<p>RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.</p>Fórmula:C31H35N3O8SPureza:98.77% - 99.77%Cor e Forma:SolidPeso molecular:609.69Mizagliflozin
CAS:<p>Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.</p>Fórmula:C28H44N4O8Pureza:98.66% - 99.67%Cor e Forma:SolidPeso molecular:564.67Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Fórmula:C28H33ClN2·2HClPureza:98.05%Cor e Forma:Off-White PowderPeso molecular:505.95Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Fórmula:C17H25N3O2S·HClPureza:99.17% - 99.93%Cor e Forma:Beige SolidPeso molecular:371.93Lofexidine
CAS:<p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>Fórmula:C11H12Cl2N2OPureza:98.78%Cor e Forma:SolidPeso molecular:259.13S 38093
CAS:<p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>Fórmula:C17H24N2O2Pureza:99.95%Cor e Forma:SolidPeso molecular:288.38Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Fórmula:C21H25ClN2O3·C6H6O3SPureza:99.83% - 99.9%Cor e Forma:Brown Viscous LiquidPeso molecular:547.06CYM5442
CAS:<p>CYM5442 is an S1P agonist, targeting to Sphingosine.</p>Fórmula:C23H27N3O4Pureza:98.02% - 99.48%Cor e Forma:SolidPeso molecular:409.48SBI-553
CAS:<p>SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).</p>Fórmula:C26H31FN4O2Pureza:99.33%Cor e Forma:SolidPeso molecular:450.55Bremelanotide Acetate
CAS:<p>Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .</p>Fórmula:C52H72N14O12Pureza:96.72% - >99.99%Cor e Forma:SolidPeso molecular:1085.22α-MSH, amide Acetate
<p>a-MSH, amide Acetate as an endogenous neuropeptide.</p>Fórmula:C79H113N21O21SPureza:98.67%Cor e Forma:SolidPeso molecular:1724.94Chemerin-9 (149-157) acetate
<p>Chemerin-9 (149-157) acetate, a nonapeptide C-terminal fragment of chemerin, retains full protein's activity as chemerinR agonist.</p>Fórmula:C56H70N10O15Pureza:99.93%Cor e Forma:SolidPeso molecular:1123.23RFRP-1 (human) acetate(311309-25-8 free base)
<p>RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.</p>Fórmula:C69H105N19O16SPureza:96.84%Cor e Forma:SolidPeso molecular:1488.77Norfluoxetine Hydrochloride
CAS:<p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>Fórmula:C16H17ClF3NOPureza:99.71%Cor e Forma:SolidPeso molecular:331.76BMS-986020
CAS:<p>BMS-986020 (AM152) is a selective antagonist of LPA1.</p>Fórmula:C29H26N2O5Pureza:98.82% - >99.99%Cor e Forma:SolidPeso molecular:482.53Tandospirone citrate
CAS:<p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Cor e Forma:SolidPeso molecular:575.61HJC0350
CAS:<p>HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.</p>Fórmula:C15H19NO2SPureza:99.27% - 99.65%Cor e Forma:SolidPeso molecular:277.38RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29Neuropeptide FF acetate(99566-27-5 free base)
<p>Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family.</p>Fórmula:C56H80N14O12Pureza:98.03%Cor e Forma:SolidPeso molecular:1141.32Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Fórmula:C32H26N4O2·HClPureza:98.33% - 99.86%Cor e Forma:SolidPeso molecular:535.04Ro 46-2005
CAS:<p>Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).</p>Fórmula:C23H27N3O6SPureza:98.02% - 98.8%Cor e Forma:SolidPeso molecular:473.54SORT-PGRN interaction inhibitor 1
CAS:<p>SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).</p>Fórmula:C15H18N2O2Pureza:98.72%Cor e Forma:SolidPeso molecular:258.32MDL 100009
CAS:<p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>Fórmula:C22H28FNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:373.46Cotadutide acetate
<p>Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.</p>Fórmula:C169H256N42O57Pureza:98.28%Cor e Forma:SolidPeso molecular:3788.14Bosentan
