GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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RS-127445 hydrochloride
CAS:<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Fórmula:C17H17ClFN3Pureza:99.48%Cor e Forma:SolidPeso molecular:317.79BisfluoroModafinil
CAS:<p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>Fórmula:C15H13F2NO2SPureza:99.19%Cor e Forma:SolidPeso molecular:309.33BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Cor e Forma:SolidPeso molecular:479.87CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Fórmula:C58H69F3N12O16S2Pureza:99.7%Cor e Forma:SolidPeso molecular:1311.36Cinacalcet hydrochloride
CAS:<p>Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-</p>Fórmula:C22H23ClF3NPureza:99.96% - >99.99%Cor e Forma:Off-White To Tan SolidPeso molecular:393.87Neuropeptide S (Rat) acetate
<p>Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.</p>Fórmula:C97H164N34O29Pureza:95.36%Cor e Forma:SolidPeso molecular:2270.59JNJ-10229570
CAS:<p>JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland</p>Fórmula:C22H19N3O2SPureza:98.41%Cor e Forma:SolidPeso molecular:389.47ACTH 11-24 acetate(4237-93-8 free base)
CAS:<p>ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.</p>Fórmula:C79H138N24O18Pureza:>99.99%Cor e Forma:SolidPeso molecular:1712.12TG4-155
CAS:<p>TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.</p>Fórmula:C23H26N2O4Pureza:97.2%Cor e Forma:SolidPeso molecular:394.46NGB 2904
CAS:<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Fórmula:C28H29Cl2N3OPureza:98.79%Cor e Forma:SolidPeso molecular:494.46Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Fórmula:C129H207N45O41S3Pureza:98.24%Cor e Forma:SolidPeso molecular:3140.5Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Fórmula:C21H25ClN2O3Pureza:99.75%Cor e Forma:SolidPeso molecular:388.89Vilanterol trifenatate
CAS:<p>Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)</p>Fórmula:C44H49Cl2NO7Pureza:99.51% - >99.99%Cor e Forma:SolidPeso molecular:774.77BAR501
CAS:<p>BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。</p>Fórmula:C26H46O3Pureza:99.29% - 99.68%Cor e Forma:SolidPeso molecular:406.64Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Fórmula:C14H20F6N4O7Pureza:98.18%Cor e Forma:SolidPeso molecular:470.32Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Fórmula:C63H104N22O17SPureza:98.33%Cor e Forma:SolidPeso molecular:1473.72MHP
CAS:<p>MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.</p>Fórmula:C16H23NO4Pureza:98.58%Cor e Forma:SolidPeso molecular:293.36Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Fórmula:C18H25N·H3O4PPureza:99.65%Cor e Forma:SolidPeso molecular:353.4ML401
CAS:<p>ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .</p>Fórmula:C20H20BrClN2OPureza:99.13%Cor e Forma:SolidPeso molecular:419.74Fexofenadine
CAS:<p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>Fórmula:C32H39NO4Pureza:99.35%Cor e Forma:White To Off-White SolidPeso molecular:501.66Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Fórmula:C19H16F2N8O2Pureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:426.38ML-031
CAS:<p>ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.</p>Fórmula:C19H20N2O3Pureza:99.21%Cor e Forma:SolidPeso molecular:324.37Exo-1
CAS:<p>Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, as</p>Fórmula:C15H12FNO3Pureza:99.45%Cor e Forma:SolidPeso molecular:273.265-Iodotubercidin
CAS:<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Fórmula:C11H13IN4O4Pureza:99.98%Cor e Forma:Tan SolidPeso molecular:392.15Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Fórmula:C40H55N7O11SPureza:99.84% - >99.99%Cor e Forma:White PowderPeso molecular:841.97GR-73632
CAS:<p>Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).</p>Fórmula:C40H59N7O6SPureza:99.68%Cor e Forma:SolidPeso molecular:766Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Fórmula:C24H32ClNO6Pureza:99.73%Cor e Forma:Colorless LiquidPeso molecular:465.97Protease-Activated Receptor-4 diTFA
<p>Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist</p>Fórmula:C37H48F6N8O11Pureza:98.54%Cor e Forma:SolidPeso molecular:894.81Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Fórmula:C149H234N40O47SPureza:98% - 99.65%Cor e Forma:SolidPeso molecular:3369.76Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Fórmula:C14H22ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:299.80TGR5 Receptor Agonist
CAS:TGR5 is a potent TGR5(GPCR19) agonist.Fórmula:C18H14Cl2N2O2Pureza:99.77% - ≥95%Cor e Forma:SolidPeso molecular:361.22[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