CAS:<p>Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.</p>Fórmula:C27H29N5O6SPureza:99.74% - 99.84%Cor e Forma:Pale Yellow To Off-White SolidPeso molecular:551.614Neuropeptide SF(mouse,rat) acetate
<p>Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.</p>Fórmula:C42H69N13O12Pureza:98.37%Cor e Forma:SolidPeso molecular:948.08CJC-1295 acetate(863288-34-0 free base)
<p>CJC-1295 acetate is a synthetic GHRH analogue and GHS.</p>Fórmula:C154H256N44O44Pureza:97.29%Cor e Forma:SolidPeso molecular:3428.01CP 376395
CAS:<p>CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.</p>Fórmula:C21H30N2OPureza:99.86% - 99.94%Cor e Forma:SolidPeso molecular:326.48Substance P 1-9 aceate
<p>Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.</p>Fórmula:C54H81N15O14Pureza:99.01%Cor e Forma:SolidPeso molecular:1164.31Protease-Activated Receptor-1, PAR-1 Agonist acetate
<p>PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.</p>Fórmula:C37H62N10O11Pureza:98.1800%Cor e Forma:SolidPeso molecular:822.95Etilevodopa hydrochloride
CAS:<p>Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.</p>Fórmula:C11H16ClNO4Pureza:95.00%Cor e Forma:SolidPeso molecular:261.7Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Fórmula:C184H282N50O60SPureza:97.71% - 99.78%Cor e Forma:SolidPeso molecular:4186.57Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Fórmula:C18H13F6NO4SPureza:97.68% - 99.69%Cor e Forma:SolidPeso molecular:453.36Galanin (1-16), mouse, porcine, rat
CAS:<p>Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.</p>Fórmula:C78H116N20O21Pureza:98.65%Cor e Forma:White PowderPeso molecular:1669.88(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Fórmula:C14H20ClNO3Pureza:97.76%Cor e Forma:SolidPeso molecular:285.77Montelukast sodium
CAS:<p>Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.</p>Fórmula:C35H35ClNNaO3SPureza:99.14% - 99.89%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:608.17RFRP3(human) acetate(311309-27-0 free base)
<p>RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.</p>Fórmula:C47H76N14O12Pureza:97.09%Cor e Forma:SolidPeso molecular:1029.19Dexmedetomidine
CAS:<p>Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.</p>Fórmula:C13H16N2Pureza:99% - >99.99%Cor e Forma:SolidPeso molecular:200.28Prucalopride Succinate
CAS:<p>Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).</p>Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Cor e Forma:SolidPeso molecular:485.96AM211
CAS:<p>AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)</p>Fórmula:C27H27F3N2O4Pureza:≥95%Cor e Forma:SolidPeso molecular:500.51nifenalol.HCl
CAS:<p>Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.</p>Fórmula:C11H17ClN2O3Pureza:99.96%Cor e Forma:SolidPeso molecular:260.72GW627368
CAS:<p>GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.</p>Fórmula:C30H28N2O6SPureza:99.75% - 99.92%Cor e Forma:SolidPeso molecular:544.62Flibanserin
CAS:<p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Cor e Forma:White PowderPeso molecular:390.41-Oleoyl lysophosphatidic acid sodium
CAS:<p>1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2</p>Fórmula:C21H40O7P·NaPureza:98.75% - 99.24%Cor e Forma:SolidPeso molecular:458.51BAY 41-2272
CAS:<p>BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.</p>Fórmula:C20H17FN6Pureza:99.54%Cor e Forma:SolidPeso molecular:360.39SB-200646
CAS:<p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>Fórmula:C15H14N4OPureza:99.61%Cor e Forma:SolidPeso molecular:266.3Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Fórmula:C21H28N2O2·2ClHPureza:99.73%Cor e Forma:SolidPeso molecular:413.39ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Fórmula:C17H11N3O6SPureza:97.74%Cor e Forma:SolidPeso molecular:385.35Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFórmula:C29H27F2N7O5SPureza:98.64% - 99.97%Cor e Forma:SolidPeso molecular:623.63Obestatin (rat) acetate