<p>Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.</p>Fórmula:C81H113N19O14Pureza:97.68%Cor e Forma:SolidPeso molecular:1576.91Terutroban
CAS:<p>Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.</p>Fórmula:C20H22ClNO4SPureza:99.53%Cor e Forma:SolidPeso molecular:407.91Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Fórmula:C10H17N3S·2HCl·H2OPureza:99.68%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:302.26Vanoxerine dihydrochloride
CAS:<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Fórmula:C28H34Cl2F2N2OPureza:98.16% - 98.35%Cor e Forma:White SolidPeso molecular:523.49Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Fórmula:C25H26Cl3N7OPureza:99.79% - ≥95%Cor e Forma:SolidPeso molecular:546.88Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Fórmula:C21H30N4O4Pureza:99.52%Cor e Forma:SolidPeso molecular:402.49Bombesin acetate(31362-50-2 free base)
CAS:<p>Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).</p>Fórmula:C73H114N24O20SPureza:98.44%Cor e Forma:SolidPeso molecular:1679.92SB-649868
CAS:<p>SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).</p>Fórmula:C26H24FN3O3SPureza:99.53%Cor e Forma:SolidPeso molecular:477.55BCTC
CAS:<p>BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)</p>Fórmula:C20H25ClN4OPureza:99.21%Cor e Forma:SolidPeso molecular:372.89Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Fórmula:C32H41N5O10Pureza:97.69%Cor e Forma:SolidPeso molecular:655.7Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFórmula:C29H27F2N7O5SPureza:98.64% - 99.97%Cor e Forma:SolidPeso molecular:623.63Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Fórmula:C25H25Cl2N7OPureza:99.43%Cor e Forma:SolidPeso molecular:510.42Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Fórmula:C19H25NOSPureza:98.08% - 99.59%Cor e Forma:SolidPeso molecular:315.47(R)-Propranolol hydrochloride
CAS:<p>(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.</p>Fórmula:C16H22ClNO2Pureza:98.63% - 99.01%Cor e Forma:SolidPeso molecular:295.8Spexin acetate(1370290-58-6 free base)
<p>Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.</p>Fórmula:C76H117N19O22SPureza:95.43%Cor e Forma:SolidPeso molecular:1680.94Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Fórmula:C17H18ClN3OPureza:99.95%Cor e Forma:SolidPeso molecular:315.8Montelukast
CAS:<p>Montelukast (Singular), oral asthma med, linked to rare liver injury.</p>Fórmula:C35H36ClNO3SPureza:98.56% - >99.99%Cor e Forma:SolidPeso molecular:586.18Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Fórmula:C28H37N3O3Pureza:99.86% - >99.99%Cor e Forma:SolidPeso molecular:463.61Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Fórmula:C21H35ClN2O5Pureza:99.33%Cor e Forma:SolidPeso molecular:430.97ML 154
CAS:<p>ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.</p>Fórmula:C29H26BrN2PSPureza:99.53%Cor e Forma:SolidPeso molecular:545.47Atrasentan
CAS:<p>Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.</p>Fórmula:C29H38N2O6Pureza:97.65% - 99.08%Cor e Forma:SolidPeso molecular:510.62Metiamide
CAS:<p>Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .</p>Fórmula:C9H16N4S2Pureza:97.41%Cor e Forma:SolidPeso molecular:244.38BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Fórmula:C59H83N13O14S2Pureza:99.7%Cor e Forma:SolidPeso molecular:1262.5LY2828360
CAS:<p>LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.</p>Fórmula:C22H27ClN6OPureza:98.45% - 99.51%Cor e Forma:SolidPeso molecular:426.94RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Fórmula:C67H109N19O19Pureza:99.87%Cor e Forma:SolidPeso molecular:1484.71AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Fórmula:C15H11ClFN5Pureza:99.15% - 99.90%Cor e Forma:SolidPeso molecular:315.73carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Fórmula:C24H31N3O2SPureza:98.06%Cor e Forma:SolidPeso molecular:425.59FAUC-365
CAS:<p>FAUC-365 is a D3 dopamine receptor agonist.</p>Fórmula:C23H25Cl2N3OSPureza:99.62%Cor e Forma:SolidPeso molecular:462.44AVN-492
CAS:<p>AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).</p>Fórmula:C17H21N5O2SPureza:99.81%Cor e Forma:SolidPeso molecular:359.45EST64454 Maleic acid salt
CAS:<p>EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.</p>Fórmula:C22H26F2N4O6Pureza:97.54%Cor e Forma:SolidPeso molecular:480.46γ-L-Glutamyl-L-alanine
CAS:<p>γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).</p>Fórmula:C8H14N2O5Pureza:99.49%Cor e Forma:SolidPeso molecular:218.21ML 10302
CAS:<p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>Fórmula:C15H21ClN2O3Cor e Forma:SolidPeso molecular:312.79TRAP-6 amide acetate