<p>Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).</p>Fórmula:C114H174N34O31Pureza:99.05%Cor e Forma:SolidPeso molecular:2516.81Spexin acetate(1370290-58-6 free base)
<p>Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.</p>Fórmula:C76H117N19O22SPureza:95.43%Cor e Forma:SolidPeso molecular:1680.94Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Fórmula:C21H35ClN2O5Pureza:99.33%Cor e Forma:SolidPeso molecular:430.97AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Fórmula:C23H31ClN2O2Pureza:99.71%Cor e Forma:SolidPeso molecular:402.96Melanotan (MT)-II
CAS:<p>Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).</p>Fórmula:C50H69N15O9Pureza:>99.99%Cor e Forma:SolidPeso molecular:1024.18FAUC-365
CAS:<p>FAUC-365 is a D3 dopamine receptor agonist.</p>Fórmula:C23H25Cl2N3OSPureza:99.62%Cor e Forma:SolidPeso molecular:462.44AVN-492
CAS:<p>AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).</p>Fórmula:C17H21N5O2SPureza:99.81%Cor e Forma:SolidPeso molecular:359.45Vorapaxar sulfate
CAS:<p>Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.</p>Fórmula:C29H35FN2O8SPureza:99.9% - >99.99%Cor e Forma:SolidPeso molecular:590.66Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Fórmula:C19H26N4O4SPureza:98%Cor e Forma:SolidPeso molecular:406.5Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Fórmula:C16H15N7OPureza:97.25% - 97.36%Cor e Forma:SolidPeso molecular:321.34γ-Mangostin
CAS:<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Fórmula:C23H24O6Pureza:98.55% - 99.08%Cor e Forma:SolidPeso molecular:396.43VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Fórmula:C13H15ClN4Pureza:99.66%Cor e Forma:SolidPeso molecular:262.74Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Fórmula:C28H33ClN2Cor e Forma:SolidPeso molecular:433.03Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Cor e Forma:SolidPeso molecular:492.68Ramosetron
CAS:<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Fórmula:C17H17N3OPureza:98.84%Cor e Forma:SolidPeso molecular:279.34Nonapeptide-1 acetate salt (158563-45-2 free base)
<p>Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)</p>Fórmula:C63H91N15O11SPureza:98.26%Cor e Forma:SolidPeso molecular:1266.58SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Fórmula:C10H14ClN3·HClPureza:99.89%Cor e Forma:SolidPeso molecular:248.15BP 897
CAS:<p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>Fórmula:C26H31N3O2Pureza:99.44%Cor e Forma:SolidPeso molecular:417.54Alloxazine
CAS:<p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>Fórmula:C10H6N4O2Pureza:99.75%Cor e Forma:SolidPeso molecular:214.18Hemopressin (rat) acetate(568588-77-2 free base)
<p>Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.</p>Fórmula:C5H81N13O14Pureza:99.37%Cor e Forma:SolidPeso molecular:1148.31Droxidopa
CAS:<p>Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.</p>Fórmula:C9H11NO5Pureza:97.27% - 99.88%Cor e Forma:SolidPeso molecular:213.19TC-G-1008
CAS:<p>TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).</p>Fórmula:C18H19ClN6O2SPureza:97.37% - 99%Cor e Forma:SolidPeso molecular:418.9NPS-2143 hydrochloride
CAS:<p>NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.</p>Fórmula:C24H25ClN2O2·HClPureza:99.38% - 99.67%Cor e Forma:SolidPeso molecular:445.38AF38469
CAS:AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Fórmula:C15H11F3N2O3Pureza:99.18%Cor e Forma:SolidPeso molecular:324.25Adenosine amine congener
CAS:<p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>Fórmula:C28H32N8O6Pureza:97.86%Cor e Forma:SolidPeso molecular:576.6Exenatide
CAS:<p>Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.</p>Fórmula:C186H286N50O62SPureza:99.42%Cor e Forma:SolidPeso molecular:4247Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Fórmula:C32H44F3N3O2SPureza:98.14%Cor e Forma:SolidPeso molecular:591.77Amezinium methylsulfate
CAS:<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Fórmula:C12H15N3O5SPureza:99.64%Cor e Forma:SolidPeso molecular:313.33Levobetaxolol hydrochloride
CAS:<p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>Fórmula:C18H29NO3·HClPureza:98.80% - 99.69%Cor e Forma:SolidPeso molecular:343.89FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Fórmula:C18H19ClN4Pureza:99.84%Cor e Forma:SolidPeso molecular:326.82Eptapirone
CAS:<p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>Fórmula:C16H23N7O2Pureza:99.39% - 99.65%Cor e Forma:SolidPeso molecular:345.4(E)-3,4,5-Trimethoxycinnamic acid
CAS:<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Fórmula:C12H14O5Pureza:99.83%Cor e Forma:SolidPeso molecular:238.24Loxiglumide
CAS:<p>Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.</p>Fórmula:C21H30Cl2N2O5Pureza:97.55% - 99.81%Cor e Forma:SolidPeso molecular:461.38Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Fórmula:C23H25ClN2OPureza:98.86% - 99.85%Cor e Forma:SolidPeso molecular:380.91BETP
CAS:<p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>Fórmula:C20H17F3N2O2SPureza:98.51%Cor e Forma:SolidPeso molecular:406.42Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
<p>Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to</p>Fórmula:C49H70N12O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1035.15Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Fórmula:C25H29N9O3Pureza:98.02% - 99.68%Cor e Forma:SolidPeso molecular:503.56AM1241
CAS:<p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>Fórmula:C22H22IN3O3Pureza:98.937% - 99.1%Cor e Forma:SolidPeso molecular:503.33[Sar9] Substance P acetate(77128-75-7 free base)
<p>[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.</p>Fórmula:C66H104N18O15SPureza:96.67%Cor e Forma:SolidPeso molecular:1421.71Ponesimod
CAS:<p>Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.</p>Fórmula:C23H25ClN2O4SPureza:99.42% - 99.96%Cor e Forma:SolidPeso molecular:460.97HCGRP-(8-37) acetate
<p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>Fórmula:C141H234N44O40Pureza:99.29%Cor e Forma:SolidPeso molecular:3185.64Ibrolipim
CAS:<p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>Fórmula:C19H20BrN2O4PPureza:98.04%Cor e Forma:SolidPeso molecular:451.25Amitriptyline
CAS:<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Fórmula:C20H23NPureza:98.24% - 99.64%Cor e Forma:Crystals SolidPeso molecular:277.4Siramesine
CAS:<p>Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent</p>Fórmula:C30H31FN2OPureza:98%Cor e Forma:SolidPeso molecular:454.58[Sar9,Met(O2)11]-Substance P acetate
<p>[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.</p>Fórmula:C66H106N18O18SPureza:>99.99%Cor e Forma:SolidPeso molecular:1471.75BD 1008 dihydrobromide
CAS:<p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>Fórmula:C15H24Br2Cl2N2Pureza:97.81%Cor e Forma:SolidPeso molecular:463.08Almotriptan
CAS:<p>Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.</p>Fórmula:C17H25N3O2SPureza:99.85%Cor e Forma:Light Yellow Or White PowerPeso molecular:335.46[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:<p>Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).</p>Fórmula:C39H65N9O9Pureza:>99.99%Cor e Forma:SolidPeso molecular:803.99FAUC 346
CAS:<p>FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.</p>Fórmula:C24H29N3O2SPureza:99.46%Cor e Forma:SolidPeso molecular:423.57
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