<p>TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].</p>Fórmula:C36H61N11O10Pureza:98.55%Cor e Forma:SolidPeso molecular:807.94BML-190
CAS:<p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。</p>Fórmula:C23H23ClN2O4Pureza:97.70%Cor e Forma:SolidPeso molecular:426.891-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Fórmula:C13H13NO5Pureza:99.55%Cor e Forma:SolidPeso molecular:263.25Opromazine hydrochloride
CAS:<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Fórmula:C17H20Cl2N2OSPureza:98.03%Cor e Forma:SolidPeso molecular:371.32Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Fórmula:C32H29F5N3NaO5Pureza:99.71%Cor e Forma:SolidPeso molecular:653.57Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Fórmula:C19H26N4O4SPureza:98%Cor e Forma:SolidPeso molecular:406.5Melitracen
CAS:<p>Melitracen is a tricyclic antidepressant.</p>Fórmula:C21H25NCor e Forma:SolidPeso molecular:291.43Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Fórmula:C25H37NO4Pureza:98% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:415.57IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Fórmula:C23H27N5O2Pureza:97.05%Cor e Forma:SolidPeso molecular:405.49Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Fórmula:C40H67N7O10Pureza:99.95%Cor e Forma:SolidPeso molecular:805.9Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Fórmula:C16H15N7OPureza:97.25% - 97.36%Cor e Forma:SolidPeso molecular:321.34(±)-Ibipinabant
CAS:<p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>Fórmula:C23H20Cl2N4O2SPureza:99.28% - 99.83%Cor e Forma:SolidPeso molecular:487.4Lidamidine Hydrochloride
CAS:<p>Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.</p>Fórmula:C11H17ClN4OCor e Forma:SolidPeso molecular:256.73Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Fórmula:C18H22ClNOPureza:99.44% - 99.85%Cor e Forma:SolidPeso molecular:303.83Sarpogrelate
CAS:<p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>Fórmula:C24H31NO6Cor e Forma:SolidPeso molecular:429.51PD-168077 maleate
CAS:<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Fórmula:C24H26N4O5Pureza:99.13%Cor e Forma:SolidPeso molecular:450.49Butyrophenone
CAS:<p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>Fórmula:C10H12OPureza:99.84%Cor e Forma:Colourless To Yellow LiquidPeso molecular:148.2Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Fórmula:C24H27ClO6Pureza:97.37%Cor e Forma:SolidPeso molecular:446.92Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Fórmula:C28H33ClN2Cor e Forma:SolidPeso molecular:433.034-Methylhistamine hydrochloride
CAS:<p>Compound with imidazole ring & amine group; inhibits copper enzymes, affects gene expression.</p>Fórmula:C6H12ClN3Pureza:95%Cor e Forma:SolidPeso molecular:161.633Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Cor e Forma:SolidPeso molecular:492.68PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:301.21UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Fórmula:C52H68N10O14S2Pureza:99.78%Cor e Forma:SolidPeso molecular:1121.29Ramosetron
CAS:<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Fórmula:C17H17N3OPureza:98.84%Cor e Forma:SolidPeso molecular:279.34SSR240612
CAS:<p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>Fórmula:C42H53ClN4O7SPureza:98.59% - 99.16%Cor e Forma:SolidPeso molecular:793.41Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Cor e Forma:SolidPeso molecular:233.18Droxidopa hydrochloride
CAS:<p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>Fórmula:C9H12ClNO5Cor e Forma:SolidPeso molecular:249.65Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Fórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48Alloxazine
CAS:<p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>Fórmula:C10H6N4O2Pureza:99.75%Cor e Forma:SolidPeso molecular:214.18GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Fórmula:C21H25N3O2Pureza:98.71% - 99.858%Cor e Forma:SolidPeso molecular:351.44AP1189 acetate
CAS:<p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>Fórmula:C16H18N6O4Pureza:99.95%Cor e Forma:SolidPeso molecular:358.35Ornipressin Acetate(3397-23-7,free)
CAS:<p>Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent.</p>Fórmula:C47H67N13O124S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1102.25tcY-NH2 TFA(327177-34-4 free base)
<p>tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.</p>Fórmula:C42H50F3N7O9Pureza:>99.99%Cor e Forma:SolidPeso molecular:853.9[Sar9,Met(O2)11]-Substance P
CAS:<p>[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.</p>Fórmula:C64H100N18O15SPureza:>99.99%Cor e Forma:SolidPeso molecular:1393.66
